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JPS53101391A - 1-oxadithiacephem compounds - Google Patents

1-oxadithiacephem compounds

Info

Publication number
JPS53101391A
JPS53101391A JP1581377A JP1581377A JPS53101391A JP S53101391 A JPS53101391 A JP S53101391A JP 1581377 A JP1581377 A JP 1581377A JP 1581377 A JP1581377 A JP 1581377A JP S53101391 A JPS53101391 A JP S53101391A
Authority
JP
Japan
Prior art keywords
oxadithiacephem
compounds
carboxy
amino
protected
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP1581377A
Other languages
Japanese (ja)
Inventor
Yoshitsuru Yoshioka
Shoichiro Ageo
Yoshio Hamashima
Ikuo Kitsukawa
Shoji Tsuji
Wataru Nagata
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Shionogi and Co Ltd
Original Assignee
Shionogi and Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi and Co Ltd filed Critical Shionogi and Co Ltd
Priority to JP1581377A priority Critical patent/JPS53101391A/en
Priority to GB5339/78A priority patent/GB1557552A/en
Priority to AU33164/78A priority patent/AU514377B2/en
Priority to DK060678A priority patent/DK168217B1/en
Priority to CA296,776A priority patent/CA1099715A/en
Priority to IE298/78A priority patent/IE47711B1/en
Priority to NZ186437A priority patent/NZ186437A/en
Priority to PT67648A priority patent/PT67648B/en
Priority to ZA00780846A priority patent/ZA78846B/en
Priority to IL54044A priority patent/IL54044A/en
Priority to BG040119A priority patent/BG32855A3/en
Priority to GR55452A priority patent/GR69965B/el
Priority to FR7804162A priority patent/FR2380284A1/en
Priority to MX786846U priority patent/MX5479E/en
Priority to BG040118A priority patent/BG32854A3/en
Priority to NO780508A priority patent/NO162343C/en
Priority to ES466949A priority patent/ES466949A1/en
Priority to AT104578A priority patent/AT360152B/en
Priority to BG038671A priority patent/BG32853A3/en
Priority to PL1978204616A priority patent/PL114451B1/en
Priority to HU78SI1619A priority patent/HU177897B/en
Priority to RO78100614A priority patent/RO79886A/en
Priority to SE7801697A priority patent/SE443144B/en
Priority to CS78960A priority patent/CS196417B2/en
Priority to CS786972A priority patent/CS196420B2/en
Priority to RO78100613A priority patent/RO79398A/en
Priority to FI780474A priority patent/FI68401C/en
Priority to SU782579850A priority patent/SU833162A3/en
Priority to YU335/78A priority patent/YU41307B/en
Priority to PL1978216456A priority patent/PL117502B1/en
Priority to RO78100612A priority patent/RO78545A/en
Priority to PH20789A priority patent/PH15515A/en
Priority to BE185205A priority patent/BE863998A/en
Priority to CH167278A priority patent/CH636618A5/en
Priority to DD78203720A priority patent/DD134524A5/en
Priority to DE19782806457 priority patent/DE2806457A1/en
Priority to NL7801708A priority patent/NL191891C/en
Priority to BG040120A priority patent/BG32856A3/en
Publication of JPS53101391A publication Critical patent/JPS53101391A/en
Priority to ES475141A priority patent/ES475141A1/en
Priority to ES78475142A priority patent/ES475142A1/en
Priority to ES78475140A priority patent/ES475140A1/en
Priority to SU792706007A priority patent/SU1110386A3/en
Priority to AT617079A priority patent/AT370104B/en
Priority to PH23439A priority patent/PH15513A/en
Priority to PH23440A priority patent/PH15291A/en
Priority to PH23438A priority patent/PH15294A/en
Priority to US06/322,662 priority patent/US4366316A/en
Priority to AR22786782D priority patent/AR227867A1/en
Priority to SU823371059A priority patent/SU1041036A3/en
Priority to SU823376800A priority patent/SU1039444A3/en
Priority to US06/374,862 priority patent/US4443598A/en
Priority to YU547/83A priority patent/YU42072B/en
Priority to YU548/83A priority patent/YU42073B/en
Priority to FI833080A priority patent/FI70713C/en
Priority to FI833079A priority patent/FI833079A0/en
Priority to US06/542,520 priority patent/US4604460A/en
Priority to US06/543,664 priority patent/US4478997A/en
Priority to US06/543,940 priority patent/US4533730A/en
Priority to US06/543,939 priority patent/US4504659A/en
Priority to FI843922A priority patent/FI71154C/en
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

