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EA200200208A1 - Синергитическая композиция - Google Patents

Синергитическая композиция

Info

Publication number
EA200200208A1
EA200200208A1 EA200200208A EA200200208A EA200200208A1 EA 200200208 A1 EA200200208 A1 EA 200200208A1 EA 200200208 A EA200200208 A EA 200200208A EA 200200208 A EA200200208 A EA 200200208A EA 200200208 A1 EA200200208 A1 EA 200200208A1
Authority
EA
Eurasian Patent Office
Prior art keywords
synergy composition
synergy
composition
published
treatment
Prior art date
Application number
EA200200208A
Other languages
English (en)
Other versions
EA006685B1 (ru
Inventor
Рольф Бойме
Даниела Бундшух
Армин Хатцельманн
Кристиан Шудт
Кристиан Ваймар
Ульрих Килиан
Original Assignee
Бык Гульден Ломберг Хемише Фабрик Гмбх
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Бык Гульден Ломберг Хемише Фабрик Гмбх filed Critical Бык Гульден Ломберг Хемише Фабрик Гмбх
Publication of EA200200208A1 publication Critical patent/EA200200208A1/ru
Publication of EA006685B1 publication Critical patent/EA006685B1/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pulmonology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Seasonings (AREA)
  • Inorganic Insulating Materials (AREA)
  • Medicinal Preparation (AREA)
  • Dental Preparations (AREA)
  • Piezo-Electric Or Mechanical Vibrators, Or Delay Or Filter Circuits (AREA)
  • Lubricants (AREA)

Abstract

В заявке описано совместное применение ингибиторов PDE и агонистов β-адренорецептора для лечения заболеваний дыхательных путей.Отчет о международном поиске был опубликован 2001.09.20.
EA200200208A 1999-08-21 2000-08-11 Синергетическая композиция EA006685B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP99116447 1999-08-21
PCT/EP2000/007852 WO2001013953A2 (en) 1999-08-21 2000-08-11 Synergistic combination of pde inhibitors and beta 2 adrenoceptor agonist

Publications (2)

Publication Number Publication Date
EA200200208A1 true EA200200208A1 (ru) 2002-08-29
EA006685B1 EA006685B1 (ru) 2006-02-24

Family

ID=8238828

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200200208A EA006685B1 (ru) 1999-08-21 2000-08-11 Синергетическая композиция

Country Status (28)

Country Link
US (3) US7056936B2 (ru)
EP (3) EP1212089B1 (ru)
JP (1) JP5038568B2 (ru)
KR (1) KR100701904B1 (ru)
CN (1) CN1202865C (ru)
AT (2) ATE320800T1 (ru)
AU (1) AU777012B2 (ru)
BR (1) BRPI0013478B8 (ru)
CA (2) CA2381802C (ru)
CZ (1) CZ302882B6 (ru)
DE (2) DE60043318D1 (ru)
DK (1) DK1212089T3 (ru)
EA (1) EA006685B1 (ru)
ES (1) ES2260043T3 (ru)
HK (1) HK1047244B (ru)
HR (1) HRP20020158B1 (ru)
HU (1) HU229439B1 (ru)
IL (2) IL147688A0 (ru)
MX (1) MXPA02001830A (ru)
NO (1) NO328340B1 (ru)
NZ (1) NZ517166A (ru)
PL (1) PL200923B1 (ru)
PT (1) PT1212089E (ru)
SI (1) SI1212089T1 (ru)
SK (1) SK287231B6 (ru)
TR (2) TR200201317T2 (ru)
WO (1) WO2001013953A2 (ru)
ZA (1) ZA200201389B (ru)

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CA2381802C (en) 2010-12-07
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BRPI0013478B1 (pt) 2016-12-06
EP1671651A1 (en) 2006-06-21
HRP20020158B1 (en) 2007-08-31
US20040034087A1 (en) 2004-02-19
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ZA200201389B (en) 2002-08-21
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MXPA02001830A (es) 2002-08-12
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BRPI0013478B8 (pt) 2016-12-27
JP2003507435A (ja) 2003-02-25
KR100701904B1 (ko) 2007-04-02
ATE320800T1 (de) 2006-04-15
NO20020815L (no) 2002-02-19
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HUP0203098A2 (hu) 2003-01-28
DE60043318D1 (de) 2010-01-14
US7056936B2 (en) 2006-06-06
EP1212089A2 (en) 2002-06-12
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ATE447952T1 (de) 2009-11-15
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