HK1057557A1 - Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof - Google Patents

Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof

Info

Publication number: HK1057557A1
Authority: HK; Hong Kong
Prior art keywords: compounds; production; methods; medicaments containing; bicyclic heterocycles
Prior art date: 2000-08-26

Application number

HK04100462A

Inventor

Frank Himmelsbach

Elke Langkopf

Brigit Jung

Stefan Blech

Flavio Solca

Original Assignee

Boehringer Ingelheim Pharma

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-08-26

Filing date

2004-01-21

Publication date

2004-04-08

2004-01-21 Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma

2004-04-08 Publication of HK1057557A1 publication Critical patent/HK1057557A1/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/94—Nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pulmonology (AREA)
Oncology (AREA)
Immunology (AREA)
Dermatology (AREA)
Urology & Nephrology (AREA)
Gastroenterology & Hepatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

HK04100462A 2000-08-26 2004-01-21 Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof HK1057557A1 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE10042058A DE10042058A1 (en)	2000-08-26	2000-08-26	Bicyclic heterocycles, medicaments containing these compounds, their use and processes for their preparation
PCT/EP2001/009532 WO2002018351A1 (en)	2000-08-26	2001-08-18	Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof

Publications (1)

Publication Number	Publication Date
HK1057557A1 true HK1057557A1 (en)	2004-04-08

Family

ID=7653945

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HK04100462A HK1057557A1 (en)	2000-08-26	2004-01-21	Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof

Country Status (31)

Country	Link
EP (1)	EP1315705A1 (en)
JP (1)	JP4834282B2 (en)
KR (1)	KR100862873B1 (en)
CN (1)	CN100404517C (en)
AR (1)	AR033562A1 (en)
AU (2)	AU2001287694B2 (en)
BG (1)	BG107559A (en)
BR (1)	BR0113519A (en)
CA (1)	CA2417897C (en)
CZ (1)	CZ302567B6 (en)
DE (1)	DE10042058A1 (en)
EA (1)	EA005679B1 (en)
EC (1)	ECSP034464A (en)
EE (1)	EE05269B1 (en)
HK (1)	HK1057557A1 (en)
HR (1)	HRP20030138A2 (en)
HU (1)	HUP0300819A3 (en)
IL (2)	IL154602A0 (en)
ME (1)	MEP58708A (en)
MX (1)	MXPA03001483A (en)
MY (1)	MY126132A (en)
NO (1)	NO324866B1 (en)
NZ (1)	NZ524668A (en)
PL (1)	PL360248A1 (en)
RS (1)	RS52279B (en)
SK (1)	SK287747B6 (en)
TW (1)	TWI294422B (en)
UA (1)	UA73004C2 (en)
UY (1)	UY26903A1 (en)
WO (1)	WO2002018351A1 (en)
ZA (1)	ZA200300991B (en)

