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TN2011000272A1 - Dosage regimen for a s1p agonist - Google Patents

Dosage regimen for a s1p agonist

Info

Publication number
TN2011000272A1
TN2011000272A1 TN2011000272A TN2011000272A TN2011000272A1 TN 2011000272 A1 TN2011000272 A1 TN 2011000272A1 TN 2011000272 A TN2011000272 A TN 2011000272A TN 2011000272 A TN2011000272 A TN 2011000272A TN 2011000272 A1 TN2011000272 A1 TN 2011000272A1
Authority
TN
Tunisia
Prior art keywords
dosage regimen
agonist
dosage
daily dosage
agonists
Prior art date
Application number
TN2011000272A
Other languages
English (en)
Inventor
Robert Schmouder
Thomas Dumortier
Olivier David
Michael Looby
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41667217&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TN2011000272(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of TN2011000272A1 publication Critical patent/TN2011000272A1/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/661—Phosphorus acids or esters thereof not having P—C bonds, e.g. fosfosal, dichlorvos, malathion or mevinphos
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/06—Phosphorus compounds without P—C bonds
    • C07F9/08—Esters of oxyacids of phosphorus
    • C07F9/09—Esters of phosphoric acids
    • C07F9/10—Phosphatides, e.g. lecithin

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Emergency Medicine (AREA)
  • Transplantation (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
TN2011000272A 2008-12-22 2011-05-26 Dosage regimen for a s1p agonist TN2011000272A1 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US13967208P 2008-12-22 2008-12-22
US21853009P 2009-06-19 2009-06-19
US24671509P 2009-09-29 2009-09-29
PCT/US2009/068888 WO2010075239A1 (fr) 2008-12-22 2009-12-21 Régime posologique pour un agoniste du récepteur s1p

Publications (1)

Publication Number Publication Date
TN2011000272A1 true TN2011000272A1 (en) 2012-12-17

Family

ID=41667217

Family Applications (1)

Application Number Title Priority Date Filing Date
TN2011000272A TN2011000272A1 (en) 2008-12-22 2011-05-26 Dosage regimen for a s1p agonist

Country Status (41)

Country Link
US (11) US20100160259A1 (fr)
EP (7) EP3120844A1 (fr)
JP (7) JP2012513401A (fr)
KR (1) KR101347919B1 (fr)
CN (1) CN102264359A (fr)
AR (1) AR074826A1 (fr)
AU (1) AU2009330176C9 (fr)
BR (1) BRPI0923500A2 (fr)
CA (1) CA2747802C (fr)
CL (2) CL2011001529A1 (fr)
CO (1) CO6390117A2 (fr)
CR (1) CR20110274A (fr)
CU (1) CU20110136A7 (fr)
CY (4) CY1116990T1 (fr)
DK (3) DK3453387T3 (fr)
EA (1) EA201100978A1 (fr)
EC (1) ECSP11011222A (fr)
ES (3) ES2760607T3 (fr)
FR (1) FR20C1060I1 (fr)
HN (1) HN2011001759A (fr)
HR (3) HRP20151190T1 (fr)
HU (4) HUE048717T4 (fr)
IL (3) IL213170A0 (fr)
LT (3) LT3409274T (fr)
LU (1) LUC00183I2 (fr)
MA (1) MA32981B1 (fr)
ME (2) ME03802B (fr)
MX (2) MX2011006623A (fr)
NO (1) NO2020038I1 (fr)
NZ (1) NZ593065A (fr)
PE (1) PE20120337A1 (fr)
PL (3) PL2379067T3 (fr)
PT (3) PT3453387T (fr)
RS (2) RS59857B1 (fr)
SG (1) SG171404A1 (fr)
SI (3) SI3409274T1 (fr)
TN (1) TN2011000272A1 (fr)
TW (1) TW201028143A (fr)
UY (1) UY32352A (fr)
WO (1) WO2010075239A1 (fr)
ZA (2) ZA201103863B (fr)

