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HK1076465A1 - Pyrimidyl sulphone amide derivatives as chemokine receptor modulators - Google Patents

Pyrimidyl sulphone amide derivatives as chemokine receptor modulators

Info

Publication number
HK1076465A1
HK1076465A1 HK05108513.6A HK05108513A HK1076465A1 HK 1076465 A1 HK1076465 A1 HK 1076465A1 HK 05108513 A HK05108513 A HK 05108513A HK 1076465 A1 HK1076465 A1 HK 1076465A1
Authority
HK
Hong Kong
Prior art keywords
pyrimidyl
chemokine receptor
receptor modulators
amide derivatives
sulphone amide
Prior art date
Application number
HK05108513.6A
Other languages
English (en)
Inventor
Mark Richard Ebden
Premji Meghani
Colin Bennion
Antony Ronald Cook
Roger Victor Bonnert
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of HK1076465A1 publication Critical patent/HK1076465A1/xx

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    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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HK05108513.6A 2002-07-27 2005-09-27 Pyrimidyl sulphone amide derivatives as chemokine receptor modulators HK1076465A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0217431.6A GB0217431D0 (en) 2002-07-27 2002-07-27 Novel compounds
PCT/GB2003/003175 WO2004011443A1 (en) 2002-07-27 2003-07-23 Pyrimidyl sulphone amide derivatives as chemokine receptor modulators

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HK1076465A1 true HK1076465A1 (en) 2006-01-20

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EP (1) EP1527051B1 (zh)
JP (1) JP4619782B2 (zh)
KR (2) KR20110033313A (zh)
CN (1) CN100345829C (zh)
AR (1) AR040700A1 (zh)
AU (1) AU2003281684B2 (zh)
BR (1) BR0312967A (zh)
CA (1) CA2493785C (zh)
CO (1) CO5680479A2 (zh)
EG (1) EG25893A (zh)
ES (1) ES2392965T3 (zh)
GB (1) GB0217431D0 (zh)
HK (1) HK1076465A1 (zh)
IL (1) IL166290A0 (zh)
IS (1) IS7697A (zh)
MX (1) MXPA05000960A (zh)
MY (1) MY139561A (zh)
NO (1) NO330531B1 (zh)
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RU (1) RU2342366C2 (zh)
TW (1) TWI340038B (zh)
UA (1) UA80283C2 (zh)
WO (1) WO2004011443A1 (zh)
ZA (1) ZA200500791B (zh)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0217431D0 (en) 2002-07-27 2002-09-04 Astrazeneca Ab Novel compounds
DE60318219T2 (de) 2002-08-24 2009-01-15 Astrazeneca Ab PYRIMIDINDERIVATE ALS MODULATOREN DER AKTIVITuT VON CHEMOKINREZEPTOREN
GB0401269D0 (en) * 2004-01-21 2004-02-25 Astrazeneca Ab Compounds
US7381738B2 (en) 2004-02-19 2008-06-03 Bristol-Myers Squibb Company Substituted bicycloalkylamine derivatives as modulators of chemokine receptor activity
US7288563B2 (en) 2004-02-19 2007-10-30 Bristol-Myers Squibb Company Substituted bicycloalkylamine derivatives as modulators of chemokine receptor activity
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