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YU90901A (en)	1999-06-21	2004-07-15	Boehringer Ingelheim Pharma Gmbh. & Co.Kg.	Bicyclic heterocycles, medicaments containing these compounds, their use and methods for the production thereof
DE10042059A1 (en) *	2000-08-26	2002-03-07	Boehringer Ingelheim Pharma	Bicyclic heterocycles, medicaments containing these compounds, their use and processes for their preparation
US7019012B2 (en)	2000-12-20	2006-03-28	Boehringer Ingelheim International Pharma Gmbh & Co. Kg	Quinazoline derivatives and pharmaceutical compositions containing them
TWI324597B (en) *	2002-03-28	2010-05-11	Astrazeneca Ab	Quinazoline derivatives
US6924285B2 (en)	2002-03-30	2005-08-02	Boehringer Ingelheim Pharma Gmbh & Co.	Bicyclic heterocyclic compounds, pharmaceutical compositions containing these compounds, their use and process for preparing them
EA200701302A1 (en) *	2002-03-30	2007-12-28	Бёрингер Ингельхайм Фарма Гмбх Унд Ко. Кг	4- (N-PHYLENAMINO) QUINAZOLIN / -CHINOLINE AS THYROSINKINASE INHIBITORS
DE10214412A1 (en) *	2002-03-30	2003-10-09	Boehringer Ingelheim Pharma	Bicyclic heterocycles, pharmaceutical compositions containing these compounds, their use and process for their preparation
WO2004006846A2 (en)	2002-07-15	2004-01-22	Exelixis, Inc.	Receptor-type kinase modulators and methods of use
DE10326186A1 (en) *	2003-06-06	2004-12-23	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Bicyclic heterocycles, medicaments containing these compounds, their use and processes for their preparation
DE10334226A1 (en) *	2003-07-28	2005-02-17	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Use of tyrosine kinase inhibitors for the treatment of inflammatory processes
GB0317665D0 (en)	2003-07-29	2003-09-03	Astrazeneca Ab	Qinazoline derivatives
SI1667992T1 (en)	2003-09-19	2007-06-30	Astrazeneca Ab	Quinazoline derivatives
WO2005030140A2 (en)	2003-09-26	2005-04-07	Exelixis, Inc.	C-met modulators and methods of use
US7456189B2 (en)	2003-09-30	2008-11-25	Boehringer Ingelheim International Gmbh	Bicyclic heterocycles, medicaments containing these compounds, their use and processes for their preparation
DE10345875A1 (en) *	2003-09-30	2005-04-21	Boehringer Ingelheim Pharma	Bicyclic heterocycles, pharmaceutical compositions containing them, their use and methods of preparation
DE10350717A1 (en) *	2003-10-30	2005-06-02	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Use of tyrosine kinase inhibitors for the treatment of inflammatory processes
US20060035893A1 (en)	2004-08-07	2006-02-16	Boehringer Ingelheim International Gmbh	Pharmaceutical compositions for treatment of respiratory and gastrointestinal disorders
PE20060777A1 (en)	2004-12-24	2006-10-06	Boehringer Ingelheim Int	INDOLINONE DERIVATIVES FOR THE TREATMENT OR PREVENTION OF FIBROTIC DISEASES
KR20070107151A (en)	2005-02-26	2007-11-06	아스트라제네카 아베	Quinazoline derivatives as tyrosine kinase inhibitors
KR100673775B1 (en) *	2005-04-08	2007-01-24	엘지전자 주식회사	Home bar door of refrigerator
CA2619037A1 (en) *	2005-08-22	2007-03-01	Boehringer Ingelheim International Gmbh	Bicyclic heterocycles medicaments comprising said compounds use and method for production thereof
