SE0301373D0 - Novel compounds - Google Patents
Novel compoundsInfo
- Publication number
- SE0301373D0 SE0301373D0 SE0301373A SE0301373A SE0301373D0 SE 0301373 D0 SE0301373 D0 SE 0301373D0 SE 0301373 A SE0301373 A SE 0301373A SE 0301373 A SE0301373 A SE 0301373A SE 0301373 D0 SE0301373 D0 SE 0301373D0
- Authority
- SE
- Sweden
- Prior art keywords
- novel compounds
- imidazo
- formula
- methods
- pharmaceutical compositions
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Neurology (AREA)
- Diabetes (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Physical Education & Sports Medicine (AREA)
- Hematology (AREA)
- Dermatology (AREA)
- Rheumatology (AREA)
- Transplantation (AREA)
- Obesity (AREA)
- Pain & Pain Management (AREA)
- Endocrinology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Otolaryngology (AREA)
- Emergency Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Priority Applications (19)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0301373A SE0301373D0 (sv) | 2003-05-09 | 2003-05-09 | Novel compounds |
MXPA05012025A MXPA05012025A (es) | 2003-05-09 | 2004-05-06 | Imidazo y tiazolopiridinas como inhibidores de cinasa jak3. |
US10/556,228 US20060287355A1 (en) | 2003-05-09 | 2004-05-06 | Imidazo and thiazolopyridines as jak3 kinase inhibitors |
CA002524624A CA2524624A1 (en) | 2003-05-09 | 2004-05-06 | Imidazo and thiazolopyridines as jak3 kinase inhibitors |
BRPI0410081-6A BRPI0410081A (pt) | 2003-05-09 | 2004-05-06 | composto, composição farmacêutica, método de tratamento de uma doença ou condição mediada por jak3, e, processo para a preparação de um composto |
DK04731525T DK1625126T3 (da) | 2003-05-09 | 2004-05-06 | Imidazo- og thiazolopyridiner som JAK3-kinaseinhibitorer |
JP2006508045A JP2006525997A (ja) | 2003-05-09 | 2004-05-06 | Jak3キナーゼ阻害剤としてのイミダゾ及びチアゾロピリジン |
EP04731525A EP1625126B1 (en) | 2003-05-09 | 2004-05-06 | Imidazo and thiazolopyridines as jak3 kinase inhibitors |
AU2004236144A AU2004236144B2 (en) | 2003-05-09 | 2004-05-06 | Imidazo and thiazolopyridines as JAK3 kinase inhibitors |
SI200430618T SI1625126T1 (sl) | 2003-05-09 | 2004-05-06 | Imidazo- in tiazolopiridini kot inhibitorji JAK3-kinaze |
AT04731525T ATE384061T1 (de) | 2003-05-09 | 2004-05-06 | Imidazo- und thiazolopyridine als jak3-kinase- inhibitoren |
EP07119970A EP1887007A3 (en) | 2003-05-09 | 2004-05-06 | Imidazo- and Thiazolopyridine as JAK3 Kinase Inhibitors |
PCT/SE2004/000694 WO2004099204A1 (en) | 2003-05-09 | 2004-05-06 | Imidazo and thiazolopyridines as jak3 kinase inhibitors |
CNA200480012617XA CN1784402A (zh) | 2003-05-09 | 2004-05-06 | 用作jak3激酶抑制剂的咪唑并和噻唑并吡啶化合物 |
DE602004011330T DE602004011330T2 (de) | 2003-05-09 | 2004-05-06 | Imidazo- und thiazolopyridine als jak3-kinase-inhibitoren |
PT04731525T PT1625126E (pt) | 2003-05-09 | 2004-05-06 | Imidazo- e tiazolopiridinas como inibidores de cinase jak3 |
ES04731525T ES2298754T3 (es) | 2003-05-09 | 2004-05-06 | Imidazo- y tiazolopiridinas como inhibidores de jak3 quinasa. |