PURPOSE: 1-Oxadithiacephem cpds. I [ A is amino or protected amino; E is H or methoxy; Y is II(COB is carboxy or protected carboxy; X is H or nucleophile; Z is leaving gp.); the dotted line is α or β-bond], e.g. 7α-benzamido3-methyl-1-dithia-1-oxa-3-cephem-4-carboxylic acid benzylester.
COPYRIGHT: (C)1978,JPO&Japio
JP1581377A 1977-02-15 1977-02-15 1-oxadithiacephem compounds Pending JPS53101391A (en)

Priority Applications (60)

Application Number Priority Date Filing Date Title
JP1581377A JPS53101391A (en) 1977-02-15 1977-02-15 1-oxadithiacephem compounds
GB5339/78A GB1557552A (en) 1977-02-15 1978-02-09 1 oxadethiacepham compounds
AU33164/78A AU514377B2 (en) 1977-02-15 1978-02-09 l-OXADETHIACEPHAM COMPOUNDS
DK060678A DK168217B1 (en) 1977-02-15 1978-02-10 Process for Preparation of 1-Dethia-1-Oxacepham and Cephalosporin Compounds
CA296,776A CA1099715A (en) 1977-02-15 1978-02-10 1-oxadethiacepham compounds
IE298/78A IE47711B1 (en) 1977-02-15 1978-02-10 1-oxadethiacepham compounds
NZ186437A NZ186437A (en) 1977-02-15 1978-02-10 1-oxa-dethia-cephalosporins
PT67648A PT67648B (en) 1977-02-15 1978-02-13 Process for preparing 1-oxadethiacepham compounds
ZA00780846A ZA78846B (en) 1977-02-15 1978-02-13 1-oxadethiacepham compounds
IL54044A IL54044A (en) 1977-02-15 1978-02-13 Process for preparing 1-dethia-1-oxacepham compounds,some new compounds of this type,and method of inhibiting growth of bacteria using them
BG040119A BG32855A3 (en) 1977-02-15 1978-02-14 METHOD FOR OBTAINING 1-OXADETHIACEPHALOSPORINS
GR55452A GR69965B (en) 1977-02-15 1978-02-14
FR7804162A FR2380284A1 (en) 1977-02-15 1978-02-14 PROCESS FOR THE PREPARATION OF 1-OXADETHIACEPHAM COMPOUNDS AND THEIR USE AS ANTIBACTERIAL PRODUCTS AND AS INTERMEDIARIES FOR THE PREPARATION OF 1-DETHIA-1-OXACEPHALOSPORINS
MX786846U MX5479E (en) 1977-02-15 1978-02-14 PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 1-OXADETIACEFALOSPORINAS
BG040118A BG32854A3 (en) 1977-02-15 1978-02-14 Method for obtaining of 1- oxadethiacephalosporine
NO780508A NO162343C (en) 1977-02-15 1978-02-14 7-ACYLAMINO-1-DETIA-1-OXACEFAM COMPOUNDS SUITABLE AS INTERMEDIATE FOR THE PREPARATION OF 7BETA-ACYLAMINO-1-DETIA-1-OXACEPHALOSPORINES.
ES466949A ES466949A1 (en) 1977-02-15 1978-02-14 1-Oxadethiacepham compounds and process for producing said compounds
AT104578A AT360152B (en) 1977-02-15 1978-02-14 METHOD FOR PRODUCING 1-OXADE THIACEPHAM COMPOUNDS
BG038671A BG32853A3 (en) 1977-02-15 1978-02-14 Method for obtaining of 1- oxadethiacephalosporine
PL1978204616A PL114451B1 (en) 1977-02-15 1978-02-14 Process for preparing novel 1-oxadethiacephalosporins
HU78SI1619A HU177897B (en) 1977-02-15 1978-02-14 Process for preparing 7-amino-dethia-1-oxa-cefam- and -cefem-4-carboxylic acid derivatives resp.
RO78100614A RO79886A (en) 1977-02-15 1978-02-14 PROCEDURE FOR PREPARING FALOSPORINE 1-OXADETICATION
SE7801697A SE443144B (en) 1977-02-15 1978-02-14 INTERMEDIATES, 1-OXADETIACEFAM SOCIETIES, AND PROCEDURES FOR PRODUCING THEREOF
CS78960A CS196417B2 (en) 1977-02-15 1978-02-14 Method of producing 1-oxadethiacephamderivatives
CS786972A CS196420B2 (en) 1977-02-15 1978-02-14 Method of producing 1-dethia-1-oxacephamderivatives
RO78100613A RO79398A (en) 1977-02-15 1978-02-14 PROCESS FOR THE PREPARATION OF 1-OXA-DETHIACEPHALOSPORINS
FI780474A FI68401C (en) 1977-02-15 1978-02-14 7BETA-ACYLAMINO-7ALFA-METHOXY-3-SUBSTITUTE METADYL-1-OXADETIA-1-CEFAM-4-CARBOXYLATER ANVAENDBARA SOM MELLANPRODUKTER I FRAMSTAELLNING AV 1-DETIA-1-OXACEFALOSPORINER
