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KR970700181A - 레트로바이러스성 프로테아제 억제 화합물 제조용 합성 중간체(Synthetic intermediates for preparing retroviral protease inhibiting compounds) - Google Patents

레트로바이러스성 프로테아제 억제 화합물 제조용 합성 중간체(Synthetic intermediates for preparing retroviral protease inhibiting compounds)

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Publication number
KR970700181A
KR970700181A KR1019960703601A KR19960703601A KR970700181A KR 970700181 A KR970700181 A KR 970700181A KR 1019960703601 A KR1019960703601 A KR 1019960703601A KR 19960703601 A KR19960703601 A KR 19960703601A KR 970700181 A KR970700181 A KR 970700181A
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KR
South Korea
Prior art keywords
retroviral protease
inhibiting compounds
synthetic intermediates
protease inhibiting
preparing retroviral
Prior art date
Application number
KR1019960703601A
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English (en)
Other versions
KR100187990B1 (ko
Inventor
제이. 켐프 데일
더블유. 노벡 다니엘
렁 샴 힝
짜오 첸
제이. 소윈 토머스
에스. 레노 다니엘
알. 하이트 앤소니
제이. 쿠퍼 아서
Original Assignee
챨스 엠. 브록
애보트 라보라토리즈
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Application filed by 챨스 엠. 브록, 애보트 라보라토리즈 filed Critical 챨스 엠. 브록
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    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
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Abstract

본 발명은 레트로바이러스 프로테아제 억제 화합물 제조용 합성 중간체인 구조식
의 화합물 또는 이의 염 및 일반식
의 화합물
[여기서, R은 수소 또는 저급 알킬이다]에 관한 것이다.

Description

레트로바이러스성 프로테아제 억제 화합물 제조용 합성 중간체(Synthetic intermediates for preparing retroviral protease inhibiting compounds)
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (2)

  1. 다음 구조식의 화합물 또는 이의 염.
  2. 다음 일반식의 화합물 또는 이의 염.
    상기식에서, R은 수소 또는 저급 알킬이다.
KR1019960703601A 1992-12-29 1993-12-16 레트로바이러스성 프로테아제 억제 화합물 제조용 합성 중간체 KR100187990B1 (ko)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
US99811492A 1992-12-29 1992-12-29
US7/998,114 1992-12-29
US07/998,114 1992-12-29
US15858793A 1993-12-02 1993-12-02
US08/158,587 1993-12-02
US8/158,587 1993-12-02
KR1019940704362A KR100187613B1 (ko) 1992-12-29 1993-12-16 레트로바이러스성 프로테이제 억제 화합물, 이의 제조방법 및 이를 함유하는 약제학적 조성물
PCT/US1993/012326 WO1994014436A1 (en) 1992-12-29 1993-12-16 Retroviral protease inhibiting compounds

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KR1020017008351A KR100360964B1 (ko) 1992-12-29 1993-12-16 레트로바이러스성 프로테아제 억제 화합물의 중간체의제조방법
KR1019960703601A KR100187990B1 (ko) 1992-12-29 1993-12-16 레트로바이러스성 프로테아제 억제 화합물 제조용 합성 중간체
KR1019960703602A KR100333016B1 (ko) 1992-12-29 1993-12-16 레트로바이러스성프로테아제억제화합물,이의제조방법및이를함유하는약제학적조성물
KR1019940704362A KR100187613B1 (ko) 1992-12-29 1993-12-16 레트로바이러스성 프로테이제 억제 화합물, 이의 제조방법 및 이를 함유하는 약제학적 조성물

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KR1019940704362A KR100187613B1 (ko) 1992-12-29 1993-12-16 레트로바이러스성 프로테이제 억제 화합물, 이의 제조방법 및 이를 함유하는 약제학적 조성물

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