SE503843C2 - Förfarande för framställning av 1-etoxikarbonyloxietylestern ab 6-(D(-)-a-amino-a-fenyl-acetamido)-penicillansyra - Google Patents

Förfarande för framställning av 1-etoxikarbonyloxietylestern ab 6-(D(-)-a-amino-a-fenyl-acetamido)-penicillansyra

Info

Publication number: SE503843C2
Authority: SE; Sweden
Prior art keywords: amino; acetamido; phenyl; preparation; alpha
Prior art date: 1982-06-29

Application number

SE9100548A

Other languages

English (en)

Other versions

SE9100548D0 (sv

SE9100548L (sv

SE503843C3 (sv

Inventor

Luigi Ratti

Derek Reginald Palmer

Robert Graham Tyson

Original Assignee

Astra Laekemedel Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-06-29

Filing date

1991-02-26

Publication date

1996-09-16

1982-06-29 Priority claimed from IT22141/82A external-priority patent/IT1190897B/it

1983-01-07 Priority claimed from GB838300331A external-priority patent/GB8300331D0/en

1991-02-26 Application filed by Astra Laekemedel Ab filed Critical Astra Laekemedel Ab

1991-02-26 Publication of SE9100548D0 publication Critical patent/SE9100548D0/sv

1991-02-26 Publication of SE9100548L publication Critical patent/SE9100548L/sv

1991-02-26 Publication of SE503843C3 publication Critical patent/SE503843C3/sv

1996-09-16 Publication of SE503843C2 publication Critical patent/SE503843C2/sv

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C68/00—Preparation of esters of carbonic or haloformic acids
- C07C68/02—Preparation of esters of carbonic or haloformic acids from phosgene or haloformates
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/96—Esters of carbonic or haloformic acids
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Oncology (AREA)
Pharmacology & Pharmacy (AREA)
Communicable Diseases (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Cephalosporin Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Plural Heterocyclic Compounds (AREA)

SE9100548A 1982-06-29 1991-02-26 Förfarande för framställning av 1-etoxikarbonyloxietylestern ab 6-(D(-)-a-amino-a-fenyl-acetamido)-penicillansyra SE503843C2 (sv)

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
IT22141/82A IT1190897B (it)	1982-06-29	1982-06-29	Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico
GB8226751		1982-09-20
GB8228622		1982-10-06
GB8232629		1982-11-16
GB838300331A GB8300331D0 (en)	1983-01-07	1983-01-07	Preparation of bromo carbonates

Publications (4)

Publication Number	Publication Date
SE9100548D0 SE9100548D0 (sv)	1991-02-26
SE9100548L SE9100548L (sv)	1991-02-26
SE503843C3 SE503843C3 (sv)	1991-02-26
SE503843C2 true SE503843C2 (sv)	1996-09-16

Family

ID=27516485

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
SE8303414A SE454879B (sv)	1982-06-29	1983-06-15	Alfa-bromodietylkarbonat samt dess anvendning som mellanprodukt vid framstellning av penicillin g
SE9100548A SE503843C2 (sv)	1982-06-29	1991-02-26	Förfarande för framställning av 1-etoxikarbonyloxietylestern ab 6-(D(-)-a-amino-a-fenyl-acetamido)-penicillansyra

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
SE8303414A SE454879B (sv)	1982-06-29	1983-06-15	Alfa-bromodietylkarbonat samt dess anvendning som mellanprodukt vid framstellning av penicillin g

Country Status (23)

Country	Link
JP (2)	JPH0819052B2 (sv)
AT (1)	AT383128B (sv)
AU (1)	AU566803B2 (sv)
BG (3)	BG38336A3 (sv)
CH (2)	CH656377A5 (sv)
CY (2)	CY1520A (sv)
DD (1)	DD211561A5 (sv)
DE (2)	DE3348299C2 (sv)
DK (3)	DK160039C (sv)
FI (1)	FI79115C (sv)
FR (1)	FR2543957B1 (sv)
GB (3)	GB2168050A (sv)
GR (1)	GR78585B (sv)
HU (1)	HU191534B (sv)
IE (1)	IE56712B1 (sv)
IL (1)	IL68992A (sv)
IS (1)	IS1361B6 (sv)
NL (1)	NL194081C (sv)
NO (3)	NO157696C (sv)
NZ (1)	NZ204736A (sv)
PT (1)	PT76944B (sv)
SE (2)	SE454879B (sv)
YU (2)	YU43926B (sv)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2573756B1 (fr) *	1984-11-23	1987-01-16	Poudres & Explosifs Ste Nale	Procede de preparation des carbonates de bromo-1 ethyle et d'hydrocarbyle et nouveaux carbonates de bromo-1 ethyle et d'hydrocarbyle

