PT72090B - Process for preparing antiallergic and antiulcer 1-oxo-1h-thiazolo<3,2-a>pyrimidine-2-carboxamides - Google Patents

Process for preparing antiallergic and antiulcer 1-oxo-1h-thiazolo<3,2-a>pyrimidine-2-carboxamides

Info

Publication number: PT72090B
Authority: PT; Portugal
Prior art keywords: antiulcer; thiazolo; carboxamides; pyrimidine; oxo
Prior art date: 1979-11-23

Application number

PT72090A

Other languages

Portuguese (pt)

Other versions

PT72090A (en

Inventor

Saul Bernard Kadin

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1979-11-23

Filing date

1980-11-21

Publication date

1981-09-29

1980-11-21 Application filed by Pfizer filed Critical Pfizer

1980-12-01 Publication of PT72090A publication Critical patent/PT72090A/en

1981-09-29 Publication of PT72090B publication Critical patent/PT72090B/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/40—Unsubstituted amino or imino radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pulmonology (AREA)
Diabetes (AREA)
Hematology (AREA)
Immunology (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Dermatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Thiazole And Isothizaole Compounds (AREA)

PT72090A 1979-11-23 1980-11-21 Process for preparing antiallergic and antiulcer 1-oxo-1h-thiazolo<3,2-a>pyrimidine-2-carboxamides PT72090B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US9663179A	1979-11-23	1979-11-23

Publications (2)

Publication Number	Publication Date
PT72090A PT72090A (en)	1980-12-01
PT72090B true PT72090B (en)	1981-09-29

Family

ID=22258306

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT72090A PT72090B (en)	1979-11-23	1980-11-21	Process for preparing antiallergic and antiulcer 1-oxo-1h-thiazolo<3,2-a>pyrimidine-2-carboxamides

Country Status (35)

Country	Link
JP (1)	JPS5687586A (en)
KR (1)	KR830004322A (en)
AR (2)	AR228859A1 (en)
AT (1)	AT380883B (en)
AU (1)	AU520995B2 (en)
BE (1)	BE886319A (en)
CA (1)	CA1143731A (en)
CH (1)	CH649299A5 (en)
CS (1)	CS241476B2 (en)
DD (1)	DD154608A5 (en)
DE (2)	DE3050491C2 (en)
DK (1)	DK151811C (en)
EG (1)	EG14929A (en)
ES (1)	ES497066A0 (en)
FI (1)	FI67706C (en)
FR (1)	FR2470132A1 (en)
GB (1)	GB2063862B (en)
GR (1)	GR72132B (en)
GT (1)	GT198066458A (en)
HU (1)	HU179091B (en)
IE (1)	IE50404B1 (en)
IL (1)	IL61535A (en)
IN (1)	IN154926B (en)
IT (1)	IT1209373B (en)
LU (1)	LU82950A1 (en)
NL (1)	NL182565C (en)
NO (1)	NO803521L (en)
NZ (1)	NZ195596A (en)
PH (1)	PH16666A (en)
PL (1)	PL132354B1 (en)
PT (1)	PT72090B (en)
SE (1)	SE448732B (en)
SU (1)	SU1042620A3 (en)
YU (1)	YU41953B (en)
ZA (1)	ZA807293B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8300728D0 (en) *	1983-01-12	1983-02-16	Erba Farmitalia	Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives
US4457932A (en) *	1983-07-22	1984-07-03	Bristol-Myers Company	Anti-ulcer agents
GB8422916D0 (en) *	1984-09-11	1984-10-17	May & Baker Ltd	Compositions of matter
JP2690742B2 (en) *	1987-03-30	1997-12-17	第一製薬株式会社	Heterocyclic amine derivative
ES2087072T3 (en) *	1988-03-28	1996-07-16	Janssen Pharmaceutica Nv	AGENTS TO PRESERVE OR RESTORE SKIN HEALTH.
TWI500623B (en) *	2009-10-13	2015-09-21	Torrent Pharmaceuticals Ltd	Novel fused thiazolo and oxazolo pyrimidinones

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1331059A (en)	1971-04-19	1973-09-19	Lilly Industries Ltd	Pyrimidotriazinone compounds
US4041163A (en) *	1976-03-29	1977-08-09	Pfizer Inc.	N-(5-Tetrazolyl)-4-oxo-4H-pyrimido(2,1-b)benzothiazole-3-carboxamide antiallergy agents
DE2810863A1 (en) *	1978-03-13	1979-09-27	Boehringer Mannheim Gmbh	1-OXO-1H-PYRIMIDO ANGLE CLAMP ON 6.1-B ANGLE CLAMP ON BENZTHIAZOLE DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF
US4223031A (en) *	1978-05-05	1980-09-16	Mead Johnson & Company	Azolopyrimidinones

