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ES2123652T3 - 7-(2-aminoetil)-benzotiazolonas. - Google Patents

7-(2-aminoetil)-benzotiazolonas.

Info

Publication number
ES2123652T3
ES2123652T3 ES93913203T ES93913203T ES2123652T3 ES 2123652 T3 ES2123652 T3 ES 2123652T3 ES 93913203 T ES93913203 T ES 93913203T ES 93913203 T ES93913203 T ES 93913203T ES 2123652 T3 ES2123652 T3 ES 2123652T3
Authority
ES
Spain
Prior art keywords
independently represent
benzotiazolonas
aminoetil
membered
halogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES93913203T
Other languages
English (en)
Inventor
Roger Victor Bonnert
Roger Charles Brown
David Ranulf Cheshire
Francis Ince
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Astra Pharmaceuticals Ltd
Astra USA Inc
Original Assignee
Astra Pharmaceuticals Ltd
Astra Pharmaceutical Products Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astra Pharmaceuticals Ltd, Astra Pharmaceutical Products Inc filed Critical Astra Pharmaceuticals Ltd
Application granted granted Critical
Publication of ES2123652T3 publication Critical patent/ES2123652T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/14—Decongestants or antiallergics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Cosmetics (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Adhesives Or Adhesive Processes (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

SE DESCRIBEN COMPUESTOS DE FORMULA (I), DONDE X E Y INDEPENDIENTEMENTE REPRESENTAN -S(O)N 2, P, Q Y R INDEPENDIENTEMENTE REPRESENTAN 2 O 3, Z REPRESENTA FENIL OPCIONALMENTE SUSTITUIDO POR HALOGENO, -OR1, -NO2 O -NR2R3; O UN N, Q O S DE 5 O 6 MIEMBROS, CONTENIENDO HETEROCICLO, Y R1, R2 Y R3 INDEPENDIENTEMENTE REPRESENTAN HIDROGENO O ALQUILO C1-6, Y DERIVADOS FARMACEUTICAMENTE ACEPTABLES DE LOS MISMOS. TAMBIEN SE DESCRIBEN PROCESOS PARA SU PRODUCCION Y COMPOSICIONES FARMACEUTICAS Y METODOS DE TRATAMIENTO QUE IMPLIQUEN SU USO.
ES93913203T 1992-05-27 1993-05-27 7-(2-aminoetil)-benzotiazolonas. Expired - Lifetime ES2123652T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929211172A GB9211172D0 (en) 1992-05-27 1992-05-27 Compounds

Publications (1)

Publication Number Publication Date
ES2123652T3 true ES2123652T3 (es) 1999-01-16

Family

ID=10716059

Family Applications (1)

Application Number Title Priority Date Filing Date
ES93913203T Expired - Lifetime ES2123652T3 (es) 1992-05-27 1993-05-27 7-(2-aminoetil)-benzotiazolonas.

Country Status (31)

