ZA987114B - 3-substituted 3,4,5,7-tetrahydropyrrolol[3',4':4,5] thieno[2,3-D]pyrimidine derivatives, their preparation and use. - Google Patents

3-substituted 3,4,5,7-tetrahydropyrrolol[3',4':4,5] thieno[2,3-D]pyrimidine derivatives, their preparation and use.

Info

Publication number: ZA987114B
Authority: ZA; South Africa
Prior art keywords: tetrahydropyrrolol; thieno; substituted; preparation; pyrimidine derivatives
Prior art date: 1997-08-08

Application number

ZA9807114A

Other languages

English (en)

Inventor

Gerd Steiner

Uta Dullweber

Dorothea Starck

Alfred Bach

Karsten Wicke

Hans-Juergen Teschendorf

Francisco-Javier Garcia-Ladona

Franz Emling

Original Assignee

Basf Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-08-08

Filing date

1998-08-07

Publication date

2000-02-07

1998-08-07 Application filed by Basf Ag filed Critical Basf Ag

2000-02-07 Publication of ZA987114B publication Critical patent/ZA987114B/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Neurology (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pain & Pain Management (AREA)
Psychiatry (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

ZA9807114A 1997-08-08 1998-08-07 3-substituted 3,4,5,7-tetrahydropyrrolol[3',4':4,5] thieno[2,3-D]pyrimidine derivatives, their preparation and use. ZA987114B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE19734444A DE19734444A1 (de)	1997-08-08	1997-08-08	3-Substituierte 3,4,5,7-Tetrahydro-pyrrolo(3',4':4,5) thieno (2,3-d) pyrimidin-Derivate, ihre Herstellung und Verwendung

Publications (1)

Publication Number	Publication Date
ZA987114B true ZA987114B (en)	2000-02-07

Family

ID=7838438

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA9807114A ZA987114B (en)	1997-08-08	1998-08-07	3-substituted 3,4,5,7-tetrahydropyrrolol[3',4':4,5] thieno[2,3-D]pyrimidine derivatives, their preparation and use.

Country Status (25)

Country	Link
US (1)	US6355647B1 (xx)
EP (1)	EP1003752A1 (xx)
JP (1)	JP2001512734A (xx)
KR (1)	KR20010022658A (xx)
CN (1)	CN1267303A (xx)
AR (1)	AR016594A1 (xx)
AU (1)	AU749539B2 (xx)
BG (1)	BG104151A (xx)
BR (1)	BR9811091A (xx)
CA (1)	CA2300391A1 (xx)
CO (1)	CO4960665A1 (xx)
CZ (1)	CZ290678B6 (xx)
DE (1)	DE19734444A1 (xx)
HR (1)	HRP980435A2 (xx)
HU (1)	HUP0101311A3 (xx)
ID (1)	ID24222A (xx)
IL (1)	IL134161A0 (xx)
NO (1)	NO20000605L (xx)
NZ (1)	NZ502657A (xx)
PL (1)	PL340726A1 (xx)
SK (1)	SK1052000A3 (xx)
TR (1)	TR200000371T2 (xx)
TW (1)	TW513435B (xx)
WO (1)	WO1999007711A1 (xx)
ZA (1)	ZA987114B (xx)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US20040048874A1 (en) *	2001-05-22	2004-03-11	Bardsley Hazel Judith	New therapeutic use of 4-(2-fluorophenyl)-6-methyl-2-(1-piperazinyl)thieno[2,3-D]pyrimidine
GB0216027D0 (en) *	2002-07-10	2002-08-21	Arachnova Therapeutics Ltd	New therapeutic use
DE10259382A1 (de) *	2002-12-18	2004-07-01	Abbott Gmbh & Co. Kg	3-Substituierte 3,4-Dihydro-thieno[2,3-d]pyrimidin-4-on-Derivate, ihre Herstellung und Verwendung
WO2004062624A2 (en) *	2003-01-13	2004-07-29	Dynogen Pharmaceuticals, Inc.	Method of treating nausea, vomiting, retching or any combination thereof
NZ541008A (en) *	2003-01-13	2007-09-28	Dynogen Pharmaceuticals Inc	Method of treating functional bowel disorders
EP1539181B1 (en) *	2003-04-04	2007-06-27	Dynogen Pharmaceuticals Inc.	Method of treating lower urinary tract disorders
US20050165025A1 (en) *	2004-01-22	2005-07-28	Recordati Ireland Ltd.	Combination therapy with 5HT 1A and 5HT 1B-receptor antagonists
US7375814B2 (en) *	2005-03-11	2008-05-20	Sandia Corporation	Natural gas leak mapper
US20060293309A1 (en) *	2005-03-28	2006-12-28	Dynogen Pharmaceuticals, Inc.	Method of treating disorders and conditions using peripherally-restricted antagonists and inhibitors
WO2020183011A1 (en)	2019-03-14	2020-09-17	Institut Curie	Htr1d inhibitors and uses thereof in the treatment of cancer

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5001130A (en) *	1988-02-18	1991-03-19	Bristol-Myers Company	Psychotropic heterobicycloalkylpiperazine derivatives
US4835157A (en)	1988-03-15	1989-05-30	Ortho Pharmaceutical Corporation	Thieno- and furopyrimidine-2,4-dione piperidine derivatives as serotonin antagonists and alpha adrenergic blocking agents
DE19636769A1 (de)	1996-09-10	1998-03-12	Basf Ag	3-Substituierte Pyrido [4',3':4,5]thieno[2,3-d]pyrimidin-Derivate, ihre Herstellung und Verwendung