PL04731525T PL1625126T3 (pl) | 2003-05-09 | 2004-05-06 | Imidazo- i tiazolopirydyny jako inhibitory kinazy JAK3 |
CY20081100279T CY1107301T1 (el) | 2003-05-09 | 2008-03-12 | Ιμιδαζο και θειαζολοπυριδινες ως αναστολεις κινασης jak3 |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0301373A SE0301373D0 (sv) | 2003-05-09 | 2003-05-09 | Novel compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
SE0301373D0 true SE0301373D0 (sv) | 2003-05-09 |
Family
ID=20291271
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SE0301373A SE0301373D0 (sv) | 2003-05-09 | 2003-05-09 | Novel compounds |
Country Status (17)
Country | Link |
---|---|
US (1) | US20060287355A1 (sv) |
EP (2) | EP1887007A3 (sv) |
JP (1) | JP2006525997A (sv) |
CN (1) | CN1784402A (sv) |
AT (1) | ATE384061T1 (sv) |
AU (1) | AU2004236144B2 (sv) |
BR (1) | BRPI0410081A (sv) |
CA (1) | CA2524624A1 (sv) |
CY (1) | CY1107301T1 (sv) |
DE (1) | DE602004011330T2 (sv) |
DK (1) | DK1625126T3 (sv) |
ES (1) | ES2298754T3 (sv) |
MX (1) | MXPA05012025A (sv) |
PL (1) | PL1625126T3 (sv) |
PT (1) | PT1625126E (sv) |
SE (1) | SE0301373D0 (sv) |
WO (1) | WO2004099204A1 (sv) |
Families Citing this family (65)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE0301372D0 (sv) * | 2003-05-09 | 2003-05-09 | Astrazeneca Ab | Novel compounds |
AR054416A1 (es) | 2004-12-22 | 2007-06-27 | Incyte Corp | Pirrolo [2,3-b]piridin-4-il-aminas y pirrolo [2,3-b]pirimidin-4-il-aminas como inhibidores de las quinasas janus. composiciones farmaceuticas. |
WO2006108103A1 (en) * | 2005-04-05 | 2006-10-12 | Pharmacopeia, Inc. | Purine and imidazopyridine derivatives for immunosuppression |
US7884109B2 (en) | 2005-04-05 | 2011-02-08 | Wyeth Llc | Purine and imidazopyridine derivatives for immunosuppression |
CN102127078A (zh) | 2005-07-14 | 2011-07-20 | 安斯泰来制药株式会社 | Janus激酶3的杂环类抑制剂 |
US8163767B2 (en) | 2005-07-14 | 2012-04-24 | Astellas Pharma Inc. | Heterocyclic Janus Kinase 3 inhibitors |
EP1912639A4 (en) * | 2005-08-08 | 2011-10-12 | Janssen Pharmaceutica Nv | Thiazolopyrimidine KINASE INHIBITORS |
WO2007038215A1 (en) | 2005-09-22 | 2007-04-05 | Incyte Corporation | Tetracyclic inhibitors of janus kinases |
MX346183B (es) | 2005-12-13 | 2017-03-10 | Incyte Holdings Corp | Pirrolo[2,3-b]piridinas y pirrolo[2,3-b]pirimidinas heteroarilo-sustituidas como inhibidores de cinasas janus. |
US7989459B2 (en) | 2006-02-17 | 2011-08-02 | Pharmacopeia, Llc | Purinones and 1H-imidazopyridinones as PKC-theta inhibitors |
EP1900729A1 (en) * | 2006-09-15 | 2008-03-19 | Novartis AG | Benzoxazoles and oxazolopyridines being useful as Janus kinases inhibitors |
TW200831104A (en) | 2006-10-04 | 2008-08-01 | Pharmacopeia Inc | 6-substituted 2-(benzimidazolyl)purine and purinone derivatives for immunosuppression |
US7902187B2 (en) | 2006-10-04 | 2011-03-08 | Wyeth Llc | 6-substituted 2-(benzimidazolyl)purine and purinone derivatives for immunosuppression |
TW200837064A (en) | 2006-10-04 | 2008-09-16 | Pharmacopeia Inc | 8-substituted 2-(benzimidazolyl)purine derivatives for immunosuppression |
