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IT1269511B - Derivati di acidi ammino-solfonici , loro impiego nella sintesi di pseudopeptidi e procedimento per la loro preparazione - Google Patents

Derivati di acidi ammino-solfonici , loro impiego nella sintesi di pseudopeptidi e procedimento per la loro preparazione

Info

Publication number
IT1269511B
IT1269511B ITMI940989A ITMI940989A IT1269511B IT 1269511 B IT1269511 B IT 1269511B IT MI940989 A ITMI940989 A IT MI940989A IT MI940989 A ITMI940989 A IT MI940989A IT 1269511 B IT1269511 B IT 1269511B
Authority
IT
Italy
Prior art keywords
pseudopeptides
synthesis
amino
preparation
procedure
Prior art date
Application number
ITMI940989A
Other languages
English (en)
Inventor
Cesare Gennari
Donatella Potenza
Barbara Salom
Original Assignee
Univ Degli Studi Milano
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Degli Studi Milano filed Critical Univ Degli Studi Milano
Publication of ITMI940989A0 publication Critical patent/ITMI940989A0/it
Priority to ITMI940989A priority Critical patent/IT1269511B/it
Priority to AT95919441T priority patent/ATE174329T1/de
Priority to PCT/EP1995/001788 priority patent/WO1995031433A1/en
Priority to CN95193138A priority patent/CN1148847A/zh
Priority to AU25268/95A priority patent/AU691292B2/en
Priority to ES95919441T priority patent/ES2125617T3/es
Priority to PL95317258A priority patent/PL317258A1/xx
Priority to CA002189896A priority patent/CA2189896A1/en
Priority to JP52934895A priority patent/JP4023554B2/ja
Priority to EP95919441A priority patent/EP0759902B1/en
Priority to NZ285763A priority patent/NZ285763A/en
Priority to DE69506540T priority patent/DE69506540T2/de
Priority to US08/737,379 priority patent/US5869725A/en
Priority to KR1019960706501A priority patent/KR970703307A/ko
Priority to HU9603128A priority patent/HUT76483A/hu
Publication of ITMI940989A1 publication Critical patent/ITMI940989A1/it
Priority to MXPA/A/1996/005426A priority patent/MXPA96005426A/xx
Priority to NO964861A priority patent/NO964861L/no
Priority to FI964582A priority patent/FI964582A0/fi
Application granted granted Critical
Publication of IT1269511B publication Critical patent/IT1269511B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/63—Esters of sulfonic acids
    • C07C309/64—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms
    • C07C309/69—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms of a carbon skeleton substituted by nitrogen atoms, not being part of nitro or nitroso groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/45—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups at least one of the singly-bound nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom, e.g. N-acylaminosulfonamides
    • C07C311/47—Y being a hetero atom
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrrole Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Prodotti derivati di acidi solfonici gamma - ammino - alfa, beta insaturi, procedimento per la loro preparazione e loro impiego nella sintesi di pseudopeptidi caratterizzati dalla presenza di almeno un legame di tipo solfonammidico coniugato ad un doppio legame.
ITMI940989A 1994-05-17 1994-05-17 Derivati di acidi ammino-solfonici , loro impiego nella sintesi di pseudopeptidi e procedimento per la loro preparazione IT1269511B (it)

Priority Applications (18)

