[go: up one dir, main page]
More Web Proxy on the site http://driver.im/

NO20003273D0 - Substituerte <beta>-alaniner - Google Patents

Substituerte <beta>-alaniner

Info

Publication number
NO20003273D0
NO20003273D0 NO20003273A NO20003273A NO20003273D0 NO 20003273 D0 NO20003273 D0 NO 20003273D0 NO 20003273 A NO20003273 A NO 20003273A NO 20003273 A NO20003273 A NO 20003273A NO 20003273 D0 NO20003273 D0 NO 20003273D0
Authority
NO
Norway
Prior art keywords
beta
compounds
prodrugs
halogen
hydrogen
Prior art date
Application number
NO20003273A
Other languages
English (en)
Other versions
NO20003273L (no
Inventor
Peter Charles Astles
Neil Victor Harris
Andrew David Morley
Original Assignee
Aventis Pharma Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9727532.5A external-priority patent/GB9727532D0/en
Application filed by Aventis Pharma Ltd filed Critical Aventis Pharma Ltd
Publication of NO20003273D0 publication Critical patent/NO20003273D0/no
Publication of NO20003273L publication Critical patent/NO20003273L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24Oxygen or sulfur atoms
    • C07D207/262-Pyrrolidones
    • C07D207/2632-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms
    • C07D207/272-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C275/00Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C275/28Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C275/42Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by carboxyl groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Oncology (AREA)
  • Dermatology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrrole Compounds (AREA)
  • Polyamides (AREA)
  • Indole Compounds (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Peptides Or Proteins (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Furan Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO20003273A 1997-12-23 2000-06-22 Substituerte <beta>-alaniner NO20003273L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9727532.5A GB9727532D0 (en) 1997-12-23 1997-12-23 Chemical compounds
US9260298P 1998-07-13 1998-07-13
PCT/GB1998/003859 WO1999033789A1 (en) 1997-12-23 1998-12-23 SUBSTITUTED β-ALANINES

Publications (2)

Publication Number Publication Date
NO20003273D0 true NO20003273D0 (no) 2000-06-22
NO20003273L NO20003273L (no) 2000-06-22

Family

ID=26312873

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20003273A NO20003273L (no) 1997-12-23 2000-06-22 Substituerte <beta>-alaniner

Country Status (19)

Country Link
EP (1) EP1042279B1 (no)
JP (1) JP4555469B2 (no)
KR (1) KR20010033520A (no)
CN (1) CN1163477C (no)
AT (1) ATE289991T1 (no)
AU (1) AU747907B2 (no)
BR (1) BR9814376A (no)
CA (1) CA2316235A1 (no)
CZ (1) CZ20002342A3 (no)
DE (1) DE69829215T2 (no)
ES (1) ES2235383T3 (no)
HK (1) HK1034508A1 (no)
HU (1) HUP0101701A3 (no)
IL (1) IL136584A (no)
NO (1) NO20003273L (no)
NZ (1) NZ505363A (no)
SK (1) SK9372000A3 (no)
TR (1) TR200001947T2 (no)
WO (1) WO1999033789A1 (no)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1294576A (zh) * 1998-01-23 2001-05-09 诺瓦提斯公司 Vla-4拮抗剂
HUP0200481A3 (en) 1998-12-23 2002-12-28 Aventis Pharma Ltd West Mallin Dihydro-benzo(1,4)oxazines and tetrahydroquinoxalines, process for their preparation and pharmaceutical compositions containing them
TR200102399T2 (tr) * 1999-02-18 2002-01-21 F. Hoffmann-La Roch Ag Tiyoamid türevleri
KR20020067050A (ko) * 1999-12-28 2002-08-21 화이자 프로덕츠 인코포레이티드 염증성, 자기면역 및 호흡기 질환의 치료에 유용한브이엘에이-4 의존성 세포 결합의 비펩티드계 억제제
DE10019755A1 (de) * 2000-04-20 2001-11-08 Bayer Ag Neue Aminoaryl/cycloalkylcarbonsäuren als Integrinantagonisten
FR2812633A1 (fr) * 2000-08-04 2002-02-08 Aventis Cropscience Sa Derives de phenyl(thio)urees et phenyl(thio)carbamates fongicides
GB2367816A (en) * 2000-10-09 2002-04-17 Bayer Ag Urea- and thiourea-containing derivatives of beta-amino acids
GB2369357A (en) * 2000-10-09 2002-05-29 Bayer Ag Aliphatic, cyclic amino carboxylic acids as integrin antagonists
MXPA03003829A (es) 2000-11-04 2003-07-28 Aventis Pharma Ltd Acidos alcanoicos substituidos.
ATE524441T1 (de) 2000-12-28 2011-09-15 Daiichi Seiyaku Co Vla-4-inhibitoren
GB2377933A (en) 2001-07-06 2003-01-29 Bayer Ag Succinic acid derivatives useful as integrin antagonists
MXPA06000850A (es) 2003-07-24 2006-03-30 Daiichi Seiyaku Co Compuesto de acido ciclohexancarboxilico.
JP2008539246A (ja) * 2005-04-28 2008-11-13 フェリング ベスローテン フェンノートシャップ Ibd治療のための新規化合物の使用
JP5107724B2 (ja) 2005-12-13 2012-12-26 第一三共株式会社 Vla−4阻害薬
EP2124996A4 (en) 2007-02-20 2010-03-24 Merrimack Pharmaceuticals Inc METHODS OF TREATING MULTIPLE SCLEROSIS BY ADMINISTERING ALPHA-FETOPROTEIN COMBINED WITH INTEGRIN ANTAGONIST

