IL87698A - Pharmaceutical compositions containing azithromycin and derivatives as antiprotozoal agents - Google Patents

Pharmaceutical compositions containing azithromycin and derivatives as antiprotozoal agents

Info

Publication number: IL87698A
Authority: IL; Israel
Prior art keywords: pharmaceutical compositions; derivatives; compositions containing; antiprotozoal agents; containing azithromycin
Prior art date: 1987-09-10

Application number

IL87698A

Other languages

English (en)

Other versions

IL87698A0 (en

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-09-10

Filing date

1988-09-07

Publication date

1992-12-01

1988-09-07 Application filed by Pfizer filed Critical Pfizer

1989-02-28 Publication of IL87698A0 publication Critical patent/IL87698A0/xx

1992-12-01 Publication of IL87698A publication Critical patent/IL87698A/xx

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Molecular Biology (AREA)
Organic Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Epidemiology (AREA)
Genetics & Genomics (AREA)
Biotechnology (AREA)
Biochemistry (AREA)
Engineering & Computer Science (AREA)
Tropical Medicine & Parasitology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Plural Heterocyclic Compounds (AREA)

IL87698A 1987-09-10 1988-09-07 Pharmaceutical compositions containing azithromycin and derivatives as antiprotozoal agents IL87698A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
PCT/US1987/002317 WO1989002271A1 (fr)	1987-09-10	1987-09-10	Azithromycine et derives utilises comme agents anti-protozoaires

Publications (2)

Publication Number	Publication Date
IL87698A0 IL87698A0 (en)	1989-02-28
IL87698A true IL87698A (en)	1992-12-01

Family

ID=22202554

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL87698A IL87698A (en)	1987-09-10	1988-09-07	Pharmaceutical compositions containing azithromycin and derivatives as antiprotozoal agents

Country Status (18)

Country	Link
US (1)	US4963531A (fr)
EP (1)	EP0307128B1 (fr)
JP (1)	JPH0667847B2 (fr)
KR (1)	KR930011996B1 (fr)
AT (1)	ATE74508T1 (fr)
AU (1)	AU596029B2 (fr)
CA (1)	CA1334574C (fr)
DE (1)	DE3869880D1 (fr)
DK (1)	DK175544B1 (fr)
HU (1)	HUT47553A (fr)
IE (1)	IE61507B1 (fr)
IL (1)	IL87698A (fr)
MY (1)	MY103388A (fr)
NZ (1)	NZ226112A (fr)
PH (1)	PH26229A (fr)
PT (1)	PT88448B (fr)
WO (1)	WO1989002271A1 (fr)
ZA (1)	ZA886727B (fr)

