IL149100A0 - Heteroalkylamino-substituted bicyclic nitrogen heterocycles as inhibitors of p38 protein kinase - Google Patents

Heteroalkylamino-substituted bicyclic nitrogen heterocycles as inhibitors of p38 protein kinase

Info

Publication number: IL149100A0
Authority: IL; Israel
Prior art keywords: heteroalkylamino; inhibitors; protein kinase; substituted bicyclic; nitrogen heterocycles
Prior art date: 1999-10-21

Application number

IL14910000A

Other languages

English (en)

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-10-21

Filing date

2000-10-13

Publication date

2002-11-10

2000-10-13 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

2002-11-10 Publication of IL149100A0 publication Critical patent/IL149100A0/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Immunology (AREA)
Physical Education & Sports Medicine (AREA)
Rheumatology (AREA)
Virology (AREA)
Diabetes (AREA)
Pulmonology (AREA)
Oncology (AREA)
Neurosurgery (AREA)
Communicable Diseases (AREA)
Hematology (AREA)
Dermatology (AREA)
Orthopedic Medicine & Surgery (AREA)
Cardiology (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Ophthalmology & Optometry (AREA)
Tropical Medicine & Parasitology (AREA)
Pain & Pain Management (AREA)
Heart & Thoracic Surgery (AREA)
Hospice & Palliative Care (AREA)
Urology & Nephrology (AREA)
Molecular Biology (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Gastroenterology & Hepatology (AREA)

IL14910000A 1999-10-21 2000-10-13 Heteroalkylamino-substituted bicyclic nitrogen heterocycles as inhibitors of p38 protein kinase IL149100A0 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US16080399P	1999-10-21	1999-10-21
US21374300P	2000-06-22	2000-06-22
PCT/EP2000/010088 WO2001029042A1 (en)	1999-10-21	2000-10-13	Heteroalkylamino-substituted bicyclic nitrogen heterocycles as inhibitors of p38 protein kinase

Publications (1)

Publication Number	Publication Date
IL149100A0 true IL149100A0 (en)	2002-11-10

Family

ID=26857240

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL14910000A IL149100A0 (en)	1999-10-21	2000-10-13	Heteroalkylamino-substituted bicyclic nitrogen heterocycles as inhibitors of p38 protein kinase

Country Status (27)

Country	Link
US (1)	US6451804B1 (es)
EP (1)	EP1228070B1 (es)
JP (1)	JP3961830B2 (es)
KR (1)	KR100523120B1 (es)
CN (1)	CN1171889C (es)
AR (1)	AR026084A1 (es)
AT (1)	ATE353329T1 (es)
AU (1)	AU776250B2 (es)
BR (1)	BR0015243A (es)
CA (1)	CA2388142C (es)
CZ (1)	CZ20021744A3 (es)
DE (1)	DE60033307T2 (es)
ES (1)	ES2280247T3 (es)
HK (1)	HK1051039A1 (es)
HR (1)	HRP20020328A2 (es)
HU (1)	HUP0203564A3 (es)
IL (1)	IL149100A0 (es)
MA (1)	MA26837A1 (es)
MX (1)	MXPA02003950A (es)
NO (1)	NO20021781L (es)
NZ (1)	NZ518119A (es)
PE (1)	PE20010758A1 (es)
PL (1)	PL357502A1 (es)
RU (1)	RU2265606C2 (es)
TR (1)	TR200201057T2 (es)
WO (1)	WO2001029042A1 (es)
YU (1)	YU29102A (es)

