ES2125617T3 - Derivados de acidos aminosulfonicos, utilizacion de los mismos en la sintesis de pseudopeptidos y procedimiento para su preparacion. - Google Patents
Derivados de acidos aminosulfonicos, utilizacion de los mismos en la sintesis de pseudopeptidos y procedimiento para su preparacion.Info
- Publication number
- ES2125617T3 ES2125617T3 ES95919441T ES95919441T ES2125617T3 ES 2125617 T3 ES2125617 T3 ES 2125617T3 ES 95919441 T ES95919441 T ES 95919441T ES 95919441 T ES95919441 T ES 95919441T ES 2125617 T3 ES2125617 T3 ES 2125617T3
- Authority
- ES
- Spain
- Prior art keywords
- sub
- synthesis
- derivatives
- preparation
- same
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 239000002253 acid Substances 0.000 title abstract 2
- 150000007513 acids Chemical class 0.000 title abstract 2
- 230000015572 biosynthetic process Effects 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 238000002360 preparation method Methods 0.000 title abstract 2
- 238000003786 synthesis reaction Methods 0.000 title abstract 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical class [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- -1 AMINO GROUP Chemical group 0.000 abstract 1
- 150000001412 amines Chemical class 0.000 abstract 1
- 239000012634 fragment Substances 0.000 abstract 1
- 230000001681 protective effect Effects 0.000 abstract 1
- 150000003839 salts Chemical group 0.000 abstract 1
- 229940124530 sulfonamide Drugs 0.000 abstract 1
- 150000003456 sulfonamides Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
- C07C309/63—Esters of sulfonic acids
- C07C309/64—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms
- C07C309/69—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms of a carbon skeleton substituted by nitrogen atoms, not being part of nitro or nitroso groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/45—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups at least one of the singly-bound nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom, e.g. N-acylaminosulfonamides
- C07C311/47—Y being a hetero atom
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyrrole Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
DERIVADOS DE ACIDOS SULFONICOS GAMMA-AMINO-ALFA-BETAINSATURADOS DE FORMULA (I), DONDE R SE ELIGE ENTRE HIDROGENO, FRAGMENTOS CORRESPONDIENTES A CADENAS LATERALES DE AMINOACIDOS NATURALES, SUSTITUIDOS O NO SUSTITUIDOS: CADENAS DE ALQUILO LINEALES, RAMIFICADOS O CICLICOS; CADENAS DE ARILALQUILO; GRUPOS ARILO O HETEROAROMATICOS; Y INDICA HIDROGENO, INCLUYENDO POSIBLES FORMAS SALINAS DE LA CORRESPONDIENTE AMINA; O CUALQUIER GRUPO PROTECTOR NORMALMENTE UTILIZADO PARA LA PROTECCION DEL GRUPO AMINO; X INDICA CL, OH, OCH{SUB,2}CH{SUB,3}, OCH{SUB,3}, ONBU{SUB,4}, NHCH{SUB,2}PH; PROCESO PARA LA PREPARACION DE LOS MISMOS Y SU UTILIZACION EN LA SINTESIS DE PSEUDOPEPTIDOS CARACTERIZADA POR LA PRESENCIA DE AL MENOS UN ENLACE DE TIPO SULFONAMIDA CONJUGADA CON UN DOBLE ENLACE.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ITMI940989A IT1269511B (it) | 1994-05-17 | 1994-05-17 | Derivati di acidi ammino-solfonici , loro impiego nella sintesi di pseudopeptidi e procedimento per la loro preparazione |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2125617T3 true ES2125617T3 (es) | 1999-03-01 |
Family
ID=11368917
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES95919441T Expired - Lifetime ES2125617T3 (es) | 1994-05-17 | 1995-05-11 | Derivados de acidos aminosulfonicos, utilizacion de los mismos en la sintesis de pseudopeptidos y procedimiento para su preparacion. |
Country Status (17)
Country | Link |
---|---|
US (1) | US5869725A (es) |
EP (1) | EP0759902B1 (es) |
JP (1) | JP4023554B2 (es) |
KR (1) | KR970703307A (es) |
CN (1) | CN1148847A (es) |
AT (1) | ATE174329T1 (es) |
AU (1) | AU691292B2 (es) |
CA (1) | CA2189896A1 (es) |
DE (1) | DE69506540T2 (es) |
ES (1) | ES2125617T3 (es) |
FI (1) | FI964582A0 (es) |
HU (1) | HUT76483A (es) |
IT (1) | IT1269511B (es) |
NO (1) | NO964861L (es) |
