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RS61897B9 - Pirolo[2,3-d]pirimidinil, pirolo[2,3-b]pirazinil i pirolo[2,3-d]piridinil akrilamidi - Google Patents

Pirolo[2,3-d]pirimidinil, pirolo[2,3-b]pirazinil i pirolo[2,3-d]piridinil akrilamidi

Info

Publication number
RS61897B9
RS61897B9 RS20210657A RSP20210657A RS61897B9 RS 61897 B9 RS61897 B9 RS 61897B9 RS 20210657 A RS20210657 A RS 20210657A RS P20210657 A RSP20210657 A RS P20210657A RS 61897 B9 RS61897 B9 RS 61897B9
Authority
RS
Serbia
Prior art keywords
pyrrolo
pyrazinyl
pyrimidinyl
acrylamides
pyridinyl
Prior art date
Application number
RS20210657A
Other languages
English (en)
Inventor
Matthew Frank Brown
Agustin Casimiro-Garcia
Ye Che
Jotham Wadsworth Coe
Mark Edward Flanagan
Adam Matthew Gilbert
Matthew Merrill Hayward
Jonathan David Langille
Justin Ian Montgomery
Jean-Baptiste Telliez
Atli Thorarensen
Rayomand Jal Unwalla
John I Trujillo
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=52144776&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RS61897(B9) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of RS61897B1 publication Critical patent/RS61897B1/sr
Publication of RS61897B9 publication Critical patent/RS61897B9/sr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
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    • A61K31/33—Heterocyclic compounds
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
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RS20210657A 2013-12-05 2014-11-20 Pirolo[2,3-d]pirimidinil, pirolo[2,3-b]pirazinil i pirolo[2,3-d]piridinil akrilamidi RS61897B9 (sr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361912074P 2013-12-05 2013-12-05
EP17200940.9A EP3318565B1 (en) 2013-12-05 2014-11-20 Pyrrolo[2,3-d]pyrimidinyl, pyrrolo[2,3-b]pyrazinyl and pyrrolo[2,3-d]pyridinyl acrylamides

Publications (2)

Publication Number Publication Date
RS61897B1 RS61897B1 (sr) 2021-06-30
RS61897B9 true RS61897B9 (sr) 2021-09-30

Family

ID=52144776

Family Applications (2)

Application Number Title Priority Date Filing Date
RS20180008A RS56728B1 (sr) 2013-12-05 2014-11-20 Pirolo[2,3-d]pirimidinil, pirolo[2,3-b]pirazinil i pirolo[2,3-d]piridinil akrilamidi
RS20210657A RS61897B9 (sr) 2013-12-05 2014-11-20 Pirolo[2,3-d]pirimidinil, pirolo[2,3-b]pirazinil i pirolo[2,3-d]piridinil akrilamidi

Family Applications Before (1)

Application Number Title Priority Date Filing Date
RS20180008A RS56728B1 (sr) 2013-12-05 2014-11-20 Pirolo[2,3-d]pirimidinil, pirolo[2,3-b]pirazinil i pirolo[2,3-d]piridinil akrilamidi

Country Status (47)

Country Link
US (3) US9617258B2 (sr)
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JP6427599B2 (ja) * 2014-05-19 2018-11-21 チャンスー ヘンルイ メディシン カンパニー，リミテッド チロシンキナーゼ阻害剤としての置換エチニルヘテロ二環式化合物

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