ID19406A - Keaktifan anti bakterial yang memiliki ketolida 6-0-tersubstitusi - Google Patents
Keaktifan anti bakterial yang memiliki ketolida 6-0-tersubstitusiInfo
- Publication number
- ID19406A ID19406A IDP973095A ID973095A ID19406A ID 19406 A ID19406 A ID 19406A ID P973095 A IDP973095 A ID P973095A ID 973095 A ID973095 A ID 973095A ID 19406 A ID19406 A ID 19406A
- Authority
- ID
- Indonesia
- Prior art keywords
- alkyl
- substituted
- heteroaryl
- aryl
- optionally substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Saccharide Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Cephalosporin Compounds (AREA)
- Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US70777696A | 1996-09-04 | 1996-09-04 | |
US08/888,350 US5866549A (en) | 1996-09-04 | 1997-07-03 | 6-O-substituted ketolides having antibacterial activity |
Publications (1)
Publication Number | Publication Date |
---|---|
ID19406A true ID19406A (id) | 1998-07-09 |
Family
ID=27107953
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IDP973095A ID19406A (id) | 1996-09-04 | 1997-09-04 | Keaktifan anti bakterial yang memiliki ketolida 6-0-tersubstitusi |
Country Status (28)
Country | Link |
---|---|
US (4) | US6028181A (no) |
EP (5) | EP0929563B1 (no) |
JP (1) | JP4597274B2 (no) |
KR (5) | KR100576988B1 (no) |
CN (4) | CN100460415C (no) |
AT (5) | ATE296308T1 (no) |
BG (1) | BG63547B1 (no) |
BR (1) | BR9711661A (no) |
CA (1) | CA2263972C (no) |
CZ (1) | CZ300106B6 (no) |
DE (5) | DE69733723T2 (no) |
DK (5) | DK1291350T3 (no) |
ES (5) | ES2242811T3 (no) |
HK (1) | HK1021537A1 (no) |
HR (5) | HRP970473B1 (no) |
HU (1) | HU230166B1 (no) |
ID (1) | ID19406A (no) |
IL (1) | IL128681A0 (no) |
NO (1) | NO314230B1 (no) |
NZ (1) | NZ334274A (no) |
PL (1) | PL188173B1 (no) |
PT (5) | PT929563E (no) |
RO (1) | RO121473B1 (no) |
RU (1) | RU2192427C2 (no) |
SI (1) | SI20023B (no) |
SK (5) | SK285534B6 (no) |
TR (1) | TR199901127T2 (no) |
WO (1) | WO1998009978A1 (no) |
Families Citing this family (85)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6495348B1 (en) | 1993-10-07 | 2002-12-17 | Regents Of The University Of Minnesota | Mitomycin biosynthetic gene cluster |
UA51730C2 (uk) * | 1996-09-04 | 2002-12-16 | Ебботт Лабораторіз | 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців |
AP1060A (en) * | 1998-01-02 | 2002-04-23 | Pfizer Prod Inc | Novel erythromycin derivatives. |
DK0952157T3 (da) | 1998-04-24 | 2003-10-13 | Pfizer Prod Inc | 9a, 11b-dehydroderivater af 9-oxim-3-keto-6-0-methylerythromycin |
US6265202B1 (en) | 1998-06-26 | 2001-07-24 | Regents Of The University Of Minnesota | DNA encoding methymycin and pikromycin |
FR2780977B1 (fr) * | 1998-07-09 | 2000-09-01 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
FR2792637B1 (fr) * | 1999-04-26 | 2001-06-01 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
JP4573925B2 (ja) | 1998-07-09 | 2010-11-04 | アベンティス・ファーマ・ソシエテ・アノニム | 新規のエリスロマイシン誘導体、その製造方法及びその薬剤としての使用 |
FR2785612A1 (fr) * | 1998-11-10 | 2000-05-12 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
AU5995299A (en) * | 1998-11-03 | 2000-05-22 | Pfizer Products Inc. | Novel macrolide antibiotics |
ATE266036T1 (de) * | 1999-03-15 | 2004-05-15 | Abbott Lab | 6-o-substitutierte makroliden mit antibakterieller wirkung |