NZ (1) | NZ285763A (es) |
PL (1) | PL317258A1 (es) |
WO (1) | WO1995031433A1 (es) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6214799B1 (en) | 1996-05-14 | 2001-04-10 | Agouron Pharmaceuticals, Inc. | Antipicornaviral compounds and methods for their use and preparation |
US6020371A (en) * | 1997-03-28 | 2000-02-01 | Agouron Pharmaceuticals, Inc. | Antipicornaviral compounds compositions containing them and methods for their use |
US6331554B1 (en) | 1997-03-28 | 2001-12-18 | Agouron Pharmaceuticals, Inc. | Antipicornaviral compounds, compositions containing them, and methods for their use |
US5962487A (en) * | 1997-12-16 | 1999-10-05 | Agouron Pharmaceuticals, Inc. | Antipicornaviral compounds and methods for their use and preparation |
BR9910573A (pt) | 1998-04-30 | 2001-01-16 | Agouron Pharma | Compostos antipicornavirais, preparação e uso dos mesmos |
WO1999062880A1 (en) | 1998-06-03 | 1999-12-09 | Gpi Nil Holdings, Inc. | N-linked sulfonamides of n-heterocyclic carboxylic acids or carboxylic acid isosteres |
US6358928B1 (en) | 1999-11-22 | 2002-03-19 | Enzyme Systems Products | Peptidyl sulfonyl imidazolides as selective inhibitors of serine proteases |
PA8507801A1 (es) | 1999-12-03 | 2002-08-26 | Agouron Pharma | Compuestos y composiciones antipicornavirales, sus usos farmaceuticos y los materiales para su sintesis |
PA8515201A1 (es) | 2000-04-14 | 2002-10-24 | Agouron Pharma | Compuestos y composiciones antipicornavirales; sus usos farmaceuticos y los materiales para su sintesis |
IL153431A0 (en) | 2000-06-14 | 2003-07-06 | Agouron Pharma | Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis |
JPWO2002074299A1 (ja) * | 2000-12-27 | 2004-07-08 | 味の素株式会社 | TNFα産生抑制剤 |
-
1994
- 1994-05-17 IT ITMI940989A patent/IT1269511B/it active IP Right Grant
-
1995
- 1995-05-11 ES ES95919441T patent/ES2125617T3/es not_active Expired - Lifetime
- 1995-05-11 CN CN95193138A patent/CN1148847A/zh active Pending
- 1995-05-11 DE DE69506540T patent/DE69506540T2/de not_active Expired - Fee Related
- 1995-05-11 WO PCT/EP1995/001788 patent/WO1995031433A1/en active IP Right Grant
- 1995-05-11 JP JP52934895A patent/JP4023554B2/ja not_active Expired - Fee Related
- 1995-05-11 AT AT95919441T patent/ATE174329T1/de not_active IP Right Cessation
- 1995-05-11 CA CA002189896A patent/CA2189896A1/en not_active Abandoned
- 1995-05-11 KR KR1019960706501A patent/KR970703307A/ko not_active Application Discontinuation
- 1995-05-11 PL PL95317258A patent/PL317258A1/xx unknown
- 1995-05-11 EP EP95919441A patent/EP0759902B1/en not_active Expired - Lifetime
- 1995-05-11 US US08/737,379 patent/US5869725A/en not_active Expired - Fee Related
- 1995-05-11 NZ NZ285763A patent/NZ285763A/en unknown
- 1995-05-11 AU AU25268/95A patent/AU691292B2/en not_active Expired - Fee Related
- 1995-05-11 HU HU9603128A patent/HUT76483A/hu unknown
-
1996
- 1996-11-15 FI FI964582A patent/FI964582A0/fi not_active Application Discontinuation
- 1996-11-15 NO NO964861A patent/NO964861L/no unknown
Also Published As
Publication number | Publication date |
---|---|
MX9605426A (es) | 1998-05-31 |
ITMI940989A0 (it) | 1994-05-17 |
NO964861L (no) | 1997-01-16 |
EP0759902B1 (en) | 1998-12-09 |
HU9603128D0 (en) | 1997-01-28 |
US5869725A (en) | 1999-02-09 |
KR970703307A (ko) | 1997-07-03 |
ATE174329T1 (de) | 1998-12-15 |
JPH10500123A (ja) | 1998-01-06 |
AU2526895A (en) | 1995-12-05 |
AU691292B2 (en) | 1998-05-14 |
DE69506540T2 (de) | 1999-06-02 |
FI964582A (fi) | 1996-11-15 |
NO964861D0 (no) | 1996-11-15 |
DE69506540D1 (de) | 1999-01-21 |
IT1269511B (it) | 1997-04-01 |
NZ285763A (en) | 1997-10-24 |
JP4023554B2 (ja) | 2007-12-19 |
WO1995031433A1 (en) | 1995-11-23 |
CA2189896A1 (en) | 1995-11-23 |
ITMI940989A1 (it) | 1995-11-17 |
EP0759902A1 (en) | 1997-03-05 |
HUT76483A (en) | 1997-09-29 |
CN1148847A (zh) | 1997-04-30 |
PL317258A1 (en) | 1997-04-01 |
FI964582A0 (fi) | 1996-11-15 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG2A | Definitive protection |
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