JP5492565B2 (ja) | 2006-12-22 | 2014-05-14 | インサイト・コーポレイション | Janusキナーゼ阻害剤としての置換複素環 |
ES2627221T3 (es) | 2006-12-28 | 2017-07-27 | Rigel Pharmaceuticals, Inc. | Compuestos de heterocicloalquiloxibenzamida N-sustituidos y métodos de uso |
WO2008084861A1 (ja) * | 2007-01-12 | 2008-07-17 | Astellas Pharma Inc. | 縮合ピリジン化合物 |
CL2008001709A1 (es) | 2007-06-13 | 2008-11-03 | Incyte Corp | Compuestos derivados de pirrolo [2,3-b]pirimidina, moduladores de quinasas jak; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como cancer, psoriasis, artritis reumatoide, entre otras. |
HUE029236T2 (en) | 2007-06-13 | 2017-02-28 | Incyte Holdings Corp | (R) -3- (4- (7H-Pyrrolo [2,3-d] pyrimidin-4-yl) -1H-pyrazol-1-yl) -3-cyclopentylpropanenitrile Crystalline salts of Janus kinase inhibitor |
WO2009001021A1 (en) * | 2007-06-26 | 2008-12-31 | Chroma Therapeutics Ltd. | Imidazopyridine derivatives useful as enzyme inhibitors for the treatment of cell proliferative and autoimmune diseases |
KR101580482B1 (ko) | 2007-11-16 | 2015-12-28 | 인사이트 홀딩스 코포레이션 | 야누스 키나제 억제제로서의 4-피라졸릴-n-아릴피리미딘-2-아민 및 4-피라졸릴-n-헤테로아릴피리미딘-2-아민 |
BRPI0819529A2 (pt) * | 2007-12-19 | 2015-05-26 | Genentech Inc | "composto de fórmula i, composição farmacêutica, método para inibir o crescimento celular anormal ou tratar um distúrbio hiperproliferativo em um mamífero e método para tratar uma doença inflamatória em um mamífero" |
RU2498985C2 (ru) * | 2007-12-19 | 2013-11-20 | Дженентек, Инк. | 8-анилиноимидазопиридины и способы их использования |
PL2288610T3 (pl) | 2008-03-11 | 2017-12-29 | Incyte Holdings Corporation | Azetydynowe i cyklobutanowe pochodne jako inhibitory jak |
NZ599853A (en) * | 2008-04-11 | 2012-08-31 | Janssen Pharmaceutica Nv | Process for the preparation of meso-N-[(3-endo)-8-benzyl-8-azabicyclo[3.2.1]oct-3-yl]acetamide and its derivatives |
US8871753B2 (en) | 2008-04-24 | 2014-10-28 | Incyte Corporation | Macrocyclic compounds and their use as kinase inhibitors |
WO2009151910A2 (en) * | 2008-05-25 | 2009-12-17 | Wyeth | Combination product of receptor tyrosine kinase inhibitor and fatty acid synthase inhibitor for treating cancer |
EP2361902A4 (en) * | 2008-11-21 | 2012-04-25 | Astellas Pharma Inc | 4,6-DIAMINONICOTINSÄUREAMIDVERBINDUNG |
WO2010085597A1 (en) | 2009-01-23 | 2010-07-29 | Incyte Corporation | Macrocyclic compounds and their use as kinase inhibitors |
PT2432472T (pt) | 2009-05-22 | 2019-12-09 | Incyte Holdings Corp | 3-[4-(7h-pirrolo[2,3-d]pirimidin-4-il)-1h-pirazol-1-il]octano- ou heptano-nitrilo como inibidores de jak |
JP5775070B2 (ja) | 2009-05-22 | 2015-09-09 | インサイト・コーポレイションIncyte Corporation | ヤヌスキナーゼ阻害剤としてのピラゾール−4−イル−ピロロ[2,3−d]ピリミジンおよびピロール−3−イル−ピロロ[2,3−d]ピリミジンのN−(ヘテロ)アリール−ピロリジン誘導体 |
TW201113285A (en) | 2009-09-01 | 2011-04-16 | Incyte Corp | Heterocyclic derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors |
PL2486041T3 (pl) | 2009-10-09 | 2014-01-31 | Incyte Holdings Corp | Pochodne hydroksylowe, keto i glukuronidowe 3-(4-(7H-pirolo[2,3-d]pirymidyn-4-ylo)-1H-pirazol-1-ilo)-3-cyklopentylopropanonitrylu |
