KE3365A - New oxime derivatives of 7-aminothiazolylacetamido-cephalosporanic acid,processes for preparing them and pharmaceutical compositions incorporating them - Google Patents

New oxime derivatives of 7-aminothiazolylacetamido-cephalosporanic acid,processes for preparing them and pharmaceutical compositions incorporating them

Info

Publication number: KE3365A
Authority: KE; Kenya
Prior art keywords: aminothiazolylacetamido; preparing; processes; pharmaceutical compositions; cephalosporanic acid
Prior art date: 1976-01-23

Application number

KE3365A

Other languages

English (en)

Original Assignee

Roussel Uclaf

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-01-23

Filing date

1984-01-11

Publication date

1984-02-03

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27250574&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KE3365(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1976-01-23 Priority claimed from FR7601834A external-priority patent/FR2346014A1/fr

1976-06-11 Priority claimed from FR7617743A external-priority patent/FR2361893A2/fr

1976-08-18 Priority claimed from FR7625051A external-priority patent/FR2361894A2/fr

1984-01-11 Application filed by Roussel Uclaf filed Critical Roussel Uclaf

1984-02-03 Publication of KE3365A publication Critical patent/KE3365A/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/587—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/26—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
- C07D501/34—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group with the 7-amino radical acylated by carboxylic acids containing hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Oncology (AREA)
Pharmacology & Pharmacy (AREA)
Communicable Diseases (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Cephalosporin Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)

KE3365A 1976-01-23 1984-01-11 New oxime derivatives of 7-aminothiazolylacetamido-cephalosporanic acid,processes for preparing them and pharmaceutical compositions incorporating them KE3365A (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
FR7601834A FR2346014A1 (fr)	1976-01-23	1976-01-23	Nouvelles oximes derivees de l'acide 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
FR7617743A FR2361893A2 (fr)	1976-01-23	1976-06-11	Nouvelles oximes derivees de l'acide 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
FR7625051A FR2361894A2 (fr)	1976-01-23	1976-08-18	Nouvelles oximes derivees de l'acide 7-aminothiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments

Publications (1)

Publication Number	Publication Date
KE3365A true KE3365A (en)	1984-02-03

Family

ID=27250574

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
KE3365A KE3365A (en)	1976-01-23	1984-01-11	New oxime derivatives of 7-aminothiazolylacetamido-cephalosporanic acid,processes for preparing them and pharmaceutical compositions incorporating them

Country Status (31)

