EA004403B1 - Производные пиразолотриазинов, фармацевтические композиции, содержащие их, способы лечения - Google Patents

Производные пиразолотриазинов, фармацевтические композиции, содержащие их, способы лечения Download PDF

Info

Publication number: EA004403B1
Authority: EA; Eurasian Patent Office
Prior art keywords: denotes; compound; formula; stands; ome
Prior art date: 1996-07-24

Application number

EA199900158A

Other languages

English (en)

Russian (ru)

Other versions

EA199900158A1 (ru

Inventor

Арджириос Георгиос Арванитис

Роберт Джон Хорват

Original Assignee

Дюпон Фармасьютикалз Компани

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-07-24

Filing date

1997-07-23

Publication date

2004-04-29

1997-07-23 Application filed by Дюпон Фармасьютикалз Компани filed Critical Дюпон Фармасьютикалз Компани

1997-07-23 Priority claimed from PCT/US1997/013072 external-priority patent/WO1998003510A1/en

1997-07-23 Priority claimed from US08/899,242 external-priority patent/US6124289A/en

1999-10-28 Publication of EA199900158A1 publication Critical patent/EA199900158A1/ru

2004-04-29 Publication of EA004403B1 publication Critical patent/EA004403B1/ru

Landscapes

Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)
Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Detergent Compositions (AREA)
Coloring (AREA)

EA199900158A 1996-07-24 1997-07-23 Производные пиразолотриазинов, фармацевтические композиции, содержащие их, способы лечения EA004403B1 (ru)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US2329096P	1996-07-24	1996-07-24
US68604796A	1996-07-24	1996-07-24
PCT/US1997/013072 WO1998003510A1 (en)	1996-07-24	1997-07-23	AZOLO TRIAZINES AND PYRIMIDINES
US08/899,242 US6124289A (en)	1996-07-24	1997-07-23	Azolo triazines and pyrimidines

Publications (2)

Publication Number	Publication Date
EA199900158A1 EA199900158A1 (ru)	1999-10-28
EA004403B1 true EA004403B1 (ru)	2004-04-29

Family

ID=27362048

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EA199900158A EA004403B1 (ru)	1996-07-24	1997-07-23	Производные пиразолотриазинов, фармацевтические композиции, содержащие их, способы лечения

Country Status (15)

