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NO20062181L - Metode for fremstilling av aminokrotonylforbindelser - Google Patents

Metode for fremstilling av aminokrotonylforbindelser

Info

Publication number
NO20062181L
NO20062181L NO20062181A NO20062181A NO20062181L NO 20062181 L NO20062181 L NO 20062181L NO 20062181 A NO20062181 A NO 20062181A NO 20062181 A NO20062181 A NO 20062181A NO 20062181 L NO20062181 L NO 20062181L
Authority
NO
Norway
Prior art keywords
preparation
amino
aminocrotonyl
compounds
aminocrotonyl compounds
Prior art date
Application number
NO20062181A
Other languages
English (en)
Other versions
NO333971B1 (no
Inventor
Rainer Soyka
Juergen Schnaubelt
Christian Kulinna
Werner Rall
Peter Sieger
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34428508&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20062181(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of NO20062181L publication Critical patent/NO20062181L/no
Publication of NO333971B1 publication Critical patent/NO333971B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrrole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Oppfinnelsen angår en forbedret fremgangsmåte for fremstilling av 4-[(3klor-4-fluorfenyl)amino]-6-{[4-(N,N-dimetylamino)- l-okso-2-buten-1 -yl]ammo}-7((S)-tetrahydrofuran-3-yloksy)kinazolin og beslektede aminokrotonylforbindelser. Oppfinnelsen vedrører også et egnet salt av 4-[(3-klor-4-fluorfenyl)aminoj-6-{[4(N,N-dimetylamino)-l-okso-2-buten-l -yl]amino}-7-((S)-tetrahydrofuran-3-yloksy)kinazolin for anvendelse som en aktiv ingrediens for et medikament.
NO20062181A 2003-10-17 2006-05-15 Fremgangsmåte for fremstilling av 4-[(3-klor-4-fluorfenyl)amino]-6-{[4-(N,N-dimetylamino)-1- okso-2-buten-1-yl]amino}-7-((S)-tetrahydrofuran-3-yloksy)kinazolin NO333971B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10349113A DE10349113A1 (de) 2003-10-17 2003-10-17 Verfahren zur Herstellung von Aminocrotonylverbindungen
PCT/EP2004/011378 WO2005037824A2 (de) 2003-10-17 2004-10-12 Verfahren zur herstellung von aminocrotonylverbindungen

Publications (2)

Publication Number Publication Date
NO20062181L true NO20062181L (no) 2006-05-15
NO333971B1 NO333971B1 (no) 2013-11-04

Family

ID=34428508

Family Applications (2)

Application Number Title Priority Date Filing Date
NO20062181A NO333971B1 (no) 2003-10-17 2006-05-15 Fremgangsmåte for fremstilling av 4-[(3-klor-4-fluorfenyl)amino]-6-{[4-(N,N-dimetylamino)-1- okso-2-buten-1-yl]amino}-7-((S)-tetrahydrofuran-3-yloksy)kinazolin
NO20130663A NO335103B1 (no) 2003-10-17 2013-05-10 Forbindelse, farmasøytisk preparat inneholdende forbindelsen, anvendelse av forbindelsen samt fremgangsmåte for fremstilling derav

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO20130663A NO335103B1 (no) 2003-10-17 2013-05-10 Forbindelse, farmasøytisk preparat inneholdende forbindelsen, anvendelse av forbindelsen samt fremgangsmåte for fremstilling derav

Country Status (35)

Country Link
US (2) US20050085495A1 (no)
EP (2) EP1678165B1 (no)
JP (2) JP4594317B2 (no)
KR (2) KR101180752B1 (no)
CN (2) CN101402631A (no)
AR (1) AR046118A1 (no)
AU (2) AU2004281938B2 (no)
BR (2) BRPI0415424B8 (no)
CA (2) CA2759063C (no)
CY (2) CY1114866T1 (no)
DE (1) DE10349113A1 (no)
DK (2) DK1678165T3 (no)
EA (1) EA016624B1 (no)
EC (1) ECSP066509A (no)
ES (2) ES2563211T5 (no)
HK (1) HK1095817A1 (no)
HR (2) HRP20160246T4 (no)
HU (1) HUE028254T2 (no)
IL (2) IL174951A (no)
ME (1) ME00341B (no)
MX (2) MXPA06004076A (no)
MY (2) MY155425A (no)
NO (2) NO333971B1 (no)
NZ (2) NZ547154A (no)
PE (2) PE20100267A1 (no)
PL (2) PL1678165T3 (no)
PT (2) PT1678165E (no)
RS (3) RS60563B1 (no)
SG (1) SG139743A1 (no)
SI (2) SI2508521T2 (no)
TW (2) TWI373470B (no)
UA (2) UA91006C2 (no)
UY (2) UY28559A1 (no)
WO (1) WO2005037824A2 (no)
ZA (1) ZA200602234B (no)

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