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PA8631101A1 - Proceso de acoplamiento para la generacion de derivados reactivos de pirrol-2-carbonitrilo n-sustituidos con contenido de boro para producir biarilos - Google Patents

Proceso de acoplamiento para la generacion de derivados reactivos de pirrol-2-carbonitrilo n-sustituidos con contenido de boro para producir biarilos

Info

Publication number
PA8631101A1
PA8631101A1 PA20058631101A PA8631101A PA8631101A1 PA 8631101 A1 PA8631101 A1 PA 8631101A1 PA 20058631101 A PA20058631101 A PA 20058631101A PA 8631101 A PA8631101 A PA 8631101A PA 8631101 A1 PA8631101 A1 PA 8631101A1
Authority
PA
Panama
Prior art keywords
boro
content
pirrol
substituted
carbonitrile
Prior art date
Application number
PA20058631101A
Other languages
English (en)
Inventor
Arkadiy Zinoviy Rubezhov
Bogdan Kazimierz Wilk
Jean Louise Helom
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of PA8631101A1 publication Critical patent/PA8631101A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

SE PRESENTA UNA PREPARACION CONVENIENTE DE COMPUESTOS CON CONTENIDO DE BORO, COMPUESTOS DE PIRROLCARBONITRILO CON CONTENIDO DE BORO, COMPUESTOS DE PIRROL-2-CARBONITRILO N-SUSTITUIDOS CON CONTENIDO DE BORO Y DERIVADOS DE LOS MISMOS. LA PRESENTE INVENCION PRESENTA ASIMISMO EL USO DE ESTOS COMPUESTOS CON CONTENIDO DE BORO Y DERIVADOS DE LOS MISMOS EN REACCIONES DE ACOPLAMIENTO PARA LA PRODUCCION DE COMPUESTOS DE BIARILO.
PA20058631101A 2004-04-27 2005-04-25 Proceso de acoplamiento para la generacion de derivados reactivos de pirrol-2-carbonitrilo n-sustituidos con contenido de boro para producir biarilos PA8631101A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US56563604P 2004-04-27 2004-04-27
US64765605P 2005-01-27 2005-01-27

Publications (1)

Publication Number Publication Date
PA8631101A1 true PA8631101A1 (es) 2006-09-08

Family

ID=34967855

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20058631101A PA8631101A1 (es) 2004-04-27 2005-04-25 Proceso de acoplamiento para la generacion de derivados reactivos de pirrol-2-carbonitrilo n-sustituidos con contenido de boro para producir biarilos

Country Status (7)

Country Link
US (2) US7446211B2 (es)
AR (1) AR049631A1 (es)
PA (1) PA8631101A1 (es)
PE (1) PE20060331A1 (es)
SV (1) SV2005002092A (es)
TW (1) TW200604137A (es)
WO (1) WO2005105817A2 (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PA8631101A1 (es) 2004-04-27 2006-09-08 Wyeth Corp Proceso de acoplamiento para la generacion de derivados reactivos de pirrol-2-carbonitrilo n-sustituidos con contenido de boro para producir biarilos
AU2005238520B2 (en) 2004-04-27 2011-09-08 Wyeth Cyanopyrrole containing cyclic carbamate and thiocarbamate biaryls and methods for preparing the same
GT200500185A (es) * 2004-08-09 2006-04-10 Moduladores del receptor de progesterona que comprenden derivados de pirrol-oxindol y sus usos
WO2006020712A1 (en) * 2004-08-13 2006-02-23 Wyeth Tanaproget derivatives, metabolites, and uses thereof
BRPI0610437A2 (pt) 2005-04-28 2012-10-23 Wyeth Corp composição farmacêutica, comprimido, embalagem farmacêutica, e, processo para a preparação de uma composição farmacêutica
JP2008539254A (ja) * 2005-04-28 2008-11-13 ワイス タナプロゲットの精製形態
MX2007013469A (es) 2005-04-28 2008-01-22 Wyeth Corp Forma ii polimorfa de tanaproget.
CN101166533A (zh) 2005-04-28 2008-04-23 惠氏公司 微粉化的tanaproget和含有它的组合物
PE20070220A1 (es) 2005-07-29 2007-03-19 Wyeth Corp Proceso para la sintesis de moduladores del receptor de progesterona
US20070213526A1 (en) * 2006-03-07 2007-09-13 Wyeth Purification of progesterone receptor modulators
AU2008211047B2 (en) 2007-01-29 2013-07-25 Wako Pure Chemical Industries, Ltd. Reagent for organic synthesis reaction containing organic triol borate salt
US20080319204A1 (en) * 2007-06-25 2008-12-25 Wyeth Process for the synthesis of progesterone receptor modulators
BRPI0819571A2 (pt) * 2007-12-20 2019-09-24 Teva Womenss Health Inc "método para contracepção de emergência, pacote farmacêutico para contracepção de emergência e composição farmacêutica"
KR20240131463A (ko) 2020-05-05 2024-08-30 뉴베일런트, 아이엔씨. 헤테로방향족 거대환식 에터 화학치료제
KR102699528B1 (ko) 2020-05-05 2024-08-30 뉴베일런트, 아이엔씨. 헤테로방향족 거대환식 에터 화학치료제
EP4408844A1 (en) 2021-10-01 2024-08-07 Nuvalent, Inc. Solid forms, pharmaceutical compositions and preparation of heteroaromatic macrocyclic ether compounds

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MX9206628A (es) * 1991-11-22 1993-05-01 Boehringer Ingelheim Pharma Ester de prolinaboronato y metodo para su preparacion.
KR960704886A (ko) 1993-09-10 1996-10-09 베르너 발데크 포토크롬 화합물, 그의 제조 방법과 제조 중간체 및 그의 용도 (Photochromic Compounds, Methods and Intermediates for Producing Them and Their Use)
CA2363628A1 (en) 1999-02-22 2000-08-31 James Allen Ponasik Jr. Catalysts containing n-pyrrolyl substituted nitrogen donors
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UA73119C2 (en) 2000-04-19 2005-06-15 American Home Products Corpoir Derivatives of cyclic thiocarbamates, pharmaceutical composition including noted derivatives of cyclic thiocarbamates and active ingredients of medicines as modulators of progesterone receptors
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AU2003223930A1 (en) 2002-06-14 2003-12-31 Novo Nordisk A/S Pharmaceutical use of boronic acids and esters thereof
PA8631101A1 (es) 2004-04-27 2006-09-08 Wyeth Corp Proceso de acoplamiento para la generacion de derivados reactivos de pirrol-2-carbonitrilo n-sustituidos con contenido de boro para producir biarilos

Also Published As

Publication number Publication date
US20050272702A1 (en) 2005-12-08
WO2005105817A2 (en) 2005-11-10
SV2005002092A (es) 2005-12-13
US8129523B2 (en) 2012-03-06
US20090054663A1 (en) 2009-02-26
TW200604137A (en) 2006-02-01
PE20060331A1 (es) 2006-05-16
WO2005105817A3 (en) 2006-01-12
AR049631A1 (es) 2006-08-23
US7446211B2 (en) 2008-11-04

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