US3272781A
(en)
|
1963-08-07 |
1966-09-13 |
American Potash & Chem Corp |
Boroureas of phosphinoborine polymers
|
FR1425700A
(fr)
|
1965-02-22 |
1966-01-24 |
Basf Ag |
Composés formant des complexes métalliques et procédé pour les préparer et les utiliser
|
US4208328A
(en)
|
1978-04-27 |
1980-06-17 |
General Electric Company |
Alkyl 3,5-dihydroxy-4-(2-benzothiazolyl)benzoates
|
US4789711A
(en)
|
1986-12-02 |
1988-12-06 |
Ciba-Geigy Corporation |
Multifunctional epoxide resins
|
DE3828535A1
(de)
|
1988-08-23 |
1990-03-08 |
Basf Ag |
Benzimidazol-2-carbonsaeureanilide, ihre verwendung als lichtschutzmittel fuer organisches material und mit diesen aniliden stabilisiertes organisches material
|
US5077164A
(en)
|
1989-06-21 |
1991-12-31 |
Minolta Camera Kabushiki Kaisha |
Photosensitive member containing an azo dye
|
DE69421982T2
(de)
|
1993-09-20 |
2000-03-30 |
Fuji Photo Film Co., Ltd. |
Positiv arbeitende Photoresistzusammensetzung
|
JP3461397B2
(ja)
|
1995-01-11 |
2003-10-27 |
富士写真フイルム株式会社 |
ポジ型フオトレジスト組成物
|
JP2001505585A
(ja)
|
1996-12-16 |
2001-04-24 |
藤沢薬品工業株式会社 |
新規アミド化合物およびそれらの一酸化窒素シンターゼ阻害剤としての用途
|
JPH10316853A
(ja)
|
1997-05-15 |
1998-12-02 |
Sumitomo Bakelite Co Ltd |
半導体多層配線用層間絶縁膜樹脂組成物及び該絶縁膜の製造方法
|
JP2001519345A
(ja)
|
1997-10-02 |
2001-10-23 |
メルク エンド カムパニー インコーポレーテッド |
プレニルタンパク質トランスフェラーゼの阻害剤
|
WO1999044992A1
(fr)
|
1998-03-05 |
1999-09-10 |
Nissan Chemical Industries, Ltd. |
Composes d'anilide et herbicide
|
JP2000128987A
(ja)
|
1998-10-28 |
2000-05-09 |
Sumitomo Bakelite Co Ltd |
ポリベンゾオキサゾール前駆体及びポリベンゾオキサゾール
|
JP2000128986A
(ja)
|
1998-10-28 |
2000-05-09 |
Sumitomo Bakelite Co Ltd |
ポリベンゾオキサゾール前駆体及びポリベンゾオキサゾール
|
JP2000128984A
(ja)
|
1998-10-28 |
2000-05-09 |
Sumitomo Bakelite Co Ltd |
ポリベンゾオキサゾール前駆体及び樹脂
|
US6297351B1
(en)
|
1998-12-17 |
2001-10-02 |
Sumitomo Bakelite Company Limited |
Polybenzoxazole resin and precursor thereof
|
EP1140859A2
(fr)
|
1998-12-18 |
2001-10-10 |
Axys Pharmaceuticals, Inc. |
Derives bicycliques (hetero)aryl aryl, leur preparation et leur utilisation comme inhibiteurs de protease
|
JP2000212281A
(ja)
|
1999-01-27 |
2000-08-02 |
Sumitomo Bakelite Co Ltd |
ポリベンゾオキサゾ―ル前駆体及びポリベンゾオキサゾ―ル樹脂
|
WO2001007409A1
(fr)
|
1999-07-23 |
2001-02-01 |
Astrazeneca Uk Limited |
Derives de carbazole et leur utilisation en tant que ligands du recepteur de neuropeptide y5
|
JP2001114893A
(ja)
|
1999-10-15 |
2001-04-24 |
Sumitomo Bakelite Co Ltd |
ポリベンゾオキサゾール樹脂およびその前駆体
|
US6372907B1
(en)
|
1999-11-03 |
2002-04-16 |
Apptera Corporation |
Water-soluble rhodamine dye peptide conjugates
|
JP2001163975A
(ja)
|
1999-12-03 |
2001-06-19 |
Sumitomo Bakelite Co Ltd |
ポリベンゾオキサゾール樹脂及びその前駆体
|
CN1623984A
(zh)
|
1999-12-27 |
2005-06-08 |
日本烟草产业株式会社 |
稠环化合物及其药物用途
|
AU2001240542A1
(en)
|
2000-02-01 |
2001-08-14 |
Basf Aktiengesellschaft |
Heterocyclic compounds and their use as parp inhibitors
|
US6521618B2
(en)
|
2000-03-28 |
2003-02-18 |
Wyeth |
3-cyanoquinolines, 3-cyano-1,6-naphthyridines, and 3-cyano-1,7-naphthyridines as protein kinase inhibitors
|
AU2001249679A1
(en)
|
2000-03-31 |
2001-10-15 |
Ortho-Mcneil Pharmaceutical, Inc. |
Phenyl-substituted imidazopyridines
|
CA2405170A1
(fr)
|
2000-04-24 |
2001-11-01 |
Merck Frosst Canada & Co. |
Methode de traitement se basant sur l'utilisation de derives de phenyle et de biaryle comme inhibiteurs de prostaglandine e
|
NZ522783A
(en)
|
2000-06-28 |
2004-07-30 |
Smithkline Beecham P |
Wet milling process for pharmaceuticals with agitator or chamber having nylon with internal lubricant
|
AU2001294515A1
(en)
|
2000-08-11 |
2002-02-25 |
The Regents Of The University Of California |
Use of stat-6 inhibitors as therapeutic agents
|
EP1343785A2
(fr)
|
2000-12-13 |
2003-09-17 |
Basf Aktiengesellschaft |
Utilisation d'imidazoazines substituees, nouvelles imidazoazines, procede permettant de les produire et agents les contenant
|
US6919352B2
(en)
|
2000-12-15 |
2005-07-19 |
Smithkline Beecham Corporation |
Pyrazolopyridinyl pyridine and pyrimidine therapeutic compounds
|
SE0100567D0
(sv)
|
2001-02-20 |
2001-02-20 |
Astrazeneca Ab |
Compounds
|
ES2244772T3
(es)
|
2001-03-14 |
2005-12-16 |
Eli Lilly And Company |
Moduladores de receptores de retinoides x.