1997
- 1997-08-08 DE DE19734444A patent/DE19734444A1/de not_active Withdrawn
1998
- 1998-07-23 US US09/485,188 patent/US6355647B1/en not_active Expired - Lifetime
- 1998-07-23 AU AU90683/98A patent/AU749539B2/en not_active Ceased
- 1998-07-23 NZ NZ502657A patent/NZ502657A/en unknown
- 1998-07-23 KR KR1020007001252A patent/KR20010022658A/ko not_active Application Discontinuation
- 1998-07-23 CN CN98808009A patent/CN1267303A/zh active Pending
- 1998-07-23 JP JP2000506214A patent/JP2001512734A/ja active Pending
- 1998-07-23 PL PL98340726A patent/PL340726A1/xx not_active Application Discontinuation
- 1998-07-23 IL IL13416198A patent/IL134161A0/xx unknown
- 1998-07-23 SK SK105-2000A patent/SK1052000A3/sk unknown
- 1998-07-23 HU HU0101311A patent/HUP0101311A3/hu unknown
- 1998-07-23 TR TR2000/00371T patent/TR200000371T2/xx unknown
- 1998-07-23 CZ CZ2000462A patent/CZ290678B6/cs not_active IP Right Cessation
- 1998-07-23 ID IDW20000239A patent/ID24222A/id unknown
- 1998-07-23 WO PCT/EP1998/004633 patent/WO1999007711A1/de not_active Application Discontinuation
- 1998-07-23 BR BR9811091-8A patent/BR9811091A/pt not_active IP Right Cessation
- 1998-07-23 CA CA002300391A patent/CA2300391A1/en not_active Abandoned
- 1998-07-23 EP EP98942610A patent/EP1003752A1/de not_active Withdrawn
- 1998-08-06 HR HR19734444.5A patent/HRP980435A2/hr not_active Application Discontinuation
- 1998-08-07 AR ARP980103914A patent/AR016594A1/es not_active Application Discontinuation
- 1998-08-07 TW TW087113048A patent/TW513435B/zh active
- 1998-08-07 ZA ZA9807114A patent/ZA987114B/xx unknown
- 1998-08-10 CO CO98045546A patent/CO4960665A1/es unknown
2000
- 2000-02-07 NO NO20000605A patent/NO20000605L/no not_active Application Discontinuation
- 2000-02-10 BG BG104151A patent/BG104151A/bg unknown

Also Published As

Publication number	Publication date
NO20000605D0 (no)	2000-02-07
BR9811091A (pt)	2000-09-12
NZ502657A (en)	2001-06-29
BG104151A (bg)	2000-10-31
NO20000605L (no)	2000-02-07
WO1999007711A1 (de)	1999-02-18
CZ290678B6 (cs)	2002-09-11
AU9068398A (en)	1999-03-01
ID24222A (id)	2000-07-13
CZ2000462A3 (cs)	2000-05-17
HUP0101311A1 (hu)	2001-09-28
TR200000371T2 (tr)	2000-11-21
PL340726A1 (en)	2001-02-26
JP2001512734A (ja)	2001-08-28
EP1003752A1 (de)	2000-05-31
HRP980435A2 (en)	1999-04-30
SK1052000A3 (en)	2000-08-14
AU749539B2 (en)	2002-06-27
CN1267303A (zh)	2000-09-20
DE19734444A1 (de)	1999-02-11
AR016594A1 (es)	2001-07-25
KR20010022658A (ko)	2001-03-26
TW513435B (en)	2002-12-11
IL134161A0 (en)	2001-04-30
US6355647B1 (en)	2002-03-12
CO4960665A1 (es)	2000-09-25
CA2300391A1 (en)	1999-02-18
HUP0101311A3 (en)	2002-10-28

Publication	Publication Date	Title
AP2002002456A0 (en)	2002-06-30	Pyrazolo '4,3-d pyrimidine derivatives
ZA985121B (en)	1999-12-13	3-Substituted 3,4-dihyrothieno(2,3-d)pyrimidine derivatives their preparation and use.
HUP0103472A3 (en)	2002-12-28	Pyrrolo[2,3-d]pyrimidine derivatives and pharmaceutical compositions containing the same
ZA986250B (en)	1999-01-22	5H-thiazolo[3,2-A]pyrimidine derivatives
HUP0103836A3 (en)	2003-05-28	Pyrrolo[2,3d]pyrimidine compositions and their use
HUP0001993A3 (en)	2002-02-28	Fungicidal trifluoromethylalkylamino-triazolo [1,5a] pyrimidine derivatives, preparation and use thereof
IL128142A0 (en)	1999-11-30	3-Substituted pyrido [4',3':4,5] thieno [2,3-d] pyrimidine derivatives their preparation and their use
HUP9900607A3 (en)	1999-11-29	Pyrido[2,3-d]pyrimidine derivatives and medicinal compositions thereof
PL353366A1 (en)	2003-11-17	Pyrazolo[4,3-d]pyrimidines
ZA987114B (en)	2000-02-07	3-substituted 3,4,5,7-tetrahydropyrrolol[3',4':4,5] thieno[2,3-D]pyrimidine derivatives, their preparation and use.
ZA989664B (en)	2000-04-25	3-substituted tetrahydropyrimidinone derivatives, their preparation and use.
ZA985120B (en)	1999-12-13	3-Substituted pyrido[3',4':4,5]thieno[2,3-d]pyrimidine derivatives, their preparation and use.
ZA9811642B (en)	1999-06-24	Pyrido 1,2,4-thiadiazine derivatives their preparation and use
AU3147500A (en)	2000-10-04	Fused 1,4-thiazine-2-carbonitrile derivatives, their preparation and use
ZA200202763B (en)	2003-06-25	Pyrazolo [4,3-D] pyrimidine derivatives.