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EA200802444A1 - Стабилизированные фармацевтические композиции, содержащие фезотеродин - Google Patents

Стабилизированные фармацевтические композиции, содержащие фезотеродин

Info

Publication number
EA200802444A1
EA200802444A1 EA200802444A EA200802444A EA200802444A1 EA 200802444 A1 EA200802444 A1 EA 200802444A1 EA 200802444 A EA200802444 A EA 200802444A EA 200802444 A EA200802444 A EA 200802444A EA 200802444 A1 EA200802444 A1 EA 200802444A1
Authority
EA
Eurasian Patent Office
Prior art keywords
phesterodine
pharmaceutical compositions
compositions containing
stabilized pharmaceutical
stabilized
Prior art date
Application number
EA200802444A
Other languages
English (en)
Other versions
EA015909B1 (ru
EA015909B9 (ru
Inventor
Кристоф Арт
Ханс-Юрген Мика
Михаэль Коменда
Ханс Линднер
Фатима Бикане
Керстин Паулус
Майке Ирнгартингер
Original Assignee
Шварц Фарма Аг
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38521333&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA200802444(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Шварц Фарма Аг filed Critical Шварц Фарма Аг
Publication of EA200802444A1 publication Critical patent/EA200802444A1/ru
Publication of EA015909B1 publication Critical patent/EA015909B1/ru
Publication of EA015909B9 publication Critical patent/EA015909B9/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
    • A61K9/1623—Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A61K31/222—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin with compounds having aromatic groups, e.g. dipivefrine, ibopamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/10—Drugs for disorders of the urinary system of the bladder

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Emergency Medicine (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Urology & Nephrology (AREA)
  • Inorganic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Настоящая заявка относится к фармацевтической композиции, содержащей фезотеродин или его фармацевтически приемлемые соль или сольват и стабилизатор, выбранный из группы, состоящей из ксилита, сорбита, полидекстрозы, изомальта и декстрозы.
EA200802444A 2006-06-09 2007-06-06 Стабилизированные фармацевтические композиции, содержащие фезотеродин EA015909B9 (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP06011942 2006-06-09
EP06011941 2006-06-09
EP06011943 2006-06-09
PCT/EP2007/055582 WO2007141298A1 (en) 2006-06-09 2007-06-06 Stabilized pharmaceutical compositions comprising fesoterodine

Publications (3)

Publication Number Publication Date
EA200802444A1 true EA200802444A1 (ru) 2009-06-30
EA015909B1 EA015909B1 (ru) 2011-12-30
EA015909B9 EA015909B9 (ru) 2012-03-30

Family

ID=38521333

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200802444A EA015909B9 (ru) 2006-06-09 2007-06-06 Стабилизированные фармацевтические композиции, содержащие фезотеродин

Country Status (38)