|
JP4237497B2
(ja)
|
2001-03-30 |
2009-03-11 |
スミスクライン ビーチャム コーポレーション |
ピラゾロピリジン類、その調製方法及びその治療用化合物としての使用
|
WO2002083672A1
(fr)
|
2001-04-10 |
2002-10-24 |
Smithkline Beecham Corporation |
Composes de pyrazolopyridine antiviraux
|
JP2002316966A
(ja)
|
2001-04-19 |
2002-10-31 |
Ueno Seiyaku Oyo Kenkyusho:Kk |
ビナフトール誘導体およびその製法
|
WO2002088124A2
(fr)
|
2001-04-27 |
2002-11-07 |
Smithkline Beecham Corporation |
Composes therapeutiques
|
AR035543A1
(es)
|
2001-06-26 |
2004-06-16 |
Japan Tobacco Inc |
Agente terapeutico para la hepatitis c que comprende un compuesto de anillo condensado, compuesto de anillo condensado, composicion farmaceutica que lo comprende, compuestos de benzimidazol, tiazol y bifenilo utiles como intermediarios para producir dichos compuestos, uso del compuesto de anillo con
|
JP2005507878A
(ja)
|
2001-09-07 |
2005-03-24 |
スミスクライン ビーチャム コーポレーション |
ヘルペス感染症を治療するためのピラゾロ−ピリジン類
|
TWI320039B
(en)
|
2001-09-21 |
2010-02-01 |
|
Lactam-containing compounds and derivatives thereof as factor xa inhibitors
|
US20030143199A1
(en)
|
2001-10-09 |
2003-07-31 |
Carson Dennis A. |
Use of STAT-6 inhibitors as therapeutic agents
|
JP2005508349A
(ja)
|
2001-10-09 |
2005-03-31 |
ファルマシア アンド アップジョン カンパニー リミティド ライアビリティー カンパニー |
5−ht6受容体リガンドとしてのアリールスルホニル置換されたテトラヒドロ−およびヘキサヒドロ−カルバゾール
|
JP4024579B2
(ja)
|
2002-01-22 |
2007-12-19 |
住友ベークライト株式会社 |
プラスチック光導波路用材料及び光導波路
|
KR20040099425A
(ko)
|
2002-04-11 |
2004-11-26 |
버텍스 파마슈티칼스 인코포레이티드 |
세린 프로테아제, 특히 c형 간염 바이러스 ns3-ns4프로테아제의 억제제
|
KR20040097375A
(ko)
|
2002-04-23 |
2004-11-17 |
시오노기 앤드 컴파니, 리미티드 |
피라졸로[1, 5-에이]피리미딘 유도체 및 이를 함유한엔에이디(피)에이취 산화효소 저해제
|
JPWO2004007472A1
(ja)
|
2002-07-10 |
2005-11-17 |
小野薬品工業株式会社 |
Ccr4アンタゴニストおよびその医薬用途
|
WO2004006906A2
(fr)
|
2002-07-15 |
2004-01-22 |
Combinatorx, Incorporated |
Methodes de traitement de neoplasmes
|
JP2004059761A
(ja)
|
2002-07-30 |
2004-02-26 |
Sumitomo Bakelite Co Ltd |
ポリベンゾオキサゾール樹脂、その前駆体及びこれらを用いた光導波路材料並びに光導波路
|
US20050260126A1
(en)
|
2002-08-30 |
2005-11-24 |
Yukitsuka Kudo |
Diagnostic probes and remedies for diseases with accumulation of prion protein, and stains for prion protein
|
JP2004091369A
(ja)
|
2002-08-30 |
2004-03-25 |
Sumitomo Pharmaceut Co Ltd |
新規ビフェニル化合物
|
EP1546148A1
(fr)
|
2002-10-03 |
2005-06-29 |
SmithKline Beecham Corporation |
Composes therapeutiques a base de derives de pyrazolopyridine
|
WO2004035588A1
(fr)
|
2002-10-15 |
2004-04-29 |
Smithkline Beecham Corporation |
Composes de pyradazine utiles comme inhibiteurs de gsk-3
|
KR100624406B1
(ko)
|
2002-12-30 |
2006-09-18 |
삼성에스디아이 주식회사 |
비페닐 유도체 및 이를 채용한 유기 전계 발광 소자
|
US7320989B2
(en)
|
2003-02-28 |
2008-01-22 |
Encysive Pharmaceuticals, Inc. |
Pyridine, pyrimidine, quinoline, quinazoline, and naphthalene urotensin-II receptor antagonists
|
US7078419B2
(en)
|
2003-03-10 |
2006-07-18 |
Boehringer Ingelheim Pharmaceuticals, Inc. |
Cytokine inhibitors
|
AR043633A1
(es)
|
2003-03-20 |
2005-08-03 |
Schering Corp |
Ligandos de receptores de canabinoides
|
JP4595288B2
(ja)
|
2003-03-25 |
2010-12-08 |
住友ベークライト株式会社 |
ポリベンゾオキサゾール樹脂、その前駆体及びこれらを用いた光導波路材料並びに光導波路
|
ATE427308T1
(de)
|
2003-04-11 |
2009-04-15 |
Glenmark Pharmaceuticals Sa |
Neue heterozyklische verbindungen, die sich fur die behandlung von entzundlichen und allergischen erkrankungen eignen: verfahren zu deren herstellung und pharmazeutische zusammensetzungen,die diese enthalten
|
JP2005002330A
(ja)
|
2003-05-19 |
2005-01-06 |
Sumitomo Electric Ind Ltd |
光学樹脂材料、光学素子、光モジュール、フッ素化ポリマー前駆体及びフッ素化ポリマー
|
EP1628967B1
(fr)
|
2003-05-19 |
2014-04-09 |
Irm Llc |
Composés immunosuppresseurs et compositions
|
US20060183746A1
(en)
|
2003-06-04 |
2006-08-17 |
Currie Kevin S |
Certain imidazo[1,2-a]pyrazin-8-ylamines and method of inhibition of Bruton's tyrosine kinase by such compounds
|
US7405295B2
(en)
|
2003-06-04 |
2008-07-29 |
Cgi Pharmaceuticals, Inc. |
Certain imidazo[1,2-a]pyrazin-8-ylamines and method of inhibition of Bruton's tyrosine kinase by such compounds
|
WO2005005429A1
(fr)
|
2003-06-30 |
2005-01-20 |
Cellular Genomics, Inc. |
Certaines imidazo[1,2-a]pyrazin-8-ylamines substituees heterocycliques et methodes d'inhibition de la tyrosine kinase de bruton utilisant ces composes
|
US7276608B2
(en)
|
2003-07-11 |
2007-10-02 |
Bristol-Myers Squibb Company |
Tetrahydroquinoline derivatives as cannabinoid receptor modulators
|
US7691870B2
(en)
|
2003-07-11 |
2010-04-06 |
Merck Patent Gmbh |
Benzimidazole carboxamides as raf kinase inhibitors
|
WO2005012221A1
(fr)
|
2003-08-04 |
2005-02-10 |
Ono Pharmaceutical Co., Ltd. |
Compose d'ether de diphenyle, sa methode de preparation et d'utilisation
|
WO2005014543A1
(fr)
|
2003-08-06 |
2005-02-17 |
Japan Tobacco Inc. |
Compose a cycle condense utilise comme inhibiteur de la polymerase du vhc
|
US7504401B2
(en)
|
2003-08-29 |
2009-03-17 |
Locus Pharmaceuticals, Inc. |
Anti-cancer agents and uses thereof
|
US7749999B2
(en)
|
2003-09-11 |
2010-07-06 |
Itherx Pharmaceuticals, Inc. |
Alpha-ketoamides and derivatives thereof
|
US7449582B2
(en)
|
2003-10-08 |
2008-11-11 |
Irm Llc |
Compounds and compositions as protein kinase inhibitors
|
WO2005040135A1
(fr)
|
2003-10-24 |
2005-05-06 |
Ono Pharmaceutical Co., Ltd. |
Medicament antistress et usage medical correspondant
|
WO2005047290A2
(fr)
|
2003-11-11 |
2005-05-26 |
Cellular Genomics Inc. |
Certaines imidazo[1,2-a]pyrazin-8-ylamines, procede de fabrication et methode d'utilisation
|
WO2005063710A1
(fr)
|
2003-12-23 |
2005-07-14 |
Basf Aktiengesellschaft |
Anilides d'acide 3-trifluoromethylpicolinique et leur utilisation comme fongicides
|
CA2555402A1
(fr)
|
2004-02-12 |
2005-09-01 |
Celine Bonnefous |
Amides bipyridyles en tant que modulateurs du recepteur-5 metabotropique du glutamate
|
US20070191395A1
