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KR20070120617A - 치환된 아제티딘온 화합물을 포함하는 약제학적 조성물 - Google Patents

치환된 아제티딘온 화합물을 포함하는 약제학적 조성물 Download PDF

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Publication number
KR20070120617A
KR20070120617A KR1020077027662A KR20077027662A KR20070120617A KR 20070120617 A KR20070120617 A KR 20070120617A KR 1020077027662 A KR1020077027662 A KR 1020077027662A KR 20077027662 A KR20077027662 A KR 20077027662A KR 20070120617 A KR20070120617 A KR 20070120617A
Authority
KR
South Korea
Prior art keywords
alkyl
group
aryl
independently selected
substituted
Prior art date
Application number
KR1020077027662A
Other languages
English (en)
Korean (ko)
Inventor
해리 알. 데이비스
Original Assignee
쉐링 코포레이션
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23006987&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR20070120617(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 쉐링 코포레이션 filed Critical 쉐링 코포레이션
Publication of KR20070120617A publication Critical patent/KR20070120617A/ko

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Molecular Biology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
KR1020077027662A 2001-01-26 2002-01-25 치환된 아제티딘온 화합물을 포함하는 약제학적 조성물 KR20070120617A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US26464501P 2001-01-26 2001-01-26
US60/264,645 2001-01-26

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
KR1020037009673A Division KR100820983B1 (ko) 2001-01-26 2002-01-25 치환된 아제티딘온 화합물을 포함하는 약제학적 조성물

Publications (1)

Publication Number Publication Date
KR20070120617A true KR20070120617A (ko) 2007-12-24

Family

ID=23006987

Family Applications (2)

Application Number Title Priority Date Filing Date
KR1020077027662A KR20070120617A (ko) 2001-01-26 2002-01-25 치환된 아제티딘온 화합물을 포함하는 약제학적 조성물
KR1020037009673A KR100820983B1 (ko) 2001-01-26 2002-01-25 치환된 아제티딘온 화합물을 포함하는 약제학적 조성물

Family Applications After (1)

Application Number Title Priority Date Filing Date
KR1020037009673A KR100820983B1 (ko) 2001-01-26 2002-01-25 치환된 아제티딘온 화합물을 포함하는 약제학적 조성물

Country Status (33)

Country Link
US (2) US7417039B2 (de)
EP (1) EP1355644B1 (de)
JP (2) JP4711600B2 (de)
KR (2) KR20070120617A (de)
CN (1) CN100522159C (de)
AR (1) AR035533A1 (de)
AT (1) ATE331512T1 (de)
AU (1) AU2002243557B2 (de)
BR (1) BRPI0206641B8 (de)
CA (1) CA2434430A1 (de)
CY (1) CY1106149T1 (de)
CZ (1) CZ305202B6 (de)
DE (1) DE60212801T2 (de)
DK (1) DK1355644T3 (de)
ES (1) ES2266459T3 (de)
HK (1) HK1055679A1 (de)
HU (1) HU230435B1 (de)
IL (2) IL156422A0 (de)
ME (1) ME00145B (de)
MX (1) MXPA03006729A (de)
MY (1) MY138301A (de)
NO (1) NO333695B1 (de)
NZ (1) NZ526532A (de)
PE (1) PE20020850A1 (de)
PL (1) PL205343B1 (de)
PT (1) PT1355644E (de)
RS (1) RS50406B (de)
RU (2) RU2756946C2 (de)
SI (1) SI1355644T1 (de)
SK (1) SK287746B6 (de)
TW (1) TWI337076B (de)
WO (1) WO2002058696A2 (de)
ZA (1) ZA200305691B (de)

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YU59103A (sh) 2006-05-25
JP2007091763A (ja) 2007-04-12
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TWI337076B (en) 2011-02-11
ATE331512T1 (de) 2006-07-15
ZA200305691B (en) 2005-02-23
PL205343B1 (pl) 2010-04-30
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PT1355644E (pt) 2006-11-30
WO2002058696A3 (en) 2003-03-13
CZ20032038A3 (cs) 2003-12-17
RS50406B (sr) 2009-12-31
EP1355644B1 (de) 2006-06-28
WO2002058696A2 (en) 2002-08-01
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JP2004532186A (ja) 2004-10-21
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JP4614460B2 (ja) 2011-01-19
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US7417039B2 (en) 2008-08-26
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