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SE0202241D0 - Novel Compounds - Google Patents

Novel Compounds

Info

Publication number
SE0202241D0
SE0202241D0 SE0202241A SE0202241A SE0202241D0 SE 0202241 D0 SE0202241 D0 SE 0202241D0 SE 0202241 A SE0202241 A SE 0202241A SE 0202241 A SE0202241 A SE 0202241A SE 0202241 D0 SE0202241 D0 SE 0202241D0
Authority
SE
Sweden
Prior art keywords
novel compounds
relates
present
pharmaceutical compounds
respiratory disorders
Prior art date
Application number
SE0202241A
Other languages
English (en)
Swedish (sv)
Inventor
Simon Teague
Hitesh Sanganee
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Priority to SE0202241A priority Critical patent/SE0202241D0/xx
Publication of SE0202241D0 publication Critical patent/SE0202241D0/xx
Priority to SE0203713A priority patent/SE0203713D0/xx
Priority to TW092118486A priority patent/TW200404778A/zh
Priority to DK03764279.0T priority patent/DK1551802T3/da
Priority to MXPA05000646A priority patent/MXPA05000646A/es
Priority to JP2004521364A priority patent/JP4791729B2/ja
Priority to SI200331737T priority patent/SI1551802T1/sl
Priority to CA002492445A priority patent/CA2492445A1/en
Priority to AT03764279T priority patent/ATE450506T1/de
Priority to CNB038199718A priority patent/CN1279023C/zh
Priority to EP03764279A priority patent/EP1551802B1/en
Priority to PT03764279T priority patent/PT1551802E/pt
Priority to BR0312729-0A priority patent/BR0312729A/pt
Priority to NZ537606A priority patent/NZ537606A/en
Priority to US10/521,325 priority patent/US7723373B2/en
Priority to DE60330372T priority patent/DE60330372D1/de
Priority to ES03764279T priority patent/ES2335491T3/es
Priority to AU2003251260A priority patent/AU2003251260B2/en
Priority to PCT/SE2003/001216 priority patent/WO2004007451A1/en
Priority to AR20030102585A priority patent/AR040498A1/es
Priority to IL16612105A priority patent/IL166121A0/xx
Priority to ZA200500170A priority patent/ZA200500170B/xx
Priority to NO20050828A priority patent/NO20050828L/no
Priority to CY20101100086T priority patent/CY1109760T1/el
Priority to US12/758,348 priority patent/US20100197756A1/en
Priority to JP2010166138A priority patent/JP2010280680A/ja
Priority to JP2011043693A priority patent/JP2011116770A/ja

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404Indoles, e.g. pindolol
    • A61K31/405Indole-alkanecarboxylic acids; Derivatives thereof, e.g. tryptophan, indomethacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/14Antitussive agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/16Central respiratory analeptics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/30Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Immunology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Cardiology (AREA)
  • Virology (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Urology & Nephrology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Transplantation (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Obesity (AREA)
SE0202241A 2002-07-17 2002-07-17 Novel Compounds SE0202241D0 (sv)

Priority Applications (27)

