IL105801A - 7-(2-aminoethyl)-benzothiazolones their preparation and pharmaceutical compositions containing them - Google Patents

7-(2-aminoethyl)-benzothiazolones their preparation and pharmaceutical compositions containing them

Info

Publication number: IL105801A
Authority: IL; Israel
Prior art keywords: pharmaceutical compositions; benzothiazolones; aminoethyl; preparation; compositions containing
Prior art date: 1992-05-27

Application number

IL10580193A

Other languages

English (en)

Other versions

IL105801A0 (en

Inventor

Roger Victor Bonnert

Roger Charles Brown

David Ranulf Cheshire

Francis Ince

Original Assignee

Astra Pharma Prod

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1992-05-27

Filing date

1993-05-25

Publication date

1997-01-10

1993-05-25 Application filed by Astra Pharma Prod filed Critical Astra Pharma Prod

1993-09-22 Publication of IL105801A0 publication Critical patent/IL105801A0/xx

1997-01-10 Publication of IL105801A publication Critical patent/IL105801A/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Pulmonology (AREA)
Ophthalmology & Optometry (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Rheumatology (AREA)
Immunology (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Pain & Pain Management (AREA)
Hospice & Palliative Care (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Cosmetics (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Plural Heterocyclic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Adhesives Or Adhesive Processes (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

IL10580193A 1992-05-27 1993-05-25 7-(2-aminoethyl)-benzothiazolones their preparation and pharmaceutical compositions containing them IL105801A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB929211172A GB9211172D0 (en)	1992-05-27	1992-05-27	Compounds

Publications (2)

Publication Number	Publication Date
IL105801A0 IL105801A0 (en)	1993-09-22
IL105801A true IL105801A (en)	1997-01-10

Family

ID=10716059

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL10580193A IL105801A (en)	1992-05-27	1993-05-25	7-(2-aminoethyl)-benzothiazolones their preparation and pharmaceutical compositions containing them

Country Status (31)

Country	Link
EP (1)	EP0649418B1 (xx)
JP (1)	JP3094452B2 (xx)
KR (1)	KR100279132B1 (xx)
CN (1)	CN1036393C (xx)
AT (1)	ATE172726T1 (xx)
AU (1)	AU675649B2 (xx)
CA (1)	CA2136553C (xx)
CZ (1)	CZ286905B6 (xx)
DE (1)	DE69321835T2 (xx)
DK (1)	DK0649418T3 (xx)
DZ (1)	DZ1694A1 (xx)
ES (1)	ES2123652T3 (xx)
FI (1)	FI945538A (xx)
GB (1)	GB9211172D0 (xx)
HU (2)	HUT71124A (xx)
IL (1)	IL105801A (xx)
LV (1)	LV12443B (xx)
MA (1)	MA22895A1 (xx)
MX (1)	MX9303145A (xx)
MY (1)	MY131193A (xx)
NO (1)	NO304739B1 (xx)
NZ (1)	NZ253190A (xx)
PH (1)	PH31453A (xx)
PL (2)	PL172807B1 (xx)
RU (1)	RU2114108C1 (xx)
SG (1)	SG48068A1 (xx)
SK (1)	SK281282B6 (xx)
TW (1)	TW368501B (xx)
UA (1)	UA27901C2 (xx)
WO (1)	WO1993024473A1 (xx)
ZA (1)	ZA933648B (xx)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TW356468B (en) *	1995-09-15	1999-04-21	Astra Pharma Prod	Benzothiazolone compounds useful as beta2-adrenoreceptor and dopamine DA2 receptor agonists process for preparing same and pharmaceutical compositions containing same
GB9526511D0 (en) *	1995-12-23	1996-02-28	Astra Pharma Prod	Pharmaceutically active compounds
SE9900693D0 (sv) *	1999-02-26	1999-02-26	Astra Pharma Prod	Novel process
SE9902938D0 (sv) *	1999-08-18	1999-08-18	Astra Pharma Prod	Pharmaceutical compositions
SE9902937D0 (sv) *	1999-08-18	1999-08-18	Astra Pharma Prod	Pharmaceutical compositions
SE9902935D0 (sv) *	1999-08-18	1999-08-18	Astra Pharma Prod	Pharmaceutical compositions
SE9902936D0 (sv) *	1999-08-18	1999-08-18	Astra Pharma Prod	Pharmaceutical compositions
DE10063957A1 (de) *	2000-12-20	2002-06-27	Boehringer Ingelheim Pharma	Neue Arzneimittelkompositionen auf der Basis von Anticholinergika und Dopamin-Agonisten
PE20050130A1 (es) *	2002-08-09	2005-03-29	Novartis Ag	Compuestos organicos
GB0218629D0 (en) *	2002-08-09	2002-09-18	Novartis Ag	Organic compounds
ES2329586T3 (es)	2003-11-21	2009-11-27	Theravance, Inc.	Compuestos que tienen actividad agonista del receptor beta2 adrenergico y antagonista del receptor muscarino.
GB0426164D0 (en)	2004-11-29	2004-12-29	Novartis Ag	Organic compounds
TW200738658A (en)	2005-08-09	2007-10-16	Astrazeneca Ab	Novel compounds
TW200738659A (en) *	2005-08-29	2007-10-16	Astrazeneca Ab	Novel compounds
TW200745067A (en)	2006-03-14	2007-12-16	Astrazeneca Ab	Novel compounds
RU2455295C2 (ru) *	2006-12-20	2012-07-10	АстраЗенека AБ	4-ГИДРОКСИ-2-ОКСО-2,3-ДИГИДРО-1,3-БЕНЗОТИАЗОЛ-7-ИЛЬНЫЕ СОЕДИНЕНИЯ ДЛЯ МОДУЛЯЦИИ β2-АДРЕНОРЕЦЕПТОРНОЙ АКТИВНОСТИ
TW200833670A (en)	2006-12-20	2008-08-16	Astrazeneca Ab	Novel compounds 569
GB0702458D0 (en)	2007-02-08	2007-03-21	Astrazeneca Ab	Salts 668
GB0704000D0 (en) *	2007-03-01	2007-04-11	Astrazeneca Ab	Salts 670
JP2011524896A (ja)	2008-06-18	2011-09-08	アストラゼネカ・アクチエボラーグ	呼吸器障害の処置用のベータ２−アドレナリン受容体アゴニストとして作用するベンズオキサジノン誘導体
CN102977050B (zh) *	2012-11-20	2015-04-22	浙江工业大学	一种2-苯并噻唑二甲缩醛和2-苯并噻唑甲醛的合成方法
CN106748930B (zh) *	2016-12-05	2019-03-15	三门峡奥科化工有限公司	3-巯基-1-丙醇的制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4554284A (en) *	1984-09-12	1985-11-19	Smithkline Beckman Corporation	7-(2-Aminoethyl)-1,3-benzthia- or oxa-zol-2(3H)-ones
IE914003A1 (en) *	1990-11-20	1992-05-20	Astra Pharma Prod	Biologically Active Amines