(en)
|
2004-02-16 |
2007-08-16 |
Katsuhiro Kawakami |
Heterocyclic compounds having antifungal activity
|
GB0403864D0
(en)
|
2004-02-20 |
2004-03-24 |
Ucl Ventures |
Modulator
|
JP2005248082A
(ja)
|
2004-03-05 |
2005-09-15 |
Sumitomo Electric Ind Ltd |
ポリベンゾオキサゾール樹脂前駆体の製造方法およびポリベンゾオキサゾール樹脂の製造方法
|
AU2005221140A1
(en)
|
2004-03-08 |
2005-09-22 |
Amgen Inc. |
Therapeutic modulation of PPAR (gamma) activity
|
CA2554554A1
(fr)
|
2004-03-08 |
2005-09-22 |
The University Of North Carolina At Chapel Hill |
Nouvelles c imidazo[1,2-a]pyridines dicationique et nouvelles 5,6,7,8-tetrahydro-imidazo[1,2a]pyridines utilisee s comme agents antiprotozoaires
|
JP2007531753A
(ja)
|
2004-03-31 |
2007-11-08 |
ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ |
非イミダゾール系複素環式化合物
|
JP2005290301A
(ja)
|
2004-04-02 |
2005-10-20 |
Sumitomo Electric Ind Ltd |
ポリベンゾオキサゾール樹脂前駆体の製造方法およびポリベンゾオキサゾール樹脂の製造方法
|
WO2005099656A2
(fr)
|
2004-04-06 |
2005-10-27 |
The Procter & Gamble Company |
Composes de teinture de la keratine, compositions de teinture de la keratine contenant ces composes et leurs utilisations
|
CN1946703A
(zh)
|
2004-04-20 |
2007-04-11 |
特兰斯泰克制药公司 |
取代的噻唑和嘧啶衍生物作为黑素细胞皮质激素受体调节剂
|
DE102004021716A1
(de)
|
2004-04-30 |
2005-12-01 |
Grünenthal GmbH |
Substituierte Imidazo[1,2-a]pyridin-Verbindungen und Arzneimittel enthaltend substituierte Imidazo[1,2-a]pyridin-Verbindungen
|
CA2560387C
(fr)
|
2004-05-03 |
2013-09-24 |
Boehringer Ingelheim Pharmaceuticals, Inc. |
Inhibiteurs de cytokines
|
PE20060748A1
(es)
|
2004-09-21 |
2006-10-01 |
Smithkline Beecham Corp |
Derivados de indolcarboxamida como inhibidores de quinasa ikk2
|
BRPI0515596A
(pt)
|
2004-09-23 |
2008-07-29 |
Wyeth Corp |
composição farmacêutica usada para o tratamento e/ou prevenção de hcv, e, métodos de inibir rna polimerase ns5b de hepatite c de tratar ou prevenir infecção por hepatite c em um mamìfero
|
DE602005023333D1
(de)
|
2004-10-15 |
2010-10-14 |
Takeda Pharmaceutical |
Kinaseinhibitoren
|
WO2006053121A2
(fr)
|
2004-11-10 |
2006-05-18 |
Cgi Pharmaceuticals, Inc. |
Certaines imidazo[1,2-a] pyrazin-8-ylamines et les procédés de fabrication et d'utilisation correspondants
|
DE102004054665A1
(de)
|
2004-11-12 |
2006-05-18 |
Bayer Cropscience Gmbh |
Substituierte bi- und tricyclische Pyrazol-Derivate Verfahren zur Herstellung und Verwendung als Herbizide und Pflanzenwachstumsregulatoren
|
CA2599987A1
(fr)
|
2005-03-03 |
2006-09-08 |
Sirtris Pharmaceuticals, Inc. |
Composes heterocycliques liquefies et leur utilisation comme modulateurs de sirtuine
|
JP2008533032A
(ja)
|
2005-03-10 |
2008-08-21 |
シージーアイ ファーマシューティカルズ,インコーポレイティド |
或る種の置換アミド、その製造方法及び使用方法
|
JP2006290883A
(ja)
|
2005-03-17 |
2006-10-26 |
Nippon Nohyaku Co Ltd |
置換ヘテロ環カルボン酸アニリド誘導体、その中間体及び農園芸用薬剤並びにその使用方法
|
KR20080038278A
(ko)
|
2005-05-20 |
2008-05-06 |
어레이 바이오파마 인크. |
Raf 억제제 화합물 및 그의 사용 방법
|
US20080220968A1
(en)
|
2005-07-05 |
2008-09-11 |
Ge Healthcare Bio-Sciences Ab |
[1, 2, 4] Triazolo [1, 5-A] Pyrimidine Derivatives as Chromatographic Adsorbent for the Selective Adsorption of Igg
|
WO2007034282A2
(fr)
|
2005-09-19 |
2007-03-29 |
Pfizer Products Inc. |
Composes de biphenylimidazole utilises comme antagonistes du recepteur du c3a
|
US20070078136A1
(en)
|
2005-09-22 |
2007-04-05 |
Bristol-Myers Squibb Company |
Fused heterocyclic compounds useful as kinase modulators
|
US7723336B2
(en)
|
2005-09-22 |
2010-05-25 |
Bristol-Myers Squibb Company |
Fused heterocyclic compounds useful as kinase modulators
|
WO2007049532A1
(fr)
|
2005-10-25 |
2007-05-03 |
Shionogi & Co., Ltd. |
Derive aminodihydrothiazine
|
EP1954290B1
(fr)
|
2005-11-22 |
2012-07-25 |
Merck Sharp & Dohme Corp. |
Composes tricycliques utilises comme inhibiteurs de kinases
|
WO2007067711A2
(fr)
|
2005-12-08 |
2007-06-14 |
Amphora Discovery Corporation |
Certains types d'entites chimiques, compositions et methode de modulation de trpv1
|
JPWO2007069565A1
(ja)
|
2005-12-12 |
2009-05-21 |
小野薬品工業株式会社 |
二環式複素環化合物
|
US20090281075A1
(en)
|
2006-02-17 |
2009-11-12 |
Pharmacopeia, Inc. |
Isomeric purinones and 1h-imidazopyridinones as pkc-theta inhibitors
|
WO2007096764A2
(fr)
|
2006-02-27 |
2007-08-30 |
Glenmark Pharmaceuticals S.A. |
Dérivés d'hétéroaryles bicycliques en tant que modulateurs des récepteurs cannabinoïdes
|
US20090304821A1
(en)
|
2006-03-08 |
2009-12-10 |
Takeda Pharmaceutical Company Limited |
Pharmaceutical Combination
|
CN101410397A
(zh)
|
2006-03-31 |
2009-04-15 |
诺瓦提斯公司 |
有机化合物
|
EP2023919A4
(fr)
|
2006-05-08 |
2010-12-22 |
Molecular Neuroimaging Llc |
Composés et sondes amyloïdes de ceux-ci pour des utilisations thérapeutiques et en imagerie
|
EP2035005A4
(fr)
|
2006-06-09 |
2011-07-06 |
Kemia Inc |
Thérapie à base d'inhibiteurs de cytokine
|
US20080280891A1
(en)
|
2006-06-27 |
2008-11-13 |
Locus Pharmaceuticals, Inc. |
Anti-cancer agents and uses thereof
|
CN101790527A
(zh)
|
2006-07-20 |
2010-07-28 |
凯利普西斯公司 |
Rho激酶的苯并噻吩抑制剂
|
DE102006035018B4
(de)
|
2006-07-28 |
2009-07-23 |
Novaled Ag |
Oxazol-Triplett-Emitter für OLED-Anwendungen
|
WO2008021745A2
(fr)
|
2006-08-16 |
2008-02-21 |
Itherx Pharmaceuticals, Inc. |
Inhibiteurs de la pénétration du virus de l'hépatite c
|
TWI389895B
(zh)
|
2006-08-21 |
2013-03-21 |
Infinity Discovery Inc |
抑制bcl蛋白質與結合夥伴間之交互作用的化合物及方法
|
US7563797B2
(en)
|
2006-08-28 |
2009-07-21 |
Forest Laboratories Holding Limited |
Substituted imidazo(1,2-A)pyrimidines and imidazo(1,2-A) pyridines as cannabinoid receptor ligands
|
AR063706A1
(es)
|
2006-09-11 |
2009-02-11 |
Cgi Pharmaceuticals Inc |
Determinadas amidas sustituidas, el uso de las mismas para el tratamiento de enfermedades mediadas por la inhibicion de la actividad de btk y composiciones farmaceuticas que las comprenden.