Application Number Priority Date Filing Date Title
SE0202241A SE0202241D0 (sv) 2002-07-17 2002-07-17 Novel Compounds
SE0203713A SE0203713D0 (sv) 2002-07-17 2002-12-13 Novel compounds
TW092118486A TW200404778A (en) 2002-07-17 2003-07-07 Novel compounds
PCT/SE2003/001216 WO2004007451A1 (en) 2002-07-17 2003-07-15 Indole-3-sulphur derivatives
BR0312729-0A BR0312729A (pt) 2002-07-17 2003-07-15 Novos derivados de indol-3-enxofre
US10/521,325 US7723373B2 (en) 2002-07-17 2003-07-15 Indole-3-sulphur derivatives
JP2004521364A JP4791729B2 (ja) 2002-07-17 2003-07-15 インドール−3−硫黄誘導体
SI200331737T SI1551802T1 (sl) 2002-07-17 2003-07-15 Indol žveplovi derivati
CA002492445A CA2492445A1 (en) 2002-07-17 2003-07-15 Indole-3-sulphur derivatives
AT03764279T ATE450506T1 (de) 2002-07-17 2003-07-15 Indol-3-schwefelderivate
CNB038199718A CN1279023C (zh) 2002-07-17 2003-07-15 吲哚-3-硫衍生物
EP03764279A EP1551802B1 (en) 2002-07-17 2003-07-15 Indole-3-sulphur derivatives
PT03764279T PT1551802E (pt) 2002-07-17 2003-07-15 Derivados de indole-3-enxofre
DK03764279.0T DK1551802T3 (da) 2002-07-17 2003-07-15 Indol-3-svovlderivater
NZ537606A NZ537606A (en) 2002-07-17 2003-07-15 Indole-2-sulphur derivatives and their use to treat prostaglandin D2 mediated diseases
MXPA05000646A MXPA05000646A (es) 2002-07-17 2003-07-15 Derivados de indol-3-azufre.
DE60330372T DE60330372D1 (de) 2002-07-17 2003-07-15 Indol-3-schwefelderivate
ES03764279T ES2335491T3 (es) 2002-07-17 2003-07-15 Derivados de indol-3-azufre.
AU2003251260A AU2003251260B2 (en) 2002-07-17 2003-07-15 Indole-3-sulphur derivatives
AR20030102585A AR040498A1 (es) 2002-07-17 2003-07-17 Indoles sustituidos utiles para el tratamiento de enfermedades respiratorias
IL16612105A IL166121A0 (en) 2002-07-17 2005-01-03 Indole-3-sulphur derivatives
ZA200500170A ZA200500170B (en) 2002-07-17 2005-01-07 Indole-3-sulphur derivatives.
NO20050828A NO20050828L (no) 2002-07-17 2005-02-16 lndol-3-svovelderivater
CY20101100086T CY1109760T1 (el) 2002-07-17 2010-01-28 Παραγωγα ινδολης-3-θειου
US12/758,348 US20100197756A1 (en) 2002-07-17 2010-04-12 Indole-3-Sulphur Derivatives
JP2010166138A JP2010280680A (ja) 2002-07-17 2010-07-23 インドール−3−硫黄誘導体
JP2011043693A JP2011116770A (ja) 2002-07-17 2011-03-01 インドール−3−硫黄誘導体

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0202241A SE0202241D0 (sv) 2002-07-17 2002-07-17 Novel Compounds
SE0203713A SE0203713D0 (sv) 2002-07-17 2002-12-13 Novel compounds

Publications (1)

Publication Number Publication Date
SE0202241D0 true SE0202241D0 (sv) 2002-07-17

Family

ID=30117585

Family Applications (2)

Application Number Title Priority Date Filing Date
SE0202241A SE0202241D0 (sv) 2002-07-17 2002-07-17 Novel Compounds
SE0203713A SE0203713D0 (sv) 2002-07-17 2002-12-13 Novel compounds

Family Applications After (1)

Application Number Title Priority Date Filing Date
SE0203713A SE0203713D0 (sv) 2002-07-17 2002-12-13 Novel compounds

Country Status (23)

Country Link
US (2) US7723373B2 (xx)
EP (1) EP1551802B1 (xx)
JP (3) JP4791729B2 (xx)
CN (1) CN1279023C (xx)
AR (1) AR040498A1 (xx)
AT (1) ATE450506T1 (xx)
AU (1) AU2003251260B2 (xx)
BR (1) BR0312729A (xx)
CA (1) CA2492445A1 (xx)
CY (1) CY1109760T1 (xx)
DE (1) DE60330372D1 (xx)
DK (1) DK1551802T3 (xx)
ES (1) ES2335491T3 (xx)
IL (1) IL166121A0 (xx)
MX (1) MXPA05000646A (xx)
NO (1) NO20050828L (xx)
NZ (1) NZ537606A (xx)
PT (1) PT1551802E (xx)
SE (2) SE0202241D0 (xx)
SI (1) SI1551802T1 (xx)
TW (1) TW200404778A (xx)
WO (1) WO2004007451A1 (xx)
ZA (1) ZA200500170B (xx)

Families Citing this family (81)

