NO20001871L - Nye 3,6-hemiacetaler fra klassen 9a-azalider - Google Patents

Nye 3,6-hemiacetaler fra klassen 9a-azalider

Info

Publication number: NO20001871L
Authority: NO; Norway
Prior art keywords: group; individually; represents hydrogen; carbon atoms; individually represents
Prior art date: 1997-10-16

Application number

NO20001871A

Other languages

English (en)

Norwegian (no)

Other versions

NO20001871D0 (no

Inventor

Gabrijela Kobrehel

Gorjana Lazarevski

Mladen Vinkovic

Original Assignee

Pliva Pharm & Chem Works

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-10-16

Filing date

2000-04-11

Publication date

2000-04-17

1997-10-16 Priority claimed from HR970551A external-priority patent/HRP970551B1/xx

1998-09-10 Priority claimed from HR980497A external-priority patent/HRP980497B1/xx

2000-04-11 Application filed by Pliva Pharm & Chem Works filed Critical Pliva Pharm & Chem Works

2000-04-11 Publication of NO20001871D0 publication Critical patent/NO20001871D0/no

2000-04-17 Publication of NO20001871L publication Critical patent/NO20001871L/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Molecular Biology (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
Genetics & Genomics (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Chemical Kinetics & Catalysis (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

NO20001871A 1997-10-16 2000-04-11 Nye 3,6-hemiacetaler fra klassen 9a-azalider NO20001871L (no)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
HR970551A HRP970551B1 (en)	1997-10-16	1997-10-16	Novel o-methyl azythromycin derivatives
HR980497A HRP980497B1 (en)	1998-09-10	1998-09-10	NOVEL 3,6-HEMIKETALS FROM THE CLASS OF 9a-AZALIDES
PCT/HR1998/000005 WO1999020639A2 (en)	1997-10-16	1998-10-13	NOVEL 3,6-HEMIKETALS FROM THE CLASS OF 9a-AZALIDES

Publications (2)

Publication Number	Publication Date
NO20001871D0 NO20001871D0 (no)	2000-04-11
NO20001871L true NO20001871L (no)	2000-04-17

Family

ID=26317108

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20001871A NO20001871L (no)	1997-10-16	2000-04-11	Nye 3,6-hemiacetaler fra klassen 9a-azalider

Country Status (26)

