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PL2285410T3 - Inhibitor DPP-IV połączony z dodatkowym środkiem przeciwcukrzycowym, tabletki zawierające takie formulacje, ich zastosowanie i sposób wytwarzania - Google Patents

Inhibitor DPP-IV połączony z dodatkowym środkiem przeciwcukrzycowym, tabletki zawierające takie formulacje, ich zastosowanie i sposób wytwarzania

Info

Publication number
PL2285410T3
PL2285410T3 PL09728065T PL09728065T PL2285410T3 PL 2285410 T3 PL2285410 T3 PL 2285410T3 PL 09728065 T PL09728065 T PL 09728065T PL 09728065 T PL09728065 T PL 09728065T PL 2285410 T3 PL2285410 T3 PL 2285410T3
Authority
PL
Poland
Prior art keywords
dpp
tablets
formulations
preparation
antidiabetic agent
Prior art date
Application number
PL09728065T
Other languages
English (en)
Inventor
Thomas Friedl
Michael Braun
Kenji Egusa
Hikaru Fujita
Megumi Maruyama
Takaaki Nishioka
Original Assignee
Boehringer Ingelheim International Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39714040&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL2285410(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim International Gmbh filed Critical Boehringer Ingelheim International Gmbh
Publication of PL2285410T3 publication Critical patent/PL2285410T3/pl

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18—Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A—HUMAN NECESSITIES
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18—Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183—Amino acids, e.g. glycine, EDTA or aspartame
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    • A61K9/2022—Organic macromolecular compounds
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    • A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
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    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
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    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
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    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
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    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
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    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
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    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Inorganic Chemistry (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pain & Pain Management (AREA)
  • Child & Adolescent Psychology (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
PL09728065T 2008-04-03 2009-04-02 Inhibitor DPP-IV połączony z dodatkowym środkiem przeciwcukrzycowym, tabletki zawierające takie formulacje, ich zastosowanie i sposób wytwarzania PL2285410T3 (pl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP08154039 2008-04-03
US8734308P 2008-08-08 2008-08-08
PCT/EP2009/053978 WO2009121945A2 (en) 2008-04-03 2009-04-02 New formulations, tablets comprising such formulations, their use and process for their preparation
EP09728065.5A EP2285410B1 (en) 2008-04-03 2009-04-02 Dpp-iv inhibitor combined with a further antidiabetic agent, tablets comprising such formulations, their use and process for their preparation

Publications (1)

Publication Number Publication Date
PL2285410T3 true PL2285410T3 (pl) 2019-03-29

Family

ID=39714040

Family Applications (1)

Application Number Title Priority Date Filing Date
PL09728065T PL2285410T3 (pl) 2008-04-03 2009-04-02 Inhibitor DPP-IV połączony z dodatkowym środkiem przeciwcukrzycowym, tabletki zawierające takie formulacje, ich zastosowanie i sposób wytwarzania

Country Status (26)

Country Link
US (10) US9155705B2 (pl)
EP (3) EP2285410B1 (pl)
JP (2) JP5588428B2 (pl)
KR (3) KR101775942B1 (pl)
CN (4) CN106215190A (pl)
AR (1) AR071175A1 (pl)
AU (1) AU2009232043B2 (pl)
BR (1) BRPI0911273B8 (pl)
CA (1) CA2720450C (pl)
CO (1) CO6251277A2 (pl)
DK (1) DK2285410T3 (pl)
EA (2) EA038435B1 (pl)
EC (1) ECSP10010489A (pl)
ES (1) ES2696124T3 (pl)
HK (1) HK1149485A1 (pl)
IL (2) IL207497A0 (pl)
MA (1) MA32200B1 (pl)
MX (2) MX351232B (pl)
NZ (1) NZ587747A (pl)
PE (2) PE20091730A1 (pl)
PL (1) PL2285410T3 (pl)
TW (2) TW201509941A (pl)
UA (1) UA104136C2 (pl)
UY (1) UY31747A (pl)
WO (1) WO2009121945A2 (pl)
ZA (1) ZA201005664B (pl)

