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ES8705886A1 - Un metodo para preparar un derivadode tiazolidin-diona - Google Patents

Un metodo para preparar un derivadode tiazolidin-diona

Info

Publication number
ES8705886A1
ES8705886A1 ES550986A ES550986A ES8705886A1 ES 8705886 A1 ES8705886 A1 ES 8705886A1 ES 550986 A ES550986 A ES 550986A ES 550986 A ES550986 A ES 550986A ES 8705886 A1 ES8705886 A1 ES 8705886A1
Authority
ES
Spain
Prior art keywords
thiazolidinedione derivatives
production
therapeutic agent
hyperlipemia
diabetes
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES550986A
Other languages
English (en)
Other versions
ES550986A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Takeda Pharmaceutical Co Ltd
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=11683488&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ES8705886(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of ES8705886A1 publication Critical patent/ES8705886A1/es
Publication of ES550986A0 publication Critical patent/ES550986A0/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms
    • C07D213/30—Oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Obesity (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)

Abstract

METODO DE PREPARAR UN DERIVADO DE TIAZOLIDIN-DIONA. CONSISTE EN HIDROLIZAR UN COMPUESTO DE FORMULA (II) EN PRESENCIA DE UN ACIDO MINERAL (CLH O BRH), EN ALCANOL O SULFOXIDO DE DIMETILO, ENTRE 20 Y 150JC Y DURANTE 0,5 A 20 HORAS, PARA OBTENER UN DERIVADO DE TIAZOLIDIN-DIONA DE FORMULA (I) Y SUS SALES FARMACEUTICAMENTE ACEPTABLES.SE UTILIZAN COMO ANTIDIABETICOS EN FORMA DE TABLETAS, POLVOS O GRANULOS.
ES550986A 1985-01-19 1986-01-17 Un metodo para preparar un derivadode tiazolidin-diona Expired ES8705886A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP808585 1985-01-19

Publications (2)

Publication Number Publication Date
ES8705886A1 true ES8705886A1 (es) 1987-05-16
ES550986A0 ES550986A0 (es) 1987-05-16

Family

ID=11683488

Family Applications (1)

Application Number Title Priority Date Filing Date
ES550986A Expired ES8705886A1 (es) 1985-01-19 1986-01-17 Un metodo para preparar un derivadode tiazolidin-diona

Country Status (28)

Country Link
US (1) US4687777A (es)
EP (1) EP0193256B1 (es)
JP (1) JPS61267580A (es)
KR (1) KR920010046B1 (es)
CN (1) CN1003934B (es)
AR (1) AR240698A1 (es)
AT (1) ATE41931T1 (es)
AU (1) AU572719B2 (es)
BR (1) BR1100325A (es)
CA (1) CA1277323C (es)
CS (1) CS407991A3 (es)
DE (2) DE3662689D1 (es)
DK (2) DK21986A (es)
ES (1) ES8705886A1 (es)
FI (1) FI81098C (es)
GR (1) GR860124B (es)
HK (1) HK3692A (es)
HU (1) HU196795B (es)
IE (1) IE58928B1 (es)
LU (1) LU90719I2 (es)
LV (1) LV5779B4 (es)
MX (1) MX9202933A (es)
MY (1) MY102016A (es)
NL (1) NL300038I2 (es)
NO (1) NO163857C (es)
PT (1) PT81859B (es)
SG (1) SG105691G (es)
ZA (1) ZA86203B (es)

Families Citing this family (273)

* Cited by examiner, † Cited by third party
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ZA86203B (en) 1987-09-30
KR860005811A (ko) 1986-08-13
FI81098C (fi) 1990-09-10
KR920010046B1 (ko) 1992-11-13
MX9202933A (es) 1992-06-30
AR240698A1 (es) 1990-09-28
SG105691G (en) 1992-02-14
US4687777A (en) 1987-08-18
NO163857C (no) 1990-08-01
IE58928B1 (en) 1993-12-01
EP0193256B1 (en) 1989-04-05
CN86100411A (zh) 1986-07-16
DE10199018I2 (de) 2006-02-02
ATE41931T1 (de) 1989-04-15
NO860141L (no) 1986-07-21
HUT41775A (en) 1987-05-28
DK21986D0 (da) 1986-01-17
DE3662689D1 (en) 1989-05-11
JPH0566956B2 (es) 1993-09-22
CN1003934B (zh) 1989-04-19
ES550986A0 (es) 1987-05-16
NO163857B (no) 1990-04-23
IE860107L (en) 1986-07-19
LU90719I2 (fr) 2001-03-26
CA1277323C (en) 1990-12-04
BR1100325A (pt) 2000-06-27
NL300038I2 (nl) 2001-05-01
GR860124B (en) 1986-05-19
DK171614B1 (da) 1997-02-24
AU572719B2 (en) 1988-05-12
FI860232A (fi) 1986-07-20
CS407991A3 (en) 1992-04-15
DE10199018I1 (de) 2001-07-12
PT81859A (en) 1986-02-01
DK21986A (da) 1986-07-20
PT81859B (pt) 1988-05-27
HK3692A (en) 1992-01-17
FI860232A0 (fi) 1986-01-17
JPS61267580A (ja) 1986-11-27
HU196795B (en) 1989-01-30
LV5779B4 (lv) 1997-04-20
EP0193256A1 (en) 1986-09-03
MY102016A (en) 1992-02-29
FI81098B (fi) 1990-05-31
AU5246786A (en) 1986-07-24
LV5779A4 (lv) 1996-12-20

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