Country	Link
JP (2)	JP4704521B2 (no)
CN (3)	CN1104432C (no)
AR (1)	AR049583A2 (no)
BR (1)	BR9710544A (no)
CA (1)	CA2259583C (no)
CZ (1)	CZ299451B6 (no)
EA (1)	EA004403B1 (no)
EE (1)	EE04316B1 (no)
HR (1)	HRP970413A2 (no)
IL (4)	IL127871A0 (no)
NO (1)	NO315610B1 (no)
NZ (1)	NZ333777A (no)
PL (1)	PL195762B1 (no)
SI (1)	SI9720045B (no)
SK (1)	SK286461B6 (no)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SK287603B6 (sk) *	2001-03-13	2011-03-04	Bristol-Myers Squibb Pharma Company	4-(2-Butylamino)-2,7-dimetyl-8-(2-metyl-6-metoxypyrid-3- yl)pyrazol-[1,5-a]-1,3,5-triazín, farmaceutická kompozícia obsahujúca túto zlúčeninu, použitie tejto zlúčeniny v terapii a na prípravu farmaceutickej kompozície a výrobok obsahujúci túto zlúčeninu
WO2004110454A1 (ja) *	2003-06-13	2004-12-23	Ishihara Sangyo Kaisha, Ltd.	アデノシンＡ2ａ受容体アゴニストの投与が必要な疾患を治療又は予防するための組成物
US7329662B2 (en) *	2003-10-03	2008-02-12	Hoffmann-La Roche Inc.	Pyrazolo-pyridine
GB0519957D0 (en) *	2005-09-30	2005-11-09	Sb Pharmco Inc	Chemical compound
MY146388A (en) *	2006-09-20	2012-08-15	Lilly Co Eli	Thiazole pyrazolopyrimidines as crfi receptor antagonists
CN103694242B (zh) *	2013-12-10	2016-01-06	昆明翔昊科技有限公司	吡唑并嘧啶类化合物及其药物组合物和其在制药中的应用
CN110996943A (zh)	2017-08-14	2020-04-10	云杉生物科学公司	促肾上腺皮质激素释放因子受体拮抗剂
CN112574214B (zh) *	2019-07-30	2021-09-28	杭州阿诺生物医药科技有限公司	腺苷受体拮抗剂的制备方法
WO2022036123A1 (en)	2020-08-12	2022-02-17	Spruce Biosciences, Inc.	Methods and compositions for treating polycystic ovary syndrome
US11708372B2 (en)	2021-11-19	2023-07-25	Spruce Biosciences, Inc.	Crystalline composition of tildacerfont and methods of use and preparation thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3995039A (en) *	1975-05-27	1976-11-30	Merck & Co., Inc.	Pyrazolo [1,5-a] [1,3,5] triazines
JPS6157587A (ja) *	1984-08-29	1986-03-24	Shionogi & Co Ltd	縮合複素環誘導体および抗潰瘍剤
US4824834A (en) *	1986-10-31	1989-04-25	Otsuka Pharmaceutical Company, Limited	Pyrazolotriazine compounds
JP2691317B2 (ja) *	1989-08-25	1997-12-17	株式会社大塚製薬工場	４―ヒドロキシ―８―（３―低級アルコキシ―４―フェニルスルフィニルフェニル）ピラゾロ〔１，５―ａ〕―１，３，５―トリアジン光学活性体の塩類及びその製造方法
KR927003595A (ko) *	1990-10-09	1992-12-18	오츠카 아키히코	피리미딘 유도체, 이의 제조방법 및 안드로겐 저해제
DK0591528T3 (da) *	1991-04-22	1999-08-23	Otsuka Pharma Co Ltd	Pyrazolo[1,5-a]pyrimidinderivat og antiinflammatorisk middel, der indeholder dette
US5356897A (en) *	1991-09-09	1994-10-18	Fujisawa Pharmaceutical Co., Ltd.	3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines

1997
- 1997-07-23 BR BR9710544A patent/BR9710544A/pt not_active IP Right Cessation
- 1997-07-23 JP JP50723398A patent/JP4704521B2/ja not_active Expired - Fee Related
- 1997-07-23 EA EA199900158A patent/EA004403B1/ru not_active IP Right Cessation
- 1997-07-23 CA CA002259583A patent/CA2259583C/en not_active Expired - Lifetime
- 1997-07-23 SI SI9720045A patent/SI9720045B/sl active Search and Examination
- 1997-07-23 CN CN97196525A patent/CN1104432C/zh not_active Expired - Lifetime
- 1997-07-23 EE EEP199900019A patent/EE04316B1/xx unknown
- 1997-07-23 SK SK97-99A patent/SK286461B6/sk not_active IP Right Cessation
- 1997-07-23 CZ CZ0018499A patent/CZ299451B6/cs not_active IP Right Cessation
- 1997-07-23 NZ NZ333777A patent/NZ333777A/en not_active IP Right Cessation
- 1997-07-23 PL PL97331523A patent/PL195762B1/pl unknown
- 1997-07-23 IL IL12787197A patent/IL127871A0/xx unknown
- 1997-07-24 HR HRP970413 patent/HRP970413A2/hr not_active Application Discontinuation
1998
- 1998-12-30 IL IL127871A patent/IL127871A/en not_active IP Right Cessation
1999
- 1999-01-21 NO NO19990264A patent/NO315610B1/no not_active IP Right Cessation
2001
- 2001-05-30 CN CN 01120849 patent/CN1250223C/zh not_active Expired - Lifetime
2002
- 2002-04-25 CN CN 02118589 patent/CN1388126A/zh active Pending
- 2002-06-11 IL IL150163A patent/IL150163A/en not_active IP Right Cessation
2004
- 2004-07-23 JP JP2004216483A patent/JP4194539B2/ja not_active Expired - Fee Related
- 2004-10-12 IL IL164513A patent/IL164513A/en not_active IP Right Cessation
2005
- 2005-07-11 AR ARP050102868A patent/AR049583A2/es not_active Application Discontinuation

