IL61535A - 5-oxo-5h-thiazolo(3,2-a)pyrimidine-6-carboxylic acids and n-(5-tetrazolyl)-carboxamide derivatives thereof - Google Patents

5-oxo-5h-thiazolo(3,2-a)pyrimidine-6-carboxylic acids and n-(5-tetrazolyl)-carboxamide derivatives thereof

Info

Publication number: IL61535A
Authority: IL; Israel
Prior art keywords: thiazolo; tetrazolyl; pyrimidine; oxo; carboxylic acids
Prior art date: 1979-11-23

Application number

IL61535A

Other versions

IL61535A0 (en

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1979-11-23

Filing date

1980-11-21

Publication date

1984-06-29

1980-11-21 Application filed by Pfizer filed Critical Pfizer

1980-12-31 Publication of IL61535A0 publication Critical patent/IL61535A0/en

1984-06-29 Publication of IL61535A publication Critical patent/IL61535A/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/40—Unsubstituted amino or imino radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pulmonology (AREA)
Diabetes (AREA)
Hematology (AREA)
Immunology (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Dermatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Thiazole And Isothizaole Compounds (AREA)

IL61535A 1979-11-23 1980-11-21 5-oxo-5h-thiazolo(3,2-a)pyrimidine-6-carboxylic acids and n-(5-tetrazolyl)-carboxamide derivatives thereof IL61535A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US9663179A	1979-11-23	1979-11-23

Publications (2)

Publication Number	Publication Date
IL61535A0 IL61535A0 (en)	1980-12-31
IL61535A true IL61535A (en)	1984-06-29

Family

ID=22258306

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL61535A IL61535A (en)	1979-11-23	1980-11-21	5-oxo-5h-thiazolo(3,2-a)pyrimidine-6-carboxylic acids and n-(5-tetrazolyl)-carboxamide derivatives thereof

Country Status (35)

Country	Link
JP (1)	JPS5687586A (en)
KR (1)	KR830004322A (en)
AR (2)	AR228859A1 (en)
AT (1)	AT380883B (en)
AU (1)	AU520995B2 (en)
BE (1)	BE886319A (en)
CA (1)	CA1143731A (en)
CH (1)	CH649299A5 (en)
CS (1)	CS241476B2 (en)
DD (1)	DD154608A5 (en)
DE (2)	DE3050491C2 (en)
DK (1)	DK151811C (en)
EG (1)	EG14929A (en)
ES (1)	ES497066A0 (en)
FI (1)	FI67706C (en)
FR (1)	FR2470132A1 (en)
GB (1)	GB2063862B (en)
GR (1)	GR72132B (en)
GT (1)	GT198066458A (en)
HU (1)	HU179091B (en)
IE (1)	IE50404B1 (en)
IL (1)	IL61535A (en)
IN (1)	IN154926B (en)
IT (1)	IT1209373B (en)
LU (1)	LU82950A1 (en)
NL (1)	NL182565C (en)
NO (1)	NO803521L (en)
NZ (1)	NZ195596A (en)
PH (1)	PH16666A (en)
PL (1)	PL132354B1 (en)
PT (1)	PT72090B (en)
SE (1)	SE448732B (en)
SU (1)	SU1042620A3 (en)
YU (1)	YU41953B (en)
ZA (1)	ZA807293B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8300728D0 (en) *	1983-01-12	1983-02-16	Erba Farmitalia	Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives
US4457932A (en) *	1983-07-22	1984-07-03	Bristol-Myers Company	Anti-ulcer agents
GB8422916D0 (en) *	1984-09-11	1984-10-17	May & Baker Ltd	Compositions of matter
JP2690742B2 (en) *	1987-03-30	1997-12-17	第一製薬株式会社	Heterocyclic amine derivative
ES2087072T3 (en) *	1988-03-28	1996-07-16	Janssen Pharmaceutica Nv	AGENTS TO PRESERVE OR RESTORE SKIN HEALTH.
TWI500623B (en) *	2009-10-13	2015-09-21	Torrent Pharmaceuticals Ltd	Novel fused thiazolo and oxazolo pyrimidinones

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1331059A (en)	1971-04-19	1973-09-19	Lilly Industries Ltd	Pyrimidotriazinone compounds
US4041163A (en) *	1976-03-29	1977-08-09	Pfizer Inc.	N-(5-Tetrazolyl)-4-oxo-4H-pyrimido(2,1-b)benzothiazole-3-carboxamide antiallergy agents
DE2810863A1 (en) *	1978-03-13	1979-09-27	Boehringer Mannheim Gmbh	1-OXO-1H-PYRIMIDO ANGLE CLAMP ON 6.1-B ANGLE CLAMP ON BENZTHIAZOLE DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF
US4223031A (en) *	1978-05-05	1980-09-16	Mead Johnson & Company	Azolopyrimidinones