US6939861B2 (en) | 1999-04-16 | 2005-09-06 | Kosan Biosciences, Inc. | Amido macrolides |
US6451768B1 (en) | 1999-04-16 | 2002-09-17 | Kosan Biosciences, Inc. | Macrolide antiinfective agents |
DE60030847T2 (de) | 1999-04-16 | 2007-04-19 | Kosan Biosciences, Inc., Hayward | Antiinfektiöse makrolidderivate |
US6514944B2 (en) | 1999-04-16 | 2003-02-04 | Kosan Biosciences, Inc. | Macrolide antiinfective agents |
US6420535B1 (en) * | 1999-06-07 | 2002-07-16 | Abbott Laboratories | 6-O-carbamate ketolide derivatives |
ATE250076T1 (de) * | 1999-06-07 | 2003-10-15 | Abbott Lab | 6-o-carbamat ketolide derivate |
US6437106B1 (en) * | 1999-06-24 | 2002-08-20 | Abbott Laboratories | Process for preparing 6-o-substituted erythromycin derivatives |
US6417366B2 (en) * | 1999-06-24 | 2002-07-09 | Abbott Laboratories | Preparation of quinoline-substituted carbonate and carbamate derivatives |
EP1101769A3 (en) | 1999-11-18 | 2001-10-24 | Pfizer Products Inc. | Nitrogen containing erythromycin derivatives |
WO2003079972A2 (en) | 2002-02-22 | 2003-10-02 | New River Parmaceuticals Inc. | Active agent delivery systems and methods for protecting and administering active agents |
US6472372B1 (en) | 2000-12-06 | 2002-10-29 | Ortho-Mcneil Pharmaceuticals, Inc. | 6-O-Carbamoyl ketolide antibacterials |
CA2451391A1 (en) * | 2001-07-03 | 2003-01-16 | Chiron Corporation | C12 modified erythromycin macrolides and ketolides having antibacterial activity |
CN1589277A (zh) | 2001-09-17 | 2005-03-02 | 奥索-麦克尼尔药品公司 | 6-o-氨基甲酸酯-11,12-内酯-酮内酯抗菌剂 |
US6673774B2 (en) * | 2001-12-03 | 2004-01-06 | Enanta Pharmaceuticals, Inc. | 11-O-substituted macrolides and their descladinose derivatives |
WO2003050132A1 (en) | 2001-12-05 | 2003-06-19 | Ortho-Mcneil Pharmaceutical, Inc. | 6-o-acyl ketolide derivatives of erythromycine useful as antibacterials |
US6831068B2 (en) * | 2002-02-13 | 2004-12-14 | Abbott Laboratories | Macrolide antibacterial compounds |
US20030162729A1 (en) * | 2002-02-13 | 2003-08-28 | Zhenkun Ma | Macrolides with activity against methicillin-resistant staphylococcus aureus |
CA2476223A1 (en) * | 2002-02-13 | 2003-08-21 | Abbott Laboratories | Macrolide antibacterial compounds |
US6995143B2 (en) | 2002-02-28 | 2006-02-07 | Basilea Pharmaceutica Ag | Macrolides with antibacterial activity |
US7910558B2 (en) * | 2002-05-13 | 2011-03-22 | Enanta Pharmaceuticals, Inc. | Bridged macrocyclic compounds and processes for the preparation thereof |
US7273853B2 (en) * | 2002-05-13 | 2007-09-25 | Enanta Pharmaceuticals, Inc. | 6-11 bicyclic ketolide derivatives |
US6841664B2 (en) * | 2002-07-25 | 2005-01-11 | Enanra Pharmaceuticals, Inc. | 6,11-4-carbon bridged ketolides |
JP2005531603A (ja) * | 2002-05-31 | 2005-10-20 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | 3−デスクラジノシル−6−o−カルバモイルおよび6−o−カルボノイルマクロライド抗菌剤 |
WO2004078771A1 (ja) * | 2003-03-07 | 2004-09-16 | Taisho Pharmaceutical Co., Ltd. | 2-フルオロ-6-o-置換ケトライド誘導体 |
EP1638549A4 (en) * | 2003-03-10 | 2011-06-15 | Optimer Pharmaceuticals Inc | NEW ANTIBACTERIAL AGENTS |
CA2523541A1 (en) * | 2003-04-25 | 2004-11-11 | Chiron Corporation | Novel ketolide derivatives |
US6790835B1 (en) * | 2003-06-05 | 2004-09-14 | Enanta Pharmaceuticals, Inc. | Bicyclic macrolide derivatives |
