AU2001287694A1 - Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof - Google Patents

Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof

Info

Publication number: AU2001287694A1
Authority: AU; Australia
Prior art keywords: compounds; production; methods; medicaments containing; bicyclic heterocycles
Prior art date: 2000-08-26
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

AU2001287694A

Other versions

AU2001287694B2 (en

Inventor

Stefan Blech

Frank Himmelsbach

Birgit Jung

Elke Langkopf

Flavio Solca

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Boehringer Ingelheim Pharma GmbH and Co KG

Original Assignee

Boehringer Ingelheim Pharma GmbH and Co KG

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-08-26

Filing date

2001-08-18

Publication date

2002-06-06

2000-08-26 Priority claimed from DE10042058A external-priority patent/DE10042058A1/en

2001-08-18 Application filed by Boehringer Ingelheim Pharma GmbH and Co KG filed Critical Boehringer Ingelheim Pharma GmbH and Co KG

2002-06-06 Publication of AU2001287694A1 publication Critical patent/AU2001287694A1/en

2007-09-06 Application granted granted Critical

2007-09-06 Publication of AU2001287694B2 publication Critical patent/AU2001287694B2/en

2021-08-18 Anticipated expiration legal-status Critical

Status Ceased legal-status Critical Current

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
DE10042058.3		2000-08-26
DE10042058A DE10042058A1 (en)	2000-08-26	2000-08-26	Bicyclic heterocycles, medicaments containing these compounds, their use and processes for their preparation
PCT/EP2001/009532 WO2002018351A1 (en)	2000-08-26	2001-08-18	Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof

Publications (2)

Publication Number	Publication Date
AU2001287694A1 true AU2001287694A1 (en)	2002-06-06
AU2001287694B2 AU2001287694B2 (en)	2007-09-06

Family

ID=7653945

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
AU2001287694A Ceased AU2001287694B2 (en)	2000-08-26	2001-08-18	Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof
AU8769401A Pending AU8769401A (en)	2000-08-26	2001-08-18	Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
AU8769401A Pending AU8769401A (en)	2000-08-26	2001-08-18	Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof

Country Status (31)

Country	Link
EP (1)	EP1315705A1 (en)
JP (1)	JP4834282B2 (en)
KR (1)	KR100862873B1 (en)
CN (1)	CN100404517C (en)
AR (1)	AR033562A1 (en)
AU (2)	AU2001287694B2 (en)
BG (1)	BG107559A (en)
BR (1)	BR0113519A (en)
CA (1)	CA2417897C (en)
CZ (1)	CZ302567B6 (en)
DE (1)	DE10042058A1 (en)
EA (1)	EA005679B1 (en)
EC (1)	ECSP034464A (en)
EE (1)	EE05269B1 (en)
HK (1)	HK1057557A1 (en)
HR (1)	HRP20030138A2 (en)
HU (1)	HUP0300819A3 (en)
IL (2)	IL154602A0 (en)
ME (1)	MEP58708A (en)
MX (1)	MXPA03001483A (en)
MY (1)	MY126132A (en)
NO (1)	NO324866B1 (en)
NZ (1)	NZ524668A (en)
PL (1)	PL360248A1 (en)
RS (1)	RS52279B (en)
SK (1)	SK287747B6 (en)
TW (1)	TWI294422B (en)
UA (1)	UA73004C2 (en)
UY (1)	UY26903A1 (en)
WO (1)	WO2002018351A1 (en)
ZA (1)	ZA200300991B (en)