SU782579850A SU833162A3 (en) 1977-02-15 1978-02-14 Method of preparing 1-oxadethiacephalosporins
YU335/78A YU41307B (en) 1977-02-15 1978-02-14 Process for obtaining 1-oxadethia cepham compounds
PL1978216456A PL117502B1 (en) 1977-02-15 1978-02-14 Process for preparing 1-dethia-1-oxacephame derivatives
RO78100612A RO78545A (en) 1977-02-15 1978-02-14 PROCEDURE FOR PREPARING FALOSPORINE 1-OXADETICATION
PH20789A PH15515A (en) 1977-02-15 1978-02-15 1-oxadethiacephan compounds
BE185205A BE863998A (en) 1977-02-15 1978-02-15 1-OXADETHIACEPHAMES
CH167278A CH636618A5 (en) 1977-02-15 1978-02-15 1-Oxadethiacepham compounds, and a process for preparing them
DD78203720A DD134524A5 (en) 1977-02-15 1978-02-15 PROCESS FOR PREPARING 1-OXADETHIACEPHAM COMPOUNDS
DE19782806457 DE2806457A1 (en) 1977-02-15 1978-02-15 1-OXADETHIACEPHAM COMPOUNDS AND METHOD FOR THEIR MANUFACTURE
NL7801708A NL191891C (en) 1977-02-15 1978-02-15 Process for the preparation of 1-oxadethiacepham or cephem derivatives.
BG040120A BG32856A3 (en) 1977-02-15 1978-06-16 METHOD OF OBTAINING 1-OXADETYLACEPHALOSPORIUM
ES475141A ES475141A1 (en) 1977-02-15 1978-11-16 1-Oxadethiacepham compounds and process for producing said compounds
ES78475142A ES475142A1 (en) 1977-02-15 1978-11-16 1-Oxadethiacepham compounds and process for producing said compounds
ES78475140A ES475140A1 (en) 1977-02-15 1978-11-16 1-Oxadethiacepham compounds and process for producing said compounds
SU792706007A SU1110386A3 (en) 1977-02-15 1979-01-03 Process for preparing 1-oxadethiacephalosporins
AT617079A AT370104B (en) 1977-02-15 1979-09-19 METHOD FOR PRODUCING 1-DETHIA-1-OXACEPHEM DERIVATIVES
PH23439A PH15513A (en) 1977-02-15 1979-12-20 1-oxadethiacepham compounds
PH23440A PH15291A (en) 1977-02-15 1979-12-20 1-oxadethiacepham compounds
PH23438A PH15294A (en) 1977-02-15 1979-12-20 1-oxadethiacepham compounds
US06/322,662 US4366316A (en) 1977-02-15 1981-11-18 1-Oxadethiacepham compounds and process for producing said compounds
AR22786782D AR227867A1 (en) 1977-02-15 1982-01-01 NEW DERIVATIVES OF ACID 7-AMINO-1-DETIA-1-OXACEFAM-4-CARBOXILICO EXEMPT FROM THERAPEUTIC ACTIVITY AND USEFUL AS INTERMEDIARIES TO OBTAIN 1-OXADETIACEFALOSPORINAS AND PROCEDURE TO PREPARE THEM
SU823371059A SU1041036A3 (en) 1977-02-15 1982-01-06 Process for preparing 1-oxadethiacephalosporins
SU823376800A SU1039444A3 (en) 1977-02-15 1982-01-18 Process for preparing 1-oxadethia cephalosporin
US06/374,862 US4443598A (en) 1977-02-15 1982-05-04 1-Oxadethiacepham compounds
YU547/83A YU42072B (en) 1977-02-15 1983-03-07 Process for obtaining 1-oxadethiacepham compounds
YU548/83A YU42073B (en) 1977-02-15 1983-03-07 Process for obtaining 1-oxadethiaceptham compounds
FI833080A FI70713C (en) 1977-02-15 1983-08-30 7BETA-ACYLAMINO-1-CEFAM-FOERENINGAR ANVAENDBARA SOM MELLANPRODUKTER I FRAMSTAELLNING AV 7-ACYLAMINO-1-DETIA-1-OKSACEFALOSPORINER
FI833079A FI833079A0 (en) 1977-02-15 1983-08-30 1-dethia-1-OXACEFAMFOERENINGAR
US06/542,520 US4604460A (en) 1977-02-15 1983-10-17 1-oxadethiacepham compounds
US06/543,664 US4478997A (en) 1977-02-15 1983-10-19 1-Oxadethiacepham compounds
US06/543,940 US4533730A (en) 1977-02-15 1983-10-19 1-Oxadethiacepham compounds
US06/543,939 US4504659A (en) 1977-02-15 1983-10-19 1-Oxadethiacepham compounds
FI843922A FI71154C (en) 1977-02-15 1984-10-05 1-dethia-1-OXA-3- (1-methyl-1,2,3,4-tetrazol-5-YL) TIOMETYLCEFAM-4-KARBOXYLATER

