PH23392A - Dihydrobenzofuran-and chroman-carboxamide derivatives and their use as neuroleptics - Google Patents

Dihydrobenzofuran-and chroman-carboxamide derivatives and their use as neuroleptics

Info

Publication number: PH23392A
Authority: PH; Philippines
Prior art keywords: neuroleptics; dihydrobenzofuran; chroman; alkyl; image
Prior art date: 1986-01-30

Application number

PH34786A

Other languages

English (en)

Inventor

Jacqueline Franceschini

Josette Margarit

Original Assignee

Delagrange Lab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-01-30

Filing date

1987-01-29

Publication date

1989-07-26

1987-01-29 Application filed by Delagrange Lab filed Critical Delagrange Lab

1989-07-26 Publication of PH23392A publication Critical patent/PH23392A/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
- C07D407/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
- C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Biomedical Technology (AREA)
Public Health (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Pyrane Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Medicinal Preparation (AREA)
Hydrogenated Pyridines (AREA)
Furan Compounds (AREA)
Peptides Or Proteins (AREA)
Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
Polyamides (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

PH34786A 1986-01-30 1987-01-29 Dihydrobenzofuran-and chroman-carboxamide derivatives and their use as neuroleptics PH23392A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR8601279A FR2593504B1 (fr)	1986-01-30	1986-01-30	Nouveaux derives de dihydrobenzofuranne - et de chromane - carboxamides, leurs procedes de preparation et leur utilisation comme neuroleptiques

Publications (1)

Publication Number	Publication Date
PH23392A true PH23392A (en)	1989-07-26

Family

ID=9331629

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PH34786A PH23392A (en)	1986-01-30	1987-01-29	Dihydrobenzofuran-and chroman-carboxamide derivatives and their use as neuroleptics

Country Status (40)