|
PE20081370A1
(es)
|
2006-09-11 |
2008-11-28 |
Cgi Pharmaceuticals Inc |
Determinadas amidas sustituidas, metodo de elaboracion y metodo de uso de las mismas
|
NZ575389A
(en)
|
2006-09-11 |
2012-03-30 |
Mylan Lab Ltd |
Dibenzofuran derivatives as inhibitors of pde-4 and pde-10
|
US7838523B2
(en)
|
2006-09-11 |
2010-11-23 |
Cgi Pharmaceuticals, Inc. |
Certain substituted amides, method of making, and method of use thereof
|
JP2010502751A
(ja)
|
2006-09-11 |
2010-01-28 |
シージーアイ ファーマシューティカルズ,インコーポレイティド |
キナーゼ阻害物質、およびキナーゼ阻害物質の使用および同定方法
|
FR2906250B1
(fr)
|
2006-09-22 |
2008-10-31 |
Sanofi Aventis Sa |
Derives de 2-aryl-6phenyl-imidazo(1,2-a) pyridines, leur preparation et leur application en therapeutique
|
JP2010507674A
(ja)
|
2006-10-27 |
2010-03-11 |
ワイス エルエルシー |
マトリクスメタロプロテアーゼ阻害剤としての三環式化合物
|
CA2669266C
(fr)
|
2006-11-08 |
2014-04-29 |
Bristol-Myers Squibb Company |
Composes de pyridinone
|
GB0623209D0
(en)
|
2006-11-21 |
2007-01-03 |
F2G Ltd |
Antifungal agents
|
WO2008064318A2
(fr)
|
2006-11-22 |
2008-05-29 |
University Of Medicine And Dentistry Of New Jersey |
Composés actifs de récepteurs opioïdes périphériques
|
WO2008064317A1
(fr)
|
2006-11-22 |
2008-05-29 |
University Of Medicine And Dentistry Of New Jersey |
Composés actifs de récepteurs opioïdes lipophiles
|
EP2102177A1
(fr)
|
2006-12-14 |
2009-09-23 |
Boehringer Ingelheim International GmbH |
Benzoxasoles utiles dans le traitement de l'inflammation
|
WO2008079965A1
(fr)
|
2006-12-22 |
2008-07-03 |
Incyte Corporation |
Hétérocycles substitués servant d'inhibiteurs de janus kinases
|
EP1964840A1
(fr)
|
2007-02-28 |
2008-09-03 |
sanofi-aventis |
Imidazo[1,2-a]pyridines et leur utilisation en tant que produits pharmaceutiques
|
WO2008104077A1
(fr)
|
2007-02-28 |
2008-09-04 |
Methylgene Inc. |
Inhibiteurs à petite molécule de protéines arginine méthyltransférases (prmt)
|
EP1964841A1
(fr)
|
2007-02-28 |
2008-09-03 |
sanofi-aventis |
Imidazo[1,2-a]azine et son utilisation en tant que produit pharmaceutique
|
JP2008218327A
(ja)
|
2007-03-07 |
2008-09-18 |
Hitachi Ltd |
電解質、電解質膜、それを用いた膜電極接合体、燃料電池電源及び燃料電池電源システム
|
JP2010120852A
(ja)
|
2007-03-09 |
2010-06-03 |
Daiichi Sankyo Co Ltd |
新規なジアミド誘導体
|
WO2008114002A1
(fr)
|
2007-03-22 |
2008-09-25 |
Astrazeneca Ab |
Dérivés de quinoléine destinés au traitement de maladies inflammatoires
|
TW200902526A
(en)
|
2007-04-24 |
2009-01-16 |
Shionogi & Amp Co Ltd |
Aminodihydrothiazin derivative substituted with a cyclic group
|
JP5383483B2
(ja)
|
2007-04-24 |
2014-01-08 |
塩野義製薬株式会社 |
アルツハイマー症治療用医薬組成物
|
WO2008134553A1
(fr)
|
2007-04-26 |
2008-11-06 |
Xenon Pharmaceuticals Inc. |
Procédés de traitement de maladies associées aux canaux sodiques au moyen de composés bicycliques
|
CN101855222A
(zh)
|
2007-05-10 |
2010-10-06 |
通用电气健康护理有限公司 |
对大麻素cb2受体具有活性的咪唑并(1,2-a)吡啶和相关化合物
|
WO2009027733A1
(fr)
|
2007-08-24 |
2009-03-05 |
Astrazeneca Ab |
Dérivés de (2-pyridin-3-ylimidazo[1,2-b]pyridazin-6-yl)urée en tant qu'agents antibactériens
|
EP2188252B1
(fr)
|
2007-09-20 |
2011-04-13 |
Amgen Inc. |
Derives du 1-(4-(4-benzylbenzamido)-benzyl)azetidine-3-acide carboxylique et composes similaires en tant que modulateurs du rezepteur s1p pour le traitement de maladies immunologiques
|
CL2008002793A1
(es)
|
2007-09-20 |
2009-09-04 |
Cgi Pharmaceuticals Inc |
Compuestos derivados de amidas sustituidas, inhibidores de la actividad de btk; composicion farmaceutica que los comprende; utiles en el tratamiento del cancer, trastornos oseos, enfermedades autoinmunes, entre otras
|
DE102007048716A1
(de)
|
2007-10-11 |
2009-04-23 |
Merck Patent Gmbh |
Imidazo[1,2-a]pyrimidinderivate
|
TW200932219A
(en)
|
2007-10-24 |
2009-08-01 |
Astellas Pharma Inc |
Oxadiazolidinedione compound
|
KR20100089090A
(ko)
|
2007-10-25 |
2010-08-11 |
아스트라제네카 아베 |
세포 증식 장애의 치료에 유용한 피리딘 및 피라진 유도체
|
US7868001B2
(en)
|
2007-11-02 |
2011-01-11 |
Hutchison Medipharma Enterprises Limited |
Cytokine inhibitors
|
WO2009062059A2
(fr)
|
2007-11-08 |
2009-05-14 |
Pharmacopeia, Inc. |
Purinones et 1h-imidazopyridinones isomères comme inhibiteurs de pkc-thêta
|
JP5489296B2
(ja)
|
2007-12-13 |
2014-05-14 |
メルク・シャープ・アンド・ドーム・コーポレーション |
Janusキナーゼの阻害剤
|
RU2364597C1
(ru)
|
2007-12-14 |
2009-08-20 |
Андрей Александрович Иващенко |
ГЕТЕРОЦИКЛИЧЕСКИЕ ИНГИБИТОРЫ Hh-СИГНАЛЬНОГО КАСКАДА, ЛЕКАРСТВЕННЫЕ КОМПОЗИЦИИ НА ИХ ОСНОВЕ И СПОСОБ ЛЕЧЕНИЯ ЗАБОЛЕВАНИЙ, СВЯЗАННЫХ С АББЕРАНТНОЙ АКТИВНОСТЬЮ Hh СИГНАЛЬНОЙ СИСТЕМЫ
|
US8410145B2
(en)
|
2007-12-19 |
2013-04-02 |
Syngenta Crop Protection Llc |
Insecticidal compounds
|
AU2008345225A1
(en)
|
2007-12-21 |
2009-07-09 |
University Of Rochester |
Method for altering the lifespan of eukaryotic organisms
|
JP2011506487A
(ja)
|
2007-12-21 |
2011-03-03 |
ザ・ユニバーシティ・オブ・シドニー |
トランスロケータータンパク質リガンド
|
AU2009205072C1
(en)
|
2008-01-18 |
2016-10-13 |
Eisai R & D Management Co., Ltd. |
Condensed aminodihydrothiazine derivative
|
JP5381718B2
(ja)
|
2008-01-31 |
2014-01-08 |
コニカミノルタ株式会社 |
ハロ多環芳香族化合物及びその製造方法
|
US20110009429A1
(en)
|
2008-02-26 |
2011-01-13 |
Paul Oakley |
Heterocyclic compounds as inhibitors of cxcr2
|
EP2095818A1
(fr)
|
2008-02-29 |
2009-09-02 |
AEterna Zentaris GmbH |
Utilisation d'antagonistes LHRH dans des doses n'impliquant pas de castration
|
FR2928922B1
(fr)
|
2008-03-21 |
2010-04-23 |
Sanofi Aventis |
Derives de 2-aryl-6-phenyl-imidazo°1,2-a!pyridines polysubstitues, leur preparation et leur application en therapeutique
|
FR2928924B1
(fr)
|
2008-03-21 |
2010-04-23 |
Sanofi Aventis |
Derives polysubstitues de 6-heteroaryle-imidazo°1,2-a! pyridines, leur preparation et leur application en therapeutique
|
FR2928921B1
(fr)
|
2008-03-21 |
2010-04-23 |
Sanofi Aventis |
Derives polysubstitues de 2-aryl-6-phenyl-imidazo°1,2-a!pyridines, leur preparation et leur application en therapeutique
|
EP2271646A1
(fr)
|
2008-03-31 |
2011-01-12 |
Takeda Pharmaceutical Company Limited |
Inhibiteurs de kinase 1 de régulation de signal d'apoptose
|
KR101034351B1
(ko)
|
2008-05-14 |
2011-05-16 |
한국화학연구원 |
신규 벤즈옥사졸로 치환된 피리딘 유도체 또는 이의약학적으로 허용가능한 염, 이의 제조방법 및 이를유효성분으로 함유하는 이상세포 성장 질환의 예방 및치료용 약학적 조성물
