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TR200001542T2 - Mide fundusunu gevşetici özelliklere sahip (benzodioksan, benzofuran veya benzopiran) türevleri. - Google Patents

Mide fundusunu gevşetici özelliklere sahip (benzodioksan, benzofuran veya benzopiran) türevleri.

Info

Publication number
TR200001542T2
TR200001542T2 TR2000/01542T TR200001542T TR200001542T2 TR 200001542 T2 TR200001542 T2 TR 200001542T2 TR 2000/01542 T TR2000/01542 T TR 2000/01542T TR 200001542 T TR200001542 T TR 200001542T TR 200001542 T2 TR200001542 T2 TR 200001542T2
Authority
TR
Turkey
Prior art keywords
benzodioxane
benzopyran
benzofuran
derivatives
stomach fundus
Prior art date
Application number
TR2000/01542T
Other languages
English (en)
Inventor
Tom Bert Paul Wigerinck Piet
Gaston Verschueren Wim
Francis Josephine Schroven Marc
Frans Leopold De Bruyn Marcel
Original Assignee
Janssen Pharmaceutica N.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica N.V. filed Critical Janssen Pharmaceutica N.V.
Publication of TR200001542T2 publication Critical patent/TR200001542T2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

(Formül(I), Formül(A)); Bu bulus, formül (I)' e sahip bilesiklere, bunlarin stereokimyasal olarak izomerik bir formuna, N-oksit formuna veya farmasötik olarak kabul edilebilir bir asit ilave tuzuna iliskindir. Bahsedilen ürünlerin hazirlanmasi için islemler, bahsedilen ürünleri içeren formülasyonlar ve bunlarin özellikle bozulmus fundus gevsemesiyle iliskili durumlarin tedavisinde bir ilaç olarak kullanimi da açiklanmistir.
TR2000/01542T 1997-12-05 1998-11-27 Mide fundusunu gevşetici özelliklere sahip (benzodioksan, benzofuran veya benzopiran) türevleri. TR200001542T2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP97203808 1997-12-05

Publications (1)

Publication Number Publication Date
TR200001542T2 true TR200001542T2 (tr) 2001-01-22

Family

ID=8229014

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2000/01542T TR200001542T2 (tr) 1997-12-05 1998-11-27 Mide fundusunu gevşetici özelliklere sahip (benzodioksan, benzofuran veya benzopiran) türevleri.

Country Status (32)

Country Link
US (4) US6133277A (tr)
EP (1) EP1036073B8 (tr)
JP (1) JP2001525407A (tr)
KR (1) KR100591605B1 (tr)
CN (1) CN1155597C (tr)
AR (1) AR017195A1 (tr)
AT (1) ATE334125T1 (tr)
AU (1) AU748669B2 (tr)
BG (1) BG64624B1 (tr)
BR (1) BR9814256A (tr)
CA (1) CA2311669C (tr)
CO (1) CO5011114A1 (tr)
CZ (1) CZ297895B6 (tr)
DE (1) DE69835372T2 (tr)
EA (1) EA003365B1 (tr)
EE (1) EE04438B1 (tr)
ES (1) ES2270541T3 (tr)
HK (1) HK1028400A1 (tr)
HR (1) HRP20000340B1 (tr)
HU (1) HU224813B1 (tr)
ID (1) ID24616A (tr)
IL (1) IL136529A (tr)
MY (1) MY124586A (tr)
NO (1) NO320727B1 (tr)
NZ (1) NZ503603A (tr)
PL (1) PL191144B1 (tr)
SK (1) SK286268B6 (tr)
TR (1) TR200001542T2 (tr)
TW (1) TW577886B (tr)
UA (1) UA70308C2 (tr)
WO (1) WO1999029687A1 (tr)
ZA (1) ZA9811081B (tr)