Country Link
EP (1) EP2029134B1 (ru)
JP (2) JP4743321B2 (ru)
KR (1) KR101316773B1 (ru)
CN (1) CN101466371B (ru)
AP (1) AP2416A (ru)
AR (1) AR061289A1 (ru)
AT (1) ATE517619T1 (ru)
AU (1) AU2007255408B2 (ru)
BR (1) BRPI0712865B1 (ru)
CA (1) CA2652712C (ru)
CR (1) CR10494A (ru)
CU (1) CU23850B1 (ru)
CY (1) CY1111934T1 (ru)
DK (1) DK2029134T3 (ru)
EA (1) EA015909B9 (ru)
EC (1) ECSP089010A (ru)
ES (1) ES2370943T3 (ru)
GT (1) GT200800276A (ru)
HK (1) HK1128626A1 (ru)
HR (1) HRP20110776T1 (ru)
IL (2) IL195732A (ru)
MA (1) MA30504B1 (ru)
MX (1) MX2008015736A (ru)
MY (1) MY146574A (ru)
NI (1) NI200800318A (ru)
NL (1) NL2000690C2 (ru)
NO (1) NO341980B1 (ru)
NZ (1) NZ572616A (ru)
PE (2) PE20080331A1 (ru)
PL (1) PL2029134T3 (ru)
PT (1) PT2029134E (ru)
RS (1) RS51973B (ru)
SI (1) SI2029134T1 (ru)
TN (1) TNSN08505A1 (ru)
TW (2) TWI397409B (ru)
UY (1) UY30394A1 (ru)
WO (1) WO2007141298A1 (ru)
ZA (1) ZA200806411B (ru)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009122303A2 (en) * 2008-04-04 2009-10-08 Actavis Group Ptc Ehf Novel mandelate salt of fesoterodine
IT1392082B1 (it) * 2008-12-10 2012-02-09 Chemi Spa Nuove forme solide della fesoterodina fumarato
US9085507B2 (en) 2009-05-11 2015-07-21 Ratiopharm Gmbh Desfesoterodine in the form of a tartaric acid salt
EP2316432A1 (de) 2009-10-30 2011-05-04 ratiopharm GmbH Zusammensetzung enthaltend Fesoterodin und Ballaststoffe
EP2549985A1 (en) * 2010-03-22 2013-01-30 Cadila Healthcare Limited Stable pharmaceutical compositions comprising fesoterodine
TWI590821B (zh) 2011-01-18 2017-07-11 輝瑞有限公司 固體分子分散液
EP2508173A1 (en) 2011-04-08 2012-10-10 LEK Pharmaceuticals d.d. Stabilized pharmaceutical composition comprising fesoterodine
EP2508175A1 (en) 2011-04-08 2012-10-10 LEK Pharmaceuticals d.d. Pharmaceutical composition comprising fesoterodine or a salt or a solvate thereof
US20140199401A1 (en) * 2011-07-04 2014-07-17 Cadila Healthcare Limited Extended release pharmaceutical compositions of fesoterodine
US9440910B2 (en) * 2012-05-18 2016-09-13 Alembic Pharmaceuticals Limited Reference markers for fesoterodine fumarate
ES2674811T3 (es) * 2012-07-02 2018-07-04 Hetero Research Foundation Composiciones estables de fesoterodina
KR20240074883A (ko) 2012-11-02 2024-05-28 머레이 앤 풀 엔터프라이지즈, 리미티드 콜히친 유도체의 투여를 통한 심혈관성 병태의 치료 또는 예방
EP2986280B1 (en) 2013-04-16 2021-03-17 Murray & Poole Enterprises, Ltd. Sustained-release formulations of colchicine and methods of using same
CZ2014400A3 (cs) 2014-06-09 2015-12-16 Zentiva, K.S. Stabilizovaná formulace fesoterodinu
CN105687154A (zh) * 2014-11-27 2016-06-22 合肥信风科技开发有限公司 含非索罗定的药用组合物及其制备方法
WO2019011393A1 (en) 2017-07-12 2019-01-17 Rontis Hellas S.A. EXTENDED RELEASE PHARMACEUTICAL COMPOSITION CONTAINING FESOTERODINE AND PREPARATION METHOD THEREOF
WO2019132832A1 (en) * 2017-12-25 2019-07-04 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Tablet compositions of fesoterodine fumarate
TR201721437A2 (tr) * 2017-12-25 2019-07-22 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Fesoterodi̇ni̇n modi̇fi̇ye salim sağlayan formülasyonlari
KR102018495B1 (ko) * 2018-03-13 2019-09-05 충북대학교 산학협력단 과민성 방광의 치료를 위한 서방형의 이중층 정제 및 이의 제조방법
CA3094551C (en) 2018-04-26 2024-01-02 Rontis Hellas S.A. Extended release pharmaceutical composition containing fesoterodine and process for the preparation thereof
CN110151720B (zh) * 2019-05-09 2019-12-17 合肥信风科技开发有限公司 含非索罗定的药用组合物及其制备方法
JPWO2023145486A1 (ru) * 2022-01-28 2023-08-03