|
CA2724842A1
(fr)
|
2008-05-19 |
2009-11-26 |
Sunovion Pharmaceuticals Inc. |
Composes imidazo[1,2-a]pyridines
|
CA2726262A1
(fr)
|
2008-05-29 |
2009-12-03 |
Sirtris Pharmaceuticals, Inc. |
Imidazopyridine et analogues lies en tant que modulateurs de la sirtuine
|
EP2280946B1
(fr)
|
2008-06-05 |
2016-02-10 |
Glaxo Group Limited |
Dérivés de 4-carboxamide indazole utiles en tant qu'inhibiteurs de p13 kinases
|
EP2323665B1
(fr)
|
2008-07-24 |
2013-06-19 |
Bristol-Myers Squibb Company |
Composés hétérocycliques condensés utiles en tant que modulateurs de kinases
|
US9540322B2
(en)
|
2008-08-18 |
2017-01-10 |
Yale University |
MIF modulators
|
US9643922B2
(en)
|
2008-08-18 |
2017-05-09 |
Yale University |
MIF modulators
|
JP2011231017A
(ja)
|
2008-09-09 |
2011-11-17 |
Nissan Chem Ind Ltd |
光学活性エポキシ化合物及び光学活性スルホキシド化合物の製造方法、並びに該方法に用いる配位子、錯体及び該錯体の製造方法
|
EP2365970B1
(fr)
|
2008-11-12 |
2018-03-21 |
Gilead Connecticut, Inc. |
Pyridazinones et leur utilisation comme inhibiteurs btk
|
ES2403633T3
(es)
|
2008-12-04 |
2013-05-20 |
Proximagen Limited |
Compuestos de imidazopiridina
|
CN102325752B
(zh)
|
2008-12-19 |
2015-02-04 |
百时美施贵宝公司 |
咔唑和咔啉激酶抑制剂
|
AU2009335821A1
(en)
|
2008-12-19 |
2010-07-15 |
Bristol-Myers Squibb Company |
Carbazole carboxamide compounds useful as kinase inhibitors
|
ES2539620T3
(es)
|
2008-12-19 |
2015-07-02 |
Cephalon, Inc. |
Pirrolotriazina como inhibidor de ALK y de JAK2
|
JP5624275B2
(ja)
|
2008-12-22 |
2014-11-12 |
ユー・ディー・シー アイルランド リミテッド |
有機電界発光素子
|
RU2505540C2
(ru)
|
2008-12-23 |
2014-01-27 |
Эббви Инк. |
Антивирусные соединения
|
JP5578490B2
(ja)
|
2008-12-26 |
2014-08-27 |
味の素株式会社 |
ピラゾロピリミジン化合物
|
JP2010202530A
(ja)
|
2009-02-27 |
2010-09-16 |
Tokyo Institute Of Technology |
含ヘテロ芳香族化合物および光学材料
|
KR20100101055A
(ko)
|
2009-03-07 |
2010-09-16 |
주식회사 메디젠텍 |
세포핵에서 세포질로의 gsk3의 이동을 억제하는 화합물을 함유하는 세포핵에서 세포질로의 gsk3 이동 관련 질환의 치료 또는 예방용 약학적 조성물
|
MY159575A
(en)
|
2009-04-02 |
2017-01-13 |
Merck Serono Sa |
Dihydroorotate dehydrogenase inhibitors
|
WO2010119264A1
(fr)
|
2009-04-16 |
2010-10-21 |
Centro Nacional De Investigaciones Oncólogicas (Cnio) |
Imidazopyrazines pour une utilisation en tant qu'inhibiteurs de kinase
|
US8338441B2
(en)
|
2009-05-15 |
2012-12-25 |
Gilead Sciences, Inc. |
Inhibitors of human immunodeficiency virus replication
|
US8993604B2
(en)
|
2009-06-30 |
2015-03-31 |
Siga Technologies, Inc. |
Treatment and prevention of dengue virus infections
|
AU2010266570A1
(en)
|
2009-06-30 |
2012-01-19 |
Siga Technologies, Inc. |
Treatment and prevention of Dengue virus infections
|
TWI625121B
(zh)
|
2009-07-13 |
2018-06-01 |
基利科學股份有限公司 |
調節細胞凋亡信號之激酶的抑制劑
|
JP2011057661A
(ja)
|
2009-08-14 |
2011-03-24 |
Bayer Cropscience Ag |
殺虫性カルボキサミド類
|
UA108363C2
(uk)
|
2009-10-08 |
2015-04-27 |
|
Похідні імінотіадіазиндіоксиду як інгібітори bace, композиція на їх основі і їх застосування
|
US9095596B2
(en)
|
2009-10-15 |
2015-08-04 |
Southern Research Institute |
Treatment of neurodegenerative diseases, causation of memory enhancement, and assay for screening compounds for such
|
MX349718B
(es)
|
2009-10-16 |
2017-08-10 |
Melinta Therapeutics Inc |
Compuestos antimicrobianos y metodos para fabricar y utilizar los mismos.
|
WO2011050245A1
(fr)
|
2009-10-23 |
2011-04-28 |
Yangbo Feng |
Hétéroaryles bicycliques formant inhibiteurs de la kinase
|
WO2011078221A1
(fr)
|
2009-12-24 |
2011-06-30 |
味の素株式会社 |
Composés d'imidazopyridazine
|
US20130022629A1
(en)
*
|
2010-01-04 |
2013-01-24 |
Sharpe Arlene H |
Modulators of Immunoinhibitory Receptor PD-1, and Methods of Use Thereof
|
WO2011097607A1
(fr)
|
2010-02-08 |
2011-08-11 |
Southern Research Institute |
Traitement antiviral et dosage pour cribler des antiviraux
|
TW201136919A
(en)
|
2010-03-02 |
2011-11-01 |
Merck Sharp & Amp Dohme Corp |
Inhibitors of hepatitis C virus NS5B polymerase
|
EP2542076B1
(fr)
|
2010-03-04 |
2021-01-13 |
Merck Sharp & Dohme Corp. |
Inhibiteurs de catéchol o-méthyl transférase et utilisation associée dans le traitement de troubles psychotiques
|
SG10201502109VA
(en)
|
2010-03-18 |
2015-05-28 |
Pasteur Institut Korea |
Anti-infective compounds
|
US8410117B2
(en)
|
2010-03-26 |
2013-04-02 |
Hoffmann-La Roche Inc. |
Imidazopyrimidine derivatives
|
EP2582668B1
(fr)
|
2010-06-16 |
2016-01-13 |
Bristol-Myers Squibb Company |
Composes carboline carboxamide utiles en tant qu'inhibiteurs de kinase
|
CN102295642B
(zh)
|
2010-06-25 |
2016-04-06 |
中国人民解放军军事医学科学院毒物药物研究所 |
2-芳基咪唑并[1,2-a]吡啶-3-乙酰胺衍生物、其制备方法及用途
|
EP2402345A1
(fr)
|
2010-06-29 |
2012-01-04 |
Basf Se |
Composés pyrazoliques bicycliques condenses
|
CN101891895B
(zh)
|
2010-07-28 |
2011-11-30 |
南京航空航天大学 |
基于桥联双水杨醛结构的苯并噻唑类金属配位聚合物及其制法及应用
|
WO2012016133A2
(fr)
|
2010-07-29 |
2012-02-02 |
President And Fellows Of Harvard College |
Inhibiteurs de la ros1 kinase pour le traitement de glioblastome et d'autres cancers déficients en p53
|
US8633200B2
(en)
|
2010-09-08 |
2014-01-21 |
Bristol-Myers Squibb Company |
Inhibitors of human immunodeficiency virus replication
|
CN101993415B
(zh)
|
2010-09-15 |
2013-08-14 |
北京韩美药品有限公司 |
作为Hedgehog通路抑制剂的化合物以及包含该化合物的药物组合物及其应用
|
US8921381B2
(en)
|
2010-10-04 |
2014-12-30 |
Baruch S. Blumberg Institute |
Inhibitors of secretion of hepatitis B virus antigens
|
EP2444084A1
(fr)
|
2010-10-21 |
2012-04-25 |
Centro Nacional de Investigaciones Oncológicas (CNIO) |
Utilisation d'inhibiteurs de PI3K pour le traitement de l'obésité
|
WO2012052745A1
(fr)
|
2010-10-21 |
2012-04-26 |
Centro Nacional De Investigaciones Oncológicas (Cnio) |
Combinaisons d'inhibiteurs de pi3k avec un second agent antitumoral
|
CN103282034A
(zh)
|
2010-11-18 |
2013-09-04 |
利亘制药公司 |
造血生长因子模拟物的用途
|
UY33808A
(es)
|
2010-12-17 |
2012-07-31 |
Syngenta Participations Ag |
Compuestos insecticidas
|
TWI617559B
(zh)
|
2010-12-22 |
2018-03-11 |
江蘇恆瑞醫藥股份有限公司 |
2-芳基咪唑并[1,2-b]嗒.2-苯基咪唑并[1,2-a]吡啶,和2-苯基咪唑并[1,2-a]吡衍生物
|
EP2661433B1
(fr)
|
2011-01-04 |
2017-08-16 |
Novartis AG |
Composes d'indole ou de ses analogues utiles pour le traitement de la degenerescence maculaire liee a l'age (dma)