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JO2352B1 (en) * 2000-06-22 2006-12-12 جانسين فارماسيوتيكا ان. في Compounds for the treatment of non-adaptation of the bottom of the uterus
JO2654B1 (en) 2000-09-04 2012-06-17 شركة جانسين فارماسوتيكا ان. في Multiple aryl caroxa amides are useful as lipid - lowering agents
JO2409B1 (en) * 2000-11-21 2007-06-17 شركة جانسين فارماسوتيكا ان. في Second-phenyl carboxy amides are useful as lipid-lowering agents
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JPWO2003040382A1 (ja) * 2001-11-09 2005-03-03 株式会社カネカ 光学活性クロマン誘導体の製造法および中間体
ES2199086B1 (es) 2002-07-31 2005-06-01 Cepa Schwarz Pharma Sl Nuevos derivados de cicloalcanodionas, procedimiento para su preparacion y sus aplicaciones farmacologicas.
US7071821B2 (en) * 2003-05-14 2006-07-04 Bellsouth Intellectual Property Corporation Method and system for alerting a person to a situation
ITTO20030140U1 (it) * 2003-09-16 2005-03-17 Interfila Srl Matita cosmetica
CA2580584C (en) * 2003-09-19 2015-07-28 Galileo Pharmaceuticals, Inc. Use of alpha-tocotrienol for treatment of mitochondrial diseases
EP1687277B1 (en) 2003-11-20 2018-04-04 Janssen Pharmaceutica NV 6-alkenyl and 6-phenylalkyl substituted 2-quinolinones and 2-quinoxalinones as poly(adp-ribose) polymerase inhibitors
MXPA06005686A (es) 2003-11-20 2006-08-17 Janssen Pharmaceutica Nv 2-quinolinonas y 2-quinoxalinonas 7-fenilaquilo sustituidas como inhibidores de la poli(adp-ribosa)polimerasa.
ES2238015B1 (es) * 2004-01-30 2006-11-01 Cepa Schwarz Pharma, S.L. Derivados de cicloalcanodionas con actividad neuroprotectora.
SG154432A1 (en) * 2004-06-30 2009-08-28 Janssen Pharmaceutica Nv Quinazolinedione derivatives as parp inhibitors
CA2569826C (en) 2004-06-30 2013-07-16 Janssen Pharmaceutica N.V. Substituted 2-alkyl quinazolinone derivatives as parp inhibitors
EA014955B1 (ru) 2004-06-30 2011-04-29 Янссен Фармацевтика Н. В. Производные фталазина в качестве ингибиторов parp
DE102004032277A1 (de) * 2004-07-02 2006-01-19 Basell Polyolefine Gmbh Verfahren zur racemoselektiven Synthese von ansa-Metallocenen
PA8663501A1 (es) 2005-02-17 2006-11-09 Wyeth Wyeth Derivados de indol, benzotiofeno, benzofurano e indeno cicloalquilcondensados
KR20080008378A (ko) * 2005-04-22 2008-01-23 와이어쓰 크로만 및 크로멘 유도체 및 이의 용도
WO2008015538A2 (en) * 2006-07-31 2008-02-07 Schwarz Pharma S.L. Use of diaza- and thiaza-cycloalkanediones for preventing and/or treating pain and /or migraine
US20080033050A1 (en) * 2006-08-04 2008-02-07 Richards Patricia Allison Tewe Method of treating thermoregulatory disfunction with paroxetine
US8503431B2 (en) * 2006-08-25 2013-08-06 Wireless Wonders Ltd. Mobile phone related indirect communication system and method
WO2008107478A1 (en) 2007-03-08 2008-09-12 Janssen Pharmaceutica Nv Quinolinone derivatives as parp and tank inhibitors
JP5017703B2 (ja) * 2007-05-16 2012-09-05 住友ゴム工業株式会社 ビードエイペックスおよびタイヤ
US8404713B2 (en) 2007-10-26 2013-03-26 Janssen Pharmaceutica Nv Quinolinone derivatives as PARP inhibitors
ES2367760T3 (es) 2008-03-27 2011-11-08 Janssen Pharmaceutica, N.V. Derivados de quinazolinona como inhibidores de la polimerización de la tubulina.
AU2009228943B2 (en) 2008-03-27 2013-04-04 Janssen Pharmaceutica Nv Tetrahydrophenanthridinones and tetrahydrocyclopentaquinolinones as PARP and tubulin polymerization inhibitors
PL2817299T3 (pl) 2012-02-24 2019-12-31 Lupin Limited Podstawione związki chromanowe jako modulatory receptorów wapniowych
WO2014102592A2 (en) 2012-12-27 2014-07-03 Purdue Pharma L.P. Oxime/substituted quinoxaline-type piperidine compounds and uses thereof
DE102013207163B4 (de) 2013-04-19 2022-09-22 Adidas Ag Schuhoberteil
DE102014220087B4 (de) 2014-10-02 2016-05-12 Adidas Ag Flachgestricktes Schuhoberteil für Sportschuhe
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DE4140540A1 (de) * 1991-12-09 1993-06-17 Bayer Ag Neue azaheterocyclylmethyl-chromane
SI9300097B (en) * 1992-02-27 2001-12-31 Janssen Pharmaceutica Nv (benzodioxan, benzofuran or benzopyran) alkylamino) alkyl substituted guanidines
DE4319038A1 (de) * 1993-06-08 1994-12-15 Bayer Ag Verwendung von teilweise bekannten substituierten Chromanen als Arzneimittel, neue Wirkstoffe und Verfahren zu ihrer Herstellung
SK282402B6 (sk) * 1993-08-19 2002-01-07 Janssen Pharmaceutica N. V. Deriváty dihydrobenzopyránu, spôsob a medziprodukty na ich výrobu, ich použitie a farmaceutický prostriedok na ich báze
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US6133277A (en) 1997-12-05 2000-10-17 Janssen Pharmaceutica N.V. (Benzodioxan, benzofuran or benzopyran) derivatives having fundic relaxation properties