Families Citing this family (56)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
RO107257B1 (ro)	1987-07-09	1993-10-30	Pfizer	Procedeu de obtinere a unui dihidrat de azitromicina, cristalin
SI9011409A (en) *	1990-07-18	1995-10-31	Pliva Pharm & Chem Works	O-methyl azitromycin derivates, methods and intermediates for their preparation and methods for preparation of pharmaceuticals products which comprise them
US5912331A (en) *	1991-03-15	1999-06-15	Merck & Co., Inc.	Process for the preparation of 9-deoxo-9(Z)-hydroxyiminoerythromycin A
US5985844A (en) *	1992-03-26	1999-11-16	Merck & Co., Inc.	Homoerythromycin A derivatives modified at the 4"-and 8A-positions
US5189159A (en) *	1992-04-02	1993-02-23	Merck & Co., Inc.	8a-AZA-8a-homoerythromycin cyclic iminoethers
US5215980A (en) *	1992-01-17	1993-06-01	Merck & Co., Inc.	10-AZA-9-deoxo-11-deoxy-erythromycin A and derivatives thereof
TW271400B (fr) *	1992-07-30	1996-03-01	Pfizer
US5210235A (en) *	1992-08-26	1993-05-11	Merck & Co., Inc.	Methods of elaborating erythromycin fragments into amine-containing fragments of azalide antibiotics
US5332807A (en) *	1993-04-14	1994-07-26	Merck & Co., Inc.	Process of producing 8A- and 9A-azalide antibiotics
CA2138643A1 (fr) *	1993-05-05	1994-11-10	Jack S. Remington	Utilisation de derives rifamycine pour la fabrication d'un medicament destine au traitement de la toxoplasmose
US5529994A (en) *	1993-05-05	1996-06-25	Palo Alto Medical Foundation	Treatment for toxoplasmosis
US5795871A (en) *	1994-04-26	1998-08-18	Nobuhiro Narita	Pharmaceutical composition for treatment of non-small cell lung cancer
US5605889A (en) *	1994-04-29	1997-02-25	Pfizer Inc.	Method of administering azithromycin
AU744318B2 (en) *	1994-04-29	2002-02-21	Pfizer Inc.	Method of administering azithromycin
SK282854B6 (sk) *	1994-05-06	2002-12-03	Pfizer Inc.	Dávkovacia forma s riadeným uvoľňovaním obsahujúca azitromycín
US20030212123A1 (en) *	1997-05-05	2003-11-13	Pfizer Inc.	COX-2 selective carprofen for treating pain and inflammation in dogs
US6407074B1 (en) *	1997-06-11	2002-06-18	Pfizer Inc	C-4″-substituted macrolide derivatives
JP2003512290A (ja) *	1997-09-10	2003-04-02	メルクエンドカムパニーインコーポレーテッド	家畜抗菌剤としての８ａ−アザライド
ES2279242T3 (es) *	1997-10-16	2007-08-16	Glaxosmithkline Istrazivacki Centar Zagreb D.O.O.	Nuevos 3,6-hemicetales de la clase de las 9a-azalidas.
AU768219B2 (en) *	1998-11-30	2003-12-04	Teva Pharmaceutical Industries Ltd.	Ethanolate of azithromycin, process for manufacture, and pharmaceutical compositions thereof
US6555139B2 (en)	1999-06-28	2003-04-29	Wockhardt Europe Limited	Preparation of micron-size pharmaceutical particles by microfluidization
IT1313610B1 (it)	1999-08-09	2002-09-09	S I F I Societa Ind Farmaceuti	Processo per la preparazione di formulazioni acquose per uso oftalmico
US6608033B1 (en) *	1999-08-27	2003-08-19	Pfizer Inc.	Treatment or prevention of coccidiosis
PT1246831E (pt)	2000-01-04	2008-03-28	Teva Pharma	Método de preparação de di-hidrato de azitromicina
WO2002007736A1 (fr) *	2000-07-24	2002-01-31	Cadila Pharmaceuticals Limited	Fabrication d'une composition pharmaceutique liquide limpide d'azithromycine
CA2417353C (fr)	2000-07-25	2009-09-01	Laboratorio Silanes,S.A. De C.V.	Methode de synthese en une etape de la 7,16-desoxy-2-aza-10-o-cladinosyl-12-o-desosaminyl-4,5-dihydroxy-6-ethyl-3,5,9,11,13,15-hexamethylbicyclo(11.2.1)hexadeca-1(2)-en-8-one et de production d'une nouvelle forme de 9-desoxo-9a-methyl-9a-aza-9a-homoerythromycine a
AU2001214115A1 (en) *	2000-08-01	2002-02-13	Habil F. Khorakiwala	Process for the preparation of anhydrous azithromycin
DE60114028T2 (de) *	2000-08-23	2006-07-13	Wockhardt Ltd.	Verfahren zur herstellung von wasserfreiem azithromycin
US6949519B2 (en) *	2000-11-27	2005-09-27	Sandoz Ag	Macrolide solvates
KR100491183B1 (ko) *	2001-03-21	2005-05-25	한미약품 주식회사	아지트로마이신의 제조방법 및 이 방법에 사용되는9-데옥소-9에이-아자-9에이-호모에리트로마이신 에이의결정성 수화물
IL158591A0 (en) *	2001-05-22	2004-05-12	Pfizer Prod Inc	Crystal forms of azithromycin
EP1671979B1 (fr)	2001-05-22	2008-08-13	Pfizer Products Inc.	Nouvelle forme cristalline de l'azithromycine
US6861413B2 (en) *	2001-05-22	2005-03-01	Pfizer Inc.	Stable non-dihydrate azithromycin oral suspensions
EA200400214A1 (ru) *	2001-08-21	2004-06-24	Пфайзер Продактс Инк.	Азитромицин в виде разовой дозы
US20080149521A9 (en) *	2001-10-18	2008-06-26	Michael Pesachovich	Methods of stabilizing azithromycin
WO2003032922A2 (fr) *	2001-10-18	2003-04-24	Teva Pharmaceutical Industries Ltd.	Compositions d'azithromycine stabilisees
MXPA04005105A (es) *	2001-12-21	2004-08-19	Pfizer Prod Inc	Formulaciones de acitromicina directamente compresibles.
CN1606433A (zh) *	2001-12-21	2005-04-13	辉瑞产品公司	阿齐霉素湿法制粒法
PL372394A1 (en) *	2002-02-01	2005-07-25	Pfizer Products Inc.	Dry granulated formulations of azithromycin
ES2220229B1 (es) *	2003-05-29	2005-10-16	Quimica Sintetica, S.A.	Sales de adicion de azitromicina y acido citrico y procedimiento para su obtencion.
US20050013835A1 (en) *	2003-07-15	2005-01-20	Pfizer Inc.	Stable non-dihydrate azithromycin oral suspensions
WO2005053653A1 (fr) *	2003-12-04	2005-06-16	Pfizer Products Inc.	Procede d'atomisation/congelation faisant appel a une extrudeuse pour la preparation de compositions d'azithromycine multiparticulaires contenant de preference un poloxamere et un glyceride
EP1691787B1 (fr)	2003-12-04	2008-07-02	Pfizer Products Inc.	Procédé de fabrication de formes pharmaceutiques multiparticulaires
WO2005053639A2 (fr) *	2003-12-04	2005-06-16	Pfizer Products Inc.	Formes multiparticulaires a liberation controlee produites avec des optimiseurs de dissolution
WO2005053652A1 (fr)	2003-12-04	2005-06-16	Pfizer Products Inc.	Compositions medicamenteuses cristallines multiparticulaires contenant un poloxamere et un glyceride
US6984403B2 (en)	2003-12-04	2006-01-10	Pfizer Inc.	Azithromycin dosage forms with reduced side effects
CN1889933A (zh) *	2003-12-04	2007-01-03	辉瑞产品公司	由基于液体的工艺制备的阿奇霉素多颗粒剂型
JP2007513139A (ja) *	2003-12-04	2007-05-24	ファイザー・プロダクツ・インク	安定性の改善した多粒子組成物
EP1689368B1 (fr)	2003-12-04	2016-09-28	Bend Research, Inc	Procédé d'atomisation/congélation faisant appel à une extrudeuse pour la préparation de compositions médicamenteuses cristallines multiparticulaires
CN1295719C (zh) *	2003-12-30	2007-01-17	郑玉庆	远程智能型变压器
US7468428B2 (en)	2004-03-17	2008-12-23	App Pharmaceuticals, Llc	Lyophilized azithromycin formulation
WO2006115494A1 (fr) *	2005-04-26	2006-11-02	American Pharmaceutical Partners, Inc.	Formulation d’azithromycine lyophilisee
US20060046970A1 (en) *	2004-08-31	2006-03-02	Insite Vision Incorporated	Topical otic compositions and methods of topical treatment of prevention of otic infections
US20060198895A1 (en) *	2005-03-07	2006-09-07	Kotliar Eleonora M	Azithromycin powder for oral suspension compositions
CN100427499C (zh) *	2005-12-20	2008-10-22	山东诚创医药技术开发有限公司	一种阿奇霉素的可溶性盐及其制备方法
WO2013088274A1 (fr)	2011-12-14	2013-06-20	Wockhardt Limited	Composition d'azithromycine amorphe anhydre dépourvue de dihydrate d'azithromycine

