JPS6440467A - Novel substituted diphenylimidazole derivative - Google Patents
Novel substituted diphenylimidazole derivativeInfo
- Publication number
- JPS6440467A JPS6440467A JP19611787A JP19611787A JPS6440467A JP S6440467 A JPS6440467 A JP S6440467A JP 19611787 A JP19611787 A JP 19611787A JP 19611787 A JP19611787 A JP 19611787A JP S6440467 A JPS6440467 A JP S6440467A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- diphenylimidazole
- derivative
- compound
- novel substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
NEW MATERIAL:The substituted diphenylimidazole derivative of formula I (X is H, halogen, lower alkyl or lower alkoxy; m is 0 or 1; n is 1-4; R is heterocyclic group or cyclic amino; when n=2, R is not 2-pyridyl) and its acid addition salt. EXAMPLE:4,5-Diphenyl-2-(2-pyridylmethyl)thio-imidazole. USE:It has antiulcer and anti-inflammatory actions and is useful as a drug. It has low side effect and high safety. PREPARATION:The compound of formula I can be produced according to the reaction formula, by reacting the compound of formula II with the compound of formula III in a solvent (e.g. methanol) at 20-120 deg.C.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP19611787A JPS6440467A (en) | 1987-08-04 | 1987-08-04 | Novel substituted diphenylimidazole derivative |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP19611787A JPS6440467A (en) | 1987-08-04 | 1987-08-04 | Novel substituted diphenylimidazole derivative |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS6440467A true JPS6440467A (en) | 1989-02-10 |
Family
ID=16352523
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP19611787A Pending JPS6440467A (en) | 1987-08-04 | 1987-08-04 | Novel substituted diphenylimidazole derivative |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS6440467A (en) |
Cited By (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1991009030A1 (en) * | 1989-12-12 | 1991-06-27 | Rhone-Poulenc Sante | 2-substituted 4,5-diphenyl-imidazoles |
JPH04217963A (en) * | 1990-04-09 | 1992-08-07 | Meiji Seika Kaisha Ltd | Thiazole or imidazole derivative and antiulcer agent |
EP0522887A1 (en) * | 1991-07-12 | 1993-01-13 | Rhone-Poulenc Rorer Limited | Imidazoles as ACAT- and thromboxane TxA2 inhibitors |
EP0523941A1 (en) * | 1991-07-11 | 1993-01-20 | Rhone-Poulenc Rorer Limited | Imidazoles as ACAT inhibitor |
WO2002076951A1 (en) * | 2001-03-26 | 2002-10-03 | Beiersdorf Ag | 2-mercapto-4,5-diarylimidazole derivatives and the use thereof as cyclooxygenase inhibitors |
WO2004018458A1 (en) | 2002-08-20 | 2004-03-04 | Merckle-Gmbh | 2-thio-substituted imidazole derivatives and their use in pharmaceutics |
JP2005530799A (en) * | 2002-05-17 | 2005-10-13 | メルクル・ゲーエムベーハー | 2-thio-substituted imidazole derivatives and their use in pharmacy |
US7253191B2 (en) | 2001-02-19 | 2007-08-07 | Merckle Gmbh | 2-thio-substituted imidazole derivatives and the use thereof in the pharmaceutical industry |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS54154766A (en) * | 1978-05-24 | 1979-12-06 | Schering Ag | Novel imidazole derivative*its manufacture and medicine containing said derivative and having antiiinflammatory and antiiallergic activity |
JPS62207270A (en) * | 1986-03-06 | 1987-09-11 | Yamanouchi Pharmaceut Co Ltd | Azole compound substituted with 2-pyridylmethylthio group or 2-pyridylmethylsulfinyl group |
JPS6463575A (en) * | 1987-07-31 | 1989-03-09 | Chiesi Farma Spa | Thiomethyl and sulfinylmethyl derivative having gastric acid secretion control, manufacture and pharmaceutical composition |
-
1987
- 1987-08-04 JP JP19611787A patent/JPS6440467A/en active Pending
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS54154766A (en) * | 1978-05-24 | 1979-12-06 | Schering Ag | Novel imidazole derivative*its manufacture and medicine containing said derivative and having antiiinflammatory and antiiallergic activity |
JPS62207270A (en) * | 1986-03-06 | 1987-09-11 | Yamanouchi Pharmaceut Co Ltd | Azole compound substituted with 2-pyridylmethylthio group or 2-pyridylmethylsulfinyl group |
JPS6463575A (en) * | 1987-07-31 | 1989-03-09 | Chiesi Farma Spa | Thiomethyl and sulfinylmethyl derivative having gastric acid secretion control, manufacture and pharmaceutical composition |
Cited By (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1991009030A1 (en) * | 1989-12-12 | 1991-06-27 | Rhone-Poulenc Sante | 2-substituted 4,5-diphenyl-imidazoles |
JPH04217963A (en) * | 1990-04-09 | 1992-08-07 | Meiji Seika Kaisha Ltd | Thiazole or imidazole derivative and antiulcer agent |
EP0523941A1 (en) * | 1991-07-11 | 1993-01-20 | Rhone-Poulenc Rorer Limited | Imidazoles as ACAT inhibitor |
WO1993001183A1 (en) * | 1991-07-11 | 1993-01-21 | Rhone-Poulenc Rorer Limited | Imidazole derivative as acat inhibitor |
EP0522887A1 (en) * | 1991-07-12 | 1993-01-13 | Rhone-Poulenc Rorer Limited | Imidazoles as ACAT- and thromboxane TxA2 inhibitors |
WO1993001184A1 (en) * | 1991-07-12 | 1993-01-21 | Rhone-Poulenc Rorer Limited | Imidazoles inhibitors as acat and thromboxane txa2 |
US7253191B2 (en) | 2001-02-19 | 2007-08-07 | Merckle Gmbh | 2-thio-substituted imidazole derivatives and the use thereof in the pharmaceutical industry |
WO2002076951A1 (en) * | 2001-03-26 | 2002-10-03 | Beiersdorf Ag | 2-mercapto-4,5-diarylimidazole derivatives and the use thereof as cyclooxygenase inhibitors |
US7223781B2 (en) | 2001-03-26 | 2007-05-29 | Beiersdorf Ag | 2-mercapto-4,5-diarylimidazole derivatives and the use thereof as cyclooxygenase inhibitors |
JP2005530799A (en) * | 2002-05-17 | 2005-10-13 | メルクル・ゲーエムベーハー | 2-thio-substituted imidazole derivatives and their use in pharmacy |
WO2004018458A1 (en) | 2002-08-20 | 2004-03-04 | Merckle-Gmbh | 2-thio-substituted imidazole derivatives and their use in pharmaceutics |
US7582660B2 (en) | 2002-08-20 | 2009-09-01 | C-A-I-R Biosciences Gmbh | 2-thio-substituted imidazole derivatives and their use in pharmaceutics |
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