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US8785484B2 (en) 2008-03-17 2014-07-22 Actelion Pharmaceuticals Ltd Dosing regimen for a selective S1P1 receptor agonist
MX2011006623A (es) 2008-12-22 2011-07-12 Novartis Ag Regimen de dosificacion para un agonista de los receptores de s1p.
CN102548579A (zh) 2009-09-29 2012-07-04 诺瓦提斯公司 S1p受体调节剂的给药方案
US20110124605A1 (en) * 2009-11-20 2011-05-26 Shreeram Aradhye Use of an S1P Receptor Agonist
CN108558740B (zh) 2010-01-27 2021-10-19 艾尼纳制药公司 S1p1受体调节剂及其盐的制备方法
EA201201515A1 (ru) * 2010-05-06 2013-08-30 Новартис Аг Схема приема производных диарилсульфидов
EP2455080A1 (fr) * 2010-11-23 2012-05-23 Almirall, S.A. Agonistes de récepteur S1P1 à utiliser dans le traitement de la sclérose en plaques
FR2968556B1 (fr) 2010-12-13 2013-12-27 Centre Nat Rech Scient Inhibiteurs des infections a vih et leurs utilisations
EA026144B9 (ru) 2011-01-07 2021-10-26 Новартис Аг Твердофазная фармацевтическая композиция, содержащая гемифумаратную соль 1-{4-[1-(4-циклогексил-3-трифторметилбензилоксиимино)этил]-2-этилбензил}азетидин-3-карбоновой кислоты, и таблетка, ее содержащая
WO2012112933A1 (fr) 2011-02-18 2012-08-23 The Scripps Research Institute Différenciation dirigée de cellules précurseurs d'oligodendrocytes vers un destin cellulaire myélinisant
AR085749A1 (es) 2011-04-01 2013-10-23 Novartis Ag Formulaciones
US9592268B2 (en) 2011-05-23 2017-03-14 Cornell University Endothelium protective materials and methods of use
TW201320994A (zh) 2011-10-11 2013-06-01 Novartis Ag 投藥療程
CN104540800B (zh) 2012-08-17 2017-05-10 埃科特莱茵药品有限公司 制备(2z,5z)‑5‑(3‑氯‑4‑((r)‑2,3‑二羟基丙氧基)苯亚甲基)‑2‑(丙亚氨基)‑3‑(邻甲苯基)噻唑烷‑4‑酮的方法及在该方法中所用的中间产物
AU2014225534A1 (en) * 2013-03-06 2015-09-24 Acorda Therapeutics, Inc. Therapeutic dosing of a neuregulin or a fragment thereof for treatment or prophylaxis of heart failure
WO2015053878A1 (fr) 2013-10-11 2015-04-16 Teikoku Pharma Usa, Inc. Formulations topiques agonistes du récepteur de la sphingosine-1-phosphate et procédés d'utilisation de celles-ci
US10675254B2 (en) 2013-10-11 2020-06-09 Teikoku Seiyaku Co., Ltd. Sphingosine-1-phosphate receptor agonist iontophoretic devices and methods of using the same
KR20160141841A (ko) * 2014-04-10 2016-12-09 노파르티스 아게 Ｓ１ｐ 조절제 즉시 방출 투여 요법
EP4056179A1 (fr) 2014-12-11 2022-09-14 Actelion Pharmaceuticals Ltd Régime posologique pour ponesimod, un agoniste du récepteur s1p1 sélectif
NZ771435A (en) * 2015-01-06 2024-08-30 Arena Pharm Inc Methods of treating conditions related to the s1p1 receptor
US20180042895A1 (en) 2015-02-26 2018-02-15 Novartis Ag Treatment of autoimmune disease in a patient receiving additionally a beta-blocker
MA42807A (fr) 2015-06-22 2018-07-25 Arena Pharm Inc Sel l-arginine cristallin d'acide (r)-2-(7-(4-cyclopentyl-3-(trifluorométhyl)benzyloxy)-1,2,3,4-tétrahydrocyclo-penta[b]indol-3-yl)acétique (composé 1) pour une utilisation dans des troubles associés au récepteur de s1p1
MA47504A (fr) 2017-02-16 2019-12-25 Arena Pharm Inc Composés et méthodes de traitement de l'angiocholite biliaire primitive
US11478448B2 (en) 2017-02-16 2022-10-25 Arena Pharmaceuticals, Inc. Compounds and methods for treatment of inflammatory bowel disease with extra-intestinal manifestations
JP2023501217A (ja) 2019-10-31 2023-01-18 イドーシア ファーマシューティカルズ リミテッド Ｃｘｃｒ７アンタゴニストのｓ１ｐ１受容体調節剤との合剤
WO2021158848A1 (fr) * 2020-02-07 2021-08-12 Argentum Pharmaceuticals Llc Régime posologique d'un agoniste du récepteur s1p
US11135197B2 (en) 2020-02-07 2021-10-05 Argentum Pharmaceuticals Llc Dosage regimen of an S1P receptor modulator
CN113332435B (zh) * 2021-06-18 2022-10-18 广州中医药大学(广州中医药研究院) 鞘氨醇-1-磷酸4受体激动剂及其与真武汤联合在制备治疗慢性肾小球肾炎药物中的应用