WO2007054550A1 (en)	2005-11-11	2007-05-18	Boehringer Ingelheim International Gmbh	Quinazoline derivatives for the treatment of cancer diseases
WO2007101782A1 (en) *	2006-03-09	2007-09-13	Boehringer Ingelheim International Gmbh	Bicyclic heterocycles, medicaments containing these compounds, their use and process for preparing them
US8877764B2 (en)	2006-09-18	2014-11-04	Boehringer Ingelheim International Gmbh	Method for treating cancer harboring EGFR mutations
EP1921070A1 (en)	2006-11-10	2008-05-14	Boehringer Ingelheim Pharma GmbH & Co. KG	Bicyclic heterocycles, medicaments comprising them, their use and process for their preparation
MX2009007610A (en)	2007-02-06	2009-07-24	Boehringer Ingelheim Int	Bicyclic heterocycles, drugs containing said compounds, use thereof, and method for production thereof.
BRPI0907916A2 (en)	2008-02-07	2015-07-28	Boehringer Ingelheim Int	Spirocycle heterocycles, medicaments containing such compounds, and processes for preparing them
BRPI0912170A2 (en)	2008-05-13	2015-10-13	Astrazeneca Ab	compound, form, process for preparation thereof, pharmaceutical composition, use of a compound, and method for treating cancer in a warm-blooded animal
CA2733153C (en)	2008-08-08	2016-11-08	Boehringer Ingelheim International Gmbh	Cyclohexyloxy substituted heterocycles, pharmaceutical compositions containing these compounds and processes for preparing them
NZ618004A (en)	2009-01-16	2015-06-26	Exelixis Inc	Malate salt of n-(4-{ [6,7-bis(methyloxy)quinolin-4-yl]oxy} phenyl)-n’-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide, and crystalline forms thereof for the treatment of cancer
US9545381B2 (en)	2009-07-06	2017-01-17	Boehringer Ingelheim International Gmbh	Process for drying of BIBW2992, of its salts and of solid pharmaceutical formulations comprising this active ingredient
UA108618C2 (en)	2009-08-07	2015-05-25		APPLICATION OF C-MET-MODULATORS IN COMBINATION WITH THEMOSOLOMID AND / OR RADIATION THERAPY FOR CANCER TREATMENT
KR101317809B1 (en)	2011-06-07	2013-10-16	한미약품 주식회사	Pharmaceutical composition comprising amide derivative inhibiting the growth of cancer cell and non-metalic salt lubricant
KR20140096571A (en)	2013-01-28	2014-08-06	한미약품 주식회사	Method for preparing 1-(4-(4-(3,4-dichloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yloxy)piperidin-1-yl)prop-2-en-1-one
KR101645112B1 (en)	2013-03-06	2016-08-02	아스트라제네카 아베	Quinazoline inhibitors of activating mutant forms of epidermal growth factor receptor
US9242965B2 (en)	2013-12-31	2016-01-26	Boehringer Ingelheim International Gmbh	Process for the manufacture of (E)-4-N,N-dialkylamino crotonic acid in HX salt form and use thereof for synthesis of EGFR tyrosine kinase inhibitors
ES2776359T3 (en) *	2014-04-04	2020-07-30	H Lundbeck As	Quinazolin-thf-halogenated amines as PDE1 inhibitors
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WO2018094225A1 (en)	2016-11-17	2018-05-24	Board Of Regents, The University Of Texas System	Compounds with anti-tumor activity against cancer cells bearing egfr or her2 exon 20 mutations
CN112321814B (en) *	2020-12-30	2021-03-23	广州初曲科技有限公司	Preparation and application of gefitinib idebenone conjugate