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CA2492033A1 (en)	2002-07-09	2004-01-15	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Pharmaceutical compositions of anticholinergics and p38 kinase inhibitors in the treatment of respiratory diseases
US7196090B2 (en)	2002-07-25	2007-03-27	Warner-Lambert Company	Kinase inhibitors
ATE374201T1 (de) *	2002-08-06	2007-10-15	Hoffmann La Roche	6-alkoxypyridopyrimidine als inhibitoren der p-38-map-kinase
US7084270B2 (en) *	2002-08-14	2006-08-01	Hoffman-La Roche Inc.	Pyrimido compounds having antiproliferative activity
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US7112676B2 (en)	2002-11-04	2006-09-26	Hoffmann-La Roche Inc.	Pyrimido compounds having antiproliferative activity
JP2006514624A (ja) *	2002-11-18	2006-05-11	エフ．ホフマン−ラ　ロシュ　アーゲー	ジアジノピリミジン類
KR20050111636A (ko)	2003-04-10	2005-11-25	에프. 호프만-라 로슈 아게	피리미도 화합물
BRPI0413005A (pt) *	2003-07-29	2006-09-26	Irm Llc	compostos e composições como inibidores da proteìna cinase
US20060035893A1 (en)	2004-08-07	2006-02-16	Boehringer Ingelheim International Gmbh	Pharmaceutical compositions for treatment of respiratory and gastrointestinal disorders
JP2008509964A (ja)	2004-08-31	2008-04-03	エフ．ホフマン−ラロシュアーゲー	７−アミノ−３−フェニル−ジヒドロピリミド［４，５−ｄ］ピリミジノンのアミド誘導体、これらの製造、及びプロテインキナーゼ阻害剤としての使用
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ES2301380B1 (es)	2006-08-09	2009-06-08	Laboratorios Almirall S.A.	Nuevos derivados de 1,7-naftiridina.
ES2320955B1 (es)	2007-03-02	2010-03-16	Laboratorios Almirall S.A.	Nuevos derivados de 3-((1,2,4)triazolo(4,3-a)piridin-7-il)benzamida.
ES2329639B1 (es)	2007-04-26	2010-09-23	Laboratorios Almirall S.A.	Nuevos derivados de 4,8-difenilpoliazanaftaleno.
EP1992344A1 (en)	2007-05-18	2008-11-19	Institut Curie	P38 alpha as a therapeutic target in pathologies linked to FGFR3 mutation
GB2452696B (en) *	2007-08-02	2009-09-23	Cambridge Entpr Ltd	3-(2',2'-dimethylpropanoylamino)-tetrahydropyridin-2-one and its use in pharmaceutical compositions
EP2108641A1 (en)	2008-04-11	2009-10-14	Laboratorios Almirall, S.A.	New substituted spiro[cycloalkyl-1,3'-indo]-2'(1'H)-one derivatives and their use as p38 mitogen-activated kinase inhibitors
EP2113503A1 (en)	2008-04-28	2009-11-04	Laboratorios Almirall, S.A.	New substituted indolin-2-one derivatives and their use as p39 mitogen-activated kinase inhibitors
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EP2322176A1 (en)	2009-11-11	2011-05-18	Almirall, S.A.	New 7-phenyl-[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one derivatives
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2000
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CZ20021744A3 (cs)	2002-08-14
CN1171889C (zh)	2004-10-20
YU29102A (sh)	2004-12-31
CA2388142C (en)	2008-12-09
RU2002112753A (ru)	2004-01-20
BR0015243A (pt)	2002-07-16
ES2280247T3 (es)	2007-09-16
MA26837A1 (fr)	2004-12-20
MXPA02003950A (es)	2002-10-23
AR026084A1 (es)	2002-12-26
AU776250B2 (en)	2004-09-02
HUP0203564A2 (hu)	2003-02-28
WO2001029042A1 (en)	2001-04-26
DE60033307T2 (de)	2007-07-12
NZ518119A (en)	2004-02-27
EP1228070A1 (en)	2002-08-07
CN1382144A (zh)	2002-11-27
TR200201057T2 (tr)	2002-09-23
HUP0203564A3 (en)	2004-07-28
HRP20020328A2 (en)	2004-02-29
AU7787300A (en)	2001-04-30
RU2265606C2 (ru)	2005-12-10
ATE353329T1 (de)	2007-02-15
KR20020038963A (ko)	2002-05-24
CA2388142A1 (en)	2001-04-26
KR100523120B1 (ko)	2005-10-20
JP2003512378A (ja)	2003-04-02
DE60033307D1 (en)	2007-03-22
JP3961830B2 (ja)	2007-08-22
NO20021781D0 (no)	2002-04-16
PE20010758A1 (es)	2001-07-21
EP1228070B1 (en)	2007-02-07
US6451804B1 (en)	2002-09-17
PL357502A1 (en)	2004-07-26
NO20021781L (no)	2002-04-18
HK1051039A1 (en)	2003-07-18

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