Country	Link
JP (3)	JPS52102293A (pl)
AR (1)	AR231985A1 (pl)
AT (2)	AT355205B (pl)
AU (1)	AU511680B2 (pl)
BE (1)	BE850662A (pl)
CA (1)	CA1319682C (pl)
CH (1)	CH622264A5 (pl)
CY (1)	CY1123A (pl)
DD (2)	DD128594A5 (pl)
DE (3)	DE2759895C2 (pl)
DK (1)	DK161082C (pl)
ES (2)	ES455089A1 (pl)
GB (2)	GB1580621A (pl)
GE (1)	GEP19970783B (pl)
GR (1)	GR70302B (pl)
HK (1)	HK50381A (pl)
HU (1)	HU173110B (pl)
IE (1)	IE45015B1 (pl)
IL (2)	IL51192A (pl)
IT (1)	IT1104601B (pl)
KE (1)	KE3365A (pl)
LU (1)	LU76624A1 (pl)
MX (1)	MX4407E (pl)
MY (1)	MY8500417A (pl)
NL (1)	NL7700706A (pl)
NZ (1)	NZ183150A (pl)
PL (1)	PL122698B1 (pl)
PT (1)	PT66099B (pl)
SE (2)	SE440655B (pl)
SU (1)	SU822754A3 (pl)
YU (3)	YU41060B (pl)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2408613A2 (fr) *	1977-07-19	1979-06-08	Roussel Uclaf	Nouvelles oximes derivees de l'acide 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
GB1576625A (en) *	1976-04-12	1980-10-08	Fujisawa Pharmaceutical Co	Syn isomer 3,7 disubstituted 3 cephem 4 carboxylic acid compounds and processes for the preparation thereof
DK162391C (da) *	1976-04-12	1992-03-09	Fujisawa Pharmaceutical Co	Analogifremgangsmaade til fremstilling af syn-isomerer af 3,7-disubstituerede 3-cephem-4-carboxylsyreforbindelser
GR63088B (en) *	1976-04-14	1979-08-09	Takeda Chemical Industries Ltd	Preparation process of novel cephalosporins
ZA781502B (en) *	1977-03-14	1979-09-26	Fujisawa Pharmaceutical Co	New cephem and cepham compounds and processes for preparation thereof
PH17188A (en)	1977-03-14	1984-06-14	Fujisawa Pharmaceutical Co	New cephem and cepham compounds and their pharmaceutical compositions and method of use
DE2714880A1 (de) *	1977-04-02	1978-10-26	Hoechst Ag	Cephemderivate und verfahren zu ihrer herstellung
FR2400519A1 (fr) *	1977-08-17	1979-03-16	Roussel Uclaf	Forme cristalline du sel de sodium d'un derive oximine de l'acide 7-amino-thiazolyl acetamido cephalosporanique, son procede de preparation et son application comme medicament
JPS5444695A (en) *	1977-09-13	1979-04-09	Fujisawa Pharmaceut Co Ltd	3,7-disubstituted-3-cephem-4-carboxylic acid and its salt and their preparation
FR2410655A1 (fr) *	1977-12-05	1979-06-29	Roussel Uclaf	Nouvelles oximes derivees de l'acide 3-substitue 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
JPS5498795A (en) *	1978-01-13	1979-08-03	Takeda Chem Ind Ltd	Cephalosporin derivative and its preparation
FR2387235A1 (fr) *	1978-01-23	1978-11-10	Fujisawa Pharmaceutical Co	Procede de preparation de composes d'acide 3,7-disubstitue-3-cephem-4-carboxylique et nouveaux produits ainsi obtenus, ayant une forte activite antibacterienne
FR2432521A1 (fr) *	1978-03-31	1980-02-29	Roussel Uclaf	Nouvelles oximes o-substituees derivees de l'acide 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
SE445350B (sv) *	1978-04-14	1986-06-16	Roussel Uclaf	Oximderivat av 3-azidometyl-7-amino-tiazolyl-acetamido-cefalosporansyra och dess anvendning som antibiotika
US4284631A (en) *	1978-07-31	1981-08-18	Fujisawa Pharmaceutical Co., Ltd.	7-Substituted cephem compounds and pharmaceutical antibacterial compositions containing them
FR2448543A1 (fr) *	1979-02-09	1980-09-05	Roussel Uclaf	Nouvelles oximes o-substituees par un radical comportant un ammonium quaternaire et derivees de l'acide 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
FR2461713A1 (fr) *	1979-07-19	1981-02-06	Roussel Uclaf	Nouvelles alcoyloximes substituees derivees de l'acide 7-(2-amino 4-thiazolyl) acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
FR2461712A1 (fr) *	1979-07-23	1981-02-06	Hoechst Ag	Procede de preparation de derives de cepheme
JPS57154175A (en) *	1981-03-16	1982-09-22	Mitsui Toatsu Chem Inc	2-thiazoleamine derivative, its preparation, and drug composition comprising it
FR2506307A1 (fr) *	1981-05-22	1982-11-26	Roussel Uclaf	Nouveaux derives substitues de l'acide 2-(2-amino 4-thiazolyl) 2-hydroxyimino acetique et leur procede de preparation
JPS57163386A (en) *	1981-08-13	1982-10-07	Takeda Chem Ind Ltd	Cephalosporin derivative and its production
EP0238060B1 (en)	1986-03-19	1992-01-08	Banyu Pharmaceutical Co., Ltd.	Cephalosporin derivatives, processes for their preparation and antibacterial agents
HUT53892A (en) *	1989-04-07	1990-12-28	Technologishen Kom Za Promy Mi	Process for producing synaminothiazolyl and synaminooxazolyl derivatives
CN112457271A (zh) *	2020-11-18	2021-03-09	河北合佳医药科技集团股份有限公司	一种氨噻肟酸中间体的连续流合成方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1399086A (en) *	1971-05-14	1975-06-25	Glaxo Lab Ltd	Cephalosporin compounds
GB1536281A (en) *	1975-06-09	1978-12-20	Takeda Chemical Industries Ltd	Cephem compounds
DK154939C (da)	1974-12-19	1989-06-12	Takeda Chemical Industries Ltd	Analogifremgangsmaade til fremstilling af thiazolylacetamido-cephemforbindelser eller farmaceutisk acceptable salte eller estere deraf
DE2760123C2 (de)	1976-01-23	1986-04-30	Roussel-Uclaf, Paris	7-Aminothiazolyl-syn-oxyiminoacetamidocephalosporansäuren, ihre Herstellung und sie enthaltende pharmazeutische Zusammensetzungen
JPS6011713B2 (ja)	1976-09-08	1985-03-27	武田薬品工業株式会社	セフアロスポリン誘導体およびその製造法