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CH516593A (de) *	1967-09-29	1971-12-15	Leo Pharm Prod Ltd	Verfahren zur Herstellung von neuen Estern von a-Aminobenzyl-penicillin
US3873521A (en) *	1970-09-17	1975-03-25	Astra Laekemedel Ab	Esters of {60 -amino penicillins
IE35648B1 (en) *	1970-09-25	1976-04-14	Beecham Group Ltd	Penicillins
DE2161420A1 (de) *	1970-12-30	1972-07-27	Toyama Chemical Co. Ltd., Tokio	Penicillinderivate und Verfahren zu deren Herstellung
BE784800A (fr) *	1971-06-15	1972-10-02	Yamanouchi Pharma Co Ltd	Procede de preparation de nouveaux derives esters oxymethyliques de la penicilline et de la cephalosporine
IL48514A (en) *	1972-02-15	1976-08-31	Mckenna A	Hexapeptide intermediate for the preparation of the lh-and fsh-releasing hormone
GB1425571A (en) *	1972-03-13	1976-02-18	Astra Laekemedel Ab	Penicillins and cephaosporins
GB1426869A (en) *	1972-03-13	1976-03-03	Astra Laekemedel Ab	Penicillins
GB1426717A (en) *	1972-03-13	1976-03-03	Astra Laekemedel Ab	Penicillins
SE397981B (sv) *	1973-02-19	1977-11-28	Astra Laekemedel Ab	Nya tetraalkylammoniumsalter av 6-aminopenicillansyra och av bensylpenicillin avsedda att anvendas som mellanprodukter vid framstellning av vissa estrar av 6-aminopenicillansyra och av bensylpenicillin
GB1565656A (en) *	1975-12-13	1980-04-23	Beecham Group Ltd	Preparation of substituted penicillin acid esters
GB1598568A (en) *	1977-04-19	1981-09-23	Glaxo Lab Ltd	Esters of(6r,7r)-3-carbamoyloxymethyl-7-((z)-2-(fur-2-yl)-2-methoxyiminoacetamido)-ceph-3-em-4-carboxylic acid
JPS5444694A (en) *	1977-09-06	1979-04-09	Kou Kamata	Aminobenzylpenicillin derivative
EP0098161A3 (en) *	1982-06-30	1985-04-24	Glaxo Group Limited	Cephalosporin compounds
DE3380024D1 (en) *	1982-11-04	1989-07-13	Astra Laekemedel Ab	Process for the preparation of the 1'-ethoxycarbonyloxyethyl ester of benzylpenicillin