Country	Link
US (1)	US5006570A (xx)
EP (1)	EP0231139B1 (xx)
JP (1)	JPS62277376A (xx)
KR (1)	KR870007160A (xx)
CN (2)	CN1016420B (xx)
AT (1)	ATE70063T1 (xx)
AU (1)	AU593605B2 (xx)
BE (1)	BE1000164A5 (xx)
BG (1)	BG46600A3 (xx)
CA (1)	CA1300161C (xx)
CH (1)	CH670827A5 (xx)
CS (2)	CS264288B2 (xx)
DD (1)	DD260065A5 (xx)
DE (2)	DE3702005A1 (xx)
DK (1)	DK46987A (xx)
ES (2)	ES2003671A6 (xx)
FI (1)	FI870347A (xx)
FR (1)	FR2593504B1 (xx)
GB (1)	GB2187188B (xx)
GR (2)	GR870134B (xx)
HU (1)	HU206107B (xx)
IE (1)	IE870128L (xx)
IL (1)	IL81299A (xx)
IN (2)	IN164389B (xx)
IS (1)	IS1446B6 (xx)
IT (1)	IT1205729B (xx)
LU (1)	LU86747A1 (xx)
MA (1)	MA20861A1 (xx)
NO (1)	NO168582C (xx)
NZ (1)	NZ219068A (xx)
OA (1)	OA08472A (xx)
PH (1)	PH23392A (xx)
PL (2)	PL152491B1 (xx)
PT (1)	PT84224B (xx)
SU (2)	SU1609451A3 (xx)
TN (1)	TNSN87012A1 (xx)
YU (1)	YU46185B (xx)
ZA (1)	ZA87552B (xx)
ZM (1)	ZM987A1 (xx)
ZW (1)	ZW1387A1 (xx)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2611713B1 (fr) *	1987-02-27	1990-11-30	Adir	Nouveaux derives de l'acide (dihydro-2,3 oxo-2 benzofurannyl-3)-2 acetique, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent
FR2611715B1 (fr) *	1987-02-27	1989-05-12	Adir	Nouveaux acetamides derives de la dihydro-2,3 phenyl-3 benzofurannone-2, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent
US5374637A (en) *	1989-03-22	1994-12-20	Janssen Pharmaceutica N.V.	N-(3-hydroxy-4-piperidinyl)(dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives
JP2726306B2 (ja) *	1989-04-14	1998-03-11	本田技研工業株式会社	車両の前後輪操舵装置
US5122361A (en) *	1989-04-17	1992-06-16	Trustees Of The University Of Pennsylvania	Dopamine receptor ligands and imaging agents
EP0412939A3 (en) *	1989-08-11	1991-09-04	Ciba-Geigy Ag	Certain benzopyran and benzothiopyran derivatives
US5420151A (en) *	1989-12-22	1995-05-30	Aktiebolaget Astra	Chroman derivatives
US5616610A (en) *	1989-12-22	1997-04-01	Astra Aktiebolag	(R)-5-carbamoyl-8-fluoro-3-N,N-disubstituted-amino-3,4-dihydro-2H-1-benzopyrans
GB9005014D0 (en) *	1990-03-06	1990-05-02	Janssen Pharmaceutica Nv	N.(4.piperidinyl)(dihydrobenzofuran or dihydro.2h.benzopyran)carboxamide derivatives
WO1991017144A1 (en) *	1990-05-02	1991-11-14	Yoshitomi Pharmaceutical Industries, Ltd.	Amide compound, pharmaceutical use thereof and novel 1-substituted pyrrolidinemethyl-amines
US5114947A (en) *	1990-12-27	1992-05-19	Erbamont Inc.	Method for alleviating anxiety using benzobicyclic carboxamides
MA22647A1 (fr) *	1991-09-14	1993-04-01	Smithkline Beecham Plc	Procede de preparation d'un ester ou d'un amide d'un nouveau produit .
AU667874B2 (en) *	1992-02-06	1996-04-18	Smithkline Beecham Plc	Benzopyran, benzothiopyran and benzofuran derivatives as 5-HT4 antagonists
JPH08502273A (ja) *	1992-10-13	1996-03-12	スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー	５−ｈｔ▲下４▼レセプターアンタゴニスト用複素環式エステルまたはアミド
US6127379A (en) *	1993-02-01	2000-10-03	Smithkline Beecham P.L.C.	Benzopyran, benzothiopyran and benzofuran derivatives as 5-HT4 antagonists
JP2999669B2 (ja) *	1993-08-24	2000-01-17	株式会社三和化学研究所	ベンゾ［ｂ］フランカルボキサミド誘導体、その製法及び用途
JPH0820586A (ja)	1994-07-05	1996-01-23	Sanwa Kagaku Kenkyusho Co Ltd	１−アザビシクロ［３．３．０］オクタン誘導体、その塩及び製法並びに用途
JPH0873463A (ja) *	1994-07-05	1996-03-19	Sanwa Kagaku Kenkyusho Co Ltd	ベンゾピランカルボキサミド誘導体、その塩及び製法並びに用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO1984003281A1 (en) *	1983-02-19	1984-08-30	Beecham Group Plc	Azabicycloalkyl benzamide and anilide derivatives
JPS59186969A (ja) *	1983-04-08	1984-10-23	Yoshitomi Pharmaceut Ind Ltd	ベンゾフラン−およびベンゾピランカルボキサミド誘導体
CA1297877C (en) *	1983-12-22	1992-03-24	Daniel Lednicer	Benzofurancarboxamides useful as antiemetic or antipsychotic agents
JPS63139180A (ja) *	1986-12-02	1988-06-10	Tanabe Seiyaku Co Ltd	カルボン酸誘導体