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* Cited by examiner, † Cited by third party
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US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US7501426B2 (en) 2004-02-18 2009-03-10 Boehringer Ingelheim International Gmbh 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
US7772191B2 (en) 2005-05-10 2010-08-10 Boehringer Ingelheim International Gmbh Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein
DE102005035891A1 (de) 2005-07-30 2007-02-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
EP1852108A1 (en) * 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG DPP IV inhibitor formulations
PE20110235A1 (es) 2006-05-04 2011-04-14 Boehringer Ingelheim Int Combinaciones farmaceuticas que comprenden linagliptina y metmorfina
NO347644B1 (no) 2006-05-04 2024-02-12 Boehringer Ingelheim Int Polymorfer
PE20090938A1 (es) 2007-08-16 2009-08-08 Boehringer Ingelheim Int Composicion farmaceutica que comprende un derivado de benceno sustituido con glucopiranosilo
SI2200606T1 (sl) 2007-09-10 2017-12-29 Janssen Pharmaceutica N.V. Postopek za pripravo spojin, uporabnih kot inhibitorjev SGLT
PE20091730A1 (es) * 2008-04-03 2009-12-10 Boehringer Ingelheim Int Formulaciones que comprenden un inhibidor de dpp4
UY32030A (es) 2008-08-06 2010-03-26 Boehringer Ingelheim Int "tratamiento para diabetes en pacientes inapropiados para terapia con metformina"
KR20200118243A (ko) 2008-08-06 2020-10-14 베링거 인겔하임 인터내셔날 게엠베하 메트포르민 요법이 부적합한 환자에서의 당뇨병 치료
KR20110067096A (ko) 2008-09-10 2011-06-21 베링거 인겔하임 인터내셔날 게엠베하 당뇨병 및 관련 상태를 치료하기 위한 병용 요법
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US9415016B2 (en) 2016-08-16
JP2013237707A (ja) 2013-11-28
KR20170056021A (ko) 2017-05-22
UY31747A (es) 2009-11-10
CA2720450A1 (en) 2009-10-08
EA038435B1 (ru) 2021-08-27
TW201509941A (zh) 2015-03-16
PE20091730A1 (es) 2009-12-10
TWI527816B (zh) 2016-04-01
US20240307403A1 (en) 2024-09-19
NZ587747A (en) 2013-01-25
DK2285410T3 (en) 2018-12-03
ECSP10010489A (es) 2010-10-30
JP5588428B2 (ja) 2014-09-10
US20150366812A1 (en) 2015-12-24
CN101983073A (zh) 2011-03-02
KR20160042174A (ko) 2016-04-18
UA104136C2 (ru) 2014-01-10
MX351232B (es) 2017-10-06
KR101775942B1 (ko) 2017-09-07
EA029395B1 (ru) 2018-03-30
US20110206766A1 (en) 2011-08-25
CA2720450C (en) 2017-01-03
US20170119773A1 (en) 2017-05-04
US20200069693A1 (en) 2020-03-05
EP2285410B1 (en) 2018-09-26
CO6251277A2 (es) 2011-02-21
JP5922068B2 (ja) 2016-05-24
CN106215190A (zh) 2016-12-14
PE20140960A1 (es) 2014-08-15
MA32200B1 (fr) 2011-04-01
CN103083672A (zh) 2013-05-08
US20230338386A1 (en) 2023-10-26
MX2010010819A (es) 2010-11-05
US20160310435A1 (en) 2016-10-27
CN113648422A (zh) 2021-11-16
BRPI0911273B8 (pt) 2021-05-25
EP3453403A1 (en) 2019-03-13
KR20110005690A (ko) 2011-01-18
ES2696124T3 (es) 2019-01-14
US20220378797A1 (en) 2022-12-01
WO2009121945A3 (en) 2009-12-03
AU2009232043B2 (en) 2014-09-25
IL225637A0 (en) 2013-06-27
AU2009232043A1 (en) 2009-10-08
EA201300121A1 (ru) 2014-12-30
KR101611314B1 (ko) 2016-04-11
JP2011516456A (ja) 2011-05-26
US20180289716A1 (en) 2018-10-11
HK1149485A1 (en) 2011-10-07
BRPI0911273B1 (pt) 2019-07-16
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