* Cited by examiner, † Cited by third party
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SE0201635D0 (sv) 2002-05-30 2002-05-30 Astrazeneca Ab Novel compounds
TW200307542A (en) * 2002-05-30 2003-12-16 Astrazeneca Ab Novel compounds
SE0202241D0 (sv) * 2002-07-17 2002-07-17 Astrazeneca Ab Novel Compounds
SE0301010D0 (sv) 2003-04-07 2003-04-07 Astrazeneca Ab Novel compounds
SE0301569D0 (sv) * 2003-05-27 2003-05-27 Astrazeneca Ab Novel compounds
RU2356889C2 (ru) 2003-07-17 2009-05-27 Плекссикон, Инк. Соединения, являющиеся активными по отношению к рецепторам, активируемым пролифератором пероксисом
US7348338B2 (en) 2003-07-17 2008-03-25 Plexxikon, Inc. PPAR active compounds
SE0302232D0 (sv) * 2003-08-18 2003-08-18 Astrazeneca Ab Novel Compounds
SA04250253B1 (ar) 2003-08-21 2009-11-10 استرازينيكا ايه بي احماض فينوكسي اسيتيك مستبدلة باعتبارها مركبات صيدلانية لعلاج الامراض التنفسية مثل الربو ومرض الانسداد الرئوي المزمن
CA2542716A1 (en) * 2003-10-14 2005-05-06 Oxagen Limited Compounds having crth2 antagonist activity
SE0303180D0 (sv) * 2003-11-26 2003-11-26 Astrazeneca Ab Novel compounds
SI1725553T1 (sl) 2004-03-11 2008-08-31 Actelion Pharmaceuticals Ltd Derivati tetrahidropiridoindola
GB0412914D0 (en) * 2004-06-10 2004-07-14 Oxagen Ltd Compounds
MY144903A (en) * 2004-06-17 2011-11-30 Novartis Ag Pyrrolopyridine derivatives and their use as crth2 antagonists
GB0415320D0 (en) 2004-07-08 2004-08-11 Astrazeneca Ab Novel compounds
GB0418830D0 (en) 2004-08-24 2004-09-22 Astrazeneca Ab Novel compounds
CN101052397B (zh) * 2004-08-26 2011-07-06 埃科特莱茵药品有限公司 2-硫烷基-苯并咪唑-1-基-乙酸衍生物
EP1805171A4 (en) 2004-09-21 2009-05-13 Wyeth Corp CRTH2 RECEPTOR ANTAGONISM DISPLAYING INDIGENOUS ACIDS AND APPLICATIONS THEREOF
CA2585334C (en) * 2004-10-27 2014-05-13 Janssen Pharmaceutica N.V. Indole derivatives useful as progesterone receptor modulators
UY29223A1 (es) 2004-11-23 2006-06-30 Astrazeneca Ab Ácidos fenoxiacéticos sustituidos, composiciones farmacéuticas que los contienen y procesos para su preparación
JP2008521829A (ja) * 2004-11-30 2008-06-26 プレキシコン,インコーポレーテッド Ppar活性化合物
WO2006060535A2 (en) * 2004-11-30 2006-06-08 Plexxikon, Inc. Indole derivatives for use as ppar active compounds
PL1833791T3 (pl) 2004-12-27 2011-12-30 Actelion Pharmaceuticals Ltd Pochodne 2,3,4,9-tetrahydro-1H-karbazolu jako antagonisty receptora CRTH2
GB0500604D0 (en) * 2005-01-13 2005-02-16 Astrazeneca Ab Novel process
JP5024039B2 (ja) * 2005-02-25 2012-09-12 小野薬品工業株式会社 インドール化合物およびその用途
GB0505048D0 (en) 2005-03-11 2005-04-20 Oxagen Ltd Compounds with PGD antagonist activity
ES2372701T3 (es) 2005-07-22 2012-01-25 Shionogi & Co., Ltd. Derivado de indol que tiene actividad antagonista del receptor de pgd2.
US7842692B2 (en) 2005-07-22 2010-11-30 Shionogi & Co., Ltd. Azaindole derivative having PGD2 receptor antagonistic activity
US20070027105A1 (en) 2005-07-26 2007-02-01 Alza Corporation Peroxide removal from drug delivery vehicle
EP1931658A2 (en) * 2005-09-07 2008-06-18 Plexxikon, Inc. 1 , 4 and 1 , 5-disubstituted indole derivatives for use as ppar active compounds
BRPI0615948A2 (pt) * 2005-09-07 2011-05-31 Plexxikon Inc composto ativo de ppar, sua composição, seu kit e seu uso
EP1937632A1 (en) 2005-10-06 2008-07-02 Astra Zeneca AB Novel compounds
TW200745003A (en) 2005-10-06 2007-12-16 Astrazeneca Ab Novel compounds
GB0525143D0 (en) 2005-12-09 2006-01-18 Novartis Ag Organic compounds
GB0526257D0 (en) 2005-12-22 2006-02-01 Novartis Ag Organic compounds
JP2009538289A (ja) * 2006-05-26 2009-11-05 アストラゼネカ・アクチエボラーグ ビアリールまたはヘテロアリール置換インドール
WO2007149312A2 (en) 2006-06-16 2007-12-27 The Trustees Of The University Of Pennsylvania Methods and compositions for inhibiting or reducing hair loss, acne, rosacea, prostate cancer, and bph
JP5270542B2 (ja) 2006-07-22 2013-08-21 オキサジェン リミテッド Crth2アンタゴニスト活性を有する化合物
KR101411820B1 (ko) 2006-08-07 2014-06-24 액테리온 파마슈티칼 리미티드 (3-아미노-1,2,3,4-테트라하이드로-9h-카르바졸-9-일)-아세트산 유도체
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