Application Number Priority Date Filing Date Title
ITMI940989A IT1269511B (it) 1994-05-17 1994-05-17 Derivati di acidi ammino-solfonici , loro impiego nella sintesi di pseudopeptidi e procedimento per la loro preparazione
JP52934895A JP4023554B2 (ja) 1994-05-17 1995-05-11 アミノスルホン酸の誘導体、プソイドペプチドの合成における同誘導体の利用、およびその製造法
NZ285763A NZ285763A (en) 1994-05-17 1995-05-11 Aminosulphonic acid derivatives; their preparation; use in preparing pseudopeptides; pseudopeptides
CN95193138A CN1148847A (zh) 1994-05-17 1995-05-11 氨基磺酸衍生物，它们在合成假肽中的应用及制备方法
AU25268/95A AU691292B2 (en) 1994-05-17 1995-05-11 Derivatives of aminosulfonic acids, utilization of the same in the synthesis of pseudopeptides and process for their preparation
ES95919441T ES2125617T3 (es) 1994-05-17 1995-05-11 Derivados de acidos aminosulfonicos, utilizacion de los mismos en la sintesis de pseudopeptidos y procedimiento para su preparacion.
PL95317258A PL317258A1 (en) 1994-05-17 1995-05-11 Derivatives of aminosulphonic acids, their application in synthesising pseudopeptides and method of obtaining them
CA002189896A CA2189896A1 (en) 1994-05-17 1995-05-11 Derivatives of aminosulfonic acids, utilization of the same in the synthesis of pseudopeptides and process for their preparation
AT95919441T ATE174329T1 (de) 1994-05-17 1995-05-11 Aminosulfonsäurederivate, ihre verwendung zur herstellung von pseudopeptiden und verfahren zu ihrer herstellung
EP95919441A EP0759902B1 (en) 1994-05-17 1995-05-11 Derivatives of aminosulfonic acids, utilization of the same in the synthesis of pseudopeptides and process for their preparation
PCT/EP1995/001788 WO1995031433A1 (en) 1994-05-17 1995-05-11 Derivatives of aminosulfonic acids, utilization of the same in the synthesis of pseudopeptides and process for their preparation
DE69506540T DE69506540T2 (de) 1994-05-17 1995-05-11 Aminosulfonsäurederivate, ihre verwendung zur herstellung von pseudopeptiden und verfahren zu ihrer herstellung
US08/737,379 US5869725A (en) 1994-05-17 1995-05-11 Derivatives of aminosulfonic acids, utilization of the same in the synthesis of pseudopeptides and process for their preparation
KR1019960706501A KR970703307A (ko) 1994-05-17 1995-05-11 아미노술폰산 유도체, 의사펩티드 합성으로의 용도 및 이들의 제조 방법(derivatives of aminosulfonic acids, utilization of the same in the synthesis of pseudopeptides and process for their preparation)
HU9603128A HUT76483A (en) 1994-05-17 1995-05-11 Derivatives of gamma-amino-alfa,beta-alkenyl sulfonic acids, utilization of the same in the synthesis of pseudopeptides and process for their preparation
MXPA/A/1996/005426A MXPA96005426A (en) 1994-05-17 1996-11-07 Derivatives of aminosulphonic acids, use of them in the synthesis of pseudopeptides and procedure for preparation
NO964861A NO964861L (no) 1994-05-17 1996-11-15 Derivater av aminosulfonsyrer, fremgangsmåte for fremstilling av disse samt deres anvendelse ved syntese av pseudopeptider
FI964582A FI964582A0 (fi) 1994-05-17 1996-11-15 Aminosulfonihappojohdannaisia, niiden käyttö pseudopeptidisynteesissä ja menetelmä niiden valmistamiseksi

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ITMI940989A IT1269511B (it) 1994-05-17 1994-05-17 Derivati di acidi ammino-solfonici , loro impiego nella sintesi di pseudopeptidi e procedimento per la loro preparazione

Publications (3)

Publication Number Publication Date
ITMI940989A0 ITMI940989A0 (it) 1994-05-17
ITMI940989A1 ITMI940989A1 (it) 1995-11-17
IT1269511B true IT1269511B (it) 1997-04-01

Family

ID=11368917

Family Applications (1)

Application Number Title Priority Date Filing Date
ITMI940989A IT1269511B (it) 1994-05-17 1994-05-17 Derivati di acidi ammino-solfonici , loro impiego nella sintesi di pseudopeptidi e procedimento per la loro preparazione

Country Status (17)