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DE19911509A1 (en) *	1999-03-15	2000-09-21	Boehringer Ingelheim Pharma	Bicyclic heterocycles, medicaments containing these compounds, their use and processes for their preparation

2000
- 2000-08-26 DE DE10042058A patent/DE10042058A1/en not_active Ceased
2001
- 2001-08-18 RS YU14003A patent/RS52279B/en unknown
- 2001-08-18 AU AU2001287694A patent/AU2001287694B2/en not_active Ceased
- 2001-08-18 JP JP2002523469A patent/JP4834282B2/en not_active Expired - Fee Related
- 2001-08-18 ME MEP-587/08A patent/MEP58708A/en unknown
- 2001-08-18 IL IL15460201A patent/IL154602A0/en unknown
- 2001-08-18 EA EA200300219A patent/EA005679B1/en not_active IP Right Cessation
- 2001-08-18 MX MXPA03001483A patent/MXPA03001483A/en active IP Right Grant
- 2001-08-18 CN CNB01814635XA patent/CN100404517C/en not_active Expired - Fee Related
- 2001-08-18 HU HU0300819A patent/HUP0300819A3/en unknown
- 2001-08-18 CA CA002417897A patent/CA2417897C/en not_active Expired - Fee Related
- 2001-08-18 NZ NZ524668A patent/NZ524668A/en not_active IP Right Cessation
- 2001-08-18 KR KR1020037002744A patent/KR100862873B1/en not_active IP Right Cessation
- 2001-08-18 AU AU8769401A patent/AU8769401A/en active Pending
- 2001-08-18 CZ CZ20030870A patent/CZ302567B6/en not_active IP Right Cessation
- 2001-08-18 EE EEP200300077A patent/EE05269B1/en not_active IP Right Cessation
- 2001-08-18 WO PCT/EP2001/009532 patent/WO2002018351A1/en active Application Filing
- 2001-08-18 BR BR0113519-8A patent/BR0113519A/en active Pending
- 2001-08-18 PL PL36024801A patent/PL360248A1/en not_active Application Discontinuation
- 2001-08-18 SK SK231-2003A patent/SK287747B6/en not_active IP Right Cessation
- 2001-08-18 EP EP01967285A patent/EP1315705A1/en not_active Ceased
- 2001-08-18 UA UA2003032533A patent/UA73004C2/en unknown
- 2001-08-23 UY UY26903A patent/UY26903A1/en not_active Application Discontinuation
- 2001-08-24 AR ARP010104041A patent/AR033562A1/en not_active Suspension/Interruption
- 2001-08-24 MY MYPI20013985A patent/MY126132A/en unknown
- 2001-08-24 TW TW090120905A patent/TWI294422B/en not_active IP Right Cessation
2003
- 2003-02-03 EC EC2003004464A patent/ECSP034464A/en unknown
- 2003-02-05 ZA ZA200300991A patent/ZA200300991B/en unknown
- 2003-02-14 BG BG107559A patent/BG107559A/en active Pending
- 2003-02-24 IL IL154602A patent/IL154602A/en not_active IP Right Cessation
- 2003-02-24 HR HR20030138A patent/HRP20030138A2/en not_active Application Discontinuation
- 2003-02-25 NO NO20030870A patent/NO324866B1/en not_active IP Right Cessation
2004
- 2004-01-21 HK HK04100462A patent/HK1057557A1/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
TWI294422B (en)	2008-03-11
AU2001287694B2 (en)	2007-09-06
BR0113519A (en)	2003-07-01
CN100404517C (en)	2008-07-23
HUP0300819A3 (en)	2008-03-28
ECSP034464A (en)	2003-03-31
EA005679B1 (en)	2005-04-28
AR033562A1 (en)	2003-12-26
NO20030870L (en)	2003-02-25
IL154602A0 (en)	2003-09-17
MEP58708A (en)	2011-05-10
BG107559A (en)	2003-10-31
NO20030870D0 (en)	2003-02-25
SK2312003A3 (en)	2003-10-07
WO2002018351A1 (en)	2002-03-07
EA200300219A1 (en)	2003-08-28
AU8769401A (en)	2002-03-13
CN1449390A (en)	2003-10-15
UY26903A1 (en)	2002-03-22
HRP20030138A2 (en)	2005-04-30
UA73004C2 (en)	2005-05-16
CZ302567B6 (en)	2011-07-13
SK287747B6 (en)	2011-08-04
ZA200300991B (en)	2004-04-16
DE10042058A1 (en)	2002-03-07
NZ524668A (en)	2006-06-30
NO324866B1 (en)	2007-12-17
RS52279B (en)	2012-10-31
CA2417897A1 (en)	2003-01-30
KR100862873B1 (en)	2008-10-15
MY126132A (en)	2006-09-29
PL360248A1 (en)	2004-09-06
EP1315705A1 (en)	2003-06-04
EE200300077A (en)	2004-12-15
YU14003A (en)	2006-01-16
JP2004507529A (en)	2004-03-11
HUP0300819A2 (en)	2003-09-29
MXPA03001483A (en)	2003-06-06
CA2417897C (en)	2009-03-31
EE05269B1 (en)	2010-02-15
IL154602A (en)	2008-07-08
JP4834282B2 (en)	2011-12-14
KR20030024914A (en)	2003-03-26

Publication	Publication Date	Title
HUP0300819A3 (en)	2008-03-28	Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof
IL147133A0 (en)	2002-08-14	Bicyclic heterocycles, medicaments containing these compounds, their use and methods for the production thereof
AU2001295481A1 (en)	2002-03-13	Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof
AU2001287694A1 (en)	2002-06-06	Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof
IL156552A0 (en)	2004-01-04	Diphenyl azetidinone derivatives, method for the production thereof, medicaments containing these compounds, and their use
IL156548A0 (en)	2004-01-04	Diphenyl azetidinone derivatives, method for the production thereof, medicaments containing these compounds, and their use
AU6383101A (en)	2001-10-23	Bicyclic heterocylces, medicaments containing said compounds, the use thereof and method for producing them
MXPA03000873A (en)	2003-06-06	Quinazoline derivatives, medicaments containing these compounds, their use, and methods for the production thereof.
HUS1400005I1 (en)	2017-08-28	Quinazoline derivatives, medicaments containing said compounds, their utilization and method for the production thereof
MXPA03001510A (en)	2003-06-09	Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof.
HUP0401081A3 (en)	2010-06-28	Novel 1,2-diphenzylazetidinones, method for producing the same, medicaments containing said compounds, and their use
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2013-03-15	PC	Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)	Effective date: 20120818