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Publication number
JP2019524645A5
JP2019524645A5 JP2018562308A JP2018562308A JP2019524645A5 JP 2019524645 A5 JP2019524645 A5 JP 2019524645A5 JP 2018562308 A JP2018562308 A JP 2018562308A JP 2018562308 A JP2018562308 A JP 2018562308A JP 2019524645 A5 JP2019524645 A5 JP 2019524645A5
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formula
seq
compound
amino acid
acid sequence
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JP2018562308A
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JP6843891B2 (ja
JP2019524645A (ja
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Priority claimed from PCT/US2017/035518 external-priority patent/WO2017210471A1/en
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Claims (4)

  1. 下記式の化合物。
    Figure 2019524645
     （式中、ｎは、４であり、Ａは、配列番号６６のアミノ酸配列を含む重鎖及び配列番号７３のアミノ酸配列を含む軽鎖を含むＩｇＧ１抗体である。）
  2. 下記式の化合物。
    Figure 2019524645
     （式中、ｎは、２であり、Ａは、配列番号６６のアミノ酸配列を含む重鎖及び配列番号７３のアミノ酸配列を含む軽鎖を含むＩｇＧ１抗体である。）
  3. 下記式の化合物。
    Figure 2019524645
     （式中、ｎは、４であり、Ａは、アダリムマブである。）
  4. 下記式の化合物。
    Figure 2019524645
     （式中、ｎは、２であり、Ａは、アダリムマブである。）
JP2018562308A 2016-06-02 2017-06-01 グルココルチコイド受容体アゴニスト及びこのイムノコンジュゲート Active JP6843891B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201662344948P 2016-06-02 2016-06-02
US62/344,948 2016-06-02
US201662371134P 2016-08-04 2016-08-04
US62/371,134 2016-08-04
PCT/US2017/035518 WO2017210471A1 (en) 2016-06-02 2017-06-01 Glucocorticoid receptor agonist and immunoconjugates thereof

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JP2019524645A JP2019524645A (ja) 2019-09-05
JP2019524645A5 true JP2019524645A5 (ja) 2020-05-07
JP6843891B2 JP6843891B2 (ja) 2021-03-17

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US (4) US20180126000A1 (ja)
EP (2) EP3901162A1 (ja)
JP (2) JP6843891B2 (ja)
KR (2) KR102435599B1 (ja)
CN (1) CN109476699B (ja)
AU (2) AU2017274442B2 (ja)
BR (1) BR112018074922B1 (ja)
CA (1) CA3025377A1 (ja)
CL (1) CL2018003406A1 (ja)
CO (1) CO2018012996A2 (ja)
CR (1) CR20180594A (ja)
CY (1) CY1124293T1 (ja)
DK (1) DK3464318T3 (ja)
DO (1) DOP2018000261A (ja)
EC (1) ECSP18094857A (ja)
ES (1) ES2877548T3 (ja)
HR (1) HRP20210924T1 (ja)
HU (1) HUE054804T2 (ja)
IL (1) IL263214B2 (ja)
LT (1) LT3464318T (ja)
MA (1) MA51586A (ja)
MX (2) MX2018014927A (ja)
MY (1) MY194619A (ja)
PE (1) PE20190622A1 (ja)
PH (1) PH12018502539A1 (ja)
PL (1) PL3464318T3 (ja)
PT (1) PT3464318T (ja)
RS (1) RS62040B1 (ja)
RU (1) RU2745748C2 (ja)
SG (2) SG11201810678WA (ja)
SI (1) SI3464318T1 (ja)
TW (1) TWI728118B (ja)
UA (1) UA124703C2 (ja)
UY (1) UY37269A (ja)
WO (1) WO2017210471A1 (ja)
ZA (1) ZA201808623B (ja)

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