CS207612B2 - Method of making the trans-5-aryl-2,3,4a,5,9b-hexa-hydro-1h-pyrido 4,3-b indoles - Google Patents

Method of making the trans-5-aryl-2,3,4a,5,9b-hexa-hydro-1h-pyrido 4,3-b indoles Download PDF

Info

Publication number: CS207612B2
Authority: CS; Czechoslovakia
Prior art keywords: acid; fluorophenyl; trans; pyrido; compounds
Prior art date: 1977-05-23

Application number

CS783239A

Other languages

Czech (cs)

English (en)

Inventor

Willard Mck Welch

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-05-23

Filing date

1978-05-18

Publication date

1981-08-31

1978-05-18 Application filed by Pfizer filed Critical Pfizer

1979-09-14 Priority to CS796223A priority Critical patent/CS207615B2/cs

1979-09-14 Priority to CS796221A priority patent/CS207613B2/cs

1979-09-14 Priority to CS796222A priority patent/CS207614B2/cs

1981-08-31 Publication of CS207612B2 publication Critical patent/CS207612B2/cs

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Neurosurgery (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Psychiatry (AREA)
Anesthesiology (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

CS783239A 1977-05-23 1978-05-18 Method of making the trans-5-aryl-2,3,4a,5,9b-hexa-hydro-1h-pyrido 4,3-b indoles CS207612B2 (en)

Priority Applications (3)

Application Number	Priority Date	Filing Date	Title
CS796223A CS207615B2 (cs)	1977-05-23	1979-09-14	Způsob výroby 4a,9b-trans-hexahydro;-karbolinových derivátů
CS796221A CS207613B2 (cs)	1977-05-23	1979-09-14	Způsob výroby trans-5-aryl-2,3,4,4a,5,9b-hexahydro-lH-pyrido[4,3-b]- indolů
CS796222A CS207614B2 (cs)	1977-05-23	1979-09-14	Způsob výroby 4a, 9b-trans-hexahydro-/*-karbolinových derivátů

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US79939277A	1977-05-23	1977-05-23

Publications (1)

Publication Number	Publication Date
CS207612B2 true CS207612B2 (en)	1981-08-31

Family

ID=25175793

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CS783239A CS207612B2 (en)	1977-05-23	1978-05-18	Method of making the trans-5-aryl-2,3,4a,5,9b-hexa-hydro-1h-pyrido 4,3-b indoles

Country Status (31)

Country	Link
JP (1)	JPS53144600A (ru)
AR (2)	AR217688A1 (ru)
AT (1)	AT368995B (ru)
AU (1)	AU499618B1 (ru)
BE (1)	BE867249A (ru)
CA (1)	CA1094071A (ru)
CH (1)	CH634321A5 (ru)
CS (1)	CS207612B2 (ru)
DD (4)	DD145536A5 (ru)
DE (1)	DE2822465C2 (ru)
DK (1)	DK226678A (ru)
EG (1)	EG13590A (ru)
FI (1)	FI63402C (ru)
FR (1)	FR2392023A1 (ru)
GB (1)	GB1586655A (ru)
GR (1)	GR69985B (ru)
HU (3)	HU185009B (ru)
IE (1)	IE46975B1 (ru)
IL (1)	IL54755A (ru)
IT (1)	IT1096307B (ru)
LU (1)	LU79684A1 (ru)
NL (1)	NL7804210A (ru)
NO (2)	NO150204C (ru)
NZ (1)	NZ187333A (ru)
PH (1)	PH13756A (ru)
PL (5)	PL116944B1 (ru)
PT (1)	PT68058B (ru)
SE (2)	SE441448B (ru)
SU (4)	SU873883A3 (ru)
YU (4)	YU91478A (ru)
ZA (1)	ZA782918B (ru)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4224329A (en) *	1979-01-23	1980-09-23	Pfizer Inc.	2-Substituted-trans-5-aryl-2,3,4,4a,5,9b-hexahydro-1H-pyrido[4,3-b]indoles
US4451655A (en) *	1982-05-17	1984-05-29	Pfizer Inc.	Process for preparing carboline derivatives and compounds used in their preparation
RU2106864C1 (ru) *	1995-10-23	1998-03-20	Николай Серафимович Зефиров	Средство для лечения болезни альцгеймера
SE9604786D0 (sv)	1996-12-20	1996-12-20	Astra Pharma Inc	New compounds
US6974825B1 (en)	1996-12-20	2005-12-13	Astrazeneca Canada Inc.	Compounds with analgesic effect
SE9904675D0 (sv)	1999-12-20	1999-12-20	Astra Pharma Inc	Novel compounds
SE0101769D0 (sv)	2001-05-18	2001-05-18	Astrazeneca Ab	Novel compounds
SE0101771D0 (sv)	2001-05-18	2001-05-18	Astrazeneca Ab	Novel compounds
SE0101773D0 (sv)	2001-05-18	2001-05-18	Astrazeneca Ab	Novel compounds
SE0101770D0 (sv)	2001-05-18	2001-05-18	Astrazeneca Ab	Novel compounds
DE20204239U1 (de)	2002-03-16	2002-05-29	Funke Kunststoffe GmbH, 48324 Sendenhorst	Universal-Rohrdichtung