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SI8110592A8 (en) *	1981-03-06	1996-06-30	Pliva Pharm & Chem Works	Process for preparing of n-methyl-11-aza-10-deoxo-10-dihydroerythromycine a and derivatives thereof
ZA835204B (en) *	1982-07-19	1985-02-27	Pfizer	N-methyl 11-aza-10-deoxo-10-dihydroerythromycin a,intermediates therefor and processes for their preparation
US4474768A (en) *	1982-07-19	1984-10-02	Pfizer Inc.	N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor
PH19293A (en) *	1982-11-15	1986-03-04	Pfizer	Epimeric azahomoerythromycin,pharmaceutical composition containing the same and method of use thereof
US4526889A (en) *	1982-11-15	1985-07-02	Pfizer Inc.	Epimeric azahomoerythromycin A derivative, intermediates and method of use
US4512982A (en) *	1984-04-13	1985-04-23	Pfizer Inc.	9α-Aza-9α-homoerythromycin compounds, pharmaceutical composition and therapeutic method
AU8280087A (en) *	1987-09-10	1989-04-17	Pfizer Inc.	Azithromycin and derivatives as antiprotozoal agents

1987
- 1987-09-10 WO PCT/US1987/002317 patent/WO1989002271A1/fr active Application Filing
1988
- 1988-08-16 US US07/359,676 patent/US4963531A/en not_active Expired - Lifetime
- 1988-08-29 MY MYPI88000970A patent/MY103388A/en unknown
- 1988-08-31 EP EP88308024A patent/EP0307128B1/fr not_active Expired - Lifetime
- 1988-08-31 DE DE8888308024T patent/DE3869880D1/de not_active Expired - Lifetime
- 1988-08-31 AT AT88308024T patent/ATE74508T1/de not_active IP Right Cessation
- 1988-09-07 PT PT88448A patent/PT88448B/pt not_active IP Right Cessation
- 1988-09-07 IL IL87698A patent/IL87698A/xx not_active IP Right Cessation
- 1988-09-08 KR KR1019880011575A patent/KR930011996B1/ko not_active IP Right Cessation
- 1988-09-08 CA CA000576732A patent/CA1334574C/fr not_active Expired - Fee Related
- 1988-09-09 IE IE276288A patent/IE61507B1/en not_active IP Right Cessation
- 1988-09-09 DK DK198805028A patent/DK175544B1/da not_active IP Right Cessation
- 1988-09-09 AU AU22061/88A patent/AU596029B2/en not_active Expired
- 1988-09-09 NZ NZ226112A patent/NZ226112A/en unknown
- 1988-09-09 ZA ZA886727A patent/ZA886727B/xx unknown
- 1988-09-09 PH PH37527A patent/PH26229A/en unknown
- 1988-09-09 HU HU884667A patent/HUT47553A/hu unknown
- 1988-09-10 JP JP63227353A patent/JPH0667847B2/ja not_active Expired - Fee Related

Also Published As

Publication number	Publication date
IE882762L (en)	1989-03-10
NZ226112A (en)	1997-03-24
DK502888D0 (da)	1988-09-09
DK175544B1 (da)	2004-11-29
PT88448B (pt)	1992-10-30
DE3869880D1 (de)	1992-05-14
CA1334574C (fr)	1995-02-28
DK502888A (da)	1989-03-13
ATE74508T1 (de)	1992-04-15
JPH0283326A (ja)	1990-03-23
KR930011996B1 (ko)	1993-12-23
AU596029B2 (en)	1990-04-12
EP0307128A3 (en)	1990-07-04
US4963531A (en)	1990-10-16
PH26229A (en)	1992-04-01
JPH0667847B2 (ja)	1994-08-31
PT88448A (pt)	1989-07-31
AU2206188A (en)	1989-05-11
EP0307128A2 (fr)	1989-03-15
KR890004709A (ko)	1989-05-09
WO1989002271A1 (fr)	1989-03-23
EP0307128B1 (fr)	1992-04-08
HUT47553A (en)	1989-03-28
IL87698A0 (en)	1989-02-28
ZA886727B (en)	1990-04-25
MY103388A (en)	1993-06-30
IE61507B1 (en)	1994-11-02

Publication	Publication Date	Title
IL87698A (en)	1992-12-01	Pharmaceutical compositions containing azithromycin and derivatives as antiprotozoal agents
IL86089A (en)	1992-11-15	Pharmaceutical compositions containing certain androstane-17-ones for the prophylaxis and therapy of retroviral infections
HK14294A (en)	1994-03-04	Skin improving composition containing gamma-linolenic acid or dihomo-gamma-linolenic acid
EP0296573A3 (en)	1990-07-04	Novel nucleosides, their preparation and pharmaceutical novel nucleosides, their preparation and pharmaceutical compositions compositions
EP0293751A3 (en)	1990-07-25	Taurohyodeoxycholic acid for the therapy of calculosis of the biliary tract and of biliary dyspepsia
DE3686022D1 (de)	1992-08-20	Monosaccharide enthaltende zusammensetzung zum heilen von wunden.
JPS6419066A (en)	1989-01-23	Dihydropyridineamides
GB8822546D0 (en)	1988-11-02	Antiviral combinations
ZA938478B (en)	1994-05-20	Vitamin D3 analogs
GR77719B (fr)	1984-09-25
NZ223293A (en)	1990-02-26	Beta-alkyl melatonins and pharmaceutical compositions
EP0420872A4 (en)	1992-10-21	Therapeutic uses of 2',5'-oligoadenylate derivatives
GB2177398B (en)	1989-05-04	5,6-epoxy-7-oxabicycloheptane substituted ethers useful in the treatment of thrombotic disease
IL78689A0 (en)	1986-08-31	Pharmaceutical compositions comprising dopamine agonists
CA1268468C (fr)	1990-05-01	Analogues des prostaglandines avec groupement thiabicycloheptane substitue
PT87563A (pt)	1989-05-31	Process for the preparation of vinylcephalosporins useful as medicaments
ZA887158B (en)	1989-05-30	Azachromane derivatives
AU4610689A (en)	1990-06-21	Pyridine-3-peroxycarboxylic acid monopersulfate
NZ228023A (en)	1991-10-25	24(r)-scymnol; preparatory processes and pharmaceutical compositions
DE3168544D1 (en)	1985-03-07	6,7,8,9-tetrahydro-3h-benz(e)indolamine derivatives, processes for their preparation and intermediates used therein, and pharmaceutical compositions containing the indolamine derivatives
GR3017335T3 (en)	1995-12-31	Oligophosphates with antiviral activity.
AU580646B2 (en)	1989-01-19	13``-alkyl-17``-(3-aceloxy-propyl)-gonane
GR850484B (fr)	1985-06-26
ZA881322B (en)	1988-08-23	Benzylaminoaryl-dihydropyridinelactones,process for their preparation,and their use in medicaments

Legal Events

Date	Code	Title
1999-01-26	KB	Patent renewed
2002-11-10	KB	Patent renewed
2006-10-30	KB	Patent renewed
2009-02-11	EXP	Patent expired
2010-04-14	EXP	Patent expired