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TR200800474T2 - Florfenikole aracı maddelerin hazırlanmasına ilişkin işlem. - Google Patents

Florfenikole aracı maddelerin hazırlanmasına ilişkin işlem.

Info

Publication number
TR200800474T2
TR200800474T2 TR2008/00474T TR200800474T TR200800474T2 TR 200800474 T2 TR200800474 T2 TR 200800474T2 TR 2008/00474 T TR2008/00474 T TR 2008/00474T TR 200800474 T TR200800474 T TR 200800474T TR 200800474 T2 TR200800474 T2 TR 200800474T2
Authority
TR
Turkey
Prior art keywords
preparation
intermediates
fluorfenicol
formula
florphenicol
Prior art date
Application number
TR2008/00474T
Other languages
English (en)
Inventor
B. Vashi Dhiru
C. Towson James
Original Assignee
Schering Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=24808601&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TR200800474(T2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Corporation filed Critical Schering Corporation
Publication of TR200800474T2 publication Critical patent/TR200800474T2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/28—Nitrogen atoms not forming part of a nitro radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

R ve R"' in burada belirtildiği şekilde olduğu formül (I)'in bileşiğinin hazırlanmasına yönelik bir işlem. Formül (I)' in bileşikleri, florfenikolün hazırlanmasında aracı maddeler olarak yararlıdır.
TR2008/00474T 1996-08-19 1997-08-18 Florfenikole aracı maddelerin hazırlanmasına ilişkin işlem. TR200800474T2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US08/699,271 US5663361A (en) 1996-08-19 1996-08-19 Process for preparing intermediates to florfenicol

Publications (1)

Publication Number Publication Date
TR200800474T2 true TR200800474T2 (tr) 2008-04-21

Family

ID=24808601

Family Applications (2)

Application Number Title Priority Date Filing Date
TR2008/00474T TR200800474T2 (tr) 1996-08-19 1997-08-18 Florfenikole aracı maddelerin hazırlanmasına ilişkin işlem.
TR1999/00354T TR199900354T2 (tr) 1996-08-19 1997-08-18 Florfenikole araci maddelerin hazirlanmasina iliskin islem.

Family Applications After (1)

Application Number Title Priority Date Filing Date
TR1999/00354T TR199900354T2 (tr) 1996-08-19 1997-08-18 Florfenikole araci maddelerin hazirlanmasina iliskin islem.

Country Status (31)

Country Link
US (1) US5663361A (tr)
EP (1) EP0922040B2 (tr)
JP (1) JP3274868B2 (tr)
KR (1) KR100286851B1 (tr)
CN (1) CN1097583C (tr)
AR (1) AR008298A1 (tr)
AT (1) ATE283847T1 (tr)
AU (1) AU714495B2 (tr)
BR (1) BR9711318B1 (tr)
CA (1) CA2264116C (tr)
CO (1) CO4560550A1 (tr)
CZ (1) CZ297915B6 (tr)
DE (1) DE69731835T3 (tr)
DK (1) DK0922040T3 (tr)
ES (1) ES2234026T5 (tr)
HK (1) HK1017890A1 (tr)
HU (1) HU229610B1 (tr)
ID (1) ID18047A (tr)
IL (1) IL128574A (tr)
MY (1) MY115679A (tr)
NO (1) NO312962B1 (tr)
NZ (1) NZ334111A (tr)
PE (1) PE99798A1 (tr)
PL (2) PL196454B1 (tr)
PT (1) PT922040E (tr)
SI (1) SI0922040T1 (tr)
SK (1) SK286124B6 (tr)
TR (2) TR200800474T2 (tr)
TW (1) TW381075B (tr)
WO (1) WO1998007709A1 (tr)
ZA (1) ZA977406B (tr)