1992
- 1992-05-27 GB GB929211172A patent/GB9211172D0/en active Pending
1993
- 1993-05-05 PH PH46233A patent/PH31453A/en unknown
- 1993-05-25 ZA ZA933648A patent/ZA933648B/xx unknown
- 1993-05-25 IL IL10580193A patent/IL105801A/xx not_active IP Right Cessation
- 1993-05-26 DZ DZ930063A patent/DZ1694A1/fr active
- 1993-05-26 MA MA23194A patent/MA22895A1/fr unknown
- 1993-05-26 TW TW082104181A patent/TW368501B/zh active
- 1993-05-27 EP EP93913203A patent/EP0649418B1/en not_active Expired - Lifetime
- 1993-05-27 PL PL93317714A patent/PL172807B1/pl unknown
- 1993-05-27 CA CA002136553A patent/CA2136553C/en not_active Expired - Fee Related
- 1993-05-27 HU HU9403387A patent/HUT71124A/hu unknown
- 1993-05-27 CN CN93108209A patent/CN1036393C/zh not_active Expired - Fee Related
- 1993-05-27 DK DK93913203T patent/DK0649418T3/da active
- 1993-05-27 SG SG1996006829A patent/SG48068A1/en unknown
- 1993-05-27 DE DE69321835T patent/DE69321835T2/de not_active Expired - Fee Related
- 1993-05-27 NZ NZ253190A patent/NZ253190A/en unknown
- 1993-05-27 MY MYPI93000997A patent/MY131193A/en unknown
- 1993-05-27 SK SK1433-94A patent/SK281282B6/sk unknown
- 1993-05-27 MX MX9303145A patent/MX9303145A/es not_active IP Right Cessation
- 1993-05-27 KR KR1019940704294A patent/KR100279132B1/ko not_active IP Right Cessation
- 1993-05-27 AU AU43343/93A patent/AU675649B2/en not_active Ceased
- 1993-05-27 PL PL93306303A patent/PL172904B1/pl unknown
- 1993-05-27 JP JP06500327A patent/JP3094452B2/ja not_active Expired - Fee Related
- 1993-05-27 ES ES93913203T patent/ES2123652T3/es not_active Expired - Lifetime
- 1993-05-27 UA UA94119105A patent/UA27901C2/uk unknown
- 1993-05-27 RU RU94046093A patent/RU2114108C1/ru active
- 1993-05-27 AT AT93913203T patent/ATE172726T1/de not_active IP Right Cessation
- 1993-05-27 WO PCT/GB1993/001095 patent/WO1993024473A1/en active IP Right Grant
- 1993-05-27 CZ CZ19942916A patent/CZ286905B6/cs not_active IP Right Cessation
1994
- 1994-11-24 NO NO944509A patent/NO304739B1/no not_active IP Right Cessation
- 1994-11-25 FI FI945538A patent/FI945538A/fi unknown
1995
- 1995-06-27 HU HU95P/P00462P patent/HU211947A9/hu unknown
1999
- 1999-10-28 LV LVP-99-152A patent/LV12443B/en unknown