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AR205452A1 (es) *	1973-12-06	1976-05-07	Endo Lab	Metodo para preparar nuevos trans-2, 3, 4, 4a, 5, 9b-hexahidro-5-fenil-1h-pirido(4,3-b) indoles
JPS50126699A (ru) *	1974-03-20	1975-10-04
US4001263A (en) *	1974-04-01	1977-01-04	Pfizer Inc.	5-Aryl-1,2,3,4-tetrahydro-γ-carbolines

1978
- 1978-03-30 SE SE7803625A patent/SE441448B/sv unknown
- 1978-04-17 PH PH21013A patent/PH13756A/en unknown
- 1978-04-18 YU YU00914/78A patent/YU91478A/xx unknown
- 1978-04-20 NL NL7804210A patent/NL7804210A/xx not_active Application Discontinuation
- 1978-04-24 AU AU35377/78A patent/AU499618B1/en not_active Expired
- 1978-04-25 EG EG276/78A patent/EG13590A/xx active
- 1978-04-28 AR AR271956A patent/AR217688A1/es active
- 1978-05-18 GB GB20350/78A patent/GB1586655A/en not_active Expired
- 1978-05-18 CS CS783239A patent/CS207612B2/cs unknown
- 1978-05-18 HU HU78PI626A patent/HU185009B/hu unknown
- 1978-05-18 HU HU822638A patent/HU188802B/hu unknown
- 1978-05-18 PL PL1978215923A patent/PL116944B1/pl unknown
- 1978-05-18 HU HU822639A patent/HU187782B/hu unknown
- 1978-05-18 PL PL1978215922A patent/PL114541B1/pl unknown
- 1978-05-18 SU SU782615898A patent/SU873883A3/ru active
- 1978-05-18 PL PL1978206903A patent/PL114547B1/pl unknown
- 1978-05-18 PL PL1978215921A patent/PL117107B1/pl unknown
- 1978-05-19 CA CA303,710A patent/CA1094071A/en not_active Expired
- 1978-05-19 DD DD78215015A patent/DD145536A5/de unknown
- 1978-05-19 PT PT68058A patent/PT68058B/pt unknown
- 1978-05-19 BE BE187842A patent/BE867249A/xx not_active IP Right Cessation
- 1978-05-19 DD DD78215017A patent/DD145537A5/de unknown
- 1978-05-19 DD DD78205479A patent/DD138321A5/xx unknown
- 1978-05-19 DD DD215016A patent/DD146186A5/de unknown
- 1978-05-20 GR GR56281A patent/GR69985B/el unknown
- 1978-05-22 JP JP6087278A patent/JPS53144600A/ja active Granted
- 1978-05-22 CH CH552678A patent/CH634321A5/fr not_active IP Right Cessation
- 1978-05-22 NO NO781770A patent/NO150204C/no unknown
- 1978-05-22 ZA ZA00782918A patent/ZA782918B/xx unknown
- 1978-05-22 AT AT0369678A patent/AT368995B/de not_active IP Right Cessation
- 1978-05-22 IT IT23673/78A patent/IT1096307B/it active
- 1978-05-22 DK DK226678A patent/DK226678A/da not_active Application Discontinuation
- 1978-05-22 IL IL54755A patent/IL54755A/xx unknown
- 1978-05-22 FR FR7815029A patent/FR2392023A1/fr active Granted
- 1978-05-22 IE IE1013/78A patent/IE46975B1/en unknown
- 1978-05-22 NZ NZ187333A patent/NZ187333A/en unknown
- 1978-05-22 FI FI781612A patent/FI63402C/fi not_active IP Right Cessation
- 1978-05-22 LU LU79684A patent/LU79684A1/xx unknown
- 1978-05-23 DE DE2822465A patent/DE2822465C2/de not_active Expired
1979
- 1979-04-16 AR AR276191A patent/AR221721A1/es active
- 1979-04-24 SU SU792753359A patent/SU843749A3/ru active
- 1979-04-26 SU SU792759902A patent/SU818484A3/ru active
- 1979-05-18 SU SU792763595A patent/SU841589A3/ru active
- 1979-05-18 PL PL20690379A patent/PL206903A1/xx unknown
1982
- 1982-10-01 YU YU2217/82A patent/YU40796B/xx unknown
- 1982-10-01 YU YU02218/82A patent/YU221882A/xx unknown
- 1982-10-01 YU YU02216/82A patent/YU221682A/xx unknown
1983
- 1983-05-20 NO NO831790A patent/NO151862C/no unknown
- 1983-10-27 SE SE8305917A patent/SE448459B/sv not_active IP Right Cessation

