SK9442001A3 - Imidazo[4,5-c]-pyridine-4-on-derivatives, process for the preparation thereof, use thereof and pharmaceutical composition comprising same - Google Patents

Imidazo[4,5-c]-pyridine-4-on-derivatives, process for the preparation thereof, use thereof and pharmaceutical composition comprising same Download PDF

Info

Publication number: SK9442001A3
Authority: SK; Slovakia
Prior art keywords: group; formula; compounds; salts; physiologically acceptable
Prior art date: 1999-01-08

Application number

SK944-2001A

Other languages

English (en)

Slovak (sk)

Inventor

Werner Mederski

Horst Juraszyk

Hanns Wurziger

Christos Tsaklakidis

Dieter Dorsch

Sabine Bernotat-Danielowski

Guido Melzer

Soheila Anzali

Original Assignee

Merck Patent Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-01-08

Filing date

1999-12-21

Publication date

2002-05-09

1999-12-21 Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh

2002-05-09 Publication of SK9442001A3 publication Critical patent/SK9442001A3/sk

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Hematology (AREA)
Diabetes (AREA)
Urology & Nephrology (AREA)
Vascular Medicine (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

SK944-2001A 1999-01-08 1999-12-21 Imidazo[4,5-c]-pyridine-4-on-derivatives, process for the preparation thereof, use thereof and pharmaceutical composition comprising same SK9442001A3 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE19900471A DE19900471A1 (de)	1999-01-08	1999-01-08	Imidazo[4,5c]-pyridin-4-on-derivate
PCT/EP1999/010236 WO2000040583A2 (de)	1999-01-08	1999-12-21	Imidazo[4,5-c]-pyridin-4-on-derivate

Publications (1)

Publication Number	Publication Date
SK9442001A3 true SK9442001A3 (en)	2002-05-09

Family

ID=7893790

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SK944-2001A SK9442001A3 (en)	1999-01-08	1999-12-21	Imidazo[4,5-c]-pyridine-4-on-derivatives, process for the preparation thereof, use thereof and pharmaceutical composition comprising same

Country Status (16)

Country	Link
EP (1)	EP1149099A2 (ja)
JP (1)	JP2002534429A (ja)
KR (1)	KR20010086085A (ja)
CN (1)	CN1333772A (ja)
AR (1)	AR022220A1 (ja)
AU (1)	AU3041700A (ja)
BR (1)	BR9916774A (ja)
CA (1)	CA2357771A1 (ja)
CZ (1)	CZ20012407A3 (ja)
DE (1)	DE19900471A1 (ja)
HU (1)	HUP0105054A3 (ja)
NO (1)	NO20013384D0 (ja)
PL (1)	PL349341A1 (ja)
SK (1)	SK9442001A3 (ja)
WO (1)	WO2000040583A2 (ja)
ZA (1)	ZA200106454B (ja)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2232202T3 (es)	1998-12-23	2005-05-16	Bristol-Myers Squibb Pharma Company	Heterobiciclos que contienen nitrogeno como inhibidores del factor xa.
AU2001268712A1 (en) *	2000-06-23	2002-01-08	Bristol-Myers Squibb Company	1 - (heteroaryl-phenyl) - condensed pyrazol derivatives as factor Xa inhibitors
CA2447488A1 (en)	2001-05-22	2002-11-28	Irina Jacobson	Bicyclic inhibitors of factor xa
EP1569912B1 (en)	2002-12-03	2015-04-29	Pharmacyclics, Inc.	2-(2-hydroxybiphenyl-3-yl)-1h-benzoimidazole-5-carboxamidine derivatives as factor viia inhibitors
GB0215293D0 (en)	2002-07-03	2002-08-14	Rega Foundation	Viral inhibitors
GB0225399D0 (en) *	2002-10-31	2002-12-11	Merck Sharp & Dohme	Therapeutic agents
WO2005063744A2 (en)	2003-12-22	2005-07-14	K.U. Leuven Research & Development	IMIDAZO[4,5-c]PYRIDINE COMPOUNDS AND METHODS OF ANTIVIRAL TREATMENT
SI1841765T1 (sl)	2004-12-21	2009-08-31	Gilead Sciences Inc	Imidazo(4,5-c)piridinska spojina in postopek za antivirusno zdravljenje
WO2007009883A1 (en) *	2005-07-15	2007-01-25	F. Hoffmann-La Roche Ag	Novel heteroaryl fused cyclic amines
US20070060530A1 (en)	2005-09-14	2007-03-15	Christopher Ronald J	Administration of dipeptidyl peptidase inhibitors
US8222411B2 (en)	2005-09-16	2012-07-17	Takeda Pharmaceutical Company Limited	Dipeptidyl peptidase inhibitors
WO2007112347A1 (en)	2006-03-28	2007-10-04	Takeda Pharmaceutical Company Limited	Dipeptidyl peptidase inhibitors
KR101143596B1 (ko)	2006-07-07	2012-05-11	길리애드 사이언시즈, 인코포레이티드	신규의 피리다진 화합물 및 이의 용도
TW200838536A (en)	2006-11-29	2008-10-01	Takeda Pharmaceutical	Polymorphs of succinate salt of 2-[6-(3-amino-piperidin-1-yl)-3-methyl-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-ylmethy]-4-fluor-benzonitrile and methods of use therefor
UA99466C2 (en)	2007-07-06	2012-08-27	Гилиад Сайенсиз, Инк.	Crystalline pyridazine compound
EP3180341B1 (en) *	2014-08-12	2022-04-27	Syngenta Participations AG	Pesticidally active heterocyclic derivatives with sulphur containing substituents