|
US9018395B2
(en)
|
2011-01-27 |
2015-04-28 |
Université de Montréal |
Pyrazolopyridine and pyrazolopyrimidine derivatives as melanocortin-4 receptor modulators
|
US8921368B2
(en)
|
2011-03-17 |
2014-12-30 |
Bristol-Myers Squibb Company |
Pyrrolopyridazine JAK3 inhibitors and their use for the treatment of inflammatory and autoimmune diseases
|
US9464065B2
(en)
|
2011-03-24 |
2016-10-11 |
The Scripps Research Institute |
Compounds and methods for inducing chondrogenesis
|
RU2013150349A
(ru)
|
2011-04-13 |
2015-05-20 |
Мерк Шарп И Доум Корп. |
5-замещенные иминотиазины и их моно- и диоксиды в качестве ингибиторов васе, содержащие их композиции и их применение
|
CN102796103A
(zh)
|
2011-05-23 |
2012-11-28 |
南京英派药业有限公司 |
6-(芳基甲酰)咪唑并[1,2-a]嘧啶和6-(芳基甲酰)[1,2,4]三唑并[4,3-a]嘧啶作为Hedgehog抑制剂及其应用
|
DK2713722T3
(en)
|
2011-05-31 |
2017-07-03 |
Celgene Int Ii Sarl |
Newly known GLP-1 receptor stabilizers and modulators
|
GB201109763D0
(en)
|
2011-06-10 |
2011-07-27 |
Ucl Business Plc |
Compounds
|
WO2012175991A1
(fr)
|
2011-06-24 |
2012-12-27 |
Pharminox Limited |
Composés pentacycliques fusionnés anti-prolifératifs
|
EP2729466B1
(fr)
|
2011-07-08 |
2015-08-19 |
Novartis AG |
Nouveaux dérivés de pyrrolopyrimidine
|
EP2548877A1
(fr)
|
2011-07-19 |
2013-01-23 |
MSD Oss B.V. |
Dérivés de 4-(pyridine condensée à 5 chaînons)benzamide comme inhibiteurs de BTK
|
WO2013033901A1
(fr)
|
2011-09-08 |
2013-03-14 |
Merck Sharp & Dohme Corp. |
Dérivés benzofuranes substitués par un hétérocycle et leurs procédés d'utilisation pour le traitement de maladies virales
|
WO2013040528A1
(fr)
|
2011-09-16 |
2013-03-21 |
Microbiotix, Inc. |
Composés antimicrobiens
|
WO2013043521A1
(fr)
|
2011-09-22 |
2013-03-28 |
Merck Sharp & Dohme Corp. |
Composés pyrazolopyridyle à utiliser en tant qu'inhibiteurs de l'aldostérone synthase
|
JP6040677B2
(ja)
|
2011-09-29 |
2016-12-07 |
東洋インキScホールディングス株式会社 |
太陽電池封止材用樹脂組成物
|
MX2014004479A
(es)
|
2011-10-13 |
2014-08-01 |
Novartis Ag |
Derivados de oxazina novedosos y su uso en el tratamiento de enfermedades.
|
US20140288052A1
(en)
|
2011-10-20 |
2014-09-25 |
GlaxoSmithKline, LLC |
Substituted bicyclic aza-heterocycles and analogues as sirtuin modulators
|
PH12014500855A1
(en)
|
2011-10-21 |
2014-05-19 |
Torrent Pharmaceuticals Ltd |
Novel substituted imidazopyrimidines as gpbar1 receptor modulators
|
WO2013120040A1
(fr)
|
2012-02-10 |
2013-08-15 |
Children's Medical Center Corporation |
Inhibition d'une voie ciblée pour améliorer la structure, le fonctionnement et l'activité musculaires dans la dystrophie musculaire
|
US9034882B2
(en)
|
2012-03-05 |
2015-05-19 |
Bristol-Myers Squibb Company |
Inhibitors of human immunodeficiency virus replication
|
CN104169260A
(zh)
|
2012-03-09 |
2014-11-26 |
卡尔那生物科学株式会社 |
新三嗪衍生物
|
WO2013157021A1
(fr)
|
2012-04-20 |
2013-10-24 |
Advinus Therapeutics Limited |
Composés bicycliques, compositions et applications médicinales de ceux-ci
|
JP5911638B2
(ja)
|
2012-04-20 |
2016-04-27 |
ギリアード サイエンシーズ, インコーポレイテッド |
ベンゾチアゾール−6−イル酢酸誘導体およびhiv感染を処置するためのそれらの使用
|
WO2013163404A1
(fr)
|
2012-04-27 |
2013-10-31 |
The Uab Research Foundation |
Traitement d'infections virales avec arn viraux traduits par un mécanisme non médié par l'ires
|
CN104379567A
(zh)
|
2012-06-18 |
2015-02-25 |
住友化学株式会社 |
稠合杂环化合物
|
US9630976B2
(en)
|
2012-07-03 |
2017-04-25 |
Ono Pharmaceutical Co., Ltd. |
Compound having agonistic activity on somatostatin receptor, and use thereof for medical purposes
|
GB201212513D0
(en)
|
2012-07-13 |
2012-08-29 |
Ucb Pharma Sa |
Therapeutic agents
|
JP6259823B2
(ja)
|
2012-07-13 |
2018-01-10 |
ユーシービー バイオファルマ エスピーアールエル |
Tnf活性の調節物質としてのイミダゾピリジン誘導体
|
JP2015178457A
(ja)
|
2012-07-25 |
2015-10-08 |
杏林製薬株式会社 |
ピラゾロピリジン誘導体、またはその薬理学的に許容される塩
|
US9428511B2
(en)
|
2012-09-06 |
2016-08-30 |
Bristol-Myers Squibb Company |
Imidazopyridazine JAK3 inhibitors and their use for the treatment of inflammatory and autoimmune diseases
|
MX2015003513A
(es)
|
2012-09-26 |
2015-07-17 |
Hoffmann La Roche |
Compuestos ciclicos eter pirazol-4-il-heterociclil-carboxamida y metodos de utilizacion.
|
WO2014061693A1
(fr)
|
2012-10-17 |
2014-04-24 |
塩野義製薬株式会社 |
Nouveau dérivé carbocyclique non aromatique ou hétérocyclique non aromatique
|
EP2922548A4
(fr)
|
2012-11-21 |
2016-06-01 |
Stategics Inc |
Composés triazolo-pyrimidines substitués pour la modulation de la prolifération, la différentiation et la survie cellulaires
|
JP6037804B2
(ja)
|
2012-12-03 |
2016-12-07 |
富士フイルム株式会社 |
ガス分離膜
|
SMT202000244T1
(it)
|
2013-01-15 |
2020-07-08 |
Incyte Holdings Corp |
Composti di tiazolocarbossammide e piridincarbossammide utili come inibitori di chinasi pim
|
EP2948446A1
(fr)
|
2013-01-22 |
2015-12-02 |
F. Hoffmann-La Roche AG |
Fluoro- [1,3]oxazines servant d'inhibiteurs de la bace1
|
CN103933036B
(zh)
|
2013-01-23 |
2017-10-13 |
中国人民解放军军事医学科学院毒物药物研究所 |
2‑芳基咪唑并[1,2‑α]吡啶‑3‑乙酰胺衍生物在制备防治PTSD的药物中的用途
|
US9657082B2
(en)
|
2013-01-31 |
2017-05-23 |
Thomas Jefferson University |
PD-L1 and PD-L2-based fusion proteins and uses thereof
|
WO2014133046A1
(fr)
|
2013-02-27 |
2014-09-04 |
持田製薬株式会社 |
Nouveau dérivé de pyrazole
|
AP2015008716A0
(en)
|
2013-03-08 |
2015-09-30 |
Amgen Inc |
Perfluorinated cyclopropyl fused 1,3-oxazin-2-amine compounds as beta-secretase inhibitors and methods of use
|
CN104045552B
(zh)
|
2013-03-13 |
2019-06-11 |
江苏先声药业有限公司 |
作为神经保护剂的药用化合物
|
BR112015022802A2
(pt)
|
2013-03-13 |
2017-07-18 |
Australian Nuclear Science & Tech Org |
animal não-humano transgênico, progênie do animal, método para identificação de um composto, método para seleção da especificidade ou seletividade de ligação de um composto candidato, célula, tecido ou linhagem celular imortalizada, uso da célula, tecido ou linhagem celular imortalizada, método para identificação de um composto, método para filtragem da especificidade ou seletividade de ligação de um composto candidato, e uso de um composto de fórmula geral
|
DK2968304T3
(en)
|
2013-03-14 |
2019-01-28 |
Univ Columbia |
4-PHENYLPIPERIDINES, THEIR PREPARATION AND USE.