Country	Link
US (1)	US6369035B1 (xx)
EP (2)	EP1036083B9 (xx)
JP (1)	JP2001520234A (xx)
KR (1)	KR100554549B1 (xx)
CN (1)	CN1281615C (xx)
AR (1)	AR018014A1 (xx)
AT (2)	ATE267835T1 (xx)
AU (1)	AU755315B2 (xx)
BG (1)	BG64650B1 (xx)
BR (1)	BR9812808A (xx)
CA (1)	CA2306963C (xx)
DE (2)	DE69824201T2 (xx)
DK (2)	DK1437359T3 (xx)
EE (1)	EE04681B1 (xx)
ES (2)	ES2222610T3 (xx)
HK (1)	HK1032785A1 (xx)
HU (1)	HUP0004085A3 (xx)
IL (2)	IL135648A0 (xx)
NO (1)	NO20001871L (xx)
NZ (1)	NZ503897A (xx)
PL (1)	PL191087B1 (xx)
PT (2)	PT1036083E (xx)
RU (1)	RU2220148C2 (xx)
SI (2)	SI1437359T1 (xx)
SK (1)	SK285914B6 (xx)
WO (1)	WO1999020639A2 (xx)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TR200200435T2 (tr) *	1998-11-03	2002-07-22	Pfizer Products Inc.	Yeni makrolit antibiyotikler.
KR100361397B1 (ko) *	2000-03-15	2002-11-23	한미약품공업 주식회사	에리스로마이신 에이 9-오-트로필옥심 유도체를 이용한클라리스로마이신의 제조방법
CA2476448A1 (en)	2002-02-15	2003-08-28	Sympore Gmbh	Antibiotic conjugates
WO2003070174A2 (en)	2002-02-15	2003-08-28	Sympore Gmbh	Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof
US20060099660A1 (en)	2002-02-15	2006-05-11	Synovo Gmbh	Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof
HRP20020779A2 (en)	2002-09-27	2005-02-28	Pliva-Istra�iva�ki institut d.o.o.	NEW 3-DECLADINOSYL DERIVATIVES OF 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERYTHROMICIN A 9a, 11-CYCLIC CARBAMATES
ITMI20022292A1 (it) *	2002-10-29	2004-04-30	Zambon Spa	9a-azalidi ad attivita' antiinfiammatoria.
US7435805B2 (en)	2003-05-30	2008-10-14	Glaxpsmithkline Istrazivacki	O-alkyl macrolide and azalide derivatives and regioselective process for their preparation
AU2003264910A1 (en) *	2003-05-30	2005-01-21	Pliva - Istrazivacki Institut D.O.O.	Process for selective alkylation of macrolide and azalide derivatives
US7276487B2 (en)	2003-09-23	2007-10-02	Enanta Pharmaceuticals, Inc.	9a, 11-3C-bicyclic 9a-azalide derivatives
US7468428B2 (en) *	2004-03-17	2008-12-23	App Pharmaceuticals, Llc	Lyophilized azithromycin formulation
US20060116336A1 (en) *	2004-03-17	2006-06-01	American Pharmaceutical Partners, Inc.	Lyophilized azithromycin formulation
US7402568B2 (en) *	2004-09-29	2008-07-22	Enanta Pharmaceuticals, Inc.	Bicyclic 9a-azalide derivatives
US7271155B2 (en)	2005-01-07	2007-09-18	Enanta Pharmaceuticals, Inc.	9A, 11-2C-bicyclic 9a-azalide derivatives
WO2008106225A1 (en) *	2007-02-28	2008-09-04	Rib-X Pharmaceuticals, Inc.	Macrolide compounds and methods of making and using the same
US9145436B2 (en)	2010-10-10	2015-09-29	Michael W. Burnet	Anti-inflammatory macrolides
EP2831083A4 (en) *	2012-03-27	2016-03-09	Michael W Burnet	INFLAMMATORY MAKROLIDE
JP7184520B2 (ja) *	2018-01-22	2022-12-06	旭化成株式会社	トランス型脂環式カーボネートの製造方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
YU43006B (en) *	1981-03-06	1989-02-28	Pliva Pharm & Chem Works	Process for preparing n-methyl-11-aza-10-deoxo-10-dihydro erythromycin and derivatives thereof
US4474768A (en) *	1982-07-19	1984-10-02	Pfizer Inc.	N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor
WO1989000576A1 (en) *	1987-07-09	1989-01-26	Pfizer Inc.	Azithromycin dihydrate
HU198913B (en) *	1987-09-03	1989-12-28	Pliva Pharm & Chem Works	Process for producing 10-dihydro-10-deoxo-11-aza-erythronolide a-derivatives and pharmaceutical compositions containing them as active components
WO1989002271A1 (en) *	1987-09-10	1989-03-23	Pfizer	Azithromycin and derivatives as antiprotozoal agents
SI9011409A (en) *	1990-07-18	1995-10-31	Pliva Pharm & Chem Works	O-methyl azitromycin derivates, methods and intermediates for their preparation and methods for preparation of pharmaceuticals products which comprise them
FR2691464B1 (fr) *	1992-05-21	1995-06-02	Roussel Uclaf	Nouveaux dérivés de la 1-oxa 6-azacyclopentadécane 13,15-dione, leur procédé de préparation et leur application comme médicaments.
WO1999000124A1 (en) *	1997-06-26	1999-01-07	Merck & Co., Inc.	9a-azalides, compositions containing such compounds and methods of treatment