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JP2579602B2 (ja) 1992-10-21 1997-02-05 吉富製薬株式会社 ２−アミノ−１，３−プロパンジオール化合物および免疫抑制剤
EP1315735A4 (fr) 2000-08-31 2005-04-06 Merck & Co Inc Derives de phosphates utilises en tant qu'agents immuno-regulateurs
ATE412408T1 (de) 2002-05-16 2008-11-15 Novartis Pharma Gmbh Verwendung von edg rezeptor bindenden wirkstoffen für die krebstherapie
JP4861177B2 (ja) * 2003-09-12 2012-01-25 ニューロノバ エービー 神経系の障害の処置
US20060002999A1 (en) * 2004-06-17 2006-01-05 Forest Laboratories, Inc. Immediate release formulations of 1-aminocyclohexane compounds, memantine and neramexane
EP2359821A1 (fr) * 2004-11-29 2011-08-24 Novartis AG Posologie d'un agoniste du recepteur s1p
EP1688141A1 (fr) * 2005-01-31 2006-08-09 elbion AG Utilisation de flupirtine pour le traitement de la vessie hyperactive et des maladies associées et pour le traitement du syndrome du colon irritable
EP1850689A4 (fr) * 2005-02-10 2013-05-22 G I View Ltd Techniques de deplacement d'un outil gastro-intestinal equipe d'un element de guidage
DK2952177T3 (da) * 2007-10-12 2021-04-26 Novartis Ag Sammensætninger, der omfatter sphingosin-1-phosphat (s1p)-receptormodulatorer
US8785484B2 (en) * 2008-03-17 2014-07-22 Actelion Pharmaceuticals Ltd Dosing regimen for a selective S1P1 receptor agonist
WO2009155475A1 (fr) * 2008-06-20 2009-12-23 Novartis Ag Compositions pédiatriques pour le traitement de la sclérose en plaques
BRPI0923213A2 (pt) * 2008-12-22 2016-01-26 Novaris Ag regime de dosagem de um agonista do receptor para s1p.
MX2011006623A (es) 2008-12-22 2011-07-12 Novartis Ag Regimen de dosificacion para un agonista de los receptores de s1p.

