CL2016001216A1 - Acrilamidas de pirrolo[2,3-d]pirimidinilo, pirrolo[2,3-b]pirazinilo y pirrolo[2,3-d]piridinilo. - Google Patents
Acrilamidas de pirrolo[2,3-d]pirimidinilo, pirrolo[2,3-b]pirazinilo y pirrolo[2,3-d]piridinilo.Info
- Publication number
- CL2016001216A1 CL2016001216A1 CL2016001216A CL2016001216A CL2016001216A1 CL 2016001216 A1 CL2016001216 A1 CL 2016001216A1 CL 2016001216 A CL2016001216 A CL 2016001216A CL 2016001216 A CL2016001216 A CL 2016001216A CL 2016001216 A1 CL2016001216 A1 CL 2016001216A1
- Authority
- CL
- Chile
- Prior art keywords
- pyrrolo
- pyrazinyl
- pyrimidinyl
- pirrolo
- acrylamides
- Prior art date
Links
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
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- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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Abstract
<p>ACRILAMIDAS DE PIRROLO[2,3-D]PIRIMIDINILO, PIRROLO[2,3-B]PIRAZINILO Y PIRROLO[2.3-D]PIRIDINILO; COMPOSICIÓN FARMACÉUTICA O VETERINARIA Y USO EN EL TRATAMIENTO DE ENFERMEDADES TALES COMO ARTRITIS REUMATOIDE, MIOSITIS, CROHN, ALZHEIMER, CANCER, ENTRE OTRAS.</p>
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
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US201361912074P | 2013-12-05 | 2013-12-05 |
Publications (1)
Publication Number | Publication Date |
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CL2016001216A1 true CL2016001216A1 (es) | 2017-01-20 |
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CL2016001216A CL2016001216A1 (es) | 2013-12-05 | 2016-05-20 | Acrilamidas de pirrolo[2,3-d]pirimidinilo, pirrolo[2,3-b]pirazinilo y pirrolo[2,3-d]piridinilo. |
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Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US11339167B2 (en) | 2017-12-28 | 2022-05-24 | Daewoong Pharmaceutical Co., Ltd. | Substituted piperidines as kinase inhibitors |
Families Citing this family (84)
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BR112016005881A2 (pt) * | 2013-09-18 | 2017-09-12 | Beijing Hanmi Pharmaceutical Co Ltd | composto, composição farmacêutica e uso do composto |
HUE054560T2 (hu) * | 2013-12-05 | 2021-09-28 | Pfizer | Pirrolo[2,3-d]pirimidinil, pirrolo[2,3-b]pirazinil és pirrolo[2,3-d]piridinil akrilamidok |
WO2016000615A1 (en) * | 2014-07-02 | 2016-01-07 | Sunshine Lake Pharma Co., Ltd. | Heteroaryl compounds and pharmaceutical applications thereof |
CA2958966C (en) | 2014-08-28 | 2020-01-14 | Asceneuron Sa | Substituted cyclic amines as glucosidase inhibitors |
CN105712998B (zh) * | 2014-12-05 | 2019-12-13 | 上海润诺生物科技有限公司 | 氮杂吲哚类衍生物、其制备方法及其在医药上的应用 |
US9695200B2 (en) | 2015-01-23 | 2017-07-04 | Confluence Life Sciences, Inc. | Heterocyclic ITK inhibitors for treating inflammation and cancer |
CN105837574B (zh) * | 2015-02-02 | 2018-03-02 | 四川大学 | N‑(3‑哌啶基)‑芳香胺衍生物及其制备方法和用途 |
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Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US11339167B2 (en) | 2017-12-28 | 2022-05-24 | Daewoong Pharmaceutical Co., Ltd. | Substituted piperidines as kinase inhibitors |
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