1986
- 1986-01-30 FR FR8601279A patent/FR2593504B1/fr not_active Expired
1987
- 1987-01-16 NO NO870199A patent/NO168582C/no unknown
- 1987-01-19 IL IL81299A patent/IL81299A/xx not_active IP Right Cessation
- 1987-01-20 IE IE870128A patent/IE870128L/xx unknown
- 1987-01-21 IN IN43/MAS/87A patent/IN164389B/en unknown
- 1987-01-21 IS IS3189A patent/IS1446B6/is unknown
- 1987-01-21 AU AU67855/87A patent/AU593605B2/en not_active Ceased
- 1987-01-23 DE DE19873702005 patent/DE3702005A1/de not_active Withdrawn
- 1987-01-23 ZW ZW13/87A patent/ZW1387A1/xx unknown
- 1987-01-26 ZA ZA87552A patent/ZA87552B/xx unknown
- 1987-01-27 NZ NZ219068A patent/NZ219068A/en unknown
- 1987-01-27 GR GR870134A patent/GR870134B/el unknown
- 1987-01-27 FI FI870347A patent/FI870347A/fi not_active Application Discontinuation
- 1987-01-27 MA MA21095A patent/MA20861A1/fr unknown
- 1987-01-27 YU YU11387A patent/YU46185B/sh unknown
- 1987-01-28 GB GB8701870A patent/GB2187188B/en not_active Expired
- 1987-01-28 CN CN87100978A patent/CN1016420B/zh not_active Expired
- 1987-01-28 TN TNTNSN87012A patent/TNSN87012A1/fr unknown
- 1987-01-28 BG BG078228A patent/BG46600A3/xx active Active
- 1987-01-28 LU LU86747A patent/LU86747A1/fr unknown
- 1987-01-28 CA CA000528418A patent/CA1300161C/fr not_active Expired - Lifetime
- 1987-01-28 KR KR870000673A patent/KR870007160A/ko not_active Application Discontinuation
- 1987-01-29 CH CH300/87A patent/CH670827A5/fr not_active IP Right Cessation
- 1987-01-29 ES ES8700216A patent/ES2003671A6/es not_active Expired
- 1987-01-29 DK DK046987A patent/DK46987A/da unknown
- 1987-01-29 PT PT84224A patent/PT84224B/pt not_active IP Right Cessation
- 1987-01-29 CS CS87578A patent/CS264288B2/cs unknown
- 1987-01-29 AT AT87400194T patent/ATE70063T1/de not_active IP Right Cessation
- 1987-01-29 EP EP87400194A patent/EP0231139B1/fr not_active Expired - Lifetime
- 1987-01-29 PH PH34786A patent/PH23392A/en unknown
- 1987-01-29 SU SU874028919A patent/SU1609451A3/ru active
- 1987-01-29 DE DE8787400194T patent/DE3774888D1/de not_active Expired - Lifetime
- 1987-01-29 DD DD87299591A patent/DD260065A5/de unknown
- 1987-01-29 IT IT47583/87A patent/IT1205729B/it active
- 1987-01-29 HU HU87283A patent/HU206107B/hu not_active IP Right Cessation
- 1987-01-29 ZM ZM9/87A patent/ZM987A1/xx unknown
- 1987-01-29 ES ES198787400194T patent/ES2038679T3/es not_active Expired - Lifetime
- 1987-01-29 OA OA59056A patent/OA08472A/xx unknown
- 1987-01-30 US US07/008,916 patent/US5006570A/en not_active Expired - Fee Related
- 1987-01-30 JP JP62021649A patent/JPS62277376A/ja active Pending
- 1987-01-30 PL PL1987272298A patent/PL152491B1/pl unknown
- 1987-01-30 BE BE8700065A patent/BE1000164A5/fr not_active Expired
- 1987-01-30 PL PL1987263885A patent/PL152404B1/pl unknown
1988
- 1988-01-19 CS CS88362A patent/CS264300B2/cs unknown
- 1988-05-23 IN IN343/MAS/88A patent/IN167060B/en unknown
- 1988-06-28 SU SU884355973A patent/SU1607688A3/ru active
1992
- 1992-01-04 CN CN92100139A patent/CN1062144A/zh active Pending
- 1992-01-27 GR GR920400082T patent/GR3003653T3/el unknown