1983
- 1983-06-15 IL IL68992A patent/IL68992A/xx not_active IP Right Cessation
- 1983-06-15 SE SE8303414A patent/SE454879B/sv not_active IP Right Cessation
- 1983-06-20 IE IE1445/83A patent/IE56712B1/en not_active IP Right Cessation
- 1983-06-24 DE DE3348299A patent/DE3348299C2/de not_active Expired - Lifetime
- 1983-06-24 DE DE3322783A patent/DE3322783A1/de active Granted
- 1983-06-27 GB GB08528958A patent/GB2168050A/en not_active Withdrawn
- 1983-06-28 FI FI832363A patent/FI79115C/sv not_active IP Right Cessation
- 1983-06-28 NZ NZ204736A patent/NZ204736A/en unknown
- 1983-06-28 HU HU832325A patent/HU191534B/hu unknown
- 1983-06-28 AU AU16328/83A patent/AU566803B2/en not_active Expired
- 1983-06-28 DK DK296683A patent/DK160039C/da not_active IP Right Cessation
- 1983-06-28 PT PT76944A patent/PT76944B/pt unknown
- 1983-06-28 NO NO832351A patent/NO157696C/no not_active IP Right Cessation
- 1983-06-28 GR GR71790A patent/GR78585B/el unknown
- 1983-06-28 BG BG068053A patent/BG38336A3/xx unknown
- 1983-06-28 BG BG068052A patent/BG38335A3/xx unknown
- 1983-06-28 BG BG061516A patent/BG37527A3/xx unknown
- 1983-06-28 CH CH3540/83A patent/CH656377A5/de not_active IP Right Cessation
- 1983-06-28 NL NL8302286A patent/NL194081C/nl not_active IP Right Cessation
- 1983-06-28 CH CH527585A patent/CH657620B/de not_active IP Right Cessation
- 1983-06-29 IS IS2825A patent/IS1361B6/is unknown
- 1983-06-29 AT AT0238483A patent/AT383128B/de not_active IP Right Cessation
- 1983-06-29 YU YU1415/83A patent/YU43926B/xx unknown
- 1983-06-29 DD DD83252531A patent/DD211561A5/de unknown
- 1983-12-30 FR FR8321138A patent/FR2543957B1/fr not_active Expired
1985
- 1985-03-28 NO NO851254A patent/NO851254L/no unknown
- 1985-03-28 NO NO851255A patent/NO851255L/no unknown
- 1985-09-16 GB GB08522826A patent/GB2168699B/en not_active Expired
- 1985-09-16 GB GB08522827A patent/GB2169287B/en not_active Expired
1986
- 1986-02-14 YU YU218/86A patent/YU43693B/xx unknown
1990
- 1990-04-30 DK DK106090A patent/DK167807B1/da not_active IP Right Cessation
- 1990-04-30 DK DK105990A patent/DK159821C/da not_active IP Right Cessation
- 1990-11-16 CY CY1520A patent/CY1520A/xx unknown
- 1990-11-16 CY CY1519A patent/CY1519A/xx unknown
1991
- 1991-02-26 SE SE9100548A patent/SE503843C2/sv not_active IP Right Cessation
- 1991-04-30 JP JP3124442A patent/JPH0819052B2/ja not_active Expired - Lifetime
- 1991-04-30 JP JP3124441A patent/JPH0730082B2/ja not_active Expired - Lifetime

Also Published As

Publication number	Publication date
NO851254L (no)	1983-12-30
DE3322783A1 (de)	1984-02-09
DK160039B (da)	1991-01-21
CH656377A5 (de)	1986-06-30
JPH0543583A (ja)	1993-02-23
SE454879B (sv)	1988-06-06
DK105990A (da)	1990-04-30
JPH0717918A (ja)	1995-01-20
GB2168050A (en)	1986-06-11
FI79115B (fi)	1989-07-31
DK160039C (da)	1991-06-10
DK106090A (da)	1990-04-30
IS2825A7 (is)	1984-07-08
DD211561A5 (de)	1984-07-18
IE831445L (en)	1983-12-29
AU1632883A (en)	1984-01-05
JPH0730082B2 (ja)	1995-04-05
NO157696B (no)	1988-01-25
NL194081C (nl)	2001-06-05
BG37527A3 (en)	1985-06-14
SE8303414D0 (sv)	1983-06-15
YU43926B (en)	1989-12-31
NO157696C (no)	1988-05-04
NL194081B (nl)	2001-02-01
FR2543957B1 (fr)	1986-10-24
GR78585B (sv)	1984-09-27
FR2543957A1 (fr)	1984-10-12
SE9100548D0 (sv)	1991-02-26
NO832351L (no)	1983-12-30
CH657620B (sv)	1986-09-15
GB2169287A (en)	1986-07-09
PT76944A (en)	1983-07-01
GB8528958D0 (en)	1986-01-02
DK105990D0 (da)	1990-04-30
NL8302286A (nl)	1984-01-16
NZ204736A (en)	1986-11-12
FI832363A0 (fi)	1983-06-28
NO851255L (no)	1983-12-30
BG38336A3 (en)	1985-11-15
FI79115C (sv)	1989-11-10
ATA238483A (de)	1986-10-15
FI832363L (fi)	1983-12-30
SE9100548L (sv)	1991-02-26
GB2168699B (en)	1987-04-15
DK159821B (da)	1990-12-10
JPH0819052B2 (ja)	1996-02-28
GB8522827D0 (en)	1985-10-23
CY1519A (en)	1990-11-16
SE8303414L (sv)	1983-12-30
PT76944B (en)	1986-04-09
DK159821C (da)	1991-04-29
GB2169287B (en)	1987-04-08
GB2168699A (en)	1986-06-25
YU43693B (en)	1989-10-31
AT383128B (de)	1987-05-25
DE3348299C2 (sv)	1990-12-20
IS1361B6 (is)	1989-05-25
GB8522826D0 (en)	1985-10-23
BG38335A3 (en)	1985-11-15
CY1520A (en)	1990-11-16
HU191534B (en)	1987-03-30
IE56712B1 (en)	1991-11-20
DK296683D0 (da)	1983-06-28
DK167807B1 (da)	1993-12-20
AU566803B2 (en)	1987-10-29
YU141583A (en)	1986-06-30
DE3322783C2 (sv)	1991-01-31
IL68992A (en)	1991-06-10
DK296683A (da)	1983-12-30
YU21886A (en)	1987-10-31
DK106090D0 (da)	1990-04-30