Also Published As

Publication number Publication date
HRP20000340B1 (en) 2008-12-31
MY124586A (en) 2006-06-30
CA2311669C (en) 2010-04-27
CN1280577A (zh) 2001-01-17
CO5011114A1 (es) 2001-02-28
US20030083365A1 (en) 2003-05-01
US6852714B2 (en) 2005-02-08
ZA9811081B (en) 2000-06-22
HUP0004492A3 (en) 2002-04-29
WO1999029687A8 (en) 2000-04-13
EE200000328A (et) 2001-08-15
CA2311669A1 (en) 1999-06-17
HU224813B1 (en) 2006-02-28
BG64624B1 (bg) 2005-09-30
CZ297895B6 (cs) 2007-04-25
EP1036073B8 (en) 2006-11-15
ID24616A (id) 2000-07-27
TW577886B (en) 2004-03-01
SK8032000A3 (en) 2001-02-12
HUP0004492A2 (hu) 2002-03-28
NO320727B1 (no) 2006-01-23
HRP20000340A2 (en) 2001-04-30
CN1155597C (zh) 2004-06-30
CZ20002018A3 (cs) 2000-10-11
IL136529A (en) 2003-03-12
EA200000616A1 (ru) 2000-12-25
JP2001525407A (ja) 2001-12-11
PL341007A1 (en) 2001-03-12
ATE334125T1 (de) 2006-08-15
ES2270541T3 (es) 2007-04-01
AU748669B2 (en) 2002-06-06
WO1999029687A1 (en) 1999-06-17
KR20010031010A (ko) 2001-04-16
NZ503603A (en) 2001-10-26
HK1028400A1 (en) 2001-02-16
DE69835372D1 (de) 2006-09-07
UA70308C2 (uk) 2004-10-15
AU2412799A (en) 1999-06-28
PL191144B1 (pl) 2006-03-31
US20030149093A1 (en) 2003-08-07
EE04438B1 (et) 2005-02-15
US6747045B2 (en) 2004-06-08
DE69835372T2 (de) 2007-08-09
AR017195A1 (es) 2001-08-22
US6495547B1 (en) 2002-12-17
US6133277A (en) 2000-10-17
KR100591605B1 (ko) 2006-06-20
NO20002074D0 (no) 2000-04-19
EP1036073B1 (en) 2006-07-26
EP1036073A1 (en) 2000-09-20
IL136529A0 (en) 2001-06-14
EA003365B1 (ru) 2003-04-24
SK286268B6 (sk) 2008-06-06
BR9814256A (pt) 2000-10-03
BG104372A (en) 2000-12-29
NO20002074L (no) 2000-06-02

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