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YU90901A (en)	1999-06-21	2004-07-15	Boehringer Ingelheim Pharma Gmbh. & Co.Kg.	Bicyclic heterocycles, medicaments containing these compounds, their use and methods for the production thereof
DE10042059A1 (en) *	2000-08-26	2002-03-07	Boehringer Ingelheim Pharma	Bicyclic heterocycles, medicaments containing these compounds, their use and processes for their preparation
US7019012B2 (en)	2000-12-20	2006-03-28	Boehringer Ingelheim International Pharma Gmbh & Co. Kg	Quinazoline derivatives and pharmaceutical compositions containing them
TWI324597B (en) *	2002-03-28	2010-05-11	Astrazeneca Ab	Quinazoline derivatives
US6924285B2 (en)	2002-03-30	2005-08-02	Boehringer Ingelheim Pharma Gmbh & Co.	Bicyclic heterocyclic compounds, pharmaceutical compositions containing these compounds, their use and process for preparing them
EA200701302A1 (en) *	2002-03-30	2007-12-28	Бёрингер Ингельхайм Фарма Гмбх Унд Ко. Кг	4- (N-PHYLENAMINO) QUINAZOLIN / -CHINOLINE AS THYROSINKINASE INHIBITORS
DE10214412A1 (en) *	2002-03-30	2003-10-09	Boehringer Ingelheim Pharma	Bicyclic heterocycles, pharmaceutical compositions containing these compounds, their use and process for their preparation
WO2004006846A2 (en)	2002-07-15	2004-01-22	Exelixis, Inc.	Receptor-type kinase modulators and methods of use
DE10326186A1 (en) *	2003-06-06	2004-12-23	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Bicyclic heterocycles, medicaments containing these compounds, their use and processes for their preparation
DE10334226A1 (en) *	2003-07-28	2005-02-17	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Use of tyrosine kinase inhibitors for the treatment of inflammatory processes
GB0317665D0 (en)	2003-07-29	2003-09-03	Astrazeneca Ab	Qinazoline derivatives
SI1667992T1 (en)	2003-09-19	2007-06-30	Astrazeneca Ab	Quinazoline derivatives
WO2005030140A2 (en)	2003-09-26	2005-04-07	Exelixis, Inc.	C-met modulators and methods of use
US7456189B2 (en)	2003-09-30	2008-11-25	Boehringer Ingelheim International Gmbh	Bicyclic heterocycles, medicaments containing these compounds, their use and processes for their preparation
DE10345875A1 (en) *	2003-09-30	2005-04-21	Boehringer Ingelheim Pharma	Bicyclic heterocycles, pharmaceutical compositions containing them, their use and methods of preparation
DE10350717A1 (en) *	2003-10-30	2005-06-02	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Use of tyrosine kinase inhibitors for the treatment of inflammatory processes
US20060035893A1 (en)	2004-08-07	2006-02-16	Boehringer Ingelheim International Gmbh	Pharmaceutical compositions for treatment of respiratory and gastrointestinal disorders
PE20060777A1 (en)	2004-12-24	2006-10-06	Boehringer Ingelheim Int	INDOLINONE DERIVATIVES FOR THE TREATMENT OR PREVENTION OF FIBROTIC DISEASES
KR20070107151A (en)	2005-02-26	2007-11-06	아스트라제네카 아베	Quinazoline derivatives as tyrosine kinase inhibitors
KR100673775B1 (en) *	2005-04-08	2007-01-24	엘지전자 주식회사	Home bar door of refrigerator
CA2619037A1 (en) *	2005-08-22	2007-03-01	Boehringer Ingelheim International Gmbh	Bicyclic heterocycles medicaments comprising said compounds use and method for production thereof
WO2007054550A1 (en)	2005-11-11	2007-05-18	Boehringer Ingelheim International Gmbh	Quinazoline derivatives for the treatment of cancer diseases
WO2007101782A1 (en) *	2006-03-09	2007-09-13	Boehringer Ingelheim International Gmbh	Bicyclic heterocycles, medicaments containing these compounds, their use and process for preparing them
US8877764B2 (en)	2006-09-18	2014-11-04	Boehringer Ingelheim International Gmbh	Method for treating cancer harboring EGFR mutations
EP1921070A1 (en)	2006-11-10	2008-05-14	Boehringer Ingelheim Pharma GmbH & Co. KG	Bicyclic heterocycles, medicaments comprising them, their use and process for their preparation
MX2009007610A (en)	2007-02-06	2009-07-24	Boehringer Ingelheim Int	Bicyclic heterocycles, drugs containing said compounds, use thereof, and method for production thereof.
BRPI0907916A2 (en)	2008-02-07	2015-07-28	Boehringer Ingelheim Int	Spirocycle heterocycles, medicaments containing such compounds, and processes for preparing them
BRPI0912170A2 (en)	2008-05-13	2015-10-13	Astrazeneca Ab	compound, form, process for preparation thereof, pharmaceutical composition, use of a compound, and method for treating cancer in a warm-blooded animal
CA2733153C (en)	2008-08-08	2016-11-08	Boehringer Ingelheim International Gmbh	Cyclohexyloxy substituted heterocycles, pharmaceutical compositions containing these compounds and processes for preparing them
NZ618004A (en)	2009-01-16	2015-06-26	Exelixis Inc	Malate salt of n-(4-{ [6,7-bis(methyloxy)quinolin-4-yl]oxy} phenyl)-n’-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide, and crystalline forms thereof for the treatment of cancer
US9545381B2 (en)	2009-07-06	2017-01-17	Boehringer Ingelheim International Gmbh	Process for drying of BIBW2992, of its salts and of solid pharmaceutical formulations comprising this active ingredient
UA108618C2 (en)	2009-08-07	2015-05-25		APPLICATION OF C-MET-MODULATORS IN COMBINATION WITH THEMOSOLOMID AND / OR RADIATION THERAPY FOR CANCER TREATMENT
KR101317809B1 (en)	2011-06-07	2013-10-16	한미약품 주식회사	Pharmaceutical composition comprising amide derivative inhibiting the growth of cancer cell and non-metalic salt lubricant
KR20140096571A (en)	2013-01-28	2014-08-06	한미약품 주식회사	Method for preparing 1-(4-(4-(3,4-dichloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yloxy)piperidin-1-yl)prop-2-en-1-one
KR101645112B1 (en)	2013-03-06	2016-08-02	아스트라제네카 아베	Quinazoline inhibitors of activating mutant forms of epidermal growth factor receptor
US9242965B2 (en)	2013-12-31	2016-01-26	Boehringer Ingelheim International Gmbh	Process for the manufacture of (E)-4-N,N-dialkylamino crotonic acid in HX salt form and use thereof for synthesis of EGFR tyrosine kinase inhibitors
ES2776359T3 (en) *	2014-04-04	2020-07-30	H Lundbeck As	Quinazolin-thf-halogenated amines as PDE1 inhibitors
US20170176028A1 (en)	2015-12-18	2017-06-22	Lg Electronics Inc.	Air conditioner
WO2018094225A1 (en)	2016-11-17	2018-05-24	Board Of Regents, The University Of Texas System	Compounds with anti-tumor activity against cancer cells bearing egfr or her2 exon 20 mutations
CN112321814B (en) *	2020-12-30	2021-03-23	广州初曲科技有限公司	Preparation and application of gefitinib idebenone conjugate