Also Published As

Publication number	Publication date
EP0649418A1 (en)	1995-04-26
LV12443A (en)	2000-03-20
HU211947A9 (en)	1996-01-29
FI945538A0 (fi)	1994-11-25
JPH08503923A (ja)	1996-04-30
MX9303145A (es)	1994-06-30
CZ291694A3 (en)	1995-03-15
IL105801A0 (en)	1993-09-22
EP0649418B1 (en)	1998-10-28
JP3094452B2 (ja)	2000-10-03
CN1036393C (zh)	1997-11-12
GB9211172D0 (en)	1992-07-08
NO944509D0 (no)	1994-11-24
RU2114108C1 (ru)	1998-06-27
RU94046093A (ru)	1996-09-27
FI945538A (fi)	1994-11-25
KR100279132B1 (ko)	2001-01-15
MA22895A1 (fr)	1993-12-31
DK0649418T3 (da)	1999-07-12
CN1085899A (zh)	1994-04-27
SK281282B6 (sk)	2001-02-12
SK143394A3 (en)	1995-06-07
PL172904B1 (pl)	1997-12-31
DZ1694A1 (fr)	2002-02-17
CZ286905B6 (en)	2000-08-16
PL172807B1 (pl)	1997-11-28
MY131193A (en)	2007-07-31
SG48068A1 (en)	1998-04-17
AU675649B2 (en)	1997-02-13
CA2136553A1 (en)	1993-12-09
UA27901C2 (uk)	2000-10-16
ES2123652T3 (es)	1999-01-16
CA2136553C (en)	2000-08-15
TW368501B (en)	1999-09-01
LV12443B (en)	2000-06-20
HU9403387D0 (en)	1995-02-28
PH31453A (en)	1998-11-03
ATE172726T1 (de)	1998-11-15
AU4334393A (en)	1993-12-30
HUT71124A (en)	1995-11-28
NO304739B1 (no)	1999-02-08
WO1993024473A1 (en)	1993-12-09
NZ253190A (en)	1995-12-21
ZA933648B (en)	1993-11-25
DE69321835D1 (de)	1998-12-03
NO944509L (no)	1994-11-24
DE69321835T2 (de)	1999-05-12

Publication	Publication Date	Title
IL105801A0 (en)	1993-09-22	7-(2-aminoethyl)-benzothiazolones,their preparation and pharmaceutical compositions containing them
IL96407A0 (en)	1991-08-16	Diazine derivatives
HUT53368A (en)	1990-10-28	Process for producing pyrazolo-pyridine derivatives and pharmaceutical compositions containing them
IL108602A0 (en)	1994-05-30	N-alkyl-2-substituted atp analogues, their preparation and pharmaceutical compositions containing them
NO304379B1 (no)	1998-12-07	11,21-bisfenyl-19-norpregnan-derivater, anvendelse derav og farmas°ytiske preparater inneholdende slike derivater
IL107287A (en)	2000-09-28	Heterocyclic derivatives process for their preparation and pharmaceutical compositions containing some of them
ATE170852T1 (de)	1998-09-15	Benzolsulfonamid-derivate zur behandlung der blaseninstabilität
CA2030732A1 (fr)	1991-05-25	Nouveaux derives du thiophene, leur procede de preparation et les compositions pharmaceutiques les renfermant
IL108085A0 (en)	1994-04-12	Serotoninergic ergoline derivatives their preparation and pharmacutical compositions containing them
MX9804828A (es)	1998-09-30	Benzotiazolona etanaminas biologicamente activas.
IL81337A (en)	1991-06-30	Heptanoyl-glu-asp-ala-amino acid immunostimulants,process for their preparation and pharmaceutical compositions containing them
DK283984A (da)	1984-12-12	Benzodiazepinderivater og fremgangsmaade til fremstilling deraf
ATE38982T1 (de)	1988-12-15	Guanidinmethylcyclohexancarbonsaeure-derivate, verfahren zur herstellung und pharmazeutische mittel.
ZA994817B (en)	2000-02-02	8H-thieno-[2,3-b]pyrrolizin-8-one compounds, a process for their preparation and pharmaceutical compositions containing them.

Legal Events

Date	Code	Title
1997-07-13	FF	Patent granted
1997-11-20	KB	Patent renewed
1999-10-28	KB	Patent renewed
2004-02-08	RH1	Patent not in force