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DK1156049T3 - Substituerede heterocykliske forbindelser, fremgangsmåde til fremstilling heraf og farmaceutiske sammensætninger indeholdende disse - Google Patents

Substituerede heterocykliske forbindelser, fremgangsmåde til fremstilling heraf og farmaceutiske sammensætninger indeholdende disse

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Publication number
DK1156049T3
DK1156049T3 DK01119949T DK01119949T DK1156049T3 DK 1156049 T3 DK1156049 T3 DK 1156049T3 DK 01119949 T DK01119949 T DK 01119949T DK 01119949 T DK01119949 T DK 01119949T DK 1156049 T3 DK1156049 T3 DK 1156049T3
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Prior art keywords
processes
preparation
pharmaceutical compositions
compositions containing
substituted heterocyclic
Prior art date
Application number
DK01119949T
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English (en)
Inventor
Xavier Emonds-Alt
Patrick Gueule
Didier Van Broeck
Isabelle Grossriether
Vincenzo Proietto
Original Assignee
Sanofi Aventis
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Publication date
Priority claimed from FR9501016A external-priority patent/FR2729952B1/fr
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Application granted granted Critical
Publication of DK1156049T3 publication Critical patent/DK1156049T3/da

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    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
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    • C07C215/22—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated
    • C07C215/28—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
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    • C07C233/18—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of an acyclic saturated carbon skeleton
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    • C07C255/43—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being further bound to other hetero atoms the carbon skeleton being further substituted by singly-bound oxygen atoms
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DK01119949T 1995-01-30 1996-01-30 Substituerede heterocykliske forbindelser, fremgangsmåde til fremstilling heraf og farmaceutiske sammensætninger indeholdende disse DK1156049T3 (da)

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FR9501016A FR2729952B1 (fr) 1995-01-30 1995-01-30 Composes heterocycliques substitues, procede pour leur preparation et compositions pharmaceutiques les contenant
FR9508046A FR2729953B1 (fr) 1995-01-30 1995-07-04 Composes heterocycliques substitues, procede pour leur preparation et compositions pharmaceutiques les contenant
FR9513005A FR2729954B1 (fr) 1995-01-30 1995-11-03 Composes heterocycliques substitues, procede pour leur preparation et compositions pharmaceutiques les contenant
EP96902305A EP0807111B1 (fr) 1995-01-30 1996-01-30 Composes heterocycliques substitues, procede pour leur preparation et compositions pharmaceutiques les contenant

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DK01119949T DK1156049T3 (da) 1995-01-30 1996-01-30 Substituerede heterocykliske forbindelser, fremgangsmåde til fremstilling heraf og farmaceutiske sammensætninger indeholdende disse

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FI973148A (fi) 1997-09-29
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CN1321634A (zh) 2001-11-14
CN1179954C (zh) 2004-12-15
JPH11507324A (ja) 1999-06-29
MX9705590A (es) 1997-11-29
FI973148A0 (fi) 1997-07-29
PT1156049E (pt) 2005-10-31
RU2157807C2 (ru) 2000-10-20
EP1156049A1 (fr) 2001-11-21
IL116957A (en) 1999-06-20
US5977359A (en) 1999-11-02
JP3357660B2 (ja) 2002-12-16
CA2211668C (en) 2005-09-20
JP2001172279A (ja) 2001-06-26
CN1636983A (zh) 2005-07-13
NZ301285A (en) 2000-01-28
CN1293063C (zh) 2007-01-03
DE69634806T2 (de) 2006-04-27
SI0807111T1 (en) 2003-02-28
CZ294267B6 (cs) 2004-11-10
ES2243373T3 (es) 2005-12-01
CN1502612A (zh) 2004-06-09
IL127114A (en) 2004-09-27
AU4666996A (en) 1996-08-21
NO973479D0 (no) 1997-07-29
EP1340754A1 (fr) 2003-09-03
CN1394855A (zh) 2003-02-05
NO308795B1 (no) 2000-10-30
JP3943369B2 (ja) 2007-07-11
EP1923391A1 (fr) 2008-05-21
ATE296823T1 (de) 2005-06-15
FR2729954A1 (fr) 1996-08-02
US6242637B1 (en) 2001-06-05
WO1996023787A1 (fr) 1996-08-08
JP3234228B2 (ja) 2001-12-04
EP1688416A1 (fr) 2006-08-09
FR2729954B1 (fr) 1997-08-01
IL116957A0 (en) 1996-05-14
CN1172483A (zh) 1998-02-04
CN1089764C (zh) 2002-08-28
PL192164B1 (pl) 2006-09-29
US5641777A (en) 1997-06-24
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JP2002138088A (ja) 2002-05-14
DK0807111T3 (da) 2002-12-16
ES2181866T3 (es) 2003-03-01
ATE222251T1 (de) 2002-08-15
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AR002955A1 (es) 1998-05-27
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US5869663A (en) 1999-02-09
DE69622992D1 (de) 2002-09-19
EP0807111A1 (fr) 1997-11-19
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HUP9800295A2 (hu) 1999-10-28
CA2211668A1 (en) 1996-08-08
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