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TW219935B (ja) *	1991-12-25	1994-02-01	Mitsubishi Chemicals Co Ltd
JP2001524522A (ja) *	1997-12-01	2001-12-04	メルクエンドカムパニーインコーポレーテッド	トロンビン阻害剤

1999
- 1999-01-08 DE DE19900471A patent/DE19900471A1/de not_active Withdrawn
- 1999-12-21 KR KR1020017007074A patent/KR20010086085A/ko not_active Application Discontinuation
- 1999-12-21 AU AU30417/00A patent/AU3041700A/en not_active Abandoned
- 1999-12-21 SK SK944-2001A patent/SK9442001A3/sk unknown
- 1999-12-21 WO PCT/EP1999/010236 patent/WO2000040583A2/de not_active Application Discontinuation
- 1999-12-21 CZ CZ20012407A patent/CZ20012407A3/cs unknown
- 1999-12-21 CN CN99815465A patent/CN1333772A/zh active Pending
- 1999-12-21 PL PL99349341A patent/PL349341A1/xx unknown
- 1999-12-21 JP JP2000592291A patent/JP2002534429A/ja active Pending
- 1999-12-21 HU HU0105054A patent/HUP0105054A3/hu unknown
- 1999-12-21 BR BR9916774-3A patent/BR9916774A/pt not_active Application Discontinuation
- 1999-12-21 EP EP99964639A patent/EP1149099A2/de not_active Withdrawn
- 1999-12-21 CA CA002357771A patent/CA2357771A1/en not_active Abandoned
2000
- 2000-01-07 AR ARP000100062A patent/AR022220A1/es unknown
2001
- 2001-07-06 NO NO20013384A patent/NO20013384D0/no not_active Application Discontinuation
- 2001-08-06 ZA ZA200106454A patent/ZA200106454B/en unknown

Also Published As

Publication number	Publication date
HUP0105054A3 (en)	2002-12-28
ZA200106454B (en)	2002-11-06
WO2000040583A3 (de)	2000-09-21
DE19900471A1 (de)	2000-07-13
JP2002534429A (ja)	2002-10-15
PL349341A1 (en)	2002-07-15
NO20013384L (no)	2001-07-06
WO2000040583A2 (de)	2000-07-13
EP1149099A2 (de)	2001-10-31
CZ20012407A3 (cs)	2001-12-12
CA2357771A1 (en)	2000-07-13
AU3041700A (en)	2000-07-24
NO20013384D0 (no)	2001-07-06
BR9916774A (pt)	2001-10-30
KR20010086085A (ko)	2001-09-07
AR022220A1 (es)	2002-09-04
CN1333772A (zh)	2002-01-30
HUP0105054A2 (hu)	2002-05-29

Publication	Publication Date	Title
SK9442001A3 (en)	2002-05-09	Imidazo[4,5-c]-pyridine-4-on-derivatives, process for the preparation thereof, use thereof and pharmaceutical composition comprising same
AU752574B2 (en)	2002-09-26	Imidazo(4,5-C-)-pyridine-4-one derivatives with factor XA inhibiting effect
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KR20060023154A (ko)	2006-03-13	혈전증 치료용 응고 인자 ｘａ 및 ｖｉｉａ의 저해제로서의피롤리딘-１,２-디카르복실산-１-[(４-에티닐-페닐)-아미드]-２-[(페닐)-아미드] 유도체
JP2004527514A (ja)	2004-09-09	フェニル誘導体３
SK12152001A3 (sk)	2002-03-05	Derivát pyrazol-3-ónu ako faktor Xa inhibítorov, spôsob jeho prípravy, jeho použitie a farmaceutický prostriedok, ktorý ho obsahuje
AU2002363366B2 (en)	2007-11-22	Derivatives of phenoxy-N- 4-(isothiazolidin-1,1-dioxid-2YL)pheny!-valerian- acid amide and other compounds as inhibitors of the coagulation factor XA in the treatment of thromboembolic diseases and tumors
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JP4699985B2 (ja)	2011-06-15	カルボキサミド誘導体及びその第Ｘａ因子の阻害剤としての使用
JP4567439B2 (ja)	2010-10-20	カルボン酸アミド
JP2005530754A (ja)	2005-10-13	血栓塞栓症に有効なセミカルバジド誘導体
SK2652001A3 (en)	2001-09-11	2-oxo-i(2h)-quinoline derivatives
JP2004525119A (ja)	2004-08-19	フェニル誘導体および血栓塞栓性疾患または腫瘍の処置におけるこれらの使用
MXPA01006942A (en)	2002-05-09	Imidazo[4,5-c]-pyridine-4-on-derivatives
KR20040095256A (ko)	2004-11-12	세미카르바자이드 유도체 및 항혈전제로서의 이의 용도
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