Families Citing this family (40)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1173933C (zh) * 2001-06-01 2004-11-03 中国科学院上海有机化学研究所 一种从l型取代苯丝氨酸酯制备d－（－）－苏式1－r－取代苯基－2－二氯乙酰氨基－3－氟－1－丙醇的方法
KR20040091698A (ko) * 2002-03-08 2004-10-28 쉐링-플라우 리미티드. 신규한 플로르페니콜형 항생제
MY146351A (en) * 2003-05-29 2012-08-15 Schering Plough Ltd Compositions for treating infection in cattle and swine
US7439268B2 (en) 2003-07-18 2008-10-21 Idexx Laboratories Compositions containing prodrugs of florfenicol and methods of use
US20050049210A1 (en) * 2003-08-27 2005-03-03 Idexx Laboratories, Inc. Methods for the controlled delivery of pharmacologically active compounds
US7126005B2 (en) * 2003-10-06 2006-10-24 Aurobindo Pharma Limited Process for preparing florfenicol
CA2576589C (en) 2004-08-13 2013-11-12 Schering-Plough Ltd. Pharmaceutical formulation comprising an antibiotic, a triazole and a corticosteroid
KR20070054691A (ko) 2004-09-23 2007-05-29 쉐링-프라우 리미티드 신규한 트리플루오로메탄설폰아미드 옥심 에테르 유도체를사용하여 동물의 기생충 방제
DE602005017419D1 (de) * 2004-11-19 2009-12-10 Schering Plough Ltd Kontrolle von parasiten bei tieren mittels verwendung von parasitiziden 2-phenyl-3-(1h-pyrrol-2-yl) acrylonitril-derivaten
US8680154B2 (en) * 2004-12-21 2014-03-25 Intervet International B.V. Injectable veterinary composition
JP2008545788A (ja) * 2005-06-09 2008-12-18 シェーリング−プラウ・リミテッド Ｎ−［（フェニルオキシ）フェニル］−１，１，１−トリフルオロメタンスルホンアミドおよびｎ−［（フェニルスルファニル）フェニル）］−１，１，１−トリフルオロメタンスルホンアミド誘導体による動物中の寄生生物の制御
MX2008003188A (es) * 2005-09-07 2008-03-18 Schering Plough Ltd Procedimiento para la preparacion de compuestos ester oxazolidina y su conversion a florfenicol.
US8119667B2 (en) * 2005-12-29 2012-02-21 Schering-Plough Animal Health Corporation Carbonates of fenicol antibiotics
US7518017B2 (en) 2006-02-17 2009-04-14 Idexx Laboratories Fenicol compounds and methods synthesizing 2-trifluoroacetamido-3-substituted propiophenone compounds
US20070238700A1 (en) * 2006-04-10 2007-10-11 Winzenberg Kevin N N-phenyl-1,1,1-trifluoromethanesulfonamide hydrazone derivative compounds and their usage in controlling parasites
EP2091909A1 (en) * 2006-12-13 2009-08-26 Schering-Plough Ltd. Water-soluble prodrugs of florfenicol and its analogs
EP2102154A1 (en) * 2006-12-13 2009-09-23 Schering-Plough Ltd. Water-soluble prodrugs of chloramphenicol, thiamphenicol, and analogs thereof
AR066265A1 (es) * 2007-04-27 2009-08-05 Schering Plough Ltd Compuestos y metodos para mejorar la solubilidad de florfenicol y antibioticos estructuralmente relacionados por medio del uso de ciclodextrinas. composicion. complejo. kit. metodo de tratamiento.
WO2008150406A1 (en) * 2007-05-30 2008-12-11 Schering-Plough Ltd. A process for preparing oxazoline-protected aminodiol compounds useful as intermediates to florfenicol
TWI430995B (zh) 2007-06-26 2014-03-21 Du Pont 萘異唑啉無脊椎有害動物控制劑
MX361762B (es) 2007-06-27 2018-12-17 Du Pont Metodo de control de plagas en animales.
RU2010106607A (ru) * 2007-07-25 2011-08-27 Интервет Интернэшнл Б.В. (Nl) Способ получения оксазолидин- и оксазолидинонаминодиолов
US7550625B2 (en) * 2007-10-19 2009-06-23 Idexx Laboratories Esters of florfenicol
AU2008324852A1 (en) * 2007-11-09 2009-05-14 Intervet International B.V. Fast release solid formulation, preparation and use thereof
TWI468407B (zh) 2008-02-06 2015-01-11 Du Pont 中離子農藥
JP2011529895A (ja) * 2008-07-30 2011-12-15 インターベツト・インターナシヨナル・ベー・ベー フロルフェニコール中間体として有用なオキサゾリン保護アミノジオール化合物を調製する方法
WO2011017347A2 (en) 2009-08-05 2011-02-10 E. I. Du Pont De Nemours And Company Mesoionic pesticides
UA107804C2 (en) 2009-08-05 2015-02-25 Du Pont Mixtures of pesticides mezoionnyh
JP2013501059A (ja) 2009-08-05 2013-01-10 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー メソイオン性殺虫剤
UA110924C2 (uk) 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Мезоіонні пестициди
BRPI1002023A2 (pt) 2010-03-01 2011-10-25 Nanocore Biotecnologia S A forma farmacêutica sólida de dissolução rápida para tratamento de infecções bacterianas
US8598087B2 (en) 2010-05-27 2013-12-03 E. I. Du Pont De Nemours And Company Crystalline form of 4-[5-[3-chloro-5-(trifluoromethyl)phenyl]-4, 5-dihydro-5-(trifluoromethyl)-3-isoxazolyl]-N-[2-0X0-2-[(2,2,2-trifluoroethyl)amino]ethyl]-1- naph-thalenecarboxamide
WO2012087630A1 (en) 2010-12-20 2012-06-28 E.I. Du Pont De Nemours And Company Pyridine and pyrimidine compounds for controlling invertebrate
WO2013158422A1 (en) 2012-04-17 2013-10-24 E. I. Du Pont De Nemours And Company Heterocyclic compounds for controlling invertebrate pests
CN102911133B (zh) * 2012-10-31 2014-07-02 绍兴民生医药有限公司 (4r,5r)-2-二氯甲基-4,5-二氢-5-(4-甲砜基苯基)-4-恶唑甲醇的纯化方法
CN103254147B (zh) * 2013-04-19 2016-04-06 浙江科技学院 一种d-苏式-2-(二氯甲基)-4,5-二氢-5-[对-（甲砜基）苯基]-4-噁唑甲醇的制备方法
CN106278964B (zh) * 2016-07-31 2018-01-16 浙江润康药业有限公司 氟苯尼考的制备方法
CN106631872A (zh) * 2016-12-13 2017-05-10 浙江普洛家园药业有限公司 一种氟苯尼考类似物中间体的合成方法
CN110272856B (zh) * 2019-05-08 2022-05-03 江南大学 一种表达d-苏氨酸醛缩酶的重组菌及其构建方法与应用
CN117466787B (zh) * 2023-12-28 2024-03-22 山东国邦药业有限公司 一种氟苯尼考中间体的制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2759001A (en) * 1952-03-01 1956-08-14 Parke Davis & Co Process for the production of delta2-oxazolines
US4361557A (en) * 1980-01-28 1982-11-30 Schering Corporation 1-Aryl-2-acylamido-3-fluoro-1-propanol acylates, methods for their use as anti-bacterial agents and compositions useful therefor
EP0677511A3 (en) * 1983-06-02 1996-07-24 Zambon Spa Intermediates for the production of 1-phenyl-1-hydroxy-2-amino-3-fluoropropane derivatives.
US4876352A (en) * 1988-09-14 1989-10-24 Schering Corporation Pressurized fluorination of hydroxy alkyl groups
EP0405104A1 (en) † 1989-05-15 1991-01-02 Schering Corporation Process for preparing antibacterial compounds and intermediates thereto
NZ250394A (en) * 1990-10-25 1994-10-26 Schering Corp Fluorinated and hydroxylated oxazoline compounds