1976
- 1976-12-29 SE SE7614678A patent/SE440655B/xx not_active IP Right Cessation
- 1976-12-31 IL IL51192A patent/IL51192A/xx unknown
1977
- 1977-01-15 ES ES455089A patent/ES455089A1/es not_active Expired
- 1977-01-18 SU SU772439818A patent/SU822754A3/ru active
- 1977-01-19 AR AR266241A patent/AR231985A1/es active
- 1977-01-19 YU YU137/77A patent/YU41060B/xx unknown
- 1977-01-20 IT IT47727/77A patent/IT1104601B/it active Protection Beyond IP Right Term
- 1977-01-20 MX MX775372U patent/MX4407E/es unknown
- 1977-01-21 JP JP504977A patent/JPS52102293A/ja active Granted
- 1977-01-21 GB GB2640/77A patent/GB1580621A/en not_active Expired
- 1977-01-21 DE DE2759895A patent/DE2759895C2/de not_active Expired
- 1977-01-21 NZ NZ183150A patent/NZ183150A/xx unknown
- 1977-01-21 DK DK023677A patent/DK161082C/da active
- 1977-01-21 BE BE174311A patent/BE850662A/xx not_active IP Right Cessation
- 1977-01-21 PT PT66099A patent/PT66099B/pt unknown
- 1977-01-21 CY CY1123A patent/CY1123A/xx unknown
- 1977-01-21 CH CH78777A patent/CH622264A5/fr not_active IP Right Cessation
- 1977-01-21 GB GB15561/79A patent/GB1580623A/en not_active Expired
- 1977-01-21 DE DE2702501A patent/DE2702501C2/de not_active Expired
- 1977-01-21 LU LU76624A patent/LU76624A1/xx unknown
- 1977-01-21 CA CA000270375A patent/CA1319682C/fr not_active Expired - Lifetime
- 1977-01-21 DE DE2760287A patent/DE2760287C2/de not_active Expired
- 1977-01-21 DD DD7700197036A patent/DD128594A5/xx unknown
- 1977-01-21 HU HU77RO909A patent/HU173110B/hu unknown
- 1977-01-21 DD DD7700200629A patent/DD132869A5/xx unknown
- 1977-01-22 PL PL1977195504A patent/PL122698B1/pl unknown
- 1977-01-22 GR GR52630A patent/GR70302B/el unknown
- 1977-01-24 AU AU21579/77A patent/AU511680B2/en not_active Expired
- 1977-01-24 AT AT41277A patent/AT355205B/de not_active IP Right Cessation
- 1977-01-24 NL NL7700706A patent/NL7700706A/xx not_active Application Discontinuation
- 1977-01-24 IE IE148/77A patent/IE45015B1/en not_active IP Right Cessation
1978
- 1978-02-01 ES ES466539A patent/ES466539A1/es not_active Expired
1979
- 1979-03-20 AT AT0209479A patent/AT373592B/de not_active IP Right Cessation
- 1979-05-31 IL IL57445A patent/IL57445A0/xx not_active IP Right Cessation
1981
- 1981-10-22 HK HK503/81A patent/HK50381A/xx unknown
1982
- 1982-08-26 SE SE8204893A patent/SE455307B/sv not_active IP Right Cessation
1983
- 1983-01-04 YU YU00012/83A patent/YU1283A/xx unknown
- 1983-01-04 YU YU11/83A patent/YU43143B/xx unknown
1984
- 1984-01-11 KE KE3365A patent/KE3365A/xx unknown
1985
- 1985-12-30 MY MY417/85A patent/MY8500417A/xx unknown
1990
- 1990-04-19 JP JP2101872A patent/JPH03204868A/ja active Pending
1993
- 1993-01-20 JP JP5023427A patent/JPH05247013A/ja active Pending
- 1993-09-09 GE GEAP19931537A patent/GEP19970783B/en unknown