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2002505282A (ja) * 1998-03-03 2002-02-19 塩野義製薬株式会社 ホスホリパーゼ阻害剤の［［３−（２−アミノ−１，２−ジオキソエチル）−２−エチル−１−フェニルメチル）−１ｈ−インドール−４−イル］オキシ］酢酸ナトリウムを含む薬学的組成物
EP0957073A1 (en) * 1998-05-12 1999-11-17 Schwarz Pharma Ag Novel derivatives of 3,3-diphenylpropylamines
DE29923134U1 (de) * 1999-11-16 2000-06-29 Schwarz Pharma Ag, 40789 Monheim Stabile Salze neuartiger Derviate von 3,3-Diphenylpropylaminen
DE10224107A1 (de) * 2002-05-29 2003-12-11 Gruenenthal Gmbh Kombination ausgewählter Opioide mit anderen Wirkstoffen zur Therapie der Harninkontinenz
DE10315878B4 (de) * 2003-04-08 2009-06-04 Schwarz Pharma Ag Vorrichtung zur transdermalen Verabreichung von Fesoterodin und Verwendung

Also Published As

Publication number Publication date
NI200800318A (es) 2011-01-12
ATE517619T1 (de) 2011-08-15
CA2652712C (en) 2014-04-01
EA015909B1 (ru) 2011-12-30
KR101316773B1 (ko) 2013-10-15
CU20080235A7 (es) 2011-04-26
EP2029134B1 (en) 2011-07-27
TNSN08505A1 (fr) 2010-04-14
IL220800A (en) 2015-03-31
BRPI0712865B1 (pt) 2021-08-17
RS51973B (en) 2012-02-29
HK1128626A1 (en) 2009-11-06
IL195732A (en) 2013-09-30
NL2000690A1 (nl) 2007-12-11
EA015909B9 (ru) 2012-03-30
ZA200806411B (en) 2009-05-27
PE20120476A1 (es) 2012-04-20
CR10494A (es) 2009-01-19
NZ572616A (en) 2010-11-26
WO2007141298A1 (en) 2007-12-13
CA2652712A1 (en) 2007-12-13
TWI520735B (zh) 2016-02-11
IL195732A0 (en) 2009-09-01
PT2029134E (pt) 2011-11-02
EP2029134A1 (en) 2009-03-04
GT200800276A (es) 2009-06-18
NO341980B1 (no) 2018-03-05
TWI397409B (zh) 2013-06-01
AP2416A (en) 2012-06-01
BRPI0712865A2 (pt) 2012-12-18
CU23850B1 (es) 2012-10-15
CN101466371A (zh) 2009-06-24
JP2009539802A (ja) 2009-11-19
ES2370943T3 (es) 2011-12-23
AU2007255408B2 (en) 2013-03-14
MX2008015736A (es) 2009-01-09
DK2029134T3 (da) 2011-10-17
NO20090141L (no) 2009-01-09
SI2029134T1 (sl) 2012-01-31
MY146574A (en) 2012-08-30
TW200814992A (en) 2008-04-01
JP4781489B2 (ja) 2011-09-28
CY1111934T1 (el) 2015-11-04
TW201336491A (zh) 2013-09-16
JP2011140498A (ja) 2011-07-21
PL2029134T3 (pl) 2011-12-30
KR20090026135A (ko) 2009-03-11
PE20080331A1 (es) 2008-06-19
CN101466371B (zh) 2011-10-05
AP2008004673A0 (en) 2008-12-31
NL2000690C2 (nl) 2008-04-01
MA30504B1 (fr) 2009-06-01
AU2007255408A1 (en) 2007-12-13
HRP20110776T1 (hr) 2011-11-30
AR061289A1 (es) 2008-08-20
ECSP089010A (es) 2009-01-30
UY30394A1 (es) 2007-11-30
JP4743321B2 (ja) 2011-08-10

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