Also Published As

Publication number Publication date
LT3409274T (lt) 2020-02-10
US20220142949A1 (en) 2022-05-12
DK2379067T3 (en) 2015-12-07
US20200330407A1 (en) 2020-10-22
US20140148415A1 (en) 2014-05-29
ME03594B (fr) 2020-07-20
DK3409274T3 (da) 2019-12-16
US20190091180A1 (en) 2019-03-28
CA2747802C (fr) 2021-02-09
JP7329965B2 (ja) 2023-08-21
BRPI0923500A2 (pt) 2018-05-29
IL278914A (en) 2021-01-31
MA32981B1 (fr) 2012-01-02
ES2552823T3 (es) 2015-12-02
RS59857B1 (sr) 2020-02-28
ECSP11011222A (es) 2011-08-31
US20140066657A1 (en) 2014-03-06
CY2020036I2 (el) 2021-06-25
CR20110274A (es) 2011-07-19
CO6390117A2 (es) 2012-02-29
SI3409274T1 (sl) 2020-03-31
PL2379067T3 (pl) 2016-02-29
HUE048717T2 (hu) 2020-08-28
CN102264359A (zh) 2011-11-30
EP3409274A1 (fr) 2018-12-05
EA201100978A1 (ru) 2012-01-30
PE20120337A1 (es) 2012-04-24
EP4098256A1 (fr) 2022-12-07
ZA201205942B (en) 2013-03-27
JP2017141238A (ja) 2017-08-17
SI2379067T1 (sl) 2016-01-29
WO2010075239A1 (fr) 2010-07-01
PT3409274T (pt) 2019-12-17
FR20C1060I1 (fr) 2020-12-25
JP2019167360A (ja) 2019-10-03
MX2011006623A (es) 2011-07-12
PT2379067E (pt) 2015-12-23
ES2810823T3 (es) 2021-03-09
JP2012513401A (ja) 2012-06-14
HRP20201167T1 (hr) 2020-12-11
JP2024129030A (ja) 2024-09-26
HRP20151190T1 (hr) 2016-01-01
EP3677260A1 (fr) 2020-07-08
NO2020038I1 (no) 2020-11-18
EP3120844A1 (fr) 2017-01-25
AU2009330176C9 (en) 2017-01-05
KR101347919B1 (ko) 2014-01-07
AU2009330176C1 (en) 2016-12-08
US20160081949A1 (en) 2016-03-24
JP2014144970A (ja) 2014-08-14
PL3409274T3 (pl) 2020-06-01
RS60666B1 (sr) 2020-09-30
SG171404A1 (en) 2011-07-28
IL274756A (en) 2020-07-30
HUE048717T4 (hu) 2022-02-28
US20170189353A1 (en) 2017-07-06
LT3453387T (lt) 2020-08-25
PL3453387T3 (pl) 2020-11-02
AU2009330176A1 (en) 2011-07-07
US20160263061A1 (en) 2016-09-15
UY32352A (es) 2010-07-30
ZA201103863B (en) 2012-10-31
EP3409274B1 (fr) 2019-11-20
CL2013001558A1 (es) 2013-10-25
LUC00183I2 (fr) 2024-07-01
EP2379067A1 (fr) 2011-10-26
ME03802B (fr) 2021-04-20
KR20110096175A (ko) 2011-08-29
EP2379067B1 (fr) 2015-09-02
JP2022103194A (ja) 2022-07-07
SI3453387T1 (sl) 2020-10-30
JP2016135752A (ja) 2016-07-28
MX2021010759A (es) 2022-07-19
US20100160259A1 (en) 2010-06-24
NZ593065A (en) 2012-11-30
AU2009330176B2 (en) 2014-03-06
PT3453387T (pt) 2020-08-11
HUE026869T2 (en) 2016-08-29
DK3453387T3 (da) 2020-08-10
TW201028143A (en) 2010-08-01
EP2907511A1 (fr) 2015-08-19
CA2747802A1 (fr) 2010-07-01
CY1122812T1 (el) 2021-05-05
US20110257133A1 (en) 2011-10-20
IL213170A0 (en) 2011-07-31
CY2020036I1 (el) 2021-03-12
LTPA2020005I1 (lt) 2020-12-10
HUE052048T2 (hu) 2021-04-28
CY1123255T1 (el) 2021-10-29
US20180289638A1 (en) 2018-10-11
CL2011001529A1 (es) 2012-02-24
HRP20192175T1 (hr) 2020-03-20
AR074826A1 (es) 2011-02-16
CU20110136A7 (es) 2012-01-31
EP3453387B1 (fr) 2020-06-03
CY1116990T1 (el) 2017-04-05
HN2011001759A (es) 2013-11-26
ES2760607T3 (es) 2020-05-14
HUS2000046I1 (hu) 2020-12-28
EP3453387A1 (fr) 2019-03-13

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