Also Published As

Publication number	Publication date
AT355205B (de)	1980-02-25
YU1183A (en)	1984-02-29
SU822754A3 (ru)	1981-04-15
AT373592B (de)	1984-02-10
GB1580621A (en)	1980-12-03
NL7700706A (nl)	1977-07-26
CH622264A5 (en)	1981-03-31
PT66099A (fr)	1977-02-01
PT66099B (fr)	1979-03-09
ES466539A1 (es)	1978-10-01
MX4407E (es)	1982-04-27
JPH05247013A (ja)	1993-09-24
DK23677A (da)	1977-07-24
JPS6228152B2 (pl)	1987-06-18
DE2759895C2 (de)	1986-01-16
PL122698B1 (en)	1982-08-31
ATA209479A (de)	1983-06-15
GEP19970783B (en)	1997-01-28
AU2157977A (en)	1978-08-03
CA1319682C (fr)	1993-06-29
SE455307B (sv)	1988-07-04
HK50381A (en)	1981-10-30
DE2760287C2 (pl)	1988-04-14
GB1580623A (en)	1980-12-03
DD132869A5 (de)	1978-11-15
DE2702501C2 (de)	1982-11-18
NZ183150A (en)	1979-12-11
JPS52102293A (en)	1977-08-27
CY1123A (en)	1982-02-19
ES455089A1 (es)	1978-04-16
DK161082B (da)	1991-05-27
IE45015L (en)	1977-07-23
IE45015B1 (en)	1982-06-02
BE850662A (fr)	1977-07-22
SE7614678L (sv)	1977-07-24
IL51192A (en)	1980-11-30
IL51192A0 (en)	1977-02-28
DK161082C (da)	1991-11-04
JPH03204868A (ja)	1991-09-06
DD128594A5 (de)	1977-11-30
YU13777A (en)	1983-04-30
IL57445A0 (en)	1979-09-30
AR231985A1 (es)	1985-04-30
AU511680B2 (en)	1980-08-28
YU1283A (en)	1984-02-29
YU43143B (en)	1989-04-30
SE440655B (sv)	1985-08-12
LU76624A1 (pl)	1977-08-12
GR70302B (pl)	1982-09-06
YU41060B (en)	1986-10-31
PL195504A1 (pl)	1978-03-13
SE8204893L (sv)	1982-08-26
HU173110B (hu)	1979-02-28
DE2702501A1 (de)	1977-07-28
MY8500417A (en)	1985-12-31
SE8204893D0 (sv)	1982-08-26
IT1104601B (it)	1985-10-21
ATA41277A (de)	1979-07-15