Country Link
US (1) US5869725A (it)
EP (1) EP0759902B1 (it)
JP (1) JP4023554B2 (it)
KR (1) KR970703307A (it)
CN (1) CN1148847A (it)
AT (1) ATE174329T1 (it)
AU (1) AU691292B2 (it)
CA (1) CA2189896A1 (it)
DE (1) DE69506540T2 (it)
ES (1) ES2125617T3 (it)
FI (1) FI964582A0 (it)
HU (1) HUT76483A (it)
IT (1) IT1269511B (it)
NO (1) NO964861L (it)
NZ (1) NZ285763A (it)
PL (1) PL317258A1 (it)
WO (1) WO1995031433A1 (it)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6214799B1 (en) 1996-05-14 2001-04-10 Agouron Pharmaceuticals, Inc. Antipicornaviral compounds and methods for their use and preparation
US6331554B1 (en) 1997-03-28 2001-12-18 Agouron Pharmaceuticals, Inc. Antipicornaviral compounds, compositions containing them, and methods for their use
US6020371A (en) * 1997-03-28 2000-02-01 Agouron Pharmaceuticals, Inc. Antipicornaviral compounds compositions containing them and methods for their use
US5962487A (en) * 1997-12-16 1999-10-05 Agouron Pharmaceuticals, Inc. Antipicornaviral compounds and methods for their use and preparation
EE200000621A (et) 1998-04-30 2002-06-17 Agouron Pharmaceuticals, Inc. Pikornaviirusevastased ühendid, nende valmistamine ja kasutamine
KR20010052503A (ko) 1998-06-03 2001-06-25 다니엘 피. 맥컬럼 Ｎ-헤테로사이클릭 카복실산 또는 카복실산 등입체의ｎ-결합된 설폰아미드
US6358928B1 (en) 1999-11-22 2002-03-19 Enzyme Systems Products Peptidyl sulfonyl imidazolides as selective inhibitors of serine proteases
PE20020157A1 (es) 1999-12-03 2002-02-22 Agouron Pharma Compuestos derivados de piridona como inhibidores de proteasas de picornaviral 3c, composiciones, sus usos farmaceuticos y materiales para su sintesis
PA8515201A1 (es) 2000-04-14 2002-10-24 Agouron Pharma Compuestos y composiciones antipicornavirales; sus usos farmaceuticos y los materiales para su sintesis
WO2001096297A2 (en) 2000-06-14 2001-12-20 Agouron Pharmaceuticals, Inc. Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
JPWO2002074299A1 (ja) * 2000-12-27 2004-07-08 味の素株式会社 ＴＮＦα産生抑制剤

Also Published As

Publication number Publication date
DE69506540T2 (de) 1999-06-02
US5869725A (en) 1999-02-09
AU2526895A (en) 1995-12-05
JP4023554B2 (ja) 2007-12-19
HU9603128D0 (en) 1997-01-28
HUT76483A (en) 1997-09-29
AU691292B2 (en) 1998-05-14
JPH10500123A (ja) 1998-01-06
FI964582A (fi) 1996-11-15
KR970703307A (ko) 1997-07-03
ATE174329T1 (de) 1998-12-15
NZ285763A (en) 1997-10-24
ITMI940989A1 (it) 1995-11-17
EP0759902B1 (en) 1998-12-09
FI964582A0 (fi) 1996-11-15
NO964861D0 (no) 1996-11-15
MX9605426A (es) 1998-05-31
WO1995031433A1 (en) 1995-11-23
CA2189896A1 (en) 1995-11-23
CN1148847A (zh) 1997-04-30
NO964861L (no) 1997-01-16
PL317258A1 (en) 1997-04-01
ITMI940989A0 (it) 1994-05-17
EP0759902A1 (en) 1997-03-05
DE69506540D1 (de) 1999-01-21
ES2125617T3 (es) 1999-03-01

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Legal Events

Date Code Title Description
0001 Granted
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19970418