US20040254126A1 (en) * | 2003-06-05 | 2004-12-16 | Yao-Ling Qiu | 11-12 Bicyclic erythromycin derivatives |
EP1670808A1 (en) * | 2003-09-12 | 2006-06-21 | Chiron Corporation | Antimicrobial derivatives |
GB0327720D0 (en) * | 2003-11-28 | 2003-12-31 | Biotica Tech Ltd | Erythromycins and process for their preparation |
US7414030B2 (en) * | 2004-01-07 | 2008-08-19 | Enanta Pharmaceuticals, Inc. | 6-11 Bicyclic erythromycin derivatives |
WO2005070113A2 (en) * | 2004-01-09 | 2005-08-04 | Enanta Pharmaceuticals, Inc. | 9n-substituted 6-11 bicyclic erythromycin derivatives |
US7384921B2 (en) * | 2004-02-20 | 2008-06-10 | Enanta Pharmaceuticals, Inc. | Polymorphic forms of 6-11 bicyclic ketolide derivatives |
FR2874922A1 (fr) * | 2004-07-30 | 2006-03-10 | Palumed Sa | Molecules hybrides qa ou q est une aminoquinoleine et a est un residu antibiotique, leur synthese et leurs utilisations en tant qu'agent antibacterien |
WO2006024741A2 (fr) * | 2004-07-30 | 2006-03-09 | Palumed S.A. | Molecules hybrides qa ou q est une aminoquinoleine et a est un residu antibiotique, leur synthese et leurs utilisations en tant qu'agent antibacterien |
WO2006065743A2 (en) * | 2004-12-13 | 2006-06-22 | Enanta Pharmaceuticals, Inc. | Tetracylic bicyclolides |
GEP20094834B (en) | 2004-12-21 | 2009-11-25 | Pfizer Prod Inc | Macrolides, pharmaceutical compositions containing them and their use for treatment of bacterial infections |
US20060252710A1 (en) * | 2005-05-04 | 2006-11-09 | Guoqiang Wang | 6-11 Bridged oxime erythromycin derivatives |
US7517859B2 (en) * | 2005-05-04 | 2009-04-14 | Enanta Pharmaceuticals, Inc. | Spirocyclic bicyclolides |
US7384922B2 (en) * | 2005-05-04 | 2008-06-10 | Enanta Pharmaceuticals, Inc. | 6-11 bridged oxime erythromycin derivatives |
EP1985620A4 (en) | 2006-02-07 | 2012-08-15 | Taisho Pharmaceutical Co Ltd | COMPOUND 10a-AZALIDE |
JP2010501541A (ja) | 2006-08-24 | 2010-01-21 | ウォックハート リサーチ センター | 抗菌活性を有する新規マクロライド及びケトライド |
JPWO2009019868A1 (ja) | 2007-08-06 | 2010-10-28 | 大正製薬株式会社 | 10a、12位架橋型10a−アザライド化合物 |
KR101223158B1 (ko) * | 2007-09-17 | 2013-01-17 | 이난타 파마슈티칼스, 인코포레이티드 | 6,11-다리걸친 바이아릴 매크로라이드 |
US8354383B2 (en) * | 2007-09-17 | 2013-01-15 | Enanta Pharmaceuticals, Inc. | 6,11-bridged biaryl macrolides |
US8273720B2 (en) * | 2007-09-17 | 2012-09-25 | Enanta Pharmaceuticals, Inc. | 6,11-bicyclolides: bridged biaryl macrolide derivatives |
EP2214484A4 (en) * | 2007-10-25 | 2013-01-02 | Cempra Pharmaceuticals Inc | PROCESS FOR PREPARING ANTIBACTERIAL MAKROLIDE AGENTS |
TW200946109A (en) * | 2008-05-09 | 2009-11-16 | Enanta Pharm Inc | Anti-bacterial activity of 9-hydroxy derivatives 6, 11-bicyclolides |
JPWO2009139181A1 (ja) | 2008-05-15 | 2011-09-15 | 大正製薬株式会社 | 4員環構造を有する10a−アザライド化合物 |
AU2009308181B2 (en) | 2008-10-24 | 2015-12-03 | Cempra Pharmaceuticals, Inc. | Methods for treating resistant diseases using triazole containing macrolides |
WO2010136971A1 (en) | 2009-05-27 | 2010-12-02 | Wockhardt Research Centre | Ketolide compounds having antimicrobial activity |
US9937194B1 (en) | 2009-06-12 | 2018-04-10 | Cempra Pharmaceuticals, Inc. | Compounds and methods for treating inflammatory diseases |
JP5914335B2 (ja) | 2009-09-10 | 2016-05-11 | センプラ ファーマシューティカルズ,インコーポレイテッド | マラリア、結核、及びmac病の治療方法 |
