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DK1355644T3 - Anvendelse af substituerede azetidinonforbindelser til behandling af sitosterolæmi - Google Patents

Anvendelse af substituerede azetidinonforbindelser til behandling af sitosterolæmi

Info

Publication number
DK1355644T3
DK1355644T3 DK02709050T DK02709050T DK1355644T3 DK 1355644 T3 DK1355644 T3 DK 1355644T3 DK 02709050 T DK02709050 T DK 02709050T DK 02709050 T DK02709050 T DK 02709050T DK 1355644 T3 DK1355644 T3 DK 1355644T3
Authority
DK
Denmark
Prior art keywords
sitosterolemia
treatment
substituted azetidinone
azetidinone compounds
compounds
Prior art date
Application number
DK02709050T
Other languages
English (en)
Inventor
Harry R Davis
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23006987&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK1355644(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Corp filed Critical Schering Corp
Application granted granted Critical
Publication of DK1355644T3 publication Critical patent/DK1355644T3/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • A61P31/06Antibacterial agents for tuberculosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Molecular Biology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK02709050T 2001-01-26 2002-01-25 Anvendelse af substituerede azetidinonforbindelser til behandling af sitosterolæmi DK1355644T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US26464501P 2001-01-26 2001-01-26

Publications (1)

Publication Number Publication Date
DK1355644T3 true DK1355644T3 (da) 2006-10-23

Family

ID=23006987

Family Applications (1)

Application Number Title Priority Date Filing Date
DK02709050T DK1355644T3 (da) 2001-01-26 2002-01-25 Anvendelse af substituerede azetidinonforbindelser til behandling af sitosterolæmi

Country Status (32)

Country Link
US (2) US7417039B2 (da)
EP (1) EP1355644B1 (da)
JP (2) JP4711600B2 (da)
KR (2) KR100820983B1 (da)
CN (1) CN100522159C (da)
AR (1) AR035533A1 (da)
AT (1) ATE331512T1 (da)
AU (1) AU2002243557B2 (da)
BR (1) BRPI0206641B8 (da)
CA (1) CA2434430A1 (da)
CY (1) CY1106149T1 (da)
CZ (1) CZ305202B6 (da)
DE (1) DE60212801T2 (da)
DK (1) DK1355644T3 (da)
ES (1) ES2266459T3 (da)
HU (1) HU230435B1 (da)
IL (2) IL156422A0 (da)
ME (1) ME00145B (da)
MX (1) MXPA03006729A (da)
MY (1) MY138301A (da)
NO (1) NO333695B1 (da)
NZ (1) NZ526532A (da)
PE (1) PE20020850A1 (da)
PL (1) PL205343B1 (da)
PT (1) PT1355644E (da)
RS (1) RS50406B (da)
RU (2) RU2756946C2 (da)
SI (1) SI1355644T1 (da)
SK (1) SK287746B6 (da)
TW (1) TWI337076B (da)
WO (1) WO2002058696A2 (da)
ZA (1) ZA200305691B (da)

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BRPI0206641B8 (pt) 2001-01-26 2021-05-25 Merck Sharp & Dohme uso de um inibidor da absorção de esteróis
DK1353696T3 (da) 2001-01-26 2007-04-10 Schering Corp Kombinationer af peroxisomproliferatoraktiveret receptor (PPAR)-aktivator(er) og sterolabsorptionsinhibitor(er) og behandlinger til vaskulære indikationer
PT1363668E (pt) * 2001-01-26 2007-11-07 Schering Corp Combinaçoes de sequestrante(s) de ácidos biliares e inibidor(es) de absorção de esterol e tratamento de indicações vasculares
EP1859796A3 (en) * 2001-09-21 2008-07-02 Schering Corporation Treatment of xanthoma with azetidinone derivatives as sterol absorption inhibitors
ATE411018T1 (de) * 2001-09-21 2008-10-15 Schering Corp Verfahren zur behandlung oder verhinderung von vaskulärer entzündung mit sterol-absorbierungs- inhibitor(en)
US7056906B2 (en) 2001-09-21 2006-06-06 Schering Corporation Combinations of hormone replacement therapy composition(s) and sterol absorption inhibitor(s) and treatments for vascular conditions in post-menopausal women
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EP1355644A2 (en) 2003-10-29
JP2004532186A (ja) 2004-10-21
AR035533A1 (es) 2004-06-02
ES2266459T3 (es) 2007-03-01
KR100820983B1 (ko) 2008-04-10
RS50406B (sr) 2009-12-31
JP2007091763A (ja) 2007-04-12
MY138301A (en) 2009-05-29
PE20020850A1 (es) 2002-09-21
YU59103A (sh) 2006-05-25
MXPA03006729A (es) 2003-10-24
AU2002243557B2 (en) 2006-01-05
KR20040025886A (ko) 2004-03-26
SK287746B6 (sk) 2011-08-04
US20020169134A1 (en) 2002-11-14
DE60212801T2 (de) 2007-02-01
MEP26808A (en) 2010-06-10
WO2002058696A2 (en) 2002-08-01
NZ526532A (en) 2005-01-28
CZ20032038A3 (cs) 2003-12-17
PL205343B1 (pl) 2010-04-30
BRPI0206641B1 (pt) 2017-06-20
CZ305202B6 (cs) 2015-06-10
HK1055679A1 (en) 2004-01-21
WO2002058696A3 (en) 2003-03-13
BR0206641A (pt) 2004-02-25
US20050080071A1 (en) 2005-04-14
NO333695B1 (no) 2013-08-26
IL156422A (en) 2009-06-15
BRPI0206641B8 (pt) 2021-05-25
CN1527707A (zh) 2004-09-08
KR20070120617A (ko) 2007-12-24
RU2003126187A (ru) 2005-02-20
EP1355644B1 (en) 2006-06-28
TWI337076B (en) 2011-02-11
JP4614460B2 (ja) 2011-01-19
HUP0303929A2 (hu) 2004-03-01
NO20033359D0 (no) 2003-07-25
ZA200305691B (en) 2005-02-23
CA2434430A1 (en) 2002-08-01
SI1355644T1 (sl) 2006-10-31
DE60212801D1 (de) 2006-08-10
IL156422A0 (en) 2004-01-04
ATE331512T1 (de) 2006-07-15
PT1355644E (pt) 2006-11-30
RU2007131955A (ru) 2009-02-27
CY1106149T1 (el) 2011-06-08
HU230435B1 (hu) 2016-06-28
PL364280A1 (en) 2004-12-13
US7417039B2 (en) 2008-08-26
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HUP0303929A3 (en) 2012-12-28
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RU2756946C2 (ru) 2021-10-07
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NO20033359L (no) 2003-09-25
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