Also Published As

Publication number	Publication date
NL7804210A (nl)	1978-11-27
FR2392023B1 (ru)	1980-11-07
FI63402C (fi)	1983-06-10
AR217688A1 (es)	1980-04-15
YU40796B (en)	1986-06-30
YU221782A (en)	1983-01-21
IT1096307B (it)	1985-08-26
NO150204B (no)	1984-05-28
HU188802B (en)	1986-05-28
JPS53144600A (en)	1978-12-15
PL206903A1 (pl)	1979-10-22
SE7803625L (sv)	1978-11-24
AR221721A1 (es)	1981-03-13
AU499618B1 (en)	1979-04-26
PT68058A (en)	1978-06-01
IE46975B1 (en)	1983-11-16
BE867249A (fr)	1978-11-20
NO781770L (no)	1978-11-24
DD145537A5 (de)	1980-12-17
HU187782B (en)	1986-02-28
IL54755A0 (en)	1978-07-31
SU818484A3 (ru)	1981-03-30
SU841589A3 (ru)	1981-06-23
YU221682A (en)	1983-01-21
DD145536A5 (de)	1980-12-17
SU873883A3 (ru)	1981-10-15
SE8305917L (sv)	1983-10-27
CA1094071A (en)	1981-01-20
NO150204C (no)	1984-09-05
FR2392023A1 (fr)	1978-12-22
HU185009B (en)	1984-11-28
ATA369678A (de)	1982-04-15
GB1586655A (en)	1981-03-25
DE2822465C2 (de)	1986-08-28
NO151862B (no)	1985-03-11
PH13756A (en)	1980-09-17
PL116944B1 (en)	1981-07-31
NZ187333A (en)	1984-05-31
PT68058B (en)	1979-10-24
JPS5711912B2 (ru)	1982-03-08
DD138321A5 (de)	1979-10-24
PL114541B1 (en)	1981-02-28
SU843749A3 (ru)	1981-06-30
AT368995B (de)	1982-11-25
SE448459B (sv)	1987-02-23
DD146186A5 (de)	1981-01-28
DK226678A (da)	1978-11-24
IE781013L (en)	1978-11-23
FI63402B (fi)	1983-02-28
ZA782918B (en)	1979-06-27
GR69985B (ru)	1982-07-22
CH634321A5 (en)	1983-01-31
PL114547B1 (en)	1981-02-28
PL117107B1 (en)	1981-07-31
NO831790L (no)	1978-11-24
NO151862C (no)	1985-06-19
FI781612A (fi)	1978-11-24
YU91478A (en)	1983-01-21
LU79684A1 (fr)	1979-12-06
IL54755A (en)	1981-02-27
IT7823673A0 (it)	1978-05-22
DE2822465A1 (de)	1978-11-30
SE8305917D0 (sv)	1983-10-27
YU221882A (en)	1983-01-21
SE441448B (sv)	1985-10-07
EG13590A (en)	1982-03-31

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