RU2650883C2 (ru) | 2010-03-22 | 2018-04-18 | Семпра Фармасьютикалз, Инк. | Кристаллические формы макролида и их применение |
DK2571506T3 (en) | 2010-05-20 | 2017-08-28 | Cempra Pharmaceuticals Inc | PROCEDURES FOR THE MANUFACTURE OF MACROLIDES AND KETOLIDES AND INTERMEDIATES |
US8796474B1 (en) | 2010-08-23 | 2014-08-05 | Rutgers, The State University Of New Jersey | Macrolide compounds and methods and intermediates useful for their preparation |
EP2613630A4 (en) | 2010-09-10 | 2014-01-15 | Cempra Pharmaceuticals Inc | FLUOROCETOLIDES FORMING HYDROGEN LINKS TO TREAT DISEASES |
RU2601550C2 (ru) | 2010-12-09 | 2016-11-10 | Вокхардт Лимитед | Кетолидные соединения |
AR085286A1 (es) * | 2011-02-21 | 2013-09-18 | Taisho Pharmaceutical Co Ltd | Derivado de macrolido sustituido en la posicion c-4 |
JP5718488B2 (ja) | 2011-03-01 | 2015-05-13 | ウォックハート リミテッド | ケトライド中間体の調製方法 |
EP2688900B1 (en) | 2011-03-22 | 2016-09-28 | Wockhardt Limited | Process for preparation of ketolide compounds |
CN102766089A (zh) * | 2011-05-06 | 2012-11-07 | 上海医药工业研究院 | 3-(3-喹啉基)-2-丙烯-1-卤代物及其制备方法 |
CN102766181A (zh) * | 2011-05-06 | 2012-11-07 | 上海医药工业研究院 | 6-o-取代的红霉素衍生物的制备方法 |
MX2014011537A (es) * | 2012-03-27 | 2015-02-10 | Cempra Pharmaceuticals Inc | Formulaciones parenterales para la administracion de antibioticos macrolidos. |
JP5857008B2 (ja) * | 2012-08-20 | 2016-02-10 | 大正製薬株式会社 | C−4”位置換マクロライド誘導体を含有する医薬 |
GB201217310D0 (en) | 2012-09-27 | 2012-11-14 | C10 Pharma As | Compounds |
CA2905975A1 (en) | 2013-03-14 | 2014-09-25 | Cempra Pharmaceuticals, Inc. | Methods for treating respiratory diseases and formulations therefor |
EP2968384A4 (en) | 2013-03-15 | 2017-02-15 | Cempra Pharmaceuticals, Inc. | Convergent processes for preparing macrolide antibacterial agents |
AR102810A1 (es) | 2014-08-18 | 2017-03-29 | Taisho Pharmaceutical Co Ltd | Derivado de macrólido sustituido en la posición c-4 |
JP2019533669A (ja) * | 2016-10-04 | 2019-11-21 | バイオファーマティ ソシエテ アノニム | 抗菌活性を有するケトライド |
WO2018161039A1 (en) * | 2017-03-03 | 2018-09-07 | Synovo Gmbh | Novel anti-infective and anti-inflammatory compounds |
CN109942653B (zh) * | 2019-02-27 | 2021-06-25 | 北京理工大学 | 一种红霉素衍生物及其制备方法 |
EP4069251A4 (en) * | 2019-12-02 | 2023-12-06 | Aliquantumrx, Inc. | CETHROMYCIN SALTS AND POLYMORPHS FOR THE TREATMENT OF CETHROMYCIN SALTS AND POLYMORPHS |
CN113817008B (zh) * | 2021-07-15 | 2023-05-23 | 湖州师范学院 | 新型琥珀酰基十六元大环内酯的制备方法及用途 |
Family Cites Families (22)
Publication number | Priority date | Publication date | Assignee | Title |
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KR960000434B1 (ko) * | 1986-12-17 | 1996-01-06 | 다이쇼 세이야꾸 가부시끼가이샤 | 에리스로마이신 a유도체 및 그의 제조 방법 |
WO1992006991A1 (fr) * | 1990-10-15 | 1992-04-30 | Taisho Pharmaceutical Co., Ltd. | Erythromycine modifiee en 2' ou derive de cette substance |
IL99995A (en) * | 1990-11-21 | 1997-11-20 | Roussel Uclaf | Erythromycin derivatives, their preparation and pharmaceutical compositions containing them |
KR0166096B1 (ko) * | 1990-11-28 | 1999-01-15 | 우에하라 아키라 | 6-0-메틸에리쓰로마이신 a 유도체 |
WO1993013663A1 (en) * | 1992-01-17 | 1993-07-22 | Abbott Laboratories | Method of directing biosynthesis of specific polyketides |
US5523399A (en) * | 1991-12-27 | 1996-06-04 | Taisho Pharmaceutical Co., Ltd. | 5-O-desosaminylerythronolide derivatives |