Also Published As

Publication number	Publication date
GR870134B (en)	1987-05-28
CH670827A5 (xx)	1989-07-14
SU1609451A3 (ru)	1990-11-23
GB2187188A (en)	1987-09-03
PT84224A (fr)	1987-02-01
CS264288B2 (en)	1989-06-13
ZW1387A1 (en)	1987-10-28
EP0231139B1 (fr)	1991-12-04
IT1205729B (it)	1989-03-31
KR870007160A (ko)	1987-08-17
DE3774888D1 (de)	1992-01-16
BG46600A3 (en)	1990-01-15
ZM987A1 (en)	1987-09-30
HUT47093A (en)	1989-01-30
DD260065A5 (de)	1988-09-14
EP0231139A2 (fr)	1987-08-05
EP0231139A3 (en)	1988-04-27
ATE70063T1 (de)	1991-12-15
CA1300161C (fr)	1992-05-05
HU206107B (en)	1992-08-28
ES2003671A6 (es)	1988-11-01
DK46987D0 (da)	1987-01-29
FR2593504B1 (fr)	1988-12-09
FI870347A (fi)	1987-07-31
CS57887A2 (en)	1988-09-16
MA20861A1 (fr)	1987-10-01
IN164389B (xx)	1989-03-04
NZ219068A (en)	1990-12-21
PL263885A1 (en)	1988-09-15
CN1016420B (zh)	1992-04-29
CN87100978A (zh)	1987-09-16
IT8747583A0 (it)	1987-01-29
US5006570A (en)	1991-04-09
PT84224B (pt)	1989-03-30
IS1446B6 (is)	1990-12-14
IE870128L (en)	1987-07-30
DK46987A (da)	1987-07-31
TNSN87012A1 (fr)	1990-01-01
YU11387A (en)	1988-06-30
LU86747A1 (fr)	1987-06-02
NO168582C (no)	1992-03-11
GB2187188B (en)	1989-11-08
NO168582B (no)	1991-12-02
ZA87552B (en)	1987-10-28
AU593605B2 (en)	1990-02-15
FI870347A0 (fi)	1987-01-27
DE3702005A1 (de)	1987-08-06
CS264300B2 (cs)	1989-06-13
PL152404B1 (en)	1990-12-31
IS3189A7 (is)	1987-07-31
SU1607688A3 (ru)	1990-11-15
BE1000164A5 (fr)	1988-07-05
PL272298A1 (en)	1989-02-20
PL152491B1 (en)	1990-12-31
YU46185B (sh)	1993-05-28
GR3003653T3 (xx)	1993-03-16
CS36288A2 (en)	1988-09-16
IL81299A (en)	1991-09-16
IN167060B (xx)	1990-08-25
NO870199D0 (no)	1987-01-16
CN1062144A (zh)	1992-06-24
NO870199L (no)	1987-07-31
AU6785587A (en)	1987-08-06
OA08472A (fr)	1988-07-29
ES2038679T3 (es)	1993-08-01
FR2593504A1 (fr)	1987-07-31
JPS62277376A (ja)	1987-12-02
IL81299A0 (en)	1987-08-31
GB8701870D0 (en)	1987-03-04

Publication	Publication Date	Title
ZA87552B (en)	1987-10-28	New dihydrobenzofuran-and chroman-carboxamide derivatives,processes for the preparation thereof and use thereof as neuroleptics
EP0415456A3 (en)	1991-05-29	Xanthine compounds
ATE62908T1 (de)	1991-05-15	Neue derivate von 4,5-dihydro-oxazolen, verfahren zu ihrer herstellung und ihre verwendung.
ATE37368T1 (de)	1988-10-15	Benzothiazolon-derivate, verfahren zu ihrer herstellung und sie enthaltende pharmazeutische zusammensetzungen.
AU658175B2 (en)	1995-04-06	Use of 2-iminothiazolidin-4-one derivatives as novel pharmaceutical active ingredients