1980
- 1980-09-30 DK DK413180A patent/DK151811C/en not_active IP Right Cessation
- 1980-10-15 IN IN760/DEL/80A patent/IN154926B/en unknown
- 1980-11-17 SU SU803212053A patent/SU1042620A3/en active
- 1980-11-18 AR AR283276A patent/AR228859A1/en active
- 1980-11-18 GB GB8036904A patent/GB2063862B/en not_active Expired
- 1980-11-18 CS CS807820A patent/CS241476B2/en unknown
- 1980-11-18 HU HU80802755A patent/HU179091B/en not_active IP Right Cessation
- 1980-11-19 CH CH8567/80A patent/CH649299A5/en not_active IP Right Cessation
- 1980-11-19 EG EG723/80A patent/EG14929A/en active
- 1980-11-20 GR GR63413A patent/GR72132B/el unknown
- 1980-11-20 YU YU2950/80A patent/YU41953B/en unknown
- 1980-11-20 NZ NZ195596A patent/NZ195596A/en unknown
- 1980-11-21 AT AT0570780A patent/AT380883B/en not_active IP Right Cessation
- 1980-11-21 CA CA000365258A patent/CA1143731A/en not_active Expired
- 1980-11-21 FR FR8024822A patent/FR2470132A1/en active Granted
- 1980-11-21 JP JP16450280A patent/JPS5687586A/en active Granted
- 1980-11-21 IL IL61535A patent/IL61535A/en unknown
- 1980-11-21 DE DE3050491A patent/DE3050491C2/en not_active Expired
- 1980-11-21 FI FI803628A patent/FI67706C/en not_active IP Right Cessation
- 1980-11-21 PH PH24891A patent/PH16666A/en unknown
- 1980-11-21 SE SE8008189A patent/SE448732B/en not_active IP Right Cessation
- 1980-11-21 IE IE2418/80A patent/IE50404B1/en unknown
- 1980-11-21 DE DE3043979A patent/DE3043979C2/en not_active Expired
- 1980-11-21 DD DD80225391A patent/DD154608A5/en not_active IP Right Cessation
- 1980-11-21 IT IT8026176A patent/IT1209373B/en active
- 1980-11-21 LU LU82950A patent/LU82950A1/en unknown
- 1980-11-21 GT GT198066458A patent/GT198066458A/en unknown
- 1980-11-21 AU AU64595/80A patent/AU520995B2/en not_active Ceased
- 1980-11-21 PT PT72090A patent/PT72090B/en not_active IP Right Cessation
- 1980-11-21 ZA ZA00807293A patent/ZA807293B/en unknown
- 1980-11-21 NO NO803521A patent/NO803521L/en unknown
- 1980-11-21 NL NLAANVRAGE8006362,A patent/NL182565C/en not_active IP Right Cessation
- 1980-11-21 ES ES497066A patent/ES497066A0/en active Granted
- 1980-11-22 PL PL1980228008A patent/PL132354B1/en unknown
- 1980-11-22 KR KR1019800004474A patent/KR830004322A/en unknown
- 1980-11-24 BE BE0/202915A patent/BE886319A/en not_active IP Right Cessation
1982
- 1982-09-13 AR AR290628A patent/AR231296A1/en active

Also Published As

Publication number	Publication date
DD154608A5 (en)	1982-04-07
PL132354B1 (en)	1985-02-28
AU520995B2 (en)	1982-03-11
GR72132B (en)	1983-09-19
NO803521L (en)	1981-05-25
IT1209373B (en)	1989-07-16
BE886319A (en)	1981-05-25
DE3050491C2 (en)	1985-10-10
NL8006362A (en)	1981-06-16
NL182565C (en)	1988-04-05
AT380883B (en)	1986-07-25
FR2470132B1 (en)	1983-07-29
EG14929A (en)	1989-01-30
IL61535A0 (en)	1980-12-31
ES8203363A1 (en)	1982-04-01
NL182565B (en)	1987-11-02
ATA570780A (en)	1985-12-15
DK151811C (en)	1988-06-06
FI803628L (en)	1981-05-24
KR830004322A (en)	1983-07-09
ES497066A0 (en)	1982-04-01
GB2063862B (en)	1983-06-22
LU82950A1 (en)	1981-06-04
CS782080A2 (en)	1985-06-13
PH16666A (en)	1983-12-13
JPS617432B2 (en)	1986-03-06
IL61535A (en)	1984-06-29
SE8008189L (en)	1981-05-24
YU295080A (en)	1983-06-30
IE802418L (en)	1981-05-23
AU6459580A (en)	1981-05-28
DE3043979C2 (en)	1986-08-21
FI67706C (en)	1985-05-10
AR231296A1 (en)	1984-10-31
CA1143731A (en)	1983-03-29
AR228859A1 (en)	1983-04-29
DE3043979A1 (en)	1981-09-03
PT72090A (en)	1980-12-01
NZ195596A (en)	1984-05-31
IT8026176A0 (en)	1980-11-21
PL228008A1 (en)	1981-12-11
DK413180A (en)	1981-05-24
GB2063862A (en)	1981-06-10
JPS5687586A (en)	1981-07-16
HU179091B (en)	1982-08-28
IN154926B (en)	1984-12-22
SU1042620A3 (en)	1983-09-15
GT198066458A (en)	1982-05-15
YU41953B (en)	1988-02-29
FR2470132A1 (en)	1981-05-29
ZA807293B (en)	1981-12-30
SE448732B (en)	1987-03-16
IE50404B1 (en)	1986-04-16
CS241476B2 (en)	1986-03-13
DK151811B (en)	1988-01-04
FI67706B (en)	1985-01-31
CH649299A5 (en)	1985-05-15

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PL237052A1 (en)	1983-06-20	Process for preparing novel imidazo-/1,2-a/-pyrimidines
GB2011395B (en)	1982-03-03	1,8 naphthyridine compounds and process for preparing the same
DE3371509D1 (en)	1987-06-19	Clavulone derivatives, process for preparing the same, and use of said compounds
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YU298180A (en)	1983-02-28	Process for preparing 5,10-dihydroimidazo-2,1-quinazoline
ZA804079B (en)	1981-07-29	Dihydronicotinic acid derivatives and process for the preparation thereof

Legal Events

Date	Code	Title	Description
1995-05-31	MM3A	Annulment or lapse	Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 19940330

Date

Code

Title

Description

1995-05-31

MM3A

Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19940330