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PT100514A - 3-aminoquinuclidinas substituidas e composicoes farmaceuticas que qs contem - Google Patents

3-aminoquinuclidinas substituidas e composicoes farmaceuticas que qs contem

Info

Publication number
PT100514A
PT100514A PT100514A PT10051492A PT100514A PT 100514 A PT100514 A PT 100514A PT 100514 A PT100514 A PT 100514A PT 10051492 A PT10051492 A PT 10051492A PT 100514 A PT100514 A PT 100514A
Authority
PT
Portugal
Prior art keywords
aminokinuclidins
substituted
pharmaceutical compositions
compounds
disorders
Prior art date
Application number
PT100514A
Other languages
English (en)
Other versions
PT100514B (pt
Inventor
Masami Nakane
Fumitaka Ito
Hiroaki Wakabayashi
Toshihide Kokura
Kunio Satake
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of PT100514A publication Critical patent/PT100514A/pt
Publication of PT100514B publication Critical patent/PT100514B/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Medicinal Preparation (AREA)
PT100514A 1991-05-22 1992-05-22 3-aminoquinuclidinas substituidas e composicoes farmaceuticas que qs contem PT100514B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP14682691 1991-05-22

Publications (2)

Publication Number Publication Date
PT100514A true PT100514A (pt) 1993-09-30
PT100514B PT100514B (pt) 1999-06-30

Family

ID=15416402

Family Applications (1)

Application Number Title Priority Date Filing Date
PT100514A PT100514B (pt) 1991-05-22 1992-05-22 3-aminoquinuclidinas substituidas e composicoes farmaceuticas que qs contem

Country Status (25)

Country Link
EP (1) EP0585328B1 (pt)
KR (1) KR100246065B1 (pt)
CN (1) CN1041827C (pt)
AT (1) ATE211743T1 (pt)
AU (1) AU658898B2 (pt)
BR (1) BR9206044A (pt)
CA (1) CA2109415C (pt)
CZ (1) CZ247993A3 (pt)
DE (2) DE9290057U1 (pt)
DK (1) DK0585328T3 (pt)
EG (1) EG20218A (pt)
ES (1) ES2168260T3 (pt)
FI (1) FI935134A0 (pt)
HU (1) HUT65771A (pt)
IE (1) IE921662A1 (pt)
IL (1) IL101960A (pt)
MX (1) MX9202449A (pt)
NO (1) NO305173B1 (pt)
NZ (2) NZ272941A (pt)
PL (4) PL170525B1 (pt)
PT (1) PT100514B (pt)
RU (1) RU2092486C1 (pt)
UA (1) UA26401C2 (pt)
WO (1) WO1992020676A1 (pt)
ZA (1) ZA923773B (pt)

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JP2656700B2 (ja) * 1992-10-28 1997-09-24 ファイザー製薬株式会社 置換キヌクリジン誘導体
EP0675886B1 (en) * 1992-12-10 2000-07-05 Pfizer Inc. Aminomethylene substituted non-aromatic heterocycles and use as substance p antagonists
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EP0655246A1 (en) * 1993-11-30 1995-05-31 Pfizer Inc. Substance P antagonists for the treatment of disorders caused by helicobacter pylori or other spiral urease-positive gram-negative bacteria
FR2728169A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des prurits et des dysesthesies oculaires ou palpebrales
FR2728165A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des rougeurs cutanees d'origine neurogene
FR2728166A1 (fr) 1994-12-19 1996-06-21 Oreal Composition topique contenant un antagoniste de substance p
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TW458774B (en) 1995-10-20 2001-10-11 Pfizer Antiemetic pharmaceutical compositions
FR2741262B1 (fr) 1995-11-20 1999-03-05 Oreal Utilisation d'un antagoniste de tnf-alpha pour le traitement des rougeurs cutanees d'origine neurogene
MX9706944A (es) * 1996-09-12 1998-08-30 Pfizer Quinuclidinas sustituidas con tetrazolilo como antagonistas de la sustancia p.
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CA2717509A1 (en) 2008-03-03 2009-09-11 Tiger Pharmatech Tyrosine kinase inhibitors
US9156812B2 (en) 2008-06-04 2015-10-13 Bristol-Myers Squibb Company Crystalline form of 6-[(4S)-2-methyl-4-(2-naphthyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridazin-3-amine
UA105182C2 (ru) 2008-07-03 2014-04-25 Ньюрексон, Інк. Бензоксазины, бензотиазины и родственные соединения, которые имеют ингибирующую nos активность
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US8815894B2 (en) 2009-05-12 2014-08-26 Bristol-Myers Squibb Company Crystalline forms of (S)-7-([1,2,4]triazolo[1,5-a]pyridin-6-yl)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydroisoquinoline and use thereof
MY174452A (en) 2009-10-14 2020-04-19 Schering Corp Substituted piperidines that increase p53 activity and the uses thereof
WO2011163330A1 (en) 2010-06-24 2011-12-29 Merck Sharp & Dohme Corp. Novel heterocyclic compounds as erk inhibitors
CN107090456B (zh) 2010-08-02 2022-01-18 瑟纳治疗公司 使用短干扰核酸的RNA干扰介导的联蛋白（钙粘蛋白关联蛋白质），β1基因表达的抑制
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Also Published As

Publication number Publication date
AU658898B2 (en) 1995-05-04
FI935134A (fi) 1993-11-19
DE69232334D1 (de) 2002-02-14
PL170513B1 (en) 1996-12-31
BR9206044A (pt) 1995-03-01
HUT65771A (en) 1994-07-28
DK0585328T3 (da) 2002-02-11
PL171921B1 (pl) 1997-06-30
RU2092486C1 (ru) 1997-10-10
NZ272941A (en) 1997-05-26
NZ242880A (en) 1995-10-26
EP0585328A1 (en) 1994-03-09
WO1992020676A1 (en) 1992-11-26
ES2168260T3 (es) 2002-06-16
NO934195D0 (no) 1993-11-19
ZA923773B (en) 1993-11-22
CA2109415A1 (en) 1992-11-23
IL101960A0 (en) 1994-04-12
KR100246065B1 (en) 2000-04-01
IE921662A1 (en) 1992-12-02
DE9290057U1 (de) 1994-01-05
ATE211743T1 (de) 2002-01-15
PL172069B1 (pl) 1997-07-31
AU1927592A (en) 1992-12-30
CN1068571A (zh) 1993-02-03
EG20218A (en) 1997-11-30
PT100514B (pt) 1999-06-30
FI935134A0 (fi) 1993-11-19
NO934195L (no) 1993-11-19
CA2109415C (en) 1998-12-29
EP0585328B1 (en) 2002-01-09
CZ247993A3 (en) 1994-07-13
IL101960A (en) 1999-03-12
DE69232334T2 (de) 2002-11-14
PL170525B1 (en) 1996-12-31
UA26401C2 (uk) 1999-08-30
NO305173B1 (no) 1999-04-12
MX9202449A (es) 1993-03-01
CN1041827C (zh) 1999-01-27
HU9303307D0 (en) 1994-03-28

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BB1A Laying open of patent application

Effective date: 19930415

FG3A Patent granted, date of granting

Effective date: 19990315