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SI2517710T1 - Oralne formulacije opioidnih agonistov, varne pred zlorabo - Google Patents

Oralne formulacije opioidnih agonistov, varne pred zlorabo

Info

Publication number
SI2517710T1
SI2517710T1 SI200131041T SI200131041T SI2517710T1 SI 2517710 T1 SI2517710 T1 SI 2517710T1 SI 200131041 T SI200131041 T SI 200131041T SI 200131041 T SI200131041 T SI 200131041T SI 2517710 T1 SI2517710 T1 SI 2517710T1
Authority
SI
Slovenia
Prior art keywords
tamper
opioid agonist
resistant oral
agonist formulations
oral opioid
Prior art date
Application number
SI200131041T
Other languages
English (en)
Inventor
Benjamin Oshlack
Curtis Wright
David J. Haddox
Original Assignee
Euro-Celtique S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22663996&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI2517710(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Euro-Celtique S.A. filed Critical Euro-Celtique S.A.
Publication of SI2517710T1 publication Critical patent/SI2517710T1/sl

Links

Classifications

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    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
    • A—HUMAN NECESSITIES
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
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    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
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    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
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    • A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
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    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
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    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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    • A61K9/4808—Preparations in capsules, e.g. of gelatin, of chocolate characterised by the form of the capsule or the structure of the filling; Capsules containing small tablets; Capsules with outer layer for immediate drug release
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    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
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    • A61K9/5005—Wall or coating material
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    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
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    • A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
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    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
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  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Emergency Medicine (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Otolaryngology (AREA)
  • Addiction (AREA)
  • Pain & Pain Management (AREA)
  • Physics & Mathematics (AREA)
  • Nanotechnology (AREA)
  • Optics & Photonics (AREA)
  • Inorganic Chemistry (AREA)
  • Toxicology (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SI200131041T 2000-02-08 2001-02-08 Oralne formulacije opioidnih agonistov, varne pred zlorabo SI2517710T1 (sl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US18136900P 2000-02-08 2000-02-08
EP12167170.5A EP2517710B1 (en) 2000-02-08 2001-02-08 Tamper-resistant oral opioid agonist formulations

Publications (1)

Publication Number Publication Date
SI2517710T1 true SI2517710T1 (sl) 2015-07-31

Family

ID=22663996

Family Applications (5)

Application Number Title Priority Date Filing Date
SI200130928T SI1299104T1 (sl) 2000-02-08 2001-02-08 Oralne formulacije opioidnih agonistov, varne pred zlorabo
SI200131021T SI2092936T1 (sl) 2000-02-08 2001-02-08 Oralne formulacije opioidnih antagonistov, varne pred zlorabo
SI200131041T SI2517710T1 (sl) 2000-02-08 2001-02-08 Oralne formulacije opioidnih agonistov, varne pred zlorabo
SI200131042T SI2277521T1 (sl) 2000-02-08 2001-02-08 Oralne formulacije opioidnih agonistov, varne pred zlorabo
SI200131043T SI2283842T1 (sl) 2000-02-08 2001-02-08 Oralne formulacije opioidnih agonistov, varne pred zlorabo

Family Applications Before (2)

Application Number Title Priority Date Filing Date
SI200130928T SI1299104T1 (sl) 2000-02-08 2001-02-08 Oralne formulacije opioidnih agonistov, varne pred zlorabo
SI200131021T SI2092936T1 (sl) 2000-02-08 2001-02-08 Oralne formulacije opioidnih antagonistov, varne pred zlorabo

Family Applications After (2)

Application Number Title Priority Date Filing Date
SI200131042T SI2277521T1 (sl) 2000-02-08 2001-02-08 Oralne formulacije opioidnih agonistov, varne pred zlorabo
SI200131043T SI2283842T1 (sl) 2000-02-08 2001-02-08 Oralne formulacije opioidnih agonistov, varne pred zlorabo

Country Status (35)

Country Link
US (15) US6696088B2 (sl)
EP (6) EP2092936B1 (sl)
JP (10) JP2003522144A (sl)
KR (2) KR20020071032A (sl)
CN (3) CN100563656C (sl)
AP (1) AP1665A (sl)
AT (1) ATE431145T1 (sl)
AU (2) AU776904B2 (sl)
BG (1) BG65828B1 (sl)
BR (2) BRPI0108380B8 (sl)
CA (1) CA2400567C (sl)
CY (2) CY1109270T1 (sl)
CZ (1) CZ299991B6 (sl)
DE (1) DE60138706D1 (sl)
DK (5) DK2517710T3 (sl)
EA (1) EA004876B1 (sl)
EE (1) EE05171B1 (sl)
ES (5) ES2540103T3 (sl)
GE (1) GEP20053614B (sl)
HK (3) HK1051487A1 (sl)
HU (2) HU229705B1 (sl)
IL (5) IL151057A0 (sl)
ME (1) ME00398B (sl)
MX (2) MXPA02007686A (sl)
NO (2) NO324717B1 (sl)
NZ (1) NZ520554A (sl)
OA (1) OA12215A (sl)
PL (1) PL210845B1 (sl)
PT (6) PT2092936E (sl)
RS (1) RS50407B (sl)
SI (5) SI1299104T1 (sl)
SK (1) SK287107B6 (sl)
TW (1) TWI292317B (sl)
UA (1) UA79069C2 (sl)
WO (2) WO2001058451A1 (sl)

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