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9508538D0 (en) *	1995-04-27	1995-06-14	Zeneca Ltd	Quinazoline derivatives
GB9624482D0 (en) *	1995-12-18	1997-01-15	Zeneca Phaema S A	Chemical compounds
NZ330868A (en) *	1996-02-13	2000-01-28	Zeneca Ltd	4-phenoxy, phenylthio or phenylamino substituted quinazoline derivatives ane medicaments useful as VEGF inhibitors
GB9603095D0 (en) *	1996-02-14	1996-04-10	Zeneca Ltd	Quinazoline derivatives
ES2169355T3 (en) *	1996-03-05	2002-07-01	Astrazeneca Ab	DERIVATIVES OF 4-ANILINOQUINAZOLINA.
RO121900B1 (en) *	1996-04-12	2008-07-30	Warner-Lambert Company	Irreversible inhibitors of tyrosine kinazes, pharmaceutical composition containing the same and use thereof
GB9718972D0 (en) *	1996-09-25	1997-11-12	Zeneca Ltd	Chemical compounds
DE19911509A1 (en) *	1999-03-15	2000-09-21	Boehringer Ingelheim Pharma	Bicyclic heterocycles, medicaments containing these compounds, their use and processes for their preparation

2000
- 2000-08-26 DE DE10042058A patent/DE10042058A1/en not_active Ceased
2001
- 2001-08-18 RS YU14003A patent/RS52279B/en unknown
- 2001-08-18 AU AU2001287694A patent/AU2001287694B2/en not_active Ceased
- 2001-08-18 JP JP2002523469A patent/JP4834282B2/en not_active Expired - Fee Related
- 2001-08-18 ME MEP-587/08A patent/MEP58708A/en unknown
- 2001-08-18 IL IL15460201A patent/IL154602A0/en unknown
- 2001-08-18 EA EA200300219A patent/EA005679B1/en not_active IP Right Cessation
- 2001-08-18 MX MXPA03001483A patent/MXPA03001483A/en active IP Right Grant
- 2001-08-18 CN CNB01814635XA patent/CN100404517C/en not_active Expired - Fee Related
- 2001-08-18 HU HU0300819A patent/HUP0300819A3/en unknown
- 2001-08-18 CA CA002417897A patent/CA2417897C/en not_active Expired - Fee Related
- 2001-08-18 NZ NZ524668A patent/NZ524668A/en not_active IP Right Cessation
- 2001-08-18 KR KR1020037002744A patent/KR100862873B1/en not_active IP Right Cessation
- 2001-08-18 AU AU8769401A patent/AU8769401A/en active Pending
- 2001-08-18 CZ CZ20030870A patent/CZ302567B6/en not_active IP Right Cessation
- 2001-08-18 EE EEP200300077A patent/EE05269B1/en not_active IP Right Cessation
- 2001-08-18 WO PCT/EP2001/009532 patent/WO2002018351A1/en active Application Filing
- 2001-08-18 BR BR0113519-8A patent/BR0113519A/en active Pending
- 2001-08-18 PL PL36024801A patent/PL360248A1/en not_active Application Discontinuation
- 2001-08-18 SK SK231-2003A patent/SK287747B6/en not_active IP Right Cessation
- 2001-08-18 EP EP01967285A patent/EP1315705A1/en not_active Ceased
- 2001-08-18 UA UA2003032533A patent/UA73004C2/en unknown
- 2001-08-23 UY UY26903A patent/UY26903A1/en not_active Application Discontinuation
- 2001-08-24 AR ARP010104041A patent/AR033562A1/en not_active Suspension/Interruption
- 2001-08-24 MY MYPI20013985A patent/MY126132A/en unknown
- 2001-08-24 TW TW090120905A patent/TWI294422B/en not_active IP Right Cessation
2003
- 2003-02-03 EC EC2003004464A patent/ECSP034464A/en unknown
- 2003-02-05 ZA ZA200300991A patent/ZA200300991B/en unknown
- 2003-02-14 BG BG107559A patent/BG107559A/en active Pending
- 2003-02-24 IL IL154602A patent/IL154602A/en not_active IP Right Cessation
- 2003-02-24 HR HR20030138A patent/HRP20030138A2/en not_active Application Discontinuation
- 2003-02-25 NO NO20030870A patent/NO324866B1/en not_active IP Right Cessation
2004
- 2004-01-21 HK HK04100462A patent/HK1057557A1/en not_active IP Right Cessation

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