ES2982015T3 (es) | 2010-03-10 | 2024-10-14 | Incyte Holdings Corp | Derivados de piperidin-4-IL azetidina como inhibidores de JAK1 |
TWI499421B (zh) | 2010-05-21 | 2015-09-11 | Incyte Corp | Jak抑制劑的局部製劑 |
CN103415515B (zh) | 2010-11-19 | 2015-08-26 | 因塞特公司 | 作为jak抑制剂的环丁基取代的吡咯并吡啶和吡咯并嘧啶衍生物 |
EP2640725B1 (en) | 2010-11-19 | 2015-01-07 | Incyte Corporation | Heterocyclic-substituted pyrrolopyridines and pyrrolopyrimidines as jak inhibitors |
CN103732226B (zh) | 2011-02-18 | 2016-01-06 | 诺瓦提斯药物公司 | mTOR/JAK抑制剂组合疗法 |
AR085436A1 (es) | 2011-03-17 | 2013-10-02 | Bristol Myers Squibb Co | Derivados de pirrolopiridazina inhibidores de jak3, composiciones farmaceuticas que los contienen y su uso para tratar enfermedades inflamatorias y autoinmunes |
EP2686321B1 (en) | 2011-03-17 | 2016-11-16 | Bristol-Myers Squibb Company | Pyrrolopyridazine jak3 inhibitors and their use for the treatment of inflammatory and autoimmune diseases |
WO2012125886A1 (en) * | 2011-03-17 | 2012-09-20 | Bristol-Myers Squibb Company | Pyrrolopyridazine jak3 inhibitors and their use for the treatment of inflammatory and autoimmune diseases |
CA2830882C (en) | 2011-03-22 | 2021-03-16 | Dinesh Barawkar | Substituted fused tricyclic compounds, compositions and medicinal applications thereof |
PE20140832A1 (es) | 2011-06-20 | 2014-07-14 | Incyte Corp | Derivados de azetidinil fenil, piridil o pirazinil carboxamida como inhibidores de jak |
WO2013023119A1 (en) | 2011-08-10 | 2013-02-14 | Novartis Pharma Ag | JAK P13K/mTOR COMBINATION THERAPY |
TW201313721A (zh) | 2011-08-18 | 2013-04-01 | Incyte Corp | 作為jak抑制劑之環己基氮雜環丁烷衍生物 |
UA111854C2 (uk) | 2011-09-07 | 2016-06-24 | Інсайт Холдінгс Корпорейшн | Способи і проміжні сполуки для отримання інгібіторів jak |
WO2013116291A1 (en) * | 2012-01-30 | 2013-08-08 | Cephalon, Inc. | Imidazo [4, 5 - b] pyridine derivatives as alk and jak modulators for the treatment of proliferative disorders |
TW201406761A (zh) | 2012-05-18 | 2014-02-16 | Incyte Corp | 做爲jak抑制劑之哌啶基環丁基取代之吡咯并吡啶及吡咯并嘧啶衍生物 |
EP2892899B1 (en) * | 2012-09-06 | 2018-03-21 | Bristol-Myers Squibb Company | Imidazopyridazine jak3 inhibitors and their use for the treatment of inflammatory and autoimmune diseases |
WO2014045305A1 (en) | 2012-09-21 | 2014-03-27 | Advinus Therapeutics Limited | Substituted fused tricyclic compounds, compositions and medicinal applications thereof |
AU2013344780B2 (en) | 2012-11-15 | 2018-03-01 | Incyte Holdings Corporation | Sustained-release dosage forms of ruxolitinib |
KR102366356B1 (ko) | 2013-03-06 | 2022-02-23 | 인사이트 홀딩스 코포레이션 | Jak 저해제를 제조하기 위한 방법 및 중간생성물 |
HUE049345T2 (hu) | 2013-08-07 | 2020-09-28 | Incyte Corp | Nyújtott hatóanyag-leadású dózisformák JAK1 inhibitorhoz |
US9498467B2 (en) | 2014-05-30 | 2016-11-22 | Incyte Corporation | Treatment of chronic neutrophilic leukemia (CNL) and atypical chronic myeloid leukemia (aCML) by inhibitors of JAK1 |
WO2017009751A1 (en) | 2015-07-15 | 2017-01-19 | Pfizer Inc. | Pyrimidine derivatives |
