ZA200401747B - 2-amino-6(2,4,5-substituted-phenyl)-pyridines for use as nitric oxide synthase inhibitors. - Google Patents
2-amino-6(2,4,5-substituted-phenyl)-pyridines for use as nitric oxide synthase inhibitors. Download PDFInfo
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- ZA200401747B ZA200401747B ZA200401747A ZA200401747A ZA200401747B ZA 200401747 B ZA200401747 B ZA 200401747B ZA 200401747 A ZA200401747 A ZA 200401747A ZA 200401747 A ZA200401747 A ZA 200401747A ZA 200401747 B ZA200401747 B ZA 200401747B
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- South Africa
- Prior art keywords
- disease
- ethyl
- methoxy
- pyridin
- compound
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Classifications
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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- C07—ORGANIC CHEMISTRY
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
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- Public Health (AREA)
- General Health & Medical Sciences (AREA)
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Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US32825301P | 2001-10-10 | 2001-10-10 |
Publications (1)
Publication Number | Publication Date |
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ZA200401747B true ZA200401747B (en) | 2005-03-03 |
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Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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ZA200401747A ZA200401747B (en) | 2001-10-10 | 2004-03-03 | 2-amino-6(2,4,5-substituted-phenyl)-pyridines for use as nitric oxide synthase inhibitors. |
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EP (1) | EP1434624B1 (es) |
JP (1) | JP2005506337A (es) |
KR (1) | KR20040053157A (es) |
CN (1) | CN1568207A (es) |
AP (1) | AP2004003003A0 (es) |
AR (1) | AR036763A1 (es) |
AT (1) | ATE344089T1 (es) |
BG (1) | BG108669A (es) |
BR (1) | BR0213193A (es) |
CA (1) | CA2463364A1 (es) |
CZ (1) | CZ2004450A3 (es) |
DE (1) | DE60215837T2 (es) |
DO (1) | DOP2002000467A (es) |
EA (1) | EA007074B1 (es) |
EC (1) | ECSP045055A (es) |
EE (1) | EE200400085A (es) |
ES (1) | ES2275917T3 (es) |
GT (1) | GT200200206A (es) |
HN (1) | HN2002000289A (es) |
HR (1) | HRP20040260A2 (es) |
HU (1) | HUP0401678A3 (es) |
IL (1) | IL161089A0 (es) |
IS (1) | IS7171A (es) |
MA (1) | MA27074A1 (es) |
MX (1) | MXPA04002313A (es) |
NO (1) | NO20041411L (es) |
NZ (1) | NZ531591A (es) |
OA (1) | OA12664A (es) |
PA (1) | PA8556101A1 (es) |
PE (1) | PE20030478A1 (es) |
PL (1) | PL369454A1 (es) |
SK (1) | SK1642004A3 (es) |
TN (1) | TNSN04057A1 (es) |
UY (1) | UY27476A1 (es) |
WO (1) | WO2003030993A1 (es) |
ZA (1) | ZA200401747B (es) |
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Publication number | Priority date | Publication date | Assignee | Title |
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US20030232739A1 (en) * | 2001-08-15 | 2003-12-18 | Pfizer Inc. | Pharmaceutical combinations comprising a NOS inhibitor and an NMDA receptor antagonist |
JP2008545616A (ja) * | 2005-02-21 | 2008-12-18 | プロキシマジェン エルティーディー | ジスキネジーの阻害または治療 |
AU2011347718B2 (en) * | 2010-12-24 | 2016-06-23 | Msd Oss B.V. | N-substituted azetidine derivatives |
RU2637503C1 (ru) * | 2016-12-30 | 2017-12-05 | Федеральное государственное автономное образовательное учреждение высшего образования "Национальный исследовательский Томский государственный университет" (ТГУ, НИ ТГУ) | Способ получения n2-метилдезоксигуанозина |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
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WO1997036871A1 (en) * | 1996-03-29 | 1997-10-09 | Pfizer Inc. | 6-phenylpyridyl-2-amine derivatives |
UA64740C2 (uk) * | 1997-02-10 | 2004-03-15 | Пфайзер Продактс Інк. | Похідні 2-амінопіридинів, фармацевтична композиція на їх основі (варіанти), спосіб лікування (варіанти), спосіб інгібування nos у ссавця та проміжні сполуки (варіанти) |
KR20020010916A (ko) * | 1999-05-21 | 2002-02-06 | 실버스타인 아써 에이. | Nos 억제제로서의 신규한 약학 혼합물 |
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2002
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- 2002-09-24 ES ES02775016T patent/ES2275917T3/es not_active Expired - Lifetime
- 2002-09-24 JP JP2003534022A patent/JP2005506337A/ja not_active Withdrawn
- 2002-09-24 PL PL02369454A patent/PL369454A1/xx not_active Application Discontinuation
- 2002-09-24 WO PCT/IB2002/003939 patent/WO2003030993A1/en active IP Right Grant
- 2002-09-24 CZ CZ2004450A patent/CZ2004450A3/cs unknown
- 2002-09-24 OA OA1200400093A patent/OA12664A/en unknown
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- 2002-09-24 KR KR10-2004-7005248A patent/KR20040053157A/ko not_active Application Discontinuation
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- 2002-09-24 EP EP02775016A patent/EP1434624B1/en not_active Expired - Lifetime
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- 2002-10-09 HN HN2002000289A patent/HN2002000289A/es unknown
- 2002-10-10 PA PA20028556101A patent/PA8556101A1/es unknown
- 2002-10-10 GT GT200200206A patent/GT200200206A/es unknown
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2004
- 2004-03-03 ZA ZA200401747A patent/ZA200401747B/en unknown
- 2004-03-04 IS IS7171A patent/IS7171A/is unknown
- 2004-03-17 HR HRP20040260 patent/HRP20040260A2/hr not_active Application Discontinuation
- 2004-04-02 NO NO20041411A patent/NO20041411L/no unknown
- 2004-04-06 BG BG108669A patent/BG108669A/xx unknown
- 2004-04-07 TN TNP2004000057A patent/TNSN04057A1/fr unknown
- 2004-04-08 MA MA27619A patent/MA27074A1/fr unknown
- 2004-04-08 EC EC2004005055A patent/ECSP045055A/es unknown
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