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP1581377A JPS53101391A (en) 1977-02-15 1977-02-15 1-oxadithiacephem compounds

Publications (1)

Publication Number Publication Date
JPS53101391A true JPS53101391A (en) 1978-09-04

Family

ID=11899274

Family Applications (1)

Application Number Title Priority Date Filing Date
JP1581377A Pending JPS53101391A (en) 1977-02-15 1977-02-15 1-oxadithiacephem compounds

Country Status (9)

Country Link
JP (1) JPS53101391A (en)
AT (1) AT360152B (en)
BE (1) BE863998A (en)
CS (2) CS196417B2 (en)
DD (1) DD134524A5 (en)
PL (1) PL117502B1 (en)
SU (4) SU833162A3 (en)
YU (1) YU42072B (en)
ZA (1) ZA78846B (en)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006006290A1 (en) * 2004-07-08 2006-01-19 Shionogi & Co., Ltd. PROCESS FOR PRODUCING 1-OXACEPHALOSPORIN-7α-METHOXY-3-CHLOROMETHYL DERIVATIVE
CN109485659A (en) * 2017-09-13 2019-03-19 东都股份有限公司 The preparation method of 7 alpha-alkoxy base oxacephem intermediates

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3225269A1 (en) * 1982-07-06 1984-01-12 Bayer Ag, 5090 Leverkusen METHOD FOR PRODUCING 7-AMINO-1-DETHIA-1-OXA-3-HYDROXYMETHYL-CEPHEM-4-CARBONIC ACIDS

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006006290A1 (en) * 2004-07-08 2006-01-19 Shionogi & Co., Ltd. PROCESS FOR PRODUCING 1-OXACEPHALOSPORIN-7α-METHOXY-3-CHLOROMETHYL DERIVATIVE
CN109485659A (en) * 2017-09-13 2019-03-19 东都股份有限公司 The preparation method of 7 alpha-alkoxy base oxacephem intermediates
CN109485659B (en) * 2017-09-13 2021-09-10 东都股份有限公司 Process for preparing 7 alpha-alkoxyoxycephalosporane intermediates

Also Published As

Publication number Publication date
SU1110386A3 (en) 1984-08-23
SU1039444A3 (en) 1983-08-30
CS196417B2 (en) 1980-03-31
ZA78846B (en) 1979-01-31
ATA104578A (en) 1980-05-15
BE863998A (en) 1978-05-29
PL117502B1 (en) 1981-08-31
SU833162A3 (en) 1981-05-23
SU1041036A3 (en) 1983-09-07
AT360152B (en) 1980-12-29
YU42072B (en) 1988-04-30
DD134524A5 (en) 1979-03-07
YU54783A (en) 1984-02-29
CS196420B2 (en) 1980-03-31

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