CN107513067A (zh) | 2016-06-16 | 2017-12-26 | 北京赛林泰医药技术有限公司 | 含有取代环戊基的吡咯并嘧啶化合物 |
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US3996233A (en) * | 1975-02-10 | 1976-12-07 | E. R. Squibb & Sons, Inc. | Amino derivatives of imidazo[4,5-b]pyridines |
US3953461A (en) * | 1975-03-05 | 1976-04-27 | E. R. Squibb & Sons, Inc. | Amino derivatives of thiazolo[5,4-b]pyridine-6-carboxylic acids and esters |
CA1077484A (en) * | 1975-03-05 | 1980-05-13 | E.R. Squibb And Sons | Amino derivatives of thiazolo (5,4-b) pyridine-6-carboxylic acids and esters |
US6992188B1 (en) * | 1995-12-08 | 2006-01-31 | Pfizer, Inc. | Substituted heterocyclic derivatives |
US6107300A (en) * | 1996-03-27 | 2000-08-22 | Dupont Pharmaceuticals | Arylamino fused pyrimidines |
SE0101675D0 (sv) | 2001-05-11 | 2001-05-11 | Astrazeneca Ab | Novel composition |
SE0301372D0 (sv) * | 2003-05-09 | 2003-05-09 | Astrazeneca Ab | Novel compounds |
-
2003
- 2003-05-09 SE SE0301373A patent/SE0301373D0/sv unknown
-
2004
- 2004-05-06 EP EP07119970A patent/EP1887007A3/en not_active Withdrawn
- 2004-05-06 ES ES04731525T patent/ES2298754T3/es not_active Expired - Lifetime
- 2004-05-06 DK DK04731525T patent/DK1625126T3/da active
- 2004-05-06 PL PL04731525T patent/PL1625126T3/pl unknown
- 2004-05-06 CN CNA200480012617XA patent/CN1784402A/zh active Pending
- 2004-05-06 AU AU2004236144A patent/AU2004236144B2/en not_active Ceased
- 2004-05-06 WO PCT/SE2004/000694 patent/WO2004099204A1/en active IP Right Grant
- 2004-05-06 AT AT04731525T patent/ATE384061T1/de not_active IP Right Cessation
- 2004-05-06 EP EP04731525A patent/EP1625126B1/en not_active Expired - Lifetime
- 2004-05-06 PT PT04731525T patent/PT1625126E/pt unknown
- 2004-05-06 US US10/556,228 patent/US20060287355A1/en not_active Abandoned
- 2004-05-06 JP JP2006508045A patent/JP2006525997A/ja active Pending
- 2004-05-06 MX MXPA05012025A patent/MXPA05012025A/es active IP Right Grant
- 2004-05-06 BR BRPI0410081-6A patent/BRPI0410081A/pt not_active IP Right Cessation
- 2004-05-06 CA CA002524624A patent/CA2524624A1/en not_active Abandoned
- 2004-05-06 DE DE602004011330T patent/DE602004011330T2/de not_active Expired - Fee Related
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2008
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DE602004011330T2 (de) | 2009-01-15 |
EP1625126A1 (en) | 2006-02-15 |
CA2524624A1 (en) | 2004-11-18 |
MXPA05012025A (es) | 2006-02-03 |
CN1784402A (zh) | 2006-06-07 |
EP1887007A2 (en) | 2008-02-13 |
BRPI0410081A (pt) | 2006-05-16 |
WO2004099204A1 (en) | 2004-11-18 |
EP1625126B1 (en) | 2008-01-16 |
CY1107301T1 (el) | 2012-11-21 |
ATE384061T1 (de) | 2008-02-15 |
AU2004236144A1 (en) | 2004-11-18 |
DK1625126T3 (da) | 2008-03-31 |
PL1625126T3 (pl) | 2008-07-31 |
EP1887007A3 (en) | 2008-03-26 |
PT1625126E (pt) | 2008-03-10 |
DE602004011330D1 (de) | 2008-03-06 |
ES2298754T3 (es) | 2008-05-16 |
JP2006525997A (ja) | 2006-11-16 |
US20060287355A1 (en) | 2006-12-21 |
AU2004236144B2 (en) | 2008-02-14 |
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