Publication	Publication Date	Title
IE800605L (en)	1980-09-26	Quinolines
FI892603A0 (sv)	1989-05-29	Förfarande för framställning av nya, terapeutiskt användbara 4-(kinolin-2-ylmetoxi)fenylättiksyraderivat
NO175149C (no)	1994-09-07	Analogifremgangsmåte for fremstilling av terapeutisk aktive, eventuelt ddiksyrer og -estere
NO943318L (no)	1995-03-13	Fremgangsmåte for fremstilling av eddiksyre
IS3945A (is)	1993-05-15	Aðferð til framleiðslu á ediksýruafleiðum
ATE142623T1 (de)	1996-09-15	2-substituierte chinoline, verfahren zu ihrer herstellung sowie ihre verwendung in arzneimitteln
BE881082A (nl)	1980-07-10	Werkwijze voor de bereiding van geconcentreerde natuurazijn en werkwijze voor de bereiding van azijnzuuresters
SE503843C2 (sv)	1996-09-16	Förfarande för framställning av 1-etoxikarbonyloxietylestern ab 6-(D(-)-a-amino-a-fenyl-acetamido)-penicillansyra
FI890723A0 (sv)	1989-02-15	Förfarande för framställning av kinolinkarboxylsyraderivat
JPS52128336A (en)	1977-10-27	Process for preparing metaaphenoxybenzyl alcohol and esters of alphaacyano and alphaaethynyl derivatives thereof with carboxylic acid
ES385437A1 (es)	1973-11-01	Metodo para la preparacion de nuevos derivados de acido pe-nicilanico.
SE7807225L (sv)	1978-06-26	Sett att framstella 4-hydroxicinnolin-derivat
DE3267646D1 (en)	1986-01-09	Process for the production of methyl acetate by esterifying methanol with acetic acid
DE3064719D1 (en)	1983-10-06	Process for the preparation of a polyvinyl alcohol complex compound, and polyvinylalcohol complex compound so prepared
ES8308827A1 (es)	1983-08-01	Un procedimiento para la preparacion de nuevos derivados poliprenilicos.
GB980777A (en)	1965-01-20	ª‡-amino-substituted penicillins
MY101937A (en)	1992-02-15	Process for the production of 1-ethoxycarbonyloxthyl ester of 6-(d-(-)-&-amino-&-phenylacetamido) penicillanic acid
AU545941B2 (en)	1985-08-08	Bis-esters of dicarboxylic acids with amoxicillin and certain hydroxymethylpenicillanate 1,1-dioxides
NO944336D0 (no)	1994-11-14	Enzymatisk fremgangsmåte for fremstilling av S-6-metoksy- -metyl-2-naftaleneddiksyre
JPS5711988A (en)	1982-01-21	Esterification of epipenicilin oxide
DE3775721D1 (de)	1992-02-13	Verfahren zur herstellung von veretherten 3-hydroxyvaleriansaeureestern.
ES410723A1 (es)	1976-04-01	Un procedimiento para la preparacion de nuevos derivados deacidos 6-aminopenicilanicos.
ES457577A1 (es)	1978-08-16	Un procedimiento de preparacion de nuevos compuestos de be- ta-lactama.
ES398825A1 (es)	1975-05-16	Procedimiento para la preparacion de alfa-amino-acil peni- cilinas.
NL191059C (nl)	1995-01-02	Werkwijze ter bereiding van 2-(p-fluorfenyl)-alfa-methyl-5-benzoxazolazijnzuur.

Legal Events

Date	Code	Title	Description
2003-07-29	NUG	Patent has lapsed