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6306840B1 (en) * 1995-01-23 2001-10-23 Biogen, Inc. Cell adhesion inhibitors
KR100481285B1 (ko) * 1995-08-30 2005-08-08 지.디. 썰 엘엘씨 인테그린길항제로서의메타-구아니딘,우레아,티오우레아또는아자고리아미노벤조산유도체
ES2162676T3 (es) * 1996-03-29 2002-01-01 Searle & Co Derivados de fenileno sustituidos en meta y su uso como antagonistas o inhibidores de integrina alfav,beta3.
ES2172780T3 (es) * 1996-03-29 2002-10-01 Searle & Co Derivados de acido fenilpropanoico sustituidos en para como antagonistas de integrina.
SK5462000A3 (en) * 1997-10-31 2001-02-12 Aventis Pharma Ltd Substituted anilides

Also Published As

Publication number Publication date
CA2316235A1 (en) 1999-07-08
ES2235383T3 (es) 2005-07-01
AU1771999A (en) 1999-07-19
SK9372000A3 (en) 2002-03-05
BR9814376A (pt) 2000-10-10
EP1042279A1 (en) 2000-10-11
HUP0101701A2 (hu) 2001-11-28
ATE289991T1 (de) 2005-03-15
WO1999033789A1 (en) 1999-07-08
NZ505363A (en) 2005-02-25
JP2001527061A (ja) 2001-12-25
HUP0101701A3 (en) 2003-02-28
TR200001947T2 (tr) 2001-01-22
KR20010033520A (ko) 2001-04-25
HK1034508A1 (en) 2001-10-26
DE69829215D1 (de) 2005-04-07
CZ20002342A3 (cs) 2001-11-14
NO20003273L (no) 2000-06-22
IL136584A (en) 2005-03-20
DE69829215T2 (de) 2005-07-21
CN1163477C (zh) 2004-08-25
EP1042279B1 (en) 2005-03-02
AU747907B2 (en) 2002-05-30
CN1283181A (zh) 2001-02-07
IL136584A0 (en) 2001-06-14
JP4555469B2 (ja) 2010-09-29

Similar Documents

Publication Publication Date Title
ATE289991T1 (de) Substituierte beta-alaninen
DK1027328T3 (da) Substituerede anilider
DE69523169D1 (de) Verwendung von Mangiferin oder seinen Derivaten zur kosmetischen Anwendung
TR200102959T2 (tr) İntegrin antagonistleri olarak ikame edilmiş bisiklik heteroaril bileşikleri
HUP0204496A2 (en) Novel piperidine compounds and pharmaceutical compositions containing the same and process for preparation the same
SE9604786D0 (sv) New compounds
IL151172A0 (en) Amine derivatives, their preparation and use as bax modulators
ATE270668T1 (de) Phenoxypropanolamin-derivate, ihre herstellung und therapeutische verwendung
HU9603185D0 (en) New azolidinediones as antihyperglycemic agents
FR2712591B1 (fr) Nouvelles arylpipérazines dérivées d&#39;indole, leur préparation et leur utilisation thérapeutique.
CO4820432A1 (es) Composiciones farmaceuticas para el tratamiento de rinitis que comprenden acido 2-(4-(difenilmetil)-1-piperacinil)-ace- tico o amida derivada y un compuesto seleccionado de pseudoe fedrina,fenilpropanolamina y fenilefrina
NO944892L (no) N-substituerte 3-azabicyklo (3.2.0) hepatanderivater som neuroleptika osv.
ATE126221T1 (de) Thiazolidinverbindeungen, deren herstellung und therapeutische verwendung.
HUP0102025A2 (hu) Diaril-1,3,4-oxadiazolon-származékok, ezeket tartalmazó gyógyszerkészítmények és alkalmazásuk
DE69402935D1 (de) Substituierte arylalkylaminobenzyl-aminopropanamide, ihre herstellung und verwendung als antiepileptische, neuroprotektive und antidepressive mittel
PT89082A (pt) Processo para a preparacao de novos derivados n-(23-vinblastinoilicos)do acido 1-amino-metilfosfonico
PT1068184E (pt) Derivados n-ariloxietilamina para o tratamento de depressao
EP0638564A4 (en) BENZOTHIAZOLESULFONAMIDE DERIVATIVE, PROCESS FOR PRODUCING THE SAME AND APPLICATION THEREOF.
ATE245986T1 (de) Verwendung von 8-nitro-2,3,4,5-tetrahydro-1h-3- benzazepinen zur herstellung von pharmazeutischen zusammenstellungen zur behandlung von schlafstörungen
NO950177D0 (no) Farmakologisk aktive erivater
MXPA02001861A (es) Nuevos inhbidores de la integrina alfav beta3.
BR9507668A (pt) Intermédio para preparar um composto farmaceuticamente atívo
EP1241166A4 (en) 3-MEHTYL CHROMAN AND THIOCHROME DERIVATIVES
DE69400908D1 (de) Verwendung von riluzol zum schutz gegen strahlenschäden

Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application