Country Link
EP (1) EP0649418B1 (es)
JP (1) JP3094452B2 (es)
KR (1) KR100279132B1 (es)
CN (1) CN1036393C (es)
AT (1) ATE172726T1 (es)
AU (1) AU675649B2 (es)
CA (1) CA2136553C (es)
CZ (1) CZ286905B6 (es)
DE (1) DE69321835T2 (es)
DK (1) DK0649418T3 (es)
DZ (1) DZ1694A1 (es)
ES (1) ES2123652T3 (es)
FI (1) FI945538A0 (es)
GB (1) GB9211172D0 (es)
HU (2) HUT71124A (es)
IL (1) IL105801A (es)
LV (1) LV12443B (es)
MA (1) MA22895A1 (es)
MX (1) MX9303145A (es)
MY (1) MY131193A (es)
NO (1) NO304739B1 (es)
NZ (1) NZ253190A (es)
PH (1) PH31453A (es)
PL (2) PL172904B1 (es)
RU (1) RU2114108C1 (es)
SG (1) SG48068A1 (es)
SK (1) SK281282B6 (es)
TW (1) TW368501B (es)
UA (1) UA27901C2 (es)
WO (1) WO1993024473A1 (es)
ZA (1) ZA933648B (es)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW356468B (en) * 1995-09-15 1999-04-21 Astra Pharma Prod Benzothiazolone compounds useful as beta2-adrenoreceptor and dopamine DA2 receptor agonists process for preparing same and pharmaceutical compositions containing same
GB9526511D0 (en) * 1995-12-23 1996-02-28 Astra Pharma Prod Pharmaceutically active compounds
SE9900693D0 (sv) * 1999-02-26 1999-02-26 Astra Pharma Prod Novel process
SE9902936D0 (sv) * 1999-08-18 1999-08-18 Astra Pharma Prod Pharmaceutical compositions
SE9902935D0 (sv) * 1999-08-18 1999-08-18 Astra Pharma Prod Pharmaceutical compositions
SE9902937D0 (sv) * 1999-08-18 1999-08-18 Astra Pharma Prod Pharmaceutical compositions
SE9902938D0 (sv) * 1999-08-18 1999-08-18 Astra Pharma Prod Pharmaceutical compositions
DE10063957A1 (de) * 2000-12-20 2002-06-27 Boehringer Ingelheim Pharma Neue Arzneimittelkompositionen auf der Basis von Anticholinergika und Dopamin-Agonisten
GB0218629D0 (en) * 2002-08-09 2002-09-18 Novartis Ag Organic compounds
PE20050130A1 (es) * 2002-08-09 2005-03-29 Novartis Ag Compuestos organicos
CN100569760C (zh) 2003-11-21 2009-12-16 施万制药 具有β2肾上腺素能受体激动剂和毒蕈碱性受体拮抗剂活性的化合物
GB0426164D0 (en) 2004-11-29 2004-12-29 Novartis Ag Organic compounds
TW200738658A (en) 2005-08-09 2007-10-16 Astrazeneca Ab Novel compounds
TW200738659A (en) * 2005-08-29 2007-10-16 Astrazeneca Ab Novel compounds
TW200745067A (en) 2006-03-14 2007-12-16 Astrazeneca Ab Novel compounds
TW200833670A (en) 2006-12-20 2008-08-16 Astrazeneca Ab Novel compounds 569
RU2455295C2 (ru) * 2006-12-20 2012-07-10 АстраЗенека AБ 4-ГИДРОКСИ-2-ОКСО-2,3-ДИГИДРО-1,3-БЕНЗОТИАЗОЛ-7-ИЛЬНЫЕ СОЕДИНЕНИЯ ДЛЯ МОДУЛЯЦИИ β2-АДРЕНОРЕЦЕПТОРНОЙ АКТИВНОСТИ
GB0702458D0 (en) 2007-02-08 2007-03-21 Astrazeneca Ab Salts 668
GB0704000D0 (en) * 2007-03-01 2007-04-11 Astrazeneca Ab Salts 670
EA201001747A1 (ru) 2008-06-18 2011-08-30 Астразенека Аб Бензоксазиноновые производные, действующие в качестве агониста бета-2-адренорецептора, для лечения респираторных расстройств
CN102977050B (zh) * 2012-11-20 2015-04-22 浙江工业大学 一种2-苯并噻唑二甲缩醛和2-苯并噻唑甲醛的合成方法
CN106748930B (zh) * 2016-12-05 2019-03-15 三门峡奥科化工有限公司 3-巯基-1-丙醇的制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4554284A (en) * 1984-09-12 1985-11-19 Smithkline Beckman Corporation 7-(2-Aminoethyl)-1,3-benzthia- or oxa-zol-2(3H)-ones
IE914003A1 (en) * 1990-11-20 1992-05-20 Astra Pharma Prod Biologically Active Amines

Also Published As

Publication number Publication date
CA2136553C (en) 2000-08-15
UA27901C2 (uk) 2000-10-16
CN1085899A (zh) 1994-04-27
NO944509D0 (no) 1994-11-24
KR100279132B1 (ko) 2001-01-15
PH31453A (en) 1998-11-03
SK143394A3 (en) 1995-06-07
SK281282B6 (sk) 2001-02-12
AU675649B2 (en) 1997-02-13
HU9403387D0 (en) 1995-02-28
MX9303145A (es) 1994-06-30
MA22895A1 (fr) 1993-12-31
DE69321835D1 (de) 1998-12-03
EP0649418B1 (en) 1998-10-28
NO304739B1 (no) 1999-02-08
HUT71124A (en) 1995-11-28
FI945538A (fi) 1994-11-25
AU4334393A (en) 1993-12-30
NO944509L (no) 1994-11-24
IL105801A (en) 1997-01-10
DK0649418T3 (da) 1999-07-12
SG48068A1 (en) 1998-04-17
CZ291694A3 (en) 1995-03-15
RU2114108C1 (ru) 1998-06-27
FI945538A0 (fi) 1994-11-25
CA2136553A1 (en) 1993-12-09
JP3094452B2 (ja) 2000-10-03
WO1993024473A1 (en) 1993-12-09
EP0649418A1 (en) 1995-04-26
HU211947A9 (en) 1996-01-29
IL105801A0 (en) 1993-09-22
CZ286905B6 (en) 2000-08-16
TW368501B (en) 1999-09-01
CN1036393C (zh) 1997-11-12
PL172807B1 (pl) 1997-11-28
ZA933648B (en) 1993-11-25
MY131193A (en) 2007-07-31
PL172904B1 (pl) 1997-12-31
DZ1694A1 (fr) 2002-02-17
ATE172726T1 (de) 1998-11-15
LV12443A (en) 2000-03-20
GB9211172D0 (en) 1992-07-08
JPH08503923A (ja) 1996-04-30
LV12443B (en) 2000-06-20
DE69321835T2 (de) 1999-05-12
RU94046093A (ru) 1996-09-27
NZ253190A (en) 1995-12-21

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