1980
- 1980-09-30 DK DK413180A patent/DK151811C/en not_active IP Right Cessation
- 1980-10-15 IN IN760/DEL/80A patent/IN154926B/en unknown
- 1980-11-17 SU SU803212053A patent/SU1042620A3/en active
- 1980-11-18 AR AR283276A patent/AR228859A1/en active
- 1980-11-18 GB GB8036904A patent/GB2063862B/en not_active Expired
- 1980-11-18 CS CS807820A patent/CS241476B2/en unknown
- 1980-11-18 HU HU80802755A patent/HU179091B/en not_active IP Right Cessation
- 1980-11-19 CH CH8567/80A patent/CH649299A5/en not_active IP Right Cessation
- 1980-11-19 EG EG723/80A patent/EG14929A/en active
- 1980-11-20 GR GR63413A patent/GR72132B/el unknown
- 1980-11-20 YU YU2950/80A patent/YU41953B/en unknown
- 1980-11-20 NZ NZ195596A patent/NZ195596A/en unknown
- 1980-11-21 AT AT0570780A patent/AT380883B/en not_active IP Right Cessation
- 1980-11-21 CA CA000365258A patent/CA1143731A/en not_active Expired
- 1980-11-21 FR FR8024822A patent/FR2470132A1/en active Granted
- 1980-11-21 JP JP16450280A patent/JPS5687586A/en active Granted
- 1980-11-21 IL IL61535A patent/IL61535A/en unknown
- 1980-11-21 DE DE3050491A patent/DE3050491C2/en not_active Expired
- 1980-11-21 FI FI803628A patent/FI67706C/en not_active IP Right Cessation
- 1980-11-21 PH PH24891A patent/PH16666A/en unknown
- 1980-11-21 SE SE8008189A patent/SE448732B/en not_active IP Right Cessation
- 1980-11-21 IE IE2418/80A patent/IE50404B1/en unknown
- 1980-11-21 DE DE3043979A patent/DE3043979C2/en not_active Expired
- 1980-11-21 DD DD80225391A patent/DD154608A5/en not_active IP Right Cessation
- 1980-11-21 IT IT8026176A patent/IT1209373B/en active
- 1980-11-21 LU LU82950A patent/LU82950A1/en unknown
- 1980-11-21 GT GT198066458A patent/GT198066458A/en unknown
- 1980-11-21 AU AU64595/80A patent/AU520995B2/en not_active Ceased
- 1980-11-21 PT PT72090A patent/PT72090B/en not_active IP Right Cessation
- 1980-11-21 ZA ZA00807293A patent/ZA807293B/en unknown
- 1980-11-21 NO NO803521A patent/NO803521L/en unknown
- 1980-11-21 NL NLAANVRAGE8006362,A patent/NL182565C/en not_active IP Right Cessation
- 1980-11-21 ES ES497066A patent/ES497066A0/en active Granted
- 1980-11-22 PL PL1980228008A patent/PL132354B1/en unknown
- 1980-11-22 KR KR1019800004474A patent/KR830004322A/en unknown
- 1980-11-24 BE BE0/202915A patent/BE886319A/en not_active IP Right Cessation
1982
- 1982-09-13 AR AR290628A patent/AR231296A1/en active

