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SE9702533D0 - New oral formulation - Google Patents

New oral formulation

Info

Publication number
SE9702533D0
SE9702533D0 SE9702533A SE9702533A SE9702533D0 SE 9702533 D0 SE9702533 D0 SE 9702533D0 SE 9702533 A SE9702533 A SE 9702533A SE 9702533 A SE9702533 A SE 9702533A SE 9702533 D0 SE9702533 D0 SE 9702533D0
Authority
SE
Sweden
Prior art keywords
layer
oral formulation
new oral
effervescent
excipients
Prior art date
Application number
SE9702533A
Other languages
English (en)
Inventor
Per Johan Lundberg
Mikael Thune
Original Assignee
Astra Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astra Ab filed Critical Astra Ab
Priority to SE9702533A priority Critical patent/SE9702533D0/sv
Publication of SE9702533D0 publication Critical patent/SE9702533D0/sv
Priority to JP50700999A priority patent/JP2002508781A/ja
Priority to CA002294744A priority patent/CA2294744C/en
Priority to US09/125,933 priority patent/US6284271B1/en
Priority to AT98931171T priority patent/ATE247952T1/de
Priority to AU81357/98A priority patent/AU733801B2/en
Priority to DE69817587T priority patent/DE69817587T2/de
Priority to EP98931171A priority patent/EP1014952B1/en
Priority to PCT/SE1998/001209 priority patent/WO1999001112A1/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0065—Forms with gastric retention, e.g. floating on gastric juice, adhering to gastric mucosa, expanding to prevent passage through the pylorus
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/63—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
    • A61K31/635—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0007—Effervescent
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10—Antioedematous agents; Diuretics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Medicinal Preparation (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SE9702533A 1997-07-01 1997-07-01 New oral formulation SE9702533D0 (sv)

Priority Applications (9)

Application Number Priority Date Filing Date Title
SE9702533A SE9702533D0 (sv) 1997-07-01 1997-07-01 New oral formulation
JP50700999A JP2002508781A (ja) 1997-07-01 1998-06-22 発泡性マルチユニット製剤形
CA002294744A CA2294744C (en) 1997-07-01 1998-06-22 Multiple unit effervescent dosage form
US09/125,933 US6284271B1 (en) 1997-07-01 1998-06-22 Multiple unit effervescent dosage form
AT98931171T ATE247952T1 (de) 1997-07-01 1998-06-22 Aus einer vielzahl von kleineinheiten aufgebaute brausedosisform
AU81357/98A AU733801B2 (en) 1997-07-01 1998-06-22 Multiple unit effervescent dosage form
DE69817587T DE69817587T2 (de) 1997-07-01 1998-06-22 Aus einer vielzahl von kleineinheiten aufgebaute brausedosisform
EP98931171A EP1014952B1 (en) 1997-07-01 1998-06-22 Multiple unit effervescent dosage form
PCT/SE1998/001209 WO1999001112A1 (en) 1997-07-01 1998-06-22 Multiple unit effervescent dosage form

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE9702533A SE9702533D0 (sv) 1997-07-01 1997-07-01 New oral formulation

Publications (1)

Publication Number Publication Date
SE9702533D0 true SE9702533D0 (sv) 1997-07-01

Family

ID=20407594

Family Applications (1)

Application Number Title Priority Date Filing Date
SE9702533A SE9702533D0 (sv) 1997-07-01 1997-07-01 New oral formulation

Country Status (9)

Country Link
US (1) US6284271B1 (sv)
EP (1) EP1014952B1 (sv)
JP (1) JP2002508781A (sv)
AT (1) ATE247952T1 (sv)
AU (1) AU733801B2 (sv)
CA (1) CA2294744C (sv)
DE (1) DE69817587T2 (sv)
SE (1) SE9702533D0 (sv)
WO (1) WO1999001112A1 (sv)

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US6699885B2 (en) * 1996-01-04 2004-03-02 The Curators Of The University Of Missouri Substituted benzimidazole dosage forms and methods of using same
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US9522217B2 (en) 2000-03-15 2016-12-20 Orbusneich Medical, Inc. Medical device with coating for capturing genetically-altered cells and methods for using same
US20020064555A1 (en) * 2000-09-29 2002-05-30 Dan Cullen Proton pump inhibitor formulation
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DE10111780B8 (de) * 2001-03-13 2005-02-10 Isaak Dr. Abramov Brausetablette, Pille oder Dragee, sowie das Verfahren zu ihrer Herstellung
US20030198671A1 (en) * 2001-08-10 2003-10-23 Franz G. Andrew Levothyroxine compositions having unique plasma AUC properties
US20030171436A1 (en) * 2001-10-29 2003-09-11 Franz G. Andrew Levothyroxine compositions having unique triiodothyronine Tmax properties
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US8906940B2 (en) 2004-05-25 2014-12-09 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
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US7981908B2 (en) * 2005-05-11 2011-07-19 Vecta, Ltd. Compositions and methods for inhibiting gastric acid secretion
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FR2902337B1 (fr) * 2005-12-02 2010-09-17 Vacher Dominique Comprimes a liberation immediate et leur production
AU2007266574A1 (en) * 2006-06-01 2007-12-06 Dexcel Pharma Technologies Ltd. Multiple unit pharmaceutical formulation
PL2046334T3 (pl) * 2006-07-25 2015-02-27 Vecta Ltd Kompozycje i sposoby hamowania wydzielania kwasów żołądkowych z wykorzystaniem pochodnych małych kwasów dikarboksylowych w połączeniu z PPI
AU2007323018B2 (en) * 2006-09-04 2011-02-03 Panacea Biotec Limited Programmable buoyant delivery technology
EP2068841B1 (en) * 2006-10-05 2018-09-26 Santarus, Inc. Novel formulations of proton pump inhibitors and methods of using these formulations
CN103120653B (zh) 2007-04-04 2015-09-30 希格默伊德药业有限公司 一种口服药物组合物
EP2061587A1 (en) * 2007-04-26 2009-05-27 Sigmoid Pharma Limited Manufacture of multiple minicapsules
JP2010526054A (ja) * 2007-05-01 2010-07-29 シグモイド・ファーマ・リミテッド 併用医薬組成物
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Also Published As

Publication number Publication date
AU8135798A (en) 1999-01-25
EP1014952A1 (en) 2000-07-05
CA2294744A1 (en) 1999-01-14
CA2294744C (en) 2006-10-17
EP1014952B1 (en) 2003-08-27
WO1999001112A1 (en) 1999-01-14
DE69817587T2 (de) 2004-06-24
JP2002508781A (ja) 2002-03-19
US6284271B1 (en) 2001-09-04
DE69817587D1 (de) 2003-10-02
ATE247952T1 (de) 2003-09-15
AU733801B2 (en) 2001-05-24

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