|
JP2016512558A
(ja)
|
2013-03-14 |
2016-04-28 |
ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company |
ヒト免疫不全ウイルス複製の阻害剤
|
CA2906086A1
(fr)
|
2013-03-14 |
2014-09-25 |
Celtaxsys, Inc. |
Inhibiteurs de la leucotriene a4 hydrolase
|
CA2902594C
(fr)
|
2013-03-14 |
2023-01-10 |
Curadev Pharma Private Ltd. |
Inhibiteurs de la voie de la kynurenine
|
US9308236B2
(en)
|
2013-03-15 |
2016-04-12 |
Bristol-Myers Squibb Company |
Macrocyclic inhibitors of the PD-1/PD-L1 and CD80(B7-1)/PD-L1 protein/protein interactions
|
WO2014181287A1
(fr)
|
2013-05-09 |
2014-11-13 |
Piramal Enterprises Limited |
Composés hétérocyclyliques et leurs utilisations
|
KR102273997B1
(ko)
|
2013-06-26 |
2021-07-08 |
애브비 인코포레이티드 |
Btk 억제제로서 1급 카복스아미드
|
MX2015017821A
(es)
|
2013-07-02 |
2016-04-15 |
Syngenta Participations Ag |
Heterociclos bi-o triciclicos activos como plaguicidas con sustituyentes que contienen azufre.
|
SG10201800325PA
(en)
|
2013-07-17 |
2018-02-27 |
Otsuka Pharma Co Ltd |
Cyanotriazole compounds
|
WO2015013635A2
(fr)
|
2013-07-25 |
2015-01-29 |
Dana-Farber Cancer Institute, Inc. |
Inhibiteurs des facteurs de transcription et leurs utilisations
|
EP2835375A1
(fr)
|
2013-08-09 |
2015-02-11 |
Fundació Institut Català d'Investigació Química |
Composés salphen bis et composites de matériau carboné les comprenant
|
KR101715090B1
(ko)
|
2013-08-28 |
2017-03-13 |
한국화학연구원 |
신규한 화합물 또는 이의 약학적으로 허용가능한 염, 및 이를 유효성분으로 함유하는 인플루엔자 바이러스 감염으로 인한 질환의 예방 또는 치료용 약학적 조성물
|
CA2923184A1
(fr)
|
2013-09-04 |
2015-03-12 |
Bristol-Myers Squibb Company |
Composes utiles comme immunomodulateurs
|
EP3041827B1
(fr)
|
2013-09-06 |
2018-04-18 |
Aurigene Discovery Technologies Limited |
Dérivés 1,2,4-oxadiazole utilisés comme immunomodulateurs
|
EP3385257A1
(fr)
|
2013-09-06 |
2018-10-10 |
Aurigene Discovery Technologies Limited |
Dérivés 1,3,4-oxadiazole et 1,3,4-thiadiazole servant d'immunomodulateurs
|
WO2015036927A1
(fr)
|
2013-09-10 |
2015-03-19 |
Aurigene Discovery Technologies Limited |
Dérivés peptidomimétiques d'immunomodulation
|
JP6336870B2
(ja)
|
2013-09-30 |
2018-06-06 |
日本ポリプロ株式会社 |
ビフェノール化合物及びそれを用いるオレフィン重合用触媒並びにオレフィン重合体の製造方法
|
GB201321743D0
(en)
|
2013-12-09 |
2014-01-22 |
Ucb Pharma Sa |
Therapeutic agents
|
GB201321733D0
(en)
|
2013-12-09 |
2014-01-22 |
Ucb Pharma Sa |
Therapeutic agents
|
GB201321746D0
(en)
|
2013-12-09 |
2014-01-22 |
Ucb Pharma Sa |
Therapeutic agents
|
GB201321736D0
(en)
|
2013-12-09 |
2014-01-22 |
Ucb Pharma Sa |
Therapeutic agents
|
WO2015095337A2
(fr)
|
2013-12-18 |
2015-06-25 |
The Rockefeller University |
Dérivés pyrazolo [1,5-a]pyrimidine carboxamide pour le traitement de troubles cognitifs
|
RU2016131792A
(ru)
|
2014-01-03 |
2018-02-06 |
Байер Энимэл Хельс ГмбХ |
Новые пиразолил-гетероариламиды в качестве средств для борьбы с вредителями
|
EP3105251A4
(fr)
|
2014-02-10 |
2017-11-15 |
Merck Sharp & Dohme Corp. |
Anticorps qui se lient à la protéine tau humaine et dosage pour quantifier la protéine tau humaine au moyen des anticorps
|
AU2015223121A1
(en)
|
2014-02-25 |
2016-09-01 |
Achillion Pharmaceuticals, Inc. |
Amide compounds for treatment of complement mediated disorders
|
JP6490464B2
(ja)
|
2014-03-26 |
2019-03-27 |
三井化学株式会社 |
遷移金属化合物、オレフィン重合用触媒およびオレフィン系重合体の製造方法
|
JP6554117B2
(ja)
|
2014-04-04 |
2019-07-31 |
イオメット ファーマ リミテッド |
医療で使用されるインドール誘導体
|
US9850225B2
(en)
|
2014-04-14 |
2017-12-26 |
Bristol-Myers Squibb Company |
Compounds useful as immunomodulators
|
WO2015197028A1
(fr)
|
2014-06-28 |
2015-12-30 |
Sunshine Lake Pharma Co., Ltd. |
Composés en tant qu'inhibiteurs du virus de l'hépatite c (vhc) et leurs utilisations en médecine
|
CN104211726B
(zh)
|
2014-08-11 |
2017-06-16 |
中南民族大学 |
非茂类三齿双核钛配合物、制备方法及用途
|
US20170305922A1
(en)
|
2014-09-17 |
2017-10-26 |
Epizyme, Inc. |
Carm1 inhibitors and uses thereof
|
AU2015317566B2
(en)
|
2014-09-19 |
2019-10-10 |
Mackay Medical Foundation The Presbyterian Church In Taiwan Mackay Memorial Hospital |
Benzo-heterocyclic compounds and their applications
|
EP3204382B1
(fr)
*
|
2014-10-06 |
2021-12-01 |
Merck Patent GmbH |
Composés hétéroaryle servant d'inhibiteurs de la btk, et leurs utilisations
|
WO2016094688A1
(fr)
|
2014-12-10 |
2016-06-16 |
Massachusetts Institute Of Technology |
Dérivés fusionnés de 1,3-azole utiles pour le traitement de maladies prolifératives
|
JP6853619B2
(ja)
|
2015-01-16 |
2021-03-31 |
大塚製薬株式会社 |
シアノトリアゾール化合物の医薬用途
|
DE112016000383A5
(de)
|
2015-01-20 |
2017-10-05 |
Cynora Gmbh |
Organische Moleküle, insbesondere zur Verwendung in optoelektronischen Bauelementen
|
US10071998B2
(en)
|
2015-01-20 |
2018-09-11 |
Merck Sharp & Dohme Corp. |
Iminothiadiazine dioxides bearing an amine-linked substituent as BACE inhibitors, compositions, and their use
|
WO2016156282A1
(fr)
|
2015-04-02 |
2016-10-06 |
Bayer Cropscience Aktiengesellschaft |
Nouveaux composés de triazole pour contrôler des champignons nocifs phytopathogènes
|
WO2017035405A1
(fr)
|
2015-08-26 |
2017-03-02 |
Achillion Pharmaceuticals, Inc. |
Composés amino pour le traitement de troubles immunitaires et inflammatoires
|
US10745382B2
(en)
|
2015-10-15 |
2020-08-18 |
Bristol-Myers Squibb Company |
Compounds useful as immunomodulators
|
TW201718581A
(zh)
|
2015-10-19 |
2017-06-01 |
英塞特公司 |
作為免疫調節劑之雜環化合物
|
WO2017070320A1
(fr)
|
2015-10-21 |
2017-04-27 |
University Of Pittsburgh - Of The Commonwealth System Of Higher Education |
Inhibiteurs allostériques de phényl indole de l'atpase p97
|
KR101717601B1
(ko)
|
2015-11-10 |
2017-03-20 |
한국화학연구원 |
신규한 화합물 또는 이의 약학적으로 허용가능한 염, 및 이를 유효성분으로 함유하는 인플루엔자 바이러스 감염으로 인한 질환의 예방 또는 치료용 약학적 조성물
|
DK3377488T3
(da)
|
2015-11-19 |
2022-10-03 |
Incyte Corp |
Heterocykliske forbindelser som immunomodulatorer
|
TW201726623A
(zh)
|
2015-12-17 |
2017-08-01 |
英塞特公司 |
作為免疫調節劑之雜環化合物
|
SG10202111399YA
(en)
|
2015-12-22 |
2021-11-29 |
Immatics Biotechnologies Gmbh |
Peptides and combination of peptides for use in immunotherapy against breast cancer and other cancers
|
WO2017109041A1
(fr)
|
2015-12-22 |
2017-06-29 |
Synthon B.V. |
Composition pharmaceutique comprenant du lénalidomide amorphe et un antioxydant
|
WO2017107052A1
(fr)
|
2015-12-22 |
2017-06-29 |
Merck Sharp & Dohme Corp. |
Activateurs solubles de guanylate cyclase
|
WO2017108569A1
(fr)
|
2015-12-22 |
2017-06-29 |
Syngenta Participations Ag |
Dérivés de pyrazole à activité pesticide
|
ES2844374T3
(es)
|
2015-12-22 |
2021-07-22 |
Incyte Corp |
Compuestos heterocíclicos como inmunomoduladores
|
KR101653560B1
(ko)
|
2016-02-02 |
2016-09-12 |
한국화학연구원 |
신규한 화합물 또는 이의 약학적으로 허용가능한 염, 및 이를 유효성분으로 함유하는 인플루엔자 바이러스 감염으로 인한 질환의 예방 또는 치료용 약학적 조성물
|
CN109414410B
(zh)
|
2016-04-22 |
2022-08-12 |
因赛特公司 |
Lsd1抑制剂的制剂
|
TW201808950A
(zh)
|
2016-05-06 |
2018-03-16 |
英塞特公司 |
作為免疫調節劑之雜環化合物
|
ES2905980T3
(es)
|
2016-05-26 |
2022-04-12 |
Incyte Corp |
Compuestos heterocíclicos como inmunomoduladores
|
IL263429B
(en)
|
2016-06-20 |
2022-08-01 |
Novartis Ag |
Crystalline forms of triazolopyrimidine compound
|
MX2018016295A
(es)
|
2016-06-20 |
2019-09-16 |
Elanco Us Inc |
Interferon porcino pegilado y metodos de utilizacion del mismo.
