SI3359541T1 - N-sulfonirani pirazolo(3,4 b)piridin-6-karboksamidi in postopki uporabe - Google Patents

N-sulfonirani pirazolo(3,4 b)piridin-6-karboksamidi in postopki uporabe

Info

Publication number: SI3359541T1
Authority: SI; Slovenia
Prior art keywords: sulfonylated; carboxamides; pyrazolo; pyridin; sulfonylated pyrazolo
Prior art date: 2015-10-09

Application number

SI201630965T

Other languages

English (en)

Inventor

Rhalid Akkari

Luke Jonathan Alvey

Xavier Marie Bock

Brian S. Brown

Pieter Isabelle Roger Claes

Marlon D. Cowart

Lemos Elsa De

Nicolas Desroy

Beranger Duthion

Gregory A. Gfesser

Romain Luc Marie Gosmini

Christopher Gaetan Housseman

Koen Karel Jansen

Jianguo Ji

Philip R. Kym

Jean-Michel Lefrancois

Oscar Mammoliti

Christel Jeanne Marie Menet

Nuria Merayo Merayo

Gregory John Robert Newsome

Adeline Marie Elise Palisse

Sachin V. Patel

Mathieu Rafael Pizzonero

Anurupa Shrestha

Elizabeth C. Swift

Der Plas Steven Emiel Van

Xueqing Wang

Blieck Ann De

Original Assignee

Abbvie Overseas S.A R.L.

Galapagos Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2015-10-09

Filing date

2016-10-07

Publication date

2021-01-29

2016-10-07 Application filed by Abbvie Overseas S.A R.L., Galapagos Nv filed Critical Abbvie Overseas S.A R.L.

2021-01-29 Publication of SI3359541T1 publication Critical patent/SI3359541T1/sl

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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- C07D—HETEROCYCLIC COMPOUNDS
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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Epidemiology (AREA)
Neurology (AREA)
Pulmonology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Physical Education & Sports Medicine (AREA)
Urology & Nephrology (AREA)
Diabetes (AREA)
Immunology (AREA)
Orthopedic Medicine & Surgery (AREA)
Endocrinology (AREA)
Hematology (AREA)
Hospice & Palliative Care (AREA)
Psychiatry (AREA)
Psychology (AREA)
Ophthalmology & Optometry (AREA)
Reproductive Health (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

SI201630965T 2015-10-09 2016-10-07 N-sulfonirani pirazolo(3,4 b)piridin-6-karboksamidi in postopki uporabe SI3359541T1 (sl)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US201562239647P	2015-10-09	2015-10-09
US201662309794P	2016-03-17	2016-03-17
PCT/IB2016/056029 WO2017060874A1 (en)	2015-10-09	2016-10-07	N-sulfonylated pyrazolo[3,4-b]pyridin-6-carboxamides and method of use
EP16788232.3A EP3359541B1 (en)	2015-10-09	2016-10-07	N-sulfonylated pyrazolo[3,4-b]pyridin-6-carboxamides and method of use

Publications (1)

Publication Number	Publication Date
SI3359541T1 true SI3359541T1 (sl)	2021-01-29

Family

ID=57209654

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SI201630965T SI3359541T1 (sl)	2015-10-09	2016-10-07	N-sulfonirani pirazolo(3,4 b)piridin-6-karboksamidi in postopki uporabe

Country Status (32)

Country	Link
US (4)	US9890158B2 (sl)
EP (1)	EP3359541B1 (sl)
JP (1)	JP6779992B2 (sl)
KR (1)	KR20180083323A (sl)
CN (1)	CN108513574B (sl)
AU (1)	AU2016333856C1 (sl)
BR (1)	BR112018007161B1 (sl)
CA (1)	CA3001096A1 (sl)
CL (1)	CL2018000911A1 (sl)
CO (1)	CO2018003716A2 (sl)
CR (1)	CR20180215A (sl)
CY (1)	CY1123545T1 (sl)
DK (1)	DK3359541T3 (sl)
EC (1)	ECSP18032223A (sl)
ES (1)	ES2829636T3 (sl)
HR (1)	HRP20201618T1 (sl)
HU (1)	HUE051067T2 (sl)
IL (1)	IL258553A (sl)
LT (1)	LT3359541T (sl)
MX (1)	MX2018004359A (sl)
NZ (1)	NZ741223A (sl)
PE (1)	PE20181348A1 (sl)
PH (1)	PH12018500765B1 (sl)
PL (1)	PL3359541T3 (sl)
PT (1)	PT3359541T (sl)
RU (1)	RU2724345C2 (sl)
SG (1)	SG11201802932VA (sl)
SI (1)	SI3359541T1 (sl)
TW (1)	TWI720032B (sl)
UY (1)	UY36943A (sl)
WO (1)	WO2017060874A1 (sl)
ZA (1)	ZA201802976B (sl)

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Publication number	Publication date
US20190330207A1 (en)	2019-10-31
CN108513574A (zh)	2018-09-07
JP6779992B2 (ja)	2020-11-04
PH12018500765A1 (en)	2018-10-01
ZA201802976B (en)	2019-07-31
TW201722948A (zh)	2017-07-01
US20180105522A1 (en)	2018-04-19
US9890158B2 (en)	2018-02-13
AU2016333856B2 (en)	2021-05-20
NZ741223A (en)	2023-03-31
JP2018529743A (ja)	2018-10-11
BR112018007161A2 (pt)	2018-10-30
CR20180215A (es)	2018-06-05
BR112018007161B1 (pt)	2024-01-16
EP3359541B1 (en)	2020-08-05
LT3359541T (lt)	2020-11-25
EP3359541A1 (en)	2018-08-15
US20170101405A1 (en)	2017-04-13
US20190202823A1 (en)	2019-07-04
MX2018004359A (es)	2018-05-01
CA3001096A1 (en)	2017-04-13
PT3359541T (pt)	2020-11-11
CY1123545T1 (el)	2022-03-24
HUE051067T2 (hu)	2021-01-28
CL2018000911A1 (es)	2018-08-24
UY36943A (es)	2017-05-31
PE20181348A1 (es)	2018-08-22
RU2018115722A (ru)	2019-11-12
PH12018500765B1 (en)	2018-10-01
RU2724345C2 (ru)	2020-06-23
CO2018003716A2 (es)	2018-07-19
RU2018115722A3 (sl)	2020-02-18
AU2016333856C1 (en)	2021-12-09
PL3359541T3 (pl)	2021-01-11
HRP20201618T1 (hr)	2020-12-25
DK3359541T3 (da)	2020-11-09
ECSP18032223A (es)	2018-05-31
CN108513574B (zh)	2021-01-05
TWI720032B (zh)	2021-03-01
WO2017060874A1 (en)	2017-04-13
KR20180083323A (ko)	2018-07-20
ES2829636T3 (es)	2021-06-01
AU2016333856A1 (en)	2018-04-26
US10259810B2 (en)	2019-04-16
SG11201802932VA (en)	2018-05-30
US10647717B2 (en)	2020-05-12
IL258553A (en)	2018-05-31

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