Also Published As

Publication number	Publication date
DD154608A5 (en)	1982-04-07
PL132354B1 (en)	1985-02-28
AU520995B2 (en)	1982-03-11
GR72132B (en)	1983-09-19
PT72090B (en)	1981-09-29
NO803521L (en)	1981-05-25
IT1209373B (en)	1989-07-16
BE886319A (en)	1981-05-25
DE3050491C2 (en)	1985-10-10
NL8006362A (en)	1981-06-16
NL182565C (en)	1988-04-05
AT380883B (en)	1986-07-25
FR2470132B1 (en)	1983-07-29
EG14929A (en)	1989-01-30
IL61535A0 (en)	1980-12-31
ES8203363A1 (en)	1982-04-01
NL182565B (en)	1987-11-02
ATA570780A (en)	1985-12-15
DK151811C (en)	1988-06-06
FI803628L (en)	1981-05-24
KR830004322A (en)	1983-07-09
ES497066A0 (en)	1982-04-01
GB2063862B (en)	1983-06-22
LU82950A1 (en)	1981-06-04
CS782080A2 (en)	1985-06-13
PH16666A (en)	1983-12-13
JPS617432B2 (en)	1986-03-06
SE8008189L (en)	1981-05-24
YU295080A (en)	1983-06-30
IE802418L (en)	1981-05-23
AU6459580A (en)	1981-05-28
DE3043979C2 (en)	1986-08-21
FI67706C (en)	1985-05-10
AR231296A1 (en)	1984-10-31
CA1143731A (en)	1983-03-29
AR228859A1 (en)	1983-04-29
DE3043979A1 (en)	1981-09-03
PT72090A (en)	1980-12-01
NZ195596A (en)	1984-05-31
IT8026176A0 (en)	1980-11-21
PL228008A1 (en)	1981-12-11
DK413180A (en)	1981-05-24
GB2063862A (en)	1981-06-10
JPS5687586A (en)	1981-07-16
HU179091B (en)	1982-08-28
IN154926B (en)	1984-12-22
SU1042620A3 (en)	1983-09-15
GT198066458A (en)	1982-05-15
YU41953B (en)	1988-02-29
FR2470132A1 (en)	1981-05-29
ZA807293B (en)	1981-12-30
SE448732B (en)	1987-03-16
IE50404B1 (en)	1986-04-16
CS241476B2 (en)	1986-03-13
DK151811B (en)	1988-01-04
FI67706B (en)	1985-01-31
CH649299A5 (en)	1985-05-15

Publication	Publication Date	Title
DE3072064D1 (en)	1988-02-11	Amino acid derivatives and their preparation
ZA806977B (en)	1981-10-28	7-acylamino-3-vinylcephalosporanic acid derivatives and processes for the preparation thereof
GB2066812B (en)	1983-07-27	5'-acyl-uridine derivatives and processes for the preparation thereof
PH16228A (en)	1983-08-09	Triazolo pyridazine derivatives,pharmaceutical composition containing the same and their use
ZA802155B (en)	1981-05-27	Penem-3-carboxylic acid derivatives, their preparation and use
IL58779A0 (en)	1980-02-29	1,2-dihydro-3h-pyrrolo(1,2-a)pyrrole-1-carboxylates and their preparation
IL69140A0 (en)	1983-11-30	2,3,6,7-tetrahydro-5h-thiazolo(3,2-a)pyrimidine derivatives,their preparation and their use as herbicides
IL86028A0 (en)	1988-09-30	Novel pyrrolidine-2-(1,3-dicarbonyl)derivatives,their preparation,agents containing them,and their use
ZA868752B (en)	1988-07-27	6,7,8,9-tetrahydro-10-methylpyrido(1,2-a)indol-9-amines and derivatives thereof
NZ193579A (en)	1982-09-07	2-trans-(2-arylethen-1-yl)-4-oxo-4h-pyrido (1,2-a)-pyrimid-7-ylcarboxylic acid derivatives
IL61535A (en)	1984-06-29	5-oxo-5h-thiazolo(3,2-a)pyrimidine-6-carboxylic acids and n-(5-tetrazolyl)-carboxamide derivatives thereof
GB2072660B (en)	1983-10-26	Indolo (2,3-a) quinolisine ester derivatives and preparation thereof
GB2048254B (en)	1983-05-25	19,20 -didehydro-19-hydroxy and 19-oxo-prostaglandin derivatives
IL61179A0 (en)	1980-11-30	2-amino-4-substituted-5-thiazolecarboxylic acids and their derivatives
AU513385B2 (en)	1980-11-27	5-furoyl and 5-thenoyl pyrrolo[1,2-a] pyrrole-carboxylic acid derivatives
JPS55154974A (en)	1980-12-02	Pyrazolo155c*quinazoline derivatives and their manufacture
GB1551166A (en)	1979-08-22	Pyrazolo (1,5-a)quinoxaline-3-carboxylic acid and derivatives thereof
GB2119374B (en)	1986-02-05	1,2,4-triazol-1-yl-propionitrile derivatives their preparation and use
IL60831A (en)	1985-04-30	1,2,4-benzotriazinylamino-phenoxyalkanoic acid derivatives,their preparation and their use as herbicides
DE3062022D1 (en)	1983-03-24	Dihydronicotinic acid derivatives, their preparation and use
ZA801759B (en)	1981-03-25	6-substituted-arylpyrido (2,3-d)pyrimidin-7-amines and derivatives
HUT49607A (en)	1989-10-30	Herbicides comprising n-phenyl-tetrahydrophtalimide derivatives and process for producing the active ingredients
ZA802323B (en)	1981-04-29	Clavulanic acid derivatives,their preparation and use
JPS55129286A (en)	1980-10-06	Pyrido344e**asstriazine derivatives and their manufacture
PH16300A (en)	1983-09-05	Notrothiazoline derivatives and their use as schistosonicidal agents