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EE05171B1 - Peroraalne ravimvorm, mis sisaldab opioidagonisti vabanevas vormis ja eraldatud opioidantagonisti, meetod selle valmistamiseks ning selle kasutamine meditsiinis - Google Patents

Peroraalne ravimvorm, mis sisaldab opioidagonisti vabanevas vormis ja eraldatud opioidantagonisti, meetod selle valmistamiseks ning selle kasutamine meditsiinis

Info

Publication number
EE05171B1
EE05171B1 EEP200200437A EEP200200437A EE05171B1 EE 05171 B1 EE05171 B1 EE 05171B1 EE P200200437 A EEP200200437 A EE P200200437A EE P200200437 A EEP200200437 A EE P200200437A EE 05171 B1 EE05171 B1 EE 05171B1
Authority
EE
Estonia
Prior art keywords
medicine
preparation
oral dosage
isolated
liberated
Prior art date
Application number
EEP200200437A
Other languages
English (en)
Estonian (et)
Inventor
Oshlack Benjamin
Wright Curtis
Original Assignee
Euro-Celtique, S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22663996&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EE05171(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Euro-Celtique, S.A. filed Critical Euro-Celtique, S.A.
Publication of EE200200437A publication Critical patent/EE200200437A/xx
Publication of EE05171B1 publication Critical patent/EE05171B1/xx

Links

Classifications

    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5084Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/485Morphinan derivatives, e.g. morphine, codeine
    • AHUMAN NECESSITIES
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    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0043Nose
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    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
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    • A61K9/006Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
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    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A61K9/2081Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
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    • A61K9/2806Coating materials
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    • A61K9/4808Preparations in capsules, e.g. of gelatin, of chocolate characterised by the form of the capsule or the structure of the filling; Capsules containing small tablets; Capsules with outer layer for immediate drug release
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    • A61K9/7038Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
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    • A61K9/7023Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
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    • A61K9/7038Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
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    • A61K9/7053Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
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  • Health & Medical Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Physics & Mathematics (AREA)
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  • Toxicology (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
EEP200200437A 2000-02-08 2001-02-08 Peroraalne ravimvorm, mis sisaldab opioidagonisti vabanevas vormis ja eraldatud opioidantagonisti, meetod selle valmistamiseks ning selle kasutamine meditsiinis EE05171B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US18136900P 2000-02-08 2000-02-08
PCT/US2001/004346 WO2001058451A1 (en) 2000-02-08 2001-02-08 Tamper-resistant oral opioid agonist formulations

Publications (2)

Publication Number Publication Date
EE200200437A EE200200437A (et) 2003-12-15
EE05171B1 true EE05171B1 (et) 2009-06-15

Family

ID=22663996

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200200437A EE05171B1 (et) 2000-02-08 2001-02-08 Peroraalne ravimvorm, mis sisaldab opioidagonisti vabanevas vormis ja eraldatud opioidantagonisti, meetod selle valmistamiseks ning selle kasutamine meditsiinis

Country Status (35)

Country Link
US (15) US6696088B2 (es)
EP (6) EP2092936B1 (es)
JP (10) JP2003522144A (es)
KR (2) KR20020071032A (es)
CN (3) CN100563656C (es)
AP (1) AP1665A (es)
AT (1) ATE431145T1 (es)
AU (2) AU776904B2 (es)
BG (1) BG65828B1 (es)
BR (2) BRPI0108380B8 (es)
CA (1) CA2400567C (es)
CY (2) CY1109270T1 (es)
CZ (1) CZ299991B6 (es)
DE (1) DE60138706D1 (es)
DK (5) DK2517710T3 (es)
EA (1) EA004876B1 (es)
EE (1) EE05171B1 (es)
ES (5) ES2540103T3 (es)
GE (1) GEP20053614B (es)
HK (3) HK1051487A1 (es)
HU (2) HU229705B1 (es)
IL (5) IL151057A0 (es)
ME (1) ME00398B (es)
MX (2) MXPA02007686A (es)
NO (2) NO324717B1 (es)
NZ (1) NZ520554A (es)
OA (1) OA12215A (es)
PL (1) PL210845B1 (es)
PT (6) PT2092936E (es)
RS (1) RS50407B (es)
SI (5) SI1299104T1 (es)
SK (1) SK287107B6 (es)
TW (1) TWI292317B (es)
UA (1) UA79069C2 (es)
WO (2) WO2001058451A1 (es)

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US6375957B1 (en) 1997-12-22 2002-04-23 Euro-Celtique, S.A. Opioid agonist/opioid antagonist/acetaminophen combinations
BR9813827A (pt) 1997-12-22 2000-10-10 Euro Celtique Sa Analgésico opióide aplicável em mamìferos e método para impedir o uso oral abusivo de uma formulação opióide oral
JP2001526229A (ja) * 1997-12-22 2001-12-18 ユーロ−セルティーク,エス.エイ. オピオイド投薬剤形の乱用を防止する方法
US10179130B2 (en) 1999-10-29 2019-01-15 Purdue Pharma L.P. Controlled release hydrocodone formulations
ATE526950T1 (de) 1999-10-29 2011-10-15 Euro Celtique Sa Hydrocodon-formulierungen mit gesteuerter freisetzung
MXPA02007686A (es) * 2000-02-08 2003-03-27 Euro Celtique Sa Formulaciones orales y resistentes a intervenciones de agonistas opioides..
EP2932964A1 (en) 2000-10-30 2015-10-21 Euro-Celtique S.A. Controlled release hydrocodone formulations
US7858118B2 (en) * 2001-04-11 2010-12-28 Galephar Pharmaceutical Research, Inc. Extended release composition containing Tramadol
ATE493130T1 (de) * 2001-05-11 2011-01-15 Endo Pharmaceuticals Inc Opioid enthaltende arzneiform gegen missbrauch
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