Also Published As

Publication number	Publication date
NO990264D0 (no)	1999-01-21
CZ299451B6 (cs)	2008-07-30
SK9799A3 (sk)	2005-04-01
PL331523A1 (en)	1999-07-19
NZ333777A (en)	2000-07-28
SI9720045B (sl)	2008-02-29
CN1388126A (zh)	2003-01-01
CZ18499A3 (cs)	1999-11-17
IL164513A (en)	2010-04-29
CN1104432C (zh)	2003-04-02
IL150163A (en)	2010-12-30
SI9720045A (sl)	1999-10-31
CN1250223C (zh)	2006-04-12
CA2259583C (en)	2009-11-17
AR049583A2 (es)	2006-08-16
EE04316B1 (et)	2004-06-15
BR9710544A (pt)	1999-08-17
IL164513A0 (en)	2005-12-18
HRP970413A2 (en)	1998-10-31
PL195762B1 (pl)	2007-10-31
JP2005097257A (ja)	2005-04-14
NO315610B3 (no)	2003-09-29
CN1225637A (zh)	1999-08-11
NO315610B1 (no)	2003-09-29
EE9900019A (et)	1999-08-16
JP4704521B2 (ja)	2011-06-15
CN1327793A (zh)	2001-12-26
NO990264L (no)	1999-03-10
JP4194539B2 (ja)	2008-12-10
IL127871A0 (en)	1999-10-28
EA199900158A1 (ru)	1999-10-28
JP2002513382A (ja)	2002-05-08
IL127871A (en)	2010-04-29
CA2259583A1 (en)	1998-01-29
SK286461B6 (sk)	2008-10-07

Publication	Publication Date	Title
US6060478A (en)	2000-05-09	Azolo triazines and pyrimidines
US6358950B1 (en)	2002-03-19	Azolo triazines and pyrimidines
EP0915880B1 (en)	2007-10-10	Azolo triazines and pyrimidines
US6136809A (en)	2000-10-24	Azolo triazines and pyrimidines
AU748818B2 (en)	2002-06-13	Azolo triazines and pyrimidines
US6313124B1 (en)	2001-11-06	Tetrazine bicyclic compounds
BRPI0619146A2 (pt)	2011-09-13	derivados de 4-amino-pirroltriazina substituìda úteis no tratamento de disordens e doenças hiperproliferativas associadas com angiogênesis
KR102588426B1 (ko)	2023-10-13	치환 디히드로피롤로피라졸 유도체
EA004403B1 (ru)	2004-04-29	Производные пиразолотриазинов, фармацевтические композиции, содержащие их, способы лечения
US7678793B2 (en)	2010-03-16	Azolo triazines and pyrimidines
US20030008885A1 (en)	2003-01-09	Azolo triazines and pyrimidines
AU773039B2 (en)	2004-05-13	Azolo triazines and pyrimidines
AU2002300983B2 (en)	2005-06-09	Azolo Triazines And Pyrimidines
CA2532925C (en)	2009-10-20	Azolo triazines and pyrimidines
JP2002532491A (ja)	2002-10-02	イミダゾロン類、並びに良性前立腺肥大症および他の疾患の治療におけるその使用

Legal Events

Date	Code	Title	Description
2017-08-31	MK4A	Patent expired	Designated state(s): AM AZ BY KZ KG MD TJ TM RU