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SI1275647T1 - Octahydro-2H-pyrido(1,2-a)pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them - Google Patents

Octahydro-2H-pyrido(1,2-a)pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them

Info

Publication number
SI1275647T1
SI1275647T1 SI200230005T SI200230005T SI1275647T1 SI 1275647 T1 SI1275647 T1 SI 1275647T1 SI 200230005 T SI200230005 T SI 200230005T SI 200230005 T SI200230005 T SI 200230005T SI 1275647 T1 SI1275647 T1 SI 1275647T1
Authority
SI
Slovenia
Prior art keywords
octahydro
pyrido
preparation
pharmaceutical compositions
compositions containing
Prior art date
Application number
SI200230005T
Other languages
English (en)
Slovenian (sl)
Inventor
Solo Goldstein
Guillaume Poissonnet
Jean-Gilles Parmentier
Pierre Lestage
Brian Lockhart
Original Assignee
Les Laboratoires Servier
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Les Laboratoires Servier filed Critical Les Laboratoires Servier
Publication of SI1275647T1 publication Critical patent/SI1275647T1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SI200230005T 2001-07-12 2002-07-11 Octahydro-2H-pyrido(1,2-a)pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them SI1275647T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0109260A FR2827288B1 (fr) 2001-07-12 2001-07-12 Nouveaux derives d'octahydro-2h-pyrido[1,2-a]pyrazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
EP02291745A EP1275647B1 (fr) 2001-07-12 2002-07-11 Dérivés d'octahydro-2H-pyrido[1,2-a]pyrazine, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent

Publications (1)

Publication Number Publication Date
SI1275647T1 true SI1275647T1 (en) 2004-02-29

Family

ID=8865405

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200230005T SI1275647T1 (en) 2001-07-12 2002-07-11 Octahydro-2H-pyrido(1,2-a)pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them

Country Status (25)

Country Link
US (1) US6992085B2 (xx)
EP (1) EP1275647B1 (xx)
JP (1) JP3950018B2 (xx)
KR (1) KR100485020B1 (xx)
CN (1) CN1197863C (xx)
AR (1) AR036166A1 (xx)
AT (1) ATE254124T1 (xx)
AU (1) AU2002300094B2 (xx)
BR (1) BR0202681A (xx)
CA (1) CA2394027C (xx)
DE (1) DE60200089T2 (xx)
DK (1) DK1275647T3 (xx)
EA (1) EA005160B1 (xx)
ES (1) ES2210219T3 (xx)
FR (1) FR2827288B1 (xx)
HK (1) HK1050682A1 (xx)
HU (1) HUP0202282A3 (xx)
MX (1) MXPA02006699A (xx)
NO (1) NO322966B1 (xx)
NZ (1) NZ520120A (xx)
PL (1) PL355034A1 (xx)
PT (1) PT1275647E (xx)
SI (1) SI1275647T1 (xx)
TR (1) TR200302001T4 (xx)
ZA (1) ZA200205596B (xx)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPWO2004089410A1 (ja) * 2003-04-03 2006-07-06 協和醗酵工業株式会社 神経因性疼痛の予防及び／または治療剤
MY141255A (en) * 2003-12-11 2010-03-31 Memory Pharm Corp Phosphodiesterase 4 inhibitors, including n-substituted diarylamine analogs
FR2866647B1 (fr) * 2004-02-20 2006-10-27 Servier Lab Nouveaux derives azabicycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
BRPI0512567A (pt) * 2004-06-22 2008-03-25 Pfizer Prod Inc compostos antagonistas de receptor de histamina-3 diazabicìclico e respectivas composições farmacêuticas
RU2442775C2 (ru) * 2005-07-04 2012-02-20 Хай Пойнт Фармасьютикалс, ЛЛС Антагонисты гистаминовых н3-рецепторов
US8501739B2 (en) * 2005-07-04 2013-08-06 High Point Pharmaceuticals, Llc Medicaments
DE602007011904D1 (de) * 2006-03-10 2011-02-24 Neurogen Corp Piperazinyl-oxoalkyl-tetrahydroisochinoline und verwandte analoga
KR100871691B1 (ko) 2006-10-16 2008-12-05 삼성전자주식회사 병렬 비트 테스트 방법 및 그 방법을 사용하는 반도체메모리 장치
EP3495363B1 (en) 2016-07-28 2023-08-23 Shionogi & Co., Ltd Nitrogen-containing condensed ring compounds having dopamine d3 receptor antagonistic effect
CN111801330B (zh) 2018-01-26 2024-04-05 盐野义制药株式会社 具有多巴胺d3受体拮抗作用的稠环化合物

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3388128A (en) * 1965-09-03 1968-06-11 Allan R. Day Substituted 1, 4-diazabicyclo [4. 4. 9] decanes
GB8518236D0 (en) * 1985-07-19 1985-08-29 Beecham Group Plc Compounds
WO1994006794A1 (en) * 1992-09-24 1994-03-31 National Institutes Of Health Aralkyl diazabicycloalkane derivatives for cns disorders
US6231833B1 (en) * 1999-08-05 2001-05-15 Pfizer Inc 2,7-substituted octahydro-1H-pyrido[1,2-A]pyrazine derivatives as ligands for serotonin receptors
US5731307A (en) * 1994-09-30 1998-03-24 Pfizer, Inc. Neuroleptic 2,7-disubtituted perhydro-1h-pyrido 1, 2-A!pyrazines
JP4749640B2 (ja) * 1999-07-19 2011-08-17 メルク フロスト カナダ リミテツド ピラジノン、このような化合物を含む組成物

Also Published As

Publication number Publication date
EP1275647A1 (fr) 2003-01-15
NZ520120A (en) 2004-03-26
KR20030007159A (ko) 2003-01-23
CA2394027C (fr) 2008-01-08
CA2394027A1 (fr) 2003-01-12
US20030195216A1 (en) 2003-10-16
KR100485020B1 (ko) 2005-04-25
AU2002300094B2 (en) 2007-06-14
DE60200089T2 (de) 2004-09-09
NO322966B1 (no) 2006-12-18
CN1397557A (zh) 2003-02-19
EA005160B1 (ru) 2004-12-30
BR0202681A (pt) 2003-05-06
EP1275647B1 (fr) 2003-11-12
FR2827288A1 (fr) 2003-01-17
JP3950018B2 (ja) 2007-07-25
DE60200089D1 (de) 2003-12-18
TR200302001T4 (tr) 2004-01-21
CN1197863C (zh) 2005-04-20
MXPA02006699A (es) 2005-08-16
US6992085B2 (en) 2006-01-31
JP2003064081A (ja) 2003-03-05
FR2827288B1 (fr) 2003-10-31
HU0202282D0 (xx) 2002-09-28
NO20023345D0 (no) 2002-07-11
EA200200663A1 (ru) 2003-02-27
AR036166A1 (es) 2004-08-18
ZA200205596B (en) 2003-03-27
DK1275647T3 (da) 2004-03-15
NO20023345L (no) 2003-01-13
ATE254124T1 (de) 2003-11-15
HUP0202282A2 (hu) 2003-03-28
ES2210219T3 (es) 2004-07-01
PT1275647E (pt) 2004-03-31
HK1050682A1 (en) 2003-07-04
HUP0202282A3 (en) 2003-11-28
PL355034A1 (en) 2003-01-13

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