Publication	Publication Date	Title
KE3365A (en)	1984-02-03	New oxime derivatives of 7-aminothiazolylacetamido-cephalosporanic acid,processes for preparing them and pharmaceutical compositions incorporating them
IL48642A (en)	1979-12-30	3-amino-indazolecarboxylic acid derivatives,ther preparation and pharmaceutical compositions containing them
IL49911A (en)	1979-09-30	5-benzoyl-pyrrole-2-acetic acid derivatives, their preparation and pharmaceutical compositions containing them
IL49411A0 (en)	1976-06-30	Phenylalkane-carboxylic acid derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same
IL47360A (en)	1978-12-17	-amino- and -formyl- -(p-acycloxyphenyl) acetamido-3-cephem-4-carboxylic acid derivatives,their preparation and pharmaceutical compositions containing them
IL51403A (en)	1980-09-16	5-diazinyl-1,2-dithiole-3-thione derivatives, processes for the preparation thereof and pharmaceutical compositions containing them
JPS5762288A (en)	1982-04-15	Novel oxime derivative of 7-aminothiazolylacetamidocephalosporanic acid, manufacture and pharmaceutical composition
IL50928A0 (en)	1977-01-31	New phenoxy-phenoxy-alkanecarboxylic acid derivatives,their preparation and herbicidal compositions containing them
IL50736A0 (en)	1976-12-31	Phenoxyalkylcarboxylic acid derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same
IL52466A (en)	1980-06-30	7(2-acyl-2-hydroxyiminoacetamido)-3-tetrazol-5-ylthiomethyl-3-cephem-4-carboxylic acid derivatives,their preparation and pharmaceutical compositions containing them
IL50507A0 (en)	1976-11-30	Phenoxyalkylcarboxylic acid derivatives processes for the preparation thereof and pharmaceutical compositions containing the same
GB1543004A (en)	1979-03-28	7-aminothiazolylacetamido-cephalosporanic acid derivatives processes for preparing them and pharmaceutical compositions containing them
PH13924A (en)	1980-11-04	Glavulanic acid derivatives,pharmaceutical compositions containing same and method of preparation thereof
PH12450A (en)	1979-03-08	6-substituted 5-halogen-2,3-cresotic acid derivatives process of preparation and pharmaceutical compositions containing them
IL54859A (en)	1982-01-31	Derivatives of amidinopenicillanic acid,their production and pharmaceutical compositions containing them
ZA793966B (en)	1980-08-27	N-substituted aziridine-2-carboxylic acid derivatives,processes for their preparation,and pharmaceutical compositions thereof
IL52820A (en)	1981-02-27	Acylated benzimidazole-2-methanol and-2-carboxylic acid derivatives, their preparation and pharmaceutical compositions containing them
IL52638A (en)	1980-12-31	Clivanic acid derivatives,their preparation and pharmaceutical compositions containing them
IL46543A0 (en)	1975-04-25	New phenoxyalkyl-carboxylic acid derivatives,process for the preparation thereof and pharmaceutical compositions containing the same
IL55427A (en)	1981-12-31	2-hydrazonopropionic acid derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same
IL47299A (en)	1979-01-31	3-thiomethyl-3-cephem-4-carboxylic acid derivatives,their preparation and pharmaceutical compositions containing them
IL47519A (en)	1979-03-12	7-sulphinimidoyl(sulphimidoyl)-xanthone-2-carboxylic acid derivatives, their preparation and pharmaceutical compositions containing them
IL53030A (en)	1982-11-30	Derivatives of 9-chloroprednisolone,processes for their preparation and pharmaceutical compositions containing the same
IL49208A (en)	1980-10-26	13,14-dehydro-16-fluoro prostanoic acid derivatives of the f2,a2 and e2 series,process for their preparation and pharmaceutical compositions containing same
IL51205A (en)	1981-01-30	Derivatives of 5-acyl-indane-2-carboxylic acid,their production and pharmaceutical compositions containing them