Also Published As

Publication number Publication date
JP3274868B2 (ja) 2002-04-15
KR20000068178A (ko) 2000-11-25
EP0922040A1 (en) 1999-06-16
CA2264116C (en) 2002-07-02
CZ54099A3 (cs) 1999-07-14
HUP9904166A3 (en) 2001-11-28
ZA977406B (en) 1998-02-18
DE69731835T3 (de) 2013-12-05
SK19999A3 (en) 2000-02-14
KR100286851B1 (ko) 2001-04-16
WO1998007709A1 (en) 1998-02-26
NZ334111A (en) 1999-10-28
NO990756D0 (no) 1999-02-18
PL196454B1 (pl) 2008-01-31
US5663361A (en) 1997-09-02
DE69731835D1 (de) 2005-01-05
HUP9904166A2 (hu) 2000-05-28
HK1017890A1 (en) 1999-12-03
DK0922040T3 (da) 2005-04-04
EP0922040B2 (en) 2013-07-17
ES2234026T5 (es) 2013-11-12
BR9711318A (pt) 1999-08-17
CZ297915B6 (cs) 2007-04-25
BR9711318B1 (pt) 2009-01-13
TR199900354T2 (tr) 1999-05-21
CN1233244A (zh) 1999-10-27
PE99798A1 (es) 1998-12-28
IL128574A (en) 2002-04-21
SI0922040T1 (en) 2005-02-28
AR008298A1 (es) 1999-12-29
SK286124B6 (sk) 2008-04-07
JP2000501424A (ja) 2000-02-08
IL128574A0 (en) 2000-01-31
EP0922040B1 (en) 2004-12-01
TW381075B (en) 2000-02-01
CN1097583C (zh) 2003-01-01
PT922040E (pt) 2005-02-28
MY115679A (en) 2003-08-30
NO990756L (no) 1999-02-18
CO4560550A1 (es) 1998-02-10
ID18047A (id) 1998-02-19
DE69731835T2 (de) 2005-07-21
AU714495B2 (en) 2000-01-06
NO312962B1 (no) 2002-07-22
PL198553B1 (pl) 2008-06-30
HU229610B1 (en) 2014-03-28
ATE283847T1 (de) 2004-12-15
AU4063897A (en) 1998-03-06
PL331644A1 (en) 1999-08-02
ES2234026T3 (es) 2005-06-16
CA2264116A1 (en) 1998-02-26

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