JPS559041A - Synthesis of thioketal - Google Patents
Synthesis of thioketalInfo
- Publication number
- JPS559041A JPS559041A JP8210678A JP8210678A JPS559041A JP S559041 A JPS559041 A JP S559041A JP 8210678 A JP8210678 A JP 8210678A JP 8210678 A JP8210678 A JP 8210678A JP S559041 A JPS559041 A JP S559041A
- Authority
- JP
- Japan
- Prior art keywords
- substituted
- thioketal
- butylphenol
- mercapto
- mole
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
PURPOSE: To prepare the title compound having blood cholesterol depressing activity, economically, by reacting 4-mercapto-2,6-di-t-butylphenol with acetone in the presence of a specific sulfonic acid ester.
CONSTITUTION: A thioketal of formula II is prepared by reacting 4-mercapto-2, 6-di-t-butylphenol (l mole) with acetone (0.5 mole-large excess amount) in the presence of a sulfonic acid ester of formula I (R1 is alkyl, substituted or non-substituted aryl, arylalkyl; R2 is alkyl, substituted or non-substituted arylalikyl) (0.001- 2 moles), usually in an inert solvent, usually at 40-100°C, pref. at 50-80°C.
COPYRIGHT: (C)1980,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP8210678A JPS559041A (en) | 1978-07-07 | 1978-07-07 | Synthesis of thioketal |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP8210678A JPS559041A (en) | 1978-07-07 | 1978-07-07 | Synthesis of thioketal |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS559041A true JPS559041A (en) | 1980-01-22 |
Family
ID=13765149
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP8210678A Pending JPS559041A (en) | 1978-07-07 | 1978-07-07 | Synthesis of thioketal |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS559041A (en) |
Cited By (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4560799A (en) * | 1984-02-03 | 1985-12-24 | Ciba-Geigy Corporation | Tri- and Tetra-(substituted hydroxyphenylthio) alkane and cycloalkane stabilizers and stabilized compositions |
US4719237A (en) * | 1986-01-28 | 1988-01-12 | Merrell Dow Pharmaceuticals Inc. | Cardiac antiarrythmic method employing probucol |
US4772363A (en) * | 1987-01-14 | 1988-09-20 | Merrell Dow Pharmaceuticals Inc. | Process for preparing 2,6-di-tertiarybutyl-4-mercaptophenol by electrocatalysis |
US5401883A (en) * | 1987-01-20 | 1995-03-28 | Merrell Dow Pharmaceuticals Inc. | Process for preparing 2,6-di-tertiarybutyl-4-mercaptophenol and 4,4'-isopropylidenedithio-bis-(2,6-di-tertiarybutylphenol) |
-
1978
- 1978-07-07 JP JP8210678A patent/JPS559041A/en active Pending
Cited By (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4560799A (en) * | 1984-02-03 | 1985-12-24 | Ciba-Geigy Corporation | Tri- and Tetra-(substituted hydroxyphenylthio) alkane and cycloalkane stabilizers and stabilized compositions |
US4719237A (en) * | 1986-01-28 | 1988-01-12 | Merrell Dow Pharmaceuticals Inc. | Cardiac antiarrythmic method employing probucol |
US4772363A (en) * | 1987-01-14 | 1988-09-20 | Merrell Dow Pharmaceuticals Inc. | Process for preparing 2,6-di-tertiarybutyl-4-mercaptophenol by electrocatalysis |
US5401883A (en) * | 1987-01-20 | 1995-03-28 | Merrell Dow Pharmaceuticals Inc. | Process for preparing 2,6-di-tertiarybutyl-4-mercaptophenol and 4,4'-isopropylidenedithio-bis-(2,6-di-tertiarybutylphenol) |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
JPS5278848A (en) | Preparation of novel propionic acid ester derivatives | |
IE800961L (en) | Herbicidal 5-(4-trifluoromethylphenoxy) phenyl¹oxime-o-alkanoic derivatives | |
JPS559041A (en) | Synthesis of thioketal | |
JPS54119494A (en) | Preparation of cephalosporin compound | |
JPS5517316A (en) | Preparation of thioketal compound | |
JPS54160335A (en) | Preparation of alkylated hydroxybenzoic ester | |
IE45436L (en) | 12-azaprostanoic acid derivatives | |
JPS5419946A (en) | Prostaglandin analog compound and their preparation | |
JPS5253838A (en) | Preparation of novel 16-alkyl-20-alkoxyprostadienoic acid alkyl ester derivtives | |
GB1530518A (en) | Alkyl sulphonic acid phenyl esters substituted by carboxylic acid esters | |
JPS5466651A (en) | Preparation of o-(2,6-dichloroanilino)phenylacetic acid | |
JPS55108898A (en) | 25-hydroxy-24-oxocholesterol derivative and its preparation | |
JPS5795932A (en) | Preparation of hydroquinone derivative | |
JPS55120591A (en) | Phosphinoethylmalonic acid derivative, and preparation thereof | |
JPS5242855A (en) | Process for preparation of 7_(2-alkoxycarbonylcyclopentyl+)-5-heptenoi c acid | |
ES479300A1 (en) | An alpha-methyl-4(2'-thienyl-carbonyl)phenyl acetic acid derivative, process for its preparation and its pharmaceutical use. | |
JPS5283436A (en) | Preparation of intermediates for synthesis of prostaglandin | |
JPS5444638A (en) | Production of cyclopentanecarboxylic ester derivative | |
JPS55157578A (en) | 1,2-epoxy derivative | |
JPS52118470A (en) | Dithiolane derivatives | |
JPS5283714A (en) | Novel alkyl ester derivatives of 16-alkyl-20-alkoxyprostadienoic acids | |
JPS5585587A (en) | Substituted azetidinones | |
JPS5227752A (en) | Preparation of novel (16,17-methylene) prostaglandin derivatives | |
IE46358L (en) | Prostynoic acid derivatives | |
JPS5718683A (en) | 3,8-epoxy-7-keto-6-oxabicyclo 3,2,1 octane derivative and its preparation |