1998
- 1998-10-13 DK DK04004844T patent/DK1437359T3/da active
- 1998-10-13 EP EP98946627A patent/EP1036083B9/en not_active Expired - Lifetime
- 1998-10-13 AU AU93622/98A patent/AU755315B2/en not_active Ceased
- 1998-10-13 ES ES98946627T patent/ES2222610T3/es not_active Expired - Lifetime
- 1998-10-13 PL PL340372A patent/PL191087B1/pl unknown
- 1998-10-13 IL IL13564898A patent/IL135648A0/xx not_active IP Right Cessation
- 1998-10-13 SI SI9830878T patent/SI1437359T1/sl unknown
- 1998-10-13 RU RU2000111996/04A patent/RU2220148C2/ru not_active IP Right Cessation
- 1998-10-13 BR BR9812808-6A patent/BR9812808A/pt not_active Application Discontinuation
- 1998-10-13 DE DE69824201T patent/DE69824201T2/de not_active Expired - Fee Related
- 1998-10-13 EP EP04004844A patent/EP1437359B1/en not_active Expired - Lifetime
- 1998-10-13 CN CNB988116243A patent/CN1281615C/zh not_active Expired - Fee Related
- 1998-10-13 US US09/529,642 patent/US6369035B1/en not_active Expired - Fee Related
- 1998-10-13 CA CA002306963A patent/CA2306963C/en not_active Expired - Fee Related
- 1998-10-13 WO PCT/HR1998/000005 patent/WO1999020639A2/en not_active Application Discontinuation
- 1998-10-13 ES ES04004844T patent/ES2279242T3/es not_active Expired - Lifetime
- 1998-10-13 DK DK98946627T patent/DK1036083T5/da active
- 1998-10-13 JP JP2000516980A patent/JP2001520234A/ja active Pending
- 1998-10-13 SI SI9830675T patent/SI1036083T1/xx unknown
- 1998-10-13 KR KR1020007004079A patent/KR100554549B1/ko not_active IP Right Cessation
- 1998-10-13 NZ NZ503897A patent/NZ503897A/xx unknown
- 1998-10-13 AT AT98946627T patent/ATE267835T1/de not_active IP Right Cessation
- 1998-10-13 DE DE69836697T patent/DE69836697T2/de not_active Expired - Fee Related
- 1998-10-13 PT PT98946627T patent/PT1036083E/pt unknown
- 1998-10-13 SK SK552-2000A patent/SK285914B6/sk unknown
- 1998-10-13 AT AT04004844T patent/ATE348836T1/de not_active IP Right Cessation
- 1998-10-13 EE EEP200000226A patent/EE04681B1/xx not_active IP Right Cessation
- 1998-10-13 HU HU0004085A patent/HUP0004085A3/hu unknown
- 1998-10-13 PT PT04004844T patent/PT1437359E/pt unknown
- 1998-10-16 AR ARP980105155A patent/AR018014A1/es active IP Right Grant
2000
- 2000-04-11 NO NO20001871A patent/NO20001871L/no not_active Application Discontinuation
- 2000-04-13 IL IL135648A patent/IL135648A/en unknown
- 2000-05-16 BG BG104445A patent/BG64650B1/bg unknown
2001
- 2001-05-22 HK HK01103498A patent/HK1032785A1/xx not_active IP Right Cessation

Also Published As

Publication number	Publication date
KR100554549B1 (ko)	2006-03-03
EP1036083B9 (en)	2005-01-12
DK1437359T3 (da)	2007-04-30
US6369035B1 (en)	2002-04-09
DK1036083T5 (da)	2005-04-04
EP1437359A2 (en)	2004-07-14
EE04681B1 (et)	2006-08-15
ATE267835T1 (de)	2004-06-15
HUP0004085A3 (en)	2003-05-28
KR20010031160A (ko)	2001-04-16
BG104445A (en)	2001-02-28
DE69836697D1 (de)	2007-02-01
ES2279242T3 (es)	2007-08-16
BR9812808A (pt)	2005-04-12
SI1036083T1 (en)	2004-10-31
ES2222610T3 (es)	2005-02-01
DK1036083T3 (da)	2004-09-27
DE69824201D1 (de)	2004-07-01
SI1437359T1 (sl)	2007-06-30
HUP0004085A2 (hu)	2001-04-28
JP2001520234A (ja)	2001-10-30
PL191087B1 (pl)	2006-03-31
IL135648A0 (en)	2001-05-20
EP1036083A2 (en)	2000-09-20
EP1036083B1 (en)	2004-05-26
AU755315B2 (en)	2002-12-12
CA2306963C (en)	2007-05-01
WO1999020639A2 (en)	1999-04-29
NO20001871D0 (no)	2000-04-11
EP1437359A3 (en)	2005-03-30
HK1032785A1 (en)	2001-08-03
AR018014A1 (es)	2001-10-31
DE69836697T2 (de)	2007-10-04
BG64650B1 (bg)	2005-10-31
SK5522000A3 (en)	2000-11-07
IL135648A (en)	2007-03-08
SK285914B6 (sk)	2007-11-02
RU2220148C2 (ru)	2003-12-27
PL340372A1 (en)	2001-01-29
DE69824201T2 (de)	2005-09-22
EE200000226A (et)	2001-06-15
AU9362298A (en)	1999-05-10
CA2306963A1 (en)	1999-04-29
CN1281615C (zh)	2006-10-25
WO1999020639A3 (en)	1999-07-08
PT1036083E (pt)	2004-10-29
CN1280585A (zh)	2001-01-17
NZ503897A (en)	2002-10-25
EP1437359B1 (en)	2006-12-20
PT1437359E (pt)	2007-04-30
ATE348836T1 (de)	2007-01-15

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Legal Events

Date	Code	Title	Description
2009-05-25	FC2A	Withdrawal, rejection or dismissal of laid open patent application