|
PE20190731A1
(es)
|
2016-06-20 |
2019-05-23 |
Incyte Corp |
Compuestos heterociclicos como inmunomoduladores
|
JP7054529B2
(ja)
|
2016-06-21 |
2022-04-14 |
エックス4 ファーマシューティカルズ, インコーポレイテッド |
Cxcr4阻害剤およびその使用
|
ES2930092T3
(es)
|
2016-07-14 |
2022-12-07 |
Incyte Corp |
Compuestos heterocíclicos como inmunomoduladores
|
CN109195602B
(zh)
|
2016-08-03 |
2022-01-07 |
上海齐鲁制药研究中心有限公司 |
用作免疫调节剂的对称或半对称化合物
|
US20180057486A1
(en)
|
2016-08-29 |
2018-03-01 |
Incyte Corporation |
Heterocyclic compounds as immunomodulators
|
EP3506908A1
(fr)
|
2016-08-30 |
2019-07-10 |
Tetraphase Pharmaceuticals, Inc. |
Composés de tétracycline et méthodes de traitement
|
TWI795381B
(zh)
|
2016-12-21 |
2023-03-11 |
比利時商健生藥品公司 |
作為malt1抑制劑之吡唑衍生物
|
CA3046578A1
(fr)
|
2016-12-21 |
2018-06-28 |
Acerta Pharma B.V. |
Inhibiteurs de type imidazopyrazine de tyrosine kinase de bruton
|
ES2874756T3
(es)
|
2016-12-22 |
2021-11-05 |
Incyte Corp |
Derivados de triazolo[1,5-A]piridina como inmunomoduladores
|
MD3558990T2
(ro)
|
2016-12-22 |
2023-02-28 |
Incyte Corp |
Derivați tetrahidro imidazo[4,5-c]piridină ca inductori de internalizare a PD-L1
|
US20180179179A1
(en)
|
2016-12-22 |
2018-06-28 |
Incyte Corporation |
Heterocyclic compounds as immunomodulators
|
IL292677A
(en)
|
2016-12-22 |
2022-07-01 |
Calithera Biosciences Inc |
Compositions and methods for inhibiting arginase activity
|
WO2018119263A1
(fr)
|
2016-12-22 |
2018-06-28 |
Incyte Corporation |
Composés hétérocycliques utilisés en tant qu'inducteurs de l'internalisation de pd-l1
|
EP3558963B1
(fr)
|
2016-12-22 |
2022-03-23 |
Incyte Corporation |
Composés hétéroaromatiques bicycliques utilisés en tant qu'immunomodulateurs
|
IL295660A
(en)
|
2016-12-22 |
2022-10-01 |
Incyte Corp |
Benzooxazole derivatives as immunomodulators
|
JOP20180040A1
(ar)
|
2017-04-20 |
2019-01-30 |
Gilead Sciences Inc |
مثبطات pd-1/pd-l1
|
MA49701A
(fr)
|
2017-07-28 |
2020-06-03 |
Chemocentryx Inc |
Composés immunomodulateurs
|
JP7198269B2
(ja)
|
2017-08-08 |
2022-12-28 |
ケモセントリックス,インコーポレイティド |
大員環免疫調節剤
|
EP3669872A4
(fr)
|
2017-08-18 |
2021-05-05 |
Shanghai Ennovabio Pharmaceuticals Co., Ltd. |
Composé ayant une activité inhibitrice de pd-l1, sa méthode de préparation et son utilisation
|
FI3774791T3
(fi)
|
2018-03-30 |
2023-03-21 |
Incyte Corp |
Heterosyklisiä yhdisteitä immunomodulaattoreina
|
US20210040118A1
(en)
|
2018-04-03 |
2021-02-11 |
Betta Pharmaceuticals Co., Ltd |
Immunomodulators, compositions and methods thereof
|
JP7242702B2
(ja)
|
2018-04-19 |
2023-03-20 |
ギリアード サイエンシーズ, インコーポレイテッド |
Pd-1/pd-l1阻害剤
|
CN112752756B
(zh)
|
2018-05-11 |
2024-06-25 |
因赛特公司 |
作为PD-L1免疫调节剂的四氢-咪唑并[4,5-c]吡啶衍生物
|
EP3870566A1
(fr)
|
2018-10-24 |
2021-09-01 |
Gilead Sciences, Inc. |
Inhibiteurs de pd-1/pd-l1
|
SG11202105850YA
(en)
|
2018-11-02 |
2021-07-29 |
Shanghai Maxinovel Pharmaceuticals Co Ltd |
Diphenyl-like compound, intermediate thereof, preparation method therefor, pharmaceutical composition thereof and uses thereof
|
US12187713B2
(en)
|
2019-01-31 |
2025-01-07 |
Betta Pharmaceuticals Co., Ltd |
Immunomodulators, compositions and methods thereof
|
WO2021030162A1
(fr)
|
2019-08-09 |
2021-02-18 |
Incyte Corporation |
Sels d'un inhibiteur de pd-1/pd-l1
|
PH12022550754A1
(en)
|
2019-09-30 |
2023-08-23 |
Incyte Corp |
Pyrido[3,2-d]pyrimidine compounds as immunomodulators
|
KR20220101664A
(ko)
|
2019-11-11 |
2022-07-19 |
인사이트 코포레이션 |
Pd-1/pd-l1 억제제의 염 및 결정질 형태
|
AU2021373044A1
(en)
|
2020-11-06 |
2023-06-08 |
Incyte Corporation |
Process for making a pd-1/pd-l1 inhibitor and salts and crystalline forms thereof
|
WO2022099075A1
(fr)
|
2020-11-06 |
2022-05-12 |
Incyte Corporation |
Forme cristalline d'un inhibiteur pd-1/pd-l1
|
WO2022099018A1
(fr)
|
2020-11-06 |
2022-05-12 |
Incyte Corporation |
Procédé de préparation d'un inhibiteur de pd-1/pd-l1
|
US20220193050A1
(en)
|
2020-12-18 |
2022-06-23 |
Incyte Corporation |
Oral formulation for a pd-l1 inhibitor
|