CA2093303C (en) * | 1992-04-09 | 1998-11-24 | Abraham Araya | Aluminosilicates |
EP0638584B1 (en) * | 1992-04-22 | 1996-03-20 | Taisho Pharmaceutical Co. Ltd | 5-o-desosaminylerythronolide a derivative |
FR2697524B1 (fr) * | 1992-11-05 | 1994-12-23 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
US5527780A (en) * | 1992-11-05 | 1996-06-18 | Roussel Uclaf | Erythromycin derivatives |
FR2702480B1 (fr) * | 1993-03-09 | 1995-04-28 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
FR2713226B1 (fr) * | 1993-12-03 | 1996-01-05 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
FR2718450B1 (fr) * | 1994-04-08 | 1997-01-10 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
FR2719587B1 (fr) * | 1994-05-03 | 1996-07-12 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
FR2732023B1 (fr) * | 1995-03-22 | 1997-04-30 | Roussel Uclaf | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
FR2732684B1 (fr) * | 1995-04-06 | 1997-04-30 | Roussel Uclaf | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
FR2738571B1 (fr) * | 1995-09-11 | 1997-10-17 | Roussel Uclaf | Nouveaux derives de la 5-0-desosaminyl 6-0-methyl- erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs |
ES2218604T3 (es) * | 1995-11-08 | 2004-11-16 | Abbott Laboratories | Derivados triciclicos de eritromicina. |
US6274715B1 (en) * | 1995-11-08 | 2001-08-14 | Abbott Laboratories | Tricyclic erythromycin derivatives |
UA51730C2 (uk) * | 1996-09-04 | 2002-12-16 | Ебботт Лабораторіз | 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців |
AU4472797A (en) * | 1996-10-31 | 1998-05-22 | Taisho Pharmaceutical Co., Ltd. | Erythromycin a derivatives |
US6171807B1 (en) * | 1996-11-13 | 2001-01-09 | Associates Of Cape Cod, Inc. | Detection and quantitation of endotoxin by fluorescence polarization |
-
1997
- 1997-09-02 RU RU99106778/04A patent/RU2192427C2/ru active
- 1997-09-02 KR KR1020057007117A patent/KR100576988B1/ko not_active IP Right Cessation
- 1997-09-02 EP EP97939765A patent/EP0929563B1/en not_active Expired - Lifetime
- 1997-09-02 PT PT97939765T patent/PT929563E/pt unknown
- 1997-09-02 DE DE69733723T patent/DE69733723T2/de not_active Expired - Lifetime
- 1997-09-02 AT AT02024559T patent/ATE296308T1/de active
- 1997-09-02 ES ES02024557T patent/ES2242811T3/es not_active Expired - Lifetime
- 1997-09-02 RO RO99-00228A patent/RO121473B1/ro unknown
- 1997-09-02 SK SK5083-2006A patent/SK285534B6/sk not_active IP Right Cessation
- 1997-09-02 CN CNB2005100674132A patent/CN100460415C/zh not_active Expired - Lifetime
- 1997-09-02 ES ES02024559T patent/ES2242812T3/es not_active Expired - Lifetime
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- 1997-09-02 KR KR1020057007118A patent/KR20050044816A/ko not_active Application Discontinuation
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- 1997-09-02 CN CNA2005100674147A patent/CN1680419A/zh active Pending
- 1997-09-02 DK DK02024559T patent